Showing entry for 4-Aminobutyric acid


　 　 　 　 　 　 　 　 　 　 　 　 　 　 　
General Compound Information
BXGC IdBXGC0004665
Compound Name4-Aminobutyric acid
Structure
FormulaC4H9NO2
InchiKeyBTCSSZJGUNDROE-UHFFFAOYSA-N
SMILESNCCCC(O)=O
InchiInChI=1S/C4H9NO2/c5-3-1-2-4(6)7/h1-3,5H2,(H,6,7)
IUPAC4-aminobutanoic acid
Molecular Weight103.12
Pubchem Id119
Chembl IdCHEMBL96
Targets of Information Source
DrugBank DB02530
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
P50440 BXGT010798 Glycine amidinotransferase, mitochondrial reviewed - GATM approved; investigational -
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 approved; investigational -
O75899 BXGT005161 Gamma-aminobutyric acid type B receptor subunit 2 reviewed G-protein coupled receptor GABBR2 approved; investigational -
PDB ABU
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Q99259 BXGT019915 Glutamate decarboxylase 1 reviewed GAD1 Enzyme - - - -
Q05329 BXGT012814 Glutamate decarboxylase 2 reviewed GAD2 Enzyme - - - -
P0C7B7 BXGT007447 Cys-loop ligand-gated ion channel reviewed - - - - -
Q7CX36 BXGT016948 ABC transporter, substrate binding protein (Amino acid) unreviewed Atu2422 - - - 2400 -
H2L2M6 BXGT003590 Lectin Alpha chain unreviewed - - - - -
P24627 BXGT008981 Lactotransferrin reviewed LTF - - - - -
A1R958 BXGT001033 4-aminobutyrate transaminase unreviewed gabT - - - - -
A9CGA5 BXGT001743 ABC transporter, substrate binding protein (Polyamine) unreviewed Atu4243 - - - - -
P81460 BXGT011951 Concanavalin-A reviewed - - - - -
Q6EDY6 BXGT016266 F-actin-uncapping protein LRRC16A reviewed Carmil1 - - - - -
H2L2M7 BXGT003591 Lectin Beta Chain unreviewed - - - - -
P86352 BXGT012089 Seed lectin alpha chain reviewed - - - - -
P86353 BXGT012090 Seed lectin beta chain reviewed - - - - -
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed GABBR1 G-protein coupled receptor - - - -
P55915 BXGT011133 Concanavalin-Br reviewed - - - - -
D1C7D8 BXGT002809 Pyridoxal-dependent decarboxylase unreviewed Sthe_2364 - - - - -
P0CG47 BXGT007467 Polyubiquitin-B reviewed UBB Nucleic acid binding - - - -
Q9HW93 BXGT020631 Methyl-accepting chemotaxis protein PctC reviewed pctC - - - - -
P94426 BXGT012133 HTH-type transcriptional regulatory protein GabR reviewed gabR - - - - -
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed GABRB3 Ion channel - - - -
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed GABRB2 Ion channel - - - -
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Gabra1 - - - - -
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Gabrb1 - - - - -
P50440 BXGT010798 Glycine amidinotransferase, mitochondrial reviewed GATM - - - - -
Binding DB 24183
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT010049 Heat shock factor protein 1 reviewed Hsf1 - - - >195000
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 >10000 - - -
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 38 - - -
reviewed BXGT021402 Sigma non-opioid intracellular receptor 1 reviewed Sigmar1 >10000 - - -
reviewed BXGT008440 D(1A) dopamine receptor reviewed Drd1 >10000 - - -
reviewed BXGT011367 D(2) dopamine receptor reviewed Drd2 >10000 - - -
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 33 - - -
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 77.62 - - -
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 57.54 - - -
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 21.37 - - -
reviewed BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 22.9 - - -
reviewed BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 50.11 - - -
reviewed BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 8.7 - - -
reviewed BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 77.62 - - -
reviewed BXGT001712 Gamma-aminobutyric acid receptor subunit rho-3 reviewed Ion channel GABRR3 580 - - -
reviewed BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Gabrg1 - 33 - -
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 - 40 - -
reviewed BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Gabra2 - 22 - -
reviewed BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 - 25 - -
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 - 17 - -
reviewed BXGT010618 Sodium- and chloride-dependent GABA transporter 3 reviewed Transporter SLC6A11 - 7000 - -
reviewed BXGT009432 Sodium- and chloride-dependent GABA transporter 1 reviewed Transporter SLC6A1 - 5000 - -
reviewed BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed Slc6a13 - 5000 - -
reviewed BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 - 36000 - -
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 - - - 43000
reviewed BXGT009563 Sodium- and chloride-dependent GABA transporter 3 reviewed Slc6a11 - 8128 - -
reviewed BXGT009561 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 7244 - -
reviewed BXGT009562 Sodium- and chloride-dependent GABA transporter 2 reviewed Slc6a13 - 27542 - -
reviewed BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 - - - 28000
reviewed BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 - - - 3000
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 - - - 80000
reviewed BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 - - - 1500
reviewed BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 - - - 40000
reviewed BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 - - - 50000
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 - - - 1800
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 - - - 1778
reviewed BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 - - - 270
reviewed BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 - - - 269
reviewed BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 - - - 650
reviewed BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 - - - 661
reviewed BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 - - - 920
reviewed BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 - - - 912
reviewed BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 - - - 51000
reviewed BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 - - - 800
reviewed BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 - - - 1700
reviewed BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Gabra1 - - - 10000
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 - 60 - -
reviewed BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed Slc6a13 - 2000 - -
reviewed BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed Slc6a13 - 3000 - -
reviewed BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed Gabbr1 - 30 - -
reviewed BXGT017247 Proton-coupled amino acid transporter 1 reviewed Transporter SLC36A1 4000000 - - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 1620 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 1790 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2750 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 1830 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2120 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2600 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2500 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 1800 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2880 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2150 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 1970 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2640 - -
reviewed BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 2730 - -
reviewed BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 - - - 1190
reviewed BXGT009561 Sodium- and chloride-dependent GABA transporter 1 reviewed Slc6a1 - 5000 - -
reviewed BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 - - - 530
reviewed BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 - - - 1000
CHEMBL CHEMBL96
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 100 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 100 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 100 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 100 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 100 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 100 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 100 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 100 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 100 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 100 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 100 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 100 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 100 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 100 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 100 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 100 nM
P48056 BXGT010613 Sodium- and chloride-dependent betaine transporter reviewed - Slc6a12 Inhibition '=' 95 %
P31646 BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 Inhibition '=' 95 %
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 Inhibition '=' 95 %
P31647 BXGT009560 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 Inhibition '=' 95 %
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 AC50 - - -
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 EC '=' 24 -
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 EC '=' 24 -
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 EC '=' 24 -
P38532 BXGT010049 Heat shock factor protein 1 reviewed - Hsf1 EC50 '>' 195000 nM
P10828 BXGT007624 Thyroid hormone receptor beta reviewed Nuclear receptor THRB Potency '=' 19952 nM
Q05BR4 BXGT012851 SLC16A10 protein unreviewed - SLC16A10 Activity - - -
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2120 nM
P12392 BXGT007812 Neuronal acetylcholine receptor subunit beta-4 reviewed - Chrnb4 EC50 - - -
P04757 BXGT006258 Neuronal acetylcholine receptor subunit alpha-3 reviewed - Chrna3 EC50 - - -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Relative affinity '=' 1 -
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Relative affinity '=' 1 -
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Relative affinity '=' 1 -
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Relative affinity '=' 1 -
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Relative affinity '=' 1 -
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Relative affinity '=' 1 -
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Relative affinity '=' 1 -
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Relative affinity '=' 1 -
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Relative affinity '=' 1 -
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Relative affinity '=' 1 -
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Relative affinity '=' 1 -
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Relative affinity '=' 1 -
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Relative affinity '=' 1 -
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Relative affinity '=' 1 -
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Relative affinity '=' 1 -
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Relative affinity '=' 1 -
P30531 BXGT009432 Sodium- and chloride-dependent GABA transporter 1 reviewed Transporter SLC6A1 IC50 '=' 5000 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 33 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 33 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 33 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 33 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 33 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 33 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 33 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 33 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 33 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 33 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 33 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 33 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 33 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 33 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 33 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 33 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 22 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 EC50 '=' 269 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 EC '=' 25 -
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 EC '=' 25 -
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 EC '=' 25 -
Q7Z2H8 BXGT017247 Proton-coupled amino acid transporter 1 reviewed Transporter SLC36A1 pKi '=' 0 mM
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 AC50 - - -
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT Km '=' 2500000 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 80000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 80000 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 80000 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 EC '=' 22 -
P31650 BXGT009563 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 IC50 '=' 8128 nM
O88871 BXGT005286 Gamma-aminobutyric acid type B receptor subunit 2 reviewed - Gabbr2 IC50 '=' 17 nM
Q9Z0U4 BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed - Gabbr1 IC50 '=' 17 nM
O75899 BXGT005161 Gamma-aminobutyric acid type B receptor subunit 2 reviewed G-protein coupled receptor GABBR2 Inhibition - - -
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 Inhibition - - -
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 Activity '=' 82 %
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 Activity '=' 82 %
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 Activity '=' 82 %
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE Activity '=' 82 %
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 Activity '=' 82 %
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 Activity '=' 82 %
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD Activity '=' 82 %
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP Activity '=' 82 %
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 Activity '=' 82 %
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ Activity '=' 82 %
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 Activity '=' 82 %
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 Activity '=' 82 %
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 Activity '=' 82 %
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 Activity '=' 82 %
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 Activity '=' 82 %
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 Activity '=' 82 %
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 EC50 '=' 1700 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 EC '=' 22 -
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 EC '=' 22 -
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 EC '=' 22 -
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 EC50 '=' 10000 nM
P02545 BXGT005889 Prelamin-A/C reviewed - LMNA Potency '=' 5623 nM
O88871 BXGT005286 Gamma-aminobutyric acid type B receptor subunit 2 reviewed - Gabbr2 IC50 '=' 30 nM
