| Uniprot | Drug | Mechanism | ChEMBL ID |
Target | Protein Name |
Organism | Protein Class |
Molecule Type |
First Approval |
|---|---|---|---|---|---|---|---|---|---|
| Q72547 | ABACAVIR | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1998 |
| P30968 | ABARELIX | Gonadotropin-releasing hormone receptor antagonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 2003 |
| P33681 | ABATACEPT | T-lymphocyte activation antigen CD80 inhibitor | CHEMBL2364157 | T-lymphocyte activation antigen CD80 | T-lymphocyte activation antigen CD80 | Homo sapiens | surface antigen | Protein | 2006 |
| Q72547 | ABACAVIR | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1998 |
| P30968 | ABARELIX | Gonadotropin-releasing hormone receptor antagonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 2003 |
| P33681 | ABATACEPT | T-lymphocyte activation antigen CD80 inhibitor | CHEMBL2364157 | T-lymphocyte activation antigen CD80 | T-lymphocyte activation antigen CD80 | Homo sapiens | surface antigen | Protein | 2006 |
| P42081 | ABATACEPT | T-lymphocyte activation antigen CD86 inhibitor | CHEMBL2364156 | T-lymphocyte activation antigen CD86 | T-lymphocyte activation antigen CD86 | Homo sapiens | surface antigen | Protein | 2006 |
| P05106 | ABCIXIMAB | Integrin alpha-V/beta-3 inhibitor | CHEMBL1907598 | Integrin alpha-V/beta-3 | Integrin beta-3 | Homo sapiens | membrane receptor | Antibody | 1993 |
| P05106 | ABCIXIMAB | Integrin alpha-IIb/beta-3 inhibitor | CHEMBL2093869 | Integrin alpha-IIb/beta-3 | Integrin beta-3 | Homo sapiens | membrane receptor | Antibody | 1993 |
| P05093 | ABIRATERONE ACETATE | Cytochrome P450 17A1 inhibitor | CHEMBL3522 | Cytochrome P450 17A1 | "Steroid 17-alpha-hydroxylase/17,20 lyase" | Homo sapiens | enzyme cytochrome p450 cyp_17 cyp_17a cyp_17a1 | Small molecule | 2011 |
| P60880 | ABOBOTULINUMTOXINA | Synaptosomal-associated protein 25 inhibitor | CHEMBL2364159 | Synaptosomal-associated protein 25 | Synaptosomal-associated protein 25 | Homo sapiens | cytosolic other | Unknown | 2009 |
| O00591 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| O14764 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| O15399 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| O60391 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| P14867 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P18505 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P18507 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P28472 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P31644 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P34903 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P47869 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P47870 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P48169 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P78334 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q05586 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| Q12879 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| Q13224 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| Q14957 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| Q16445 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q8N1C3 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q8TCU5 | ACAMPROSATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2004 |
| Q99928 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q9UN88 | ACAMPROSATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| O43451 | ACARBOSE | Maltase-glucoