| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
84921 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
39810 |
nM |
| Q6W5P4 |
BXGT016588 |
Neuropeptide S receptor |
reviewed |
- |
NPSR1 |
Potency |
'=' |
31622 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
35481 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Kd |
'=' |
40700 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
19952 |
nM |
| P22460 |
BXGT008774 |
Potassium voltage-gated channel subfamily A member 5 |
reviewed |
Ion channel |
KCNA5 |
IC50 |
- |
- |
- |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
IC50 |
'=' |
125000 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
707 |
nM |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
279000 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
7568 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
23934 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
12589 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Activity |
- |
- |
- |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Activity |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ke |
'=' |
1180 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
28183 |
nM |
| P06278 |
BXGT006431 |
Alpha-amylase |
reviewed |
- |
amyS |
Activity |
- |
- |
- |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
RU |
'=' |
717 |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
80000 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
4744 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
79432 |
nM |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
183000 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'>' |
30000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
25118 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
93300 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
72 |
% |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
39810 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
28183 |
nM |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ke |
'=' |
320 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
Activity |
- |
- |
- |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'=' |
546000 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
IC50 |
'=' |
310000 |
nM |
| P24298 |
BXGT008960 |
Alanine aminotransferase 1 |
reviewed |
Enzyme |
GPT |
Activity |
'=' |
103 |
U/L |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
Activity |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
36700 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Activity |
- |
- |
- |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
15848 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Activity |
- |
- |
- |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
11220 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
4100 |
nM |
| P61823 |
BXGT011385 |
Ribonuclease pancreatic |
reviewed |
- |
RNASE1 |
Inhibition |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Inhibition |
'=' |
38 |
% |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| P16098 |
BXGT008191 |
Beta-amylase |
reviewed |
- |
BMY1 |
Activity |
- |
- |
- |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'=' |
5910000 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'>' |
100000 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
28183 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
Ki |
'=' |
600 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
28183 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
28183 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
20200 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Activity |
'=' |
7 |
% |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ke |
'>' |
10000 |
nM |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
80000 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
130000 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
14125 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
92 |
% |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
37685 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
37685 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
Inhibition |
'=' |
79 |
% |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Kd |
'=' |
49200 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
IC50 |
'=' |
1700 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Ka |
'=' |
2 |
10'4/M |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'>' |
300000 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
- |
- |
- |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
Inhibition |
'=' |
52 |
% |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
98300 |
nM |
| Q02127 |
BXGT012635 |
Dihydroorotate dehydrogenase (quinone), mitochondrial |
reviewed |
Enzyme |
DHODH |
Inhibition |
'=' |
38 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
- |
- |
- |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
100000 |
nM |