Q9Z0U4 BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed - Gabbr1 IC50 '=' 30 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Ki '=' 25 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Ki '=' 25 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Ki '=' 25 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Ki '=' 25 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Ki '=' 25 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Ki '=' 25 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Ki '=' 25 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Ki '=' 25 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Ki '=' 25 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Ki '=' 25 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Ki '=' 25 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Ki '=' 25 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Ki '=' 25 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Ki '=' 25 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Ki '=' 25 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Ki '=' 25 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 Max '=' 100 -
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 Max '=' 100 -
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 Max '=' 100 -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 30 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 30 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 30 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 30 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 30 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 30 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 30 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 30 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 30 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 30 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 30 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 30 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 30 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 30 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 30 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 30 nM
O88871 BXGT005286 Gamma-aminobutyric acid type B receptor subunit 2 reviewed - Gabbr2 IC50 '=' 40 nM
Q9Z0U4 BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed - Gabbr1 IC50 '=' 40 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 EC '=' 20 -
P16305 BXGT008215 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 EC50 '=' 14300 nM
P27681 BXGT009196 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 EC50 '=' 14300 nM
P63080 BXGT011492 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 EC50 '=' 14300 nM
Q9D6F4 BXGT020259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 EC50 '=' 14300 nM
P22933 BXGT008819 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd EC50 '=' 14300 nM
P26049 BXGT009086 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 EC50 '=' 14300 nM
Q9JLF1 BXGT020834 Gamma-aminobutyric acid receptor subunit theta reviewed - Gabrq EC50 '=' 14300 nM
P62812 BXGT011459 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 EC50 '=' 14300 nM
A2AMW3 BXGT001075 Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon unreviewed - Gabre EC50 '=' 14300 nM
P22723 BXGT008798 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 EC50 '=' 14300 nM
Q9R0Y8 BXGT021410 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 EC50 '=' 14300 nM
P50571 BXGT010810 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 EC50 '=' 14300 nM
Q8QZW7 BXGT018675 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp EC50 '=' 14300 nM
P26048 BXGT009085 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 EC50 '=' 14300 nM
Q8BHJ7 BXGT017911 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 EC50 '=' 14300 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 1800 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2730 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 logEC50 '=' 1 -
P49798 BXGT010745 Regulator of G-protein signaling 4 reviewed Enzyme modulator RGS4 Potency - 376 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 logEC50 '=' 1 -
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 logEC50 '=' 1 -
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 logEC50 '=' 1 -
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 AC50 - - -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 13 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 13 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 13 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 13 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 13 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 13 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 13 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 13 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 13 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 13 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 13 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 13 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 13 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 13 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 13 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 13 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 EC '=' 25 -
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT Kcat '=' 49 /min
O89049 BXGT005293 Thioredoxin reductase 1, cytoplasmic reviewed - Txnrd1 Potency - 19952 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2750 nM
Q9UIF8 BXGT021718 Bromodomain adjacent to zinc finger domain protein 2B reviewed - BAZ2B Potency - 631 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 650 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 650 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 650 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 28183 nM
O88871 BXGT005286 Gamma-aminobutyric acid type B receptor subunit 2 reviewed - Gabbr2 Displacement '=' 100 %
Q9Z0U4 BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed - Gabbr1 Displacement '=' 100 %
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 1830 nM
P05177 BXGT006336 Cytochrome P450 1A2 reviewed Enzyme CYP1A2 AC50 '=' 31622 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 660 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 660 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 660 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 1778 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 1778 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 1778 nM
P48056 BXGT010613 Sodium- and chloride-dependent betaine transporter reviewed - Slc6a12 IC50 '=' 3000 nM
P31646 BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 IC50 '=' 3000 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 3000 nM
P31647 BXGT009560 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 IC50 '=' 3000 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 Kd '=' 1700 nM
A8MPY1 BXGT001712 Gamma-aminobutyric acid receptor subunit rho-3 reviewed Ion channel GABRR3 Kd '=' 1700 nM
P28476 BXGT009262 Gamma-aminobutyric acid receptor subunit rho-2 reviewed Ion channel GABRR2 Kd '=' 1700 nM
P23415 BXGT008864 Glycine receptor subunit alpha-1 reviewed Ion channel GLRA1 EC50 - - -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 20 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 20 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 20 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 20 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 20 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 20 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 20 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 20 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 20 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 20 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 20 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 20 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 20 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 20 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 20 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 20 nM
