| P21567 |
BXGT008664 |
Alpha-amylase |
reviewed |
- |
ALP1 |
Inhibition |
'=' |
96 |
% |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
Inhibition |
'=' |
41 |
% |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
Ki |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
IC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
Ki |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
IC50 |
- |
- |
- |
| P21567 |
BXGT008664 |
Alpha-amylase |
reviewed |
- |
ALP1 |
Inhibition |
'=' |
95 |
% |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
Ki |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
'=' |
58 |
% |
| Q5E985 |
BXGT015338 |
Hyaluronidase-1 |
reviewed |
- |
HYAL1 |
Inhibition |
- |
- |
- |
| Q8SQG8 |
BXGT018758 |
Hyaluronidase-2 |
reviewed |
- |
HYAL2 |
Inhibition |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
Ki |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
IC50 |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
Ki |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
Ki |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
IC50 |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
IC50 |
- |
- |
- |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
Ki |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
IC50 |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Ki |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
IC50 |
- |
- |
- |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
96 |
% |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Ki |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
IC50 |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
IC50 |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
IC50 |
- |
- |
- |
| P21398 |
BXGT008645 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Activity |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
IC50 |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
IC50 |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
- |
- |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
IC50 |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
IC50 |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
'=' |
55 |
% |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
Ki |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
Ki |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
Ki |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
Ki |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
IC50 |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
EC50 |
'=' |
0 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
IC50 |
- |
- |
- |
| Q9H6Z9 |
BXGT020488 |
Egl nine homolog 3 |
reviewed |
- |
EGLN3 |
Km |
'=' |
140000 |
nM |
| Q9NWT6 |
BXGT021234 |
Hypoxia-inducible factor 1-alpha inhibitor |
reviewed |
- |
HIF1AN |
Km |
'=' |
260000 |
nM |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
Ki |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
Ki |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
Ki |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ki |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
IC50 |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
IC50 |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
- |
- |
- |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
- |
- |
- |
| O14684 |
BXGT004082 |
Prostaglandin E synthase |
reviewed |
- |
PTGES |
IC50 |
- |
- |
- |
| P00689 |
BXGT005611 |
Pancreatic alpha-amylase |
reviewed |
- |
Amy2 |
IC50 |
'=' |
26500 |
nM |
| P00689 |
BXGT005611 |
Pancreatic alpha-amylase |
reviewed |
- |
Amy2 |
Ki |
'=' |
43400 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
84 |
% |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
IC50 |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
IC50 |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
IC50 |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
IC50 |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
- |
- |
- |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
IC50 |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
- |
- |
- |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
Inhibition |
'=' |
29 |
% |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
Ki |
- |
- |
- |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
Ki |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
Ki |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
IC50 |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
Ki |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Ki |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Ki |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
IC50 |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
Ki |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Ki |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Ki |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
IC50 |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
IC50 |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Ki |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
IC50 |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Ki |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Ki |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
Ki |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
IC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
IC50 |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
Ki |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
IC50 |
- |
- |
- |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
IC50 |
- |
- |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IC50 |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Ki |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
IC50 |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
- |
- |
- |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
Ki |
- |
- |
- |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
Ki |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Ki |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
- |
- |
- |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inactivation |
'=' |
50 |
% |
| P56560 |
BXGT011180 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Activity |
- |
- |
- |
| P00689 |
BXGT005611 |
Pancreatic alpha-amylase |
reviewed |
- |
Amy2 |
Inhibition |
'=' |
95 |
% |
| P04762 |
BXGT006259 |
Catalase |
reviewed |
- |
Cat |
EC50 |
'=' |
1 |
ug.mL-1 |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
Ki |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
IC50 |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
IC50 |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
- |
- |
- |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
Ki |
- |
- |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
Ki |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
'=' |
54 |
% |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Ki |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
Ki |
- |
- |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
- |
- |
- |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
Ki |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
Ki |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
IC50 |
- |
- |
- |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
IC50 |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
Ki |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
140000 |
nM |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
Ki |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
IC50 |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
Ki |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
Ki |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
- |
- |
- |
| Q9GZT9 |
BXGT020425 |
Egl nine homolog 1 |
reviewed |
- |
EGLN1 |
Km |
'=' |
180000 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
IC50 |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
Ki |
- |
- |
- |
| Q54873 |
BXGT015048 |
Hyaluronate lyase |
reviewed |
- |
SP_0314 |
IC50 |
'=' |
6000000 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
IC50 |
'=' |
32500 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Ki |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
Ki |
- |
- |
- |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
Ki |
- |
- |
- |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
IC50 |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
| P04746 |
BXGT006256 |
Pancreatic alpha-amylase |
reviewed |
- |
AMY2A |
Inhibition |
'=' |
100 |
% |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
IC50 |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
- |
- |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
- |
- |
- |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
Ki |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
IC50 |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
IC50 |
- |
- |
- |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Inhibition |
'=' |
85 |
% |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
100 |
% |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Ki |
- |
- |
- |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
Ki |
- |
- |
- |
| Q96KS0 |
BXGT019688 |
Egl nine homolog 2 |
reviewed |
- |
EGLN2 |
Km |
'=' |
170000 |
nM |
| P13674 |
BXGT007942 |
Prolyl 4-hydroxylase subunit alpha-1 |
reviewed |
- |
P4HA1 |
Km |
'=' |
300000 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
'=' |
58 |
% |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
IC50 |
- |
- |
- |
| P22985 |
BXGT008824 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
Xdh |
IC50 |
- |
- |
- |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Activity |
'=' |
75 |
% |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
IC50 |
- |
- |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IC50 |
- |
- |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
- |
- |
- |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Inhibition |
'=' |
75 |
% |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
- |
- |
- |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
IC50 |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ki |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
IC50 |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
Ki |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ki |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
IC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
IC50 |
- |
- |
- |
| P02769 |
BXGT005956 |
Serum albumin |
reviewed |
- |
ALB |
IC50 |
'=' |
155380 |
nM |
| Q29550 |
BXGT013978 |
Liver carboxylesterase |
reviewed |
- |
|
IC50 |
- |
- |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
Ki |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
IC50 |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
IC50 |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IC50 |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
Ki |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
IC50 |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Activity |
- |
- |
- |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Inhibition |
'=' |
80 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
IC50 |
- |
- |
- |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
IC50 |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
IC50 |
- |
- |
- |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
- |
- |
- |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Ki |
- |
- |
- |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Inhibition |
'=' |
50 |
% |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
'=' |
50 |
% |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
Ki |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
144000 |
nM |
| Q6P7A9 |
BXGT016460 |
Lysosomal alpha-glucosidase |
reviewed |
- |
Gaa |
IC50 |
- |
- |
- |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
Activity |
'=' |
83 |
% |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
IC50 |
- |
- |
- |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
3 |
% |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Activity |
'=' |
8 |
% |