P02791 BXGT005965 Ferritin light chain reviewed - FTL Potency '=' 316 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 EC50 '=' 1000 nM
P48056 BXGT010613 Sodium- and chloride-dependent betaine transporter reviewed - Slc6a12 IC50 '=' 2000 nM
P31646 BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 IC50 '=' 2000 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2000 nM
P31647 BXGT009560 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 IC50 '=' 2000 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 IC50 '=' 25 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 IC50 '=' 25 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 IC50 '=' 25 nM
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE IC50 '=' 25 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 IC50 '=' 25 nM
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 IC50 '=' 25 nM
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD IC50 '=' 25 nM
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP IC50 '=' 25 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 IC50 '=' 25 nM
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ IC50 '=' 25 nM
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 IC50 '=' 25 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 IC50 '=' 25 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 IC50 '=' 25 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 IC50 '=' 25 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 IC50 '=' 25 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 IC50 '=' 25 nM
Q6W5P4 BXGT016588 Neuropeptide S receptor reviewed - NPSR1 Potency '=' 31622 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 Max '=' 100 -
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 EC50 '=' 1500 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 1500 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 1500 nM
P31646 BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 IC50 '=' 5000 nM
P48066 BXGT010618 Sodium- and chloride-dependent GABA transporter 3 reviewed Transporter SLC6A11 IC50 '=' 7000 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2150 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 IC50 '=' 1450 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 IC50 '=' 1450 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 IC50 '=' 1450 nM
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE IC50 '=' 1450 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 IC50 '=' 1450 nM
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 IC50 '=' 1450 nM
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD IC50 '=' 1450 nM
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP IC50 '=' 1450 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 IC50 '=' 1450 nM
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ IC50 '=' 1450 nM
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 IC50 '=' 1450 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 IC50 '=' 1450 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 IC50 '=' 1450 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 IC50 '=' 1450 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 IC50 '=' 1450 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 IC50 '=' 1450 nM
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT Km '=' 1300000 nM
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT Kcat/Km '=' 38 /min/mM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Potency - 4109 nM
Q03164 BXGT012700 Histone-lysine N-methyltransferase 2A reviewed - KMT2A Potency '=' 79 nM
P54132 BXGT011032 Bloom syndrome protein reviewed - BLM Potency '=' 3 nM
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 36000 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 1790 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 1620 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 EC50 '=' 43000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 43000 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 43000 nM
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 39000 nM
P30531 BXGT009432 Sodium- and chloride-dependent GABA transporter 1 reviewed Transporter SLC6A1 IC50 '=' 3311 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Ki '=' 49 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Ki '=' 49 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Ki '=' 49 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Ki '=' 49 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Ki '=' 49 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Ki '=' 49 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Ki '=' 49 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Ki '=' 49 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Ki '=' 49 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Ki '=' 49 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Ki '=' 49 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Ki '=' 49 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Ki '=' 49 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Ki '=' 49 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Ki '=' 49 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Ki '=' 49 nM
P48056 BXGT010613 Sodium- and chloride-dependent betaine transporter reviewed - Slc6a12 Inhibition '=' 61 %
P31646 BXGT009559 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 Inhibition '=' 61 %
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 Inhibition '=' 61 %
P31647 BXGT009560 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 Inhibition '=' 61 %
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 9000 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 50000 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 50000 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 50000 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 50000 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 50000 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 50000 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 50000 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 50000 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 50000 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 50000 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 50000 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 50000 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 50000 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 50000 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 50000 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 50000 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 29 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 29 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 29 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 29 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 29 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 29 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 29 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 29 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 29 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 29 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 29 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 29 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 29 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 29 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 29 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 29 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 2377 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 EC50 '=' 2300 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 EC50 '=' 2300 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 EC50 '=' 2300 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 Max '=' 100 -
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT k cat '=' 49 min-1
P36544 BXGT009926 Neuronal acetylcholine receptor subunit alpha-7 reviewed - CHRNA7 EC50 - - -
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 40000 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 40000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 40000 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 920 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 920 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 920 nM
Q92830 BXGT019379 Histone acetyltransferase KAT2A reviewed - KAT2A Potency - 39810 nM
O75899 BXGT005161 Gamma-aminobutyric acid type B receptor subunit 2 reviewed G-protein coupled receptor GABBR2 IC50 '=' 25 nM
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 IC50 '=' 25 nM
P30531 BXGT009432 Sodium- and chloride-dependent GABA transporter 1 reviewed Transporter SLC6A1 IC50 '=' 3000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 logEC50 '=' 1 -
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 logEC50 '=' 1 -
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 logEC50 '=' 1 -
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 EC50 '=' 21100 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 EC50 '=' 21100 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 21100 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 EC50 '=' 21100 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 21100 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 EC50 '=' 21100 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 21100 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 21100 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 21100 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 128 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 128 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 128 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 128 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 128 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 128 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 128 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 128 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 128 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 128 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 128 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 128 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 128 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 128 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 128 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 128 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 15 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 15 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 15 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 15 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 15 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 15 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 15 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 15 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 15 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 15 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 15 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 15 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 15 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 15 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 15 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 15 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2880 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 1970 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2500 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 EC50 '=' 800 nM
O88871 BXGT005286 Gamma-aminobutyric acid type B receptor subunit 2 reviewed - Gabbr2 IC50 '=' 60 nM
Q9Z0U4 BXGT022401 Gamma-aminobutyric acid type B receptor subunit 1 reviewed - Gabbr1 IC50 '=' 60 nM
P25094 BXGT009014 Peripheral myelin protein 22 reviewed - Pmp22 Potency - 57 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Binding affinity '=' 55 spec bound mg-1
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Binding affinity '=' 55 spec bound mg-1
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Binding affinity '=' 55 spec bound mg-1
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Binding affinity '=' 55 spec bound mg-1
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Binding affinity '=' 55 spec bound mg-1
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Binding affinity '=' 55 spec bound mg-1
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Binding affinity '=' 55 spec bound mg-1
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Binding affinity '=' 55 spec bound mg-1
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Binding affinity '=' 55 spec bound mg-1
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Binding affinity '=' 55 spec bound mg-1
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Binding affinity '=' 55 spec bound mg-1
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Binding affinity '=' 55 spec bound mg-1
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Binding affinity '=' 55 spec bound mg-1
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Binding affinity '=' 55 spec bound mg-1
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Binding affinity '=' 55 spec bound mg-1
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Binding affinity '=' 55 spec bound mg-1
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2600 nM
P23978 BXGT008937 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 2640 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 Max '=' 100 -
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 EC50 '=' 3000 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 3000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 3000 nM
Q6RY99 BXGT016512 Tetraspanin unreviewed - Inhibition - - -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Inhibition - - -
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Inhibition - - -
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Inhibition - - -
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Inhibition - - -
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Inhibition - - -
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Inhibition - - -
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Inhibition - - -
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Inhibition - - -
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Inhibition - - -
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Inhibition - - -
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Inhibition - - -
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Inhibition - - -
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Inhibition - - -
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Inhibition - - -
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Inhibition - - -
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Inhibition - - -
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 Ki '=' 200 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 Ki '=' 200 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 Ki '=' 200 nM
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE Ki '=' 200 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 Ki '=' 200 nM
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 Ki '=' 200 nM
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD Ki '=' 200 nM
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP Ki '=' 200 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 Ki '=' 200 nM
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ Ki '=' 200 nM
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 Ki '=' 200 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 Ki '=' 200 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 Ki '=' 200 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 Ki '=' 200 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 Ki '=' 200 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 Ki '=' 200 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 18 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 18 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 18 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 18 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 18 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 18 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 18 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 18 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 18 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 18 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 18 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 18 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 18 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 18 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 18 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 18 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 28000 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 28000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 28000 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 2818 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 EC50 '=' 990 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 EC50 '=' 990 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 990 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 EC50 '=' 990 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 990 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 EC50 '=' 990 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 990 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 990 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 990 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Displacement '=' 100 %
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Displacement '=' 100 %
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Displacement '=' 100 %
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Displacement '=' 100 %
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Displacement '=' 100 %
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Displacement '=' 100 %
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Displacement '=' 100 %
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Displacement '=' 100 %
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Displacement '=' 100 %
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Displacement '=' 100 %
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Displacement '=' 100 %
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Displacement '=' 100 %
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Displacement '=' 100 %
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Displacement '=' 100 %
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Displacement '=' 100 %
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Displacement '=' 100 %
P50554 BXGT010809 4-aminobutyrate aminotransferase, mitochondrial reviewed - Abat Inhibition - - -
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 33 nM
P02545 BXGT005889 Prelamin-A/C reviewed - LMNA Potency '=' 7 nM
Q969S8 BXGT019613 Polyamine deacetylase HDAC10 reviewed Epigenetic regulator HDAC10 Ki '=' 8190 nM
Q9UKV0 BXGT021750 Histone deacetylase 9 reviewed Epigenetic regulator HDAC9 Ki '=' 8190 nM
P56524 BXGT011176 Histone deacetylase 4 reviewed Epigenetic regulator HDAC4 Ki '=' 8190 nM
Q96DB2 BXGT019639 Histone deacetylase 11 reviewed Epigenetic regulator HDAC11 Ki '=' 8190 nM
Q9BY41 BXGT020180 Histone deacetylase 8 reviewed Epigenetic regulator HDAC8 Ki '=' 8190 nM
Q8WUI4 BXGT018992 Histone deacetylase 7 reviewed Epigenetic regulator HDAC7 Ki '=' 8190 nM
Q9UQL6 BXGT021813 Histone deacetylase 5 reviewed Epigenetic regulator HDAC5 Ki '=' 8190 nM
Q92769 BXGT019370 Histone deacetylase 2 reviewed Epigenetic regulator HDAC2 Ki '=' 8190 nM
Q9UBN7 BXGT021658 Histone deacetylase 6 reviewed Epigenetic regulator HDAC6 Ki '=' 8190 nM
O15379 BXGT004159 Histone deacetylase 3 reviewed Epigenetic regulator HDAC3 Ki '=' 8190 nM
Q13547 BXGT013373 Histone deacetylase 1 reviewed Epigenetic regulator HDAC1 Ki '=' 8190 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 EC50 '=' 50000 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 50000 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 50000 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 Max '=' 100 -
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 912 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 912 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 912 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A EC50 - - -
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 EC50 '=' 42657 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 42657 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 42657 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 RUmax '=' 100 %
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 RUmax '=' 100 %
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 RUmax '=' 100 %
P80147 BXGT011879 4-aminobutyrate aminotransferase, mitochondrial reviewed - ABAT Km '=' 2400000 nM
P16305 BXGT008215 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Emax '=' 389 -
P27681 BXGT009196 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Emax '=' 389 -
P63080 BXGT011492 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Emax '=' 389 -
Q9D6F4 BXGT020259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Emax '=' 389 -
P22933 BXGT008819 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Emax '=' 389 -
P26049 BXGT009086 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Emax '=' 389 -
Q9JLF1 BXGT020834 Gamma-aminobutyric acid receptor subunit theta reviewed - Gabrq Emax '=' 389 -
P62812 BXGT011459 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Emax '=' 389 -
A2AMW3 BXGT001075 Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon unreviewed - Gabre Emax '=' 389 -
P22723 BXGT008798 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Emax '=' 389 -
Q9R0Y8 BXGT021410 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Emax '=' 389 -
P50571 BXGT010810 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Emax '=' 389 -
Q8QZW7 BXGT018675 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Emax '=' 389 -
P26048 BXGT009085 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Emax '=' 389 -
Q8BHJ7 BXGT017911 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Emax '=' 389 -
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 1800 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 1800 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 1800 nM
P16473 BXGT008234 Thyrotropin receptor reviewed G-protein coupled receptor TSHR Potency '=' 31622 nM
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 25000 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 GABA agonism - - -
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 GABA agonism - - -
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 GABA agonism - - -
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE GABA agonism - - -
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 GABA agonism - - -
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 GABA agonism - - -
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD GABA agonism - - -
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP GABA agonism - - -
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 GABA agonism - - -
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ GABA agonism - - -
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 GABA agonism - - -
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 GABA agonism - - -
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 GABA agonism - - -
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 GABA agonism - - -
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 GABA agonism - - -
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 GABA agonism - - -
P80404 BXGT011907 4-aminobutyrate aminotransferase, mitochondrial reviewed Enzyme ABAT Km '=' 2500000 nM
Q96QE3 BXGT019718 ATPase family AAA domain-containing protein 5 reviewed - ATAD5 Potency - 1457 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Activity - - -
P31649 BXGT009562 Sodium- and chloride-dependent GABA transporter 2 reviewed - Slc6a13 IC50 '=' 27542 nM
P31648 BXGT009561 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 7244 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 24 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 24 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 24 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 24 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 24 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 24 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 24 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 24 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 24 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 24 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 24 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 24 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 24 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 24 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 24 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 24 nM
P11308 BXGT007684 Transcriptional regulator ERG reviewed Transcription factor ERG Potency - 1122 nM
O75899 BXGT005161 Gamma-aminobutyric acid type B receptor subunit 2 reviewed G-protein coupled receptor GABBR2 EC50 '=' 530 nM
Q9UBS5 BXGT021662 Gamma-aminobutyric acid type B receptor subunit 1 reviewed G-protein coupled receptor GABBR1 EC50 '=' 530 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 EC50 '=' 51000 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 51000 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 51000 nM
O75496 BXGT005132 Geminin reviewed - GMNN Potency - 1122 nM
B2GV46 BXGT001957 Free fatty acid receptor 3 reviewed - Ffar3 EC50 - - -
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 Max '=' 100 -
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre IC50 '=' 25 nM
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq IC50 '=' 25 nM
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 IC50 '=' 25 nM
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 IC50 '=' 25 nM
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 IC50 '=' 25 nM
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 IC50 '=' 25 nM
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 IC50 '=' 25 nM
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 IC50 '=' 25 nM
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 IC50 '=' 25 nM
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 IC50 '=' 25 nM
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 IC50 '=' 25 nM
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 IC50 '=' 25 nM
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 IC50 '=' 25 nM
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd IC50 '=' 25 nM
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 IC50 '=' 25 nM
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp IC50 '=' 25 nM
P31648 BXGT009561 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 5000 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 Ki '=' 33 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 Ki '=' 33 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 Ki '=' 33 nM
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE Ki '=' 33 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 Ki '=' 33 nM
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 Ki '=' 33 nM
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD Ki '=' 33 nM
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP Ki '=' 33 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 Ki '=' 33 nM
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ Ki '=' 33 nM
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 Ki '=' 33 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 Ki '=' 33 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 Ki '=' 33 nM
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 Ki '=' 33 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 Ki '=' 33 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 Ki '=' 33 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 EC50 '=' 16500 nM
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 EC50 '=' 16500 nM
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 EC50 '=' 16500 nM
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 EC50 '=' 16500 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 16500 nM
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 EC50 '=' 16500 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 16500 nM
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 EC50 '=' 16500 nM
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 EC50 '=' 16500 nM
Q7Z2H8 BXGT017247 Proton-coupled amino acid transporter 1 reviewed Transporter SLC36A1 Ki '=' 4000000 nM
Q9Y6L6 BXGT022334 Solute carrier organic anion transporter family member 1B1 reviewed Transporter SLCO1B1 Inhibition '=' 56 %
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 3890 nM
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 181000 nM
P49798 BXGT010745 Regulator of G-protein signaling 4 reviewed Enzyme modulator RGS4 Potency - 6 nM
Q13148 BXGT013318 TAR DNA-binding protein 43 reviewed - TARDBP Potency - 35481 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 AC50 - - -
P15289 BXGT008102 Arylsulfatase A reviewed Enzyme ARSA Potency - 8492 nM
P31650 BXGT009563 Sodium- and chloride-dependent GABA transporter 3 reviewed - Slc6a11 IC50 '=' 11481 nM
Q9ES14 BXGT020314 Gamma-aminobutyric acid receptor subunit epsilon reviewed - Gabre Displacement '=' 48 %
Q91ZM7 BXGT019327 GABA theta subunit unreviewed - Gabrq Displacement '=' 48 %
P63138 BXGT011502 Gamma-aminobutyric acid receptor subunit beta-2 reviewed - Gabrb2 Displacement '=' 48 %
P63079 BXGT011491 Gamma-aminobutyric acid receptor subunit beta-3 reviewed - Gabrb3 Displacement '=' 48 %
P62813 BXGT011460 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed - Gabra1 Displacement '=' 48 %
P30191 BXGT009410 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed - Gabra6 Displacement '=' 48 %
P28473 BXGT009261 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed - Gabrg3 Displacement '=' 48 %
P28471 BXGT009259 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed - Gabra4 Displacement '=' 48 %
P23576 BXGT008885 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed - Gabra2 Displacement '=' 48 %
P23574 BXGT008884 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed - Gabrg1 Displacement '=' 48 %
P20236 BXGT008551 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed - Gabra3 Displacement '=' 48 %
P19969 BXGT008536 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed - Gabra5 Displacement '=' 48 %
P18508 BXGT008412 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed - Gabrg2 Displacement '=' 48 %
P18506 BXGT008410 Gamma-aminobutyric acid receptor subunit delta reviewed - Gabrd Displacement '=' 48 %
P15431 BXGT008122 Gamma-aminobutyric acid receptor subunit beta-1 reviewed - Gabrb1 Displacement '=' 48 %
O09028 BXGT004049 Gamma-aminobutyric acid receptor subunit pi reviewed - Gabrp Displacement '=' 48 %
P80404 BXGT011907 4-aminobutyrate aminotransferase, mitochondrial reviewed Enzyme ABAT Km '=' 1400000 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 EC50 '=' 270 nM
P24046 BXGT008943 Gamma-aminobutyric acid receptor subunit rho-1 reviewed Ion channel GABRR1 EC50 '=' 1190 nM
P18088 BXGT008378 Glutamate decarboxylase 1 reviewed - Gad1 Inhibition - - -
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 27542 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 4500 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 4500 nM
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 165958 nM
P31648 BXGT009561 Sodium- and chloride-dependent GABA transporter 1 reviewed - Slc6a1 IC50 '=' 5011 nM
Q969S8 BXGT019613 Polyamine deacetylase HDAC10 reviewed Epigenetic regulator HDAC10 Activity '=' 100 %
Q9UKV0 BXGT021750 Histone deacetylase 9 reviewed Epigenetic regulator HDAC9 Activity '=' 100 %
P56524 BXGT011176 Histone deacetylase 4 reviewed Epigenetic regulator HDAC4 Activity '=' 100 %
Q96DB2 BXGT019639 Histone deacetylase 11 reviewed Epigenetic regulator HDAC11 Activity '=' 100 %
Q9BY41 BXGT020180 Histone deacetylase 8 reviewed Epigenetic regulator HDAC8 Activity '=' 100 %
Q8WUI4 BXGT018992 Histone deacetylase 7 reviewed Epigenetic regulator HDAC7 Activity '=' 100 %
Q9UQL6 BXGT021813 Histone deacetylase 5 reviewed Epigenetic regulator HDAC5 Activity '=' 100 %
Q92769 BXGT019370 Histone deacetylase 2 reviewed Epigenetic regulator HDAC2 Activity '=' 100 %
Q9UBN7 BXGT021658 Histone deacetylase 6 reviewed Epigenetic regulator HDAC6 Activity '=' 100 %
O15379 BXGT004159 Histone deacetylase 3 reviewed Epigenetic regulator HDAC3 Activity '=' 100 %
Q13547 BXGT013373 Histone deacetylase 1 reviewed Epigenetic regulator HDAC1 Activity '=' 100 %
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 Inhibition '=' 81 %
P48065 BXGT010617 Sodium- and chloride-dependent betaine transporter reviewed Transporter SLC6A12 IC50 '=' 17782 nM
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 EC50 '=' 3400 nM
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ EC50 '=' 3400 nM
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 EC50 '=' 3400 nM
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF00012 Pineapple Ananas comosus Fruits
BXGF00016 Peanut Arachis hypogaea Nuts
BXGF00017 Burdock Arctium lappa Vegetables
BXGF00019 Tarragon Artemisia dracunculus Herbs and Spices
BXGF00056 Mandarin orange (Clementine, Tangerine) Citrus reticulata Fruits
BXGF00057 Sweet orange Citrus sinensis Fruits
BXGF00106 Mango Mangifera indica Fruits
BXGF00115 Bitter gourd Momordica charantia Gourds
BXGF00134 Common bean Phaseolus vulgaris Pulses
BXGF00135 Date Phoenix dactylifera Fruits
BXGF00139 Pepper (Spice) Piper nigrum Herbs and Spices
BXGF00141 Common pea Pisum sativum Pulses
BXGF00146 Sour cherry Prunus cerasus Fruits
BXGF00173 Garden tomato (var.) Solanum lycopersicum var. lycopersicum Vegetables
BXGF00174 Eggplant Solanum melongena Vegetables
BXGF00175 Potato Solanum tuberosum Vegetables
BXGF00186 Fenugreek Trigonella foenum-graecum Herbs and Spices
BXGF00204 Common grape Vitis vinifera Fruits
BXGF00206 Ginger Zingiber officinale Herbs and Spices
BXGF00246 Red beetroot Beta vulgaris var. rubra Vegetables
BXGF00300 Chayote Sechium edule Gourds
BXGF00310 Coconut Cocos nucifera Fruits
BXGF00337 Ginkgo nuts Ginkgo biloba Herbs and Spices
BXGF00400 French plantain Musa X paradisiaca Fruits
BXGF00440 Soursop Annona muricata Fruits
BXGF00446 Sugar apple Annona squamosa Fruits
BXGF00506 Shiitake Lentinus edodes Vegetables
BXGF00862 Phebalium ozothamnoides Phebalium ozothamnoides Others
BXGF00977 Vitex megapotamica Vitex megapotamica Human Edible Plant
BXGF01140 Angelica gigas Angelica gigas Medicinal Plant
BXGF01185 Aloe vera Aloe vera Medicinal Plant
BXGF01266 Dysoxylum lenticellatum Dysoxylum lenticellatum Others
BXGF01284 Saururus cernuus Saururus cernuus Medicinal Plant
BXGF01343 Strychnos fendleri Strychnos fendleri Others
BXGF01466 Halimeda macroloba Halimeda macroloba Others
BXGF01509 Solanum dulcamara Solanum dulcamara Medicinal Plant
BXGF01510 Cabucala madagascariensis Cabucala madagascariensis Others
BXGF01900 Aloe ferox Aloe ferox Medicinal Plant
BXGF01911 Bupleurum scorzonerifolium Bupleurum scorzonerifolium Medicinal Plant
BXGF02049 Angelica sinensis Angelica sinensis Medicinal Plant
BXGF02054 Shorea uliginosa Shorea uliginosa Others
BXGF02104 Derris reticulata Derris reticulata Others
BXGF02214 Morus bombycis Morus bombycis Medicinal Plant
BXGF02232 Gentiana arisanensis Gentiana arisanensis Others
BXGF02290 Sonchus microcarpus Sonchus microcarpus Others
BXGF02376 Ballota lanata Ballota lanata Others
BXGF02567 Lycium chinense Lycium chinense Medicinal Plant
BXGF02680 Eucalyptus ovata Eucalyptus ovata Others
BXGF02723 Hesperocyparis macrocarpa Hesperocyparis macrocarpa Others
BXGF02815 Pinellia ternata Pinellia ternata Medicinal Plant
BXGF02848 Buxus sempervirens Buxus sempervirens Medicinal Plant
BXGF03270 Aruncus dioicus Aruncus dioicus Medicinal Plant
BXGF03319 Trichosanthes kirilowii Trichosanthes kirilowii Medicinal Plant
BXGF03435 Angelica pubescens Angelica pubescens Medicinal Plant
BXGF03442 Rhaponticum carthamoides Rhaponticum carthamoides Medicinal Plant
BXGF03614 Ageratum conyzoides Ageratum conyzoides Medicinal Plant
BXGF03645 Lycium barbarum Lycium barbarum Medicinal Plant
BXGF03735 Hansenia weberbaueriana Hansenia weberbaueriana Others
BXGF03908 Hedysarum multijugum maxim Hedysarum multijugum maxim Others
BXGF03924 Kochia trichophylla Kochia trichophylla Others
BXGF04109 Saussurea costus Saussurea costus Medicinal Plant
BXGF04191 Vicia villosa Vicia villosa Medicinal Plant
BXGF04607 Morus alba Morus alba Medicinal Plant
BXGF04631 Aloe spicata Aloe spicata Medicinal Plant
BXGF04830 Artemisia oranensis Artemisia oranensis Others
BXGF04842 Angelica acutiloba Angelica acutiloba Medicinal Plant
BXGF04875 Bupleurum chinense Bupleurum chinense Medicinal Plant
BXGF04926 Aloe africana Aloe africana Medicinal Plant
BXGF04978 Isatis indigotica Isatis indigotica Medicinal Plant
BXGF04981 Bupleurum falcatum Bupleurum falcatum Medicinal Plant
BXGF05178 Lilium hansonii Lilium hansonii Medicinal Plant
BXGF05193 Piper futokadsura Piper futokadsura Others
BXGF05297 Isatis tinctoria Isatis tinctoria Medicinal Plant
BXGF05330 Arum ternatum thunb Arum ternatum thunb Others
BXGF05511 Acorus gramineus Acorus gramineus Medicinal Plant
BXGF05692 Potentilla multifida Potentilla multifida Medicinal Plant
BXGF05859 Haplopappus venetus Haplopappus venetus Others
BXGF05925 Centaurea amara Centaurea amara Others
BXGF05962 Rehmannia glutinosa Rehmannia glutinosa Medicinal Plant
BXGF05964 Citrullus lanatus subsp. vulgaris Citrullus lanatus subsp. vulgaris 0
BXGF06071 Acorus tatarinowii Acorus tatarinowii Medicinal Plant
BXGF06126 Strychnos diplotricha Strychnos diplotricha Medicinal Plant
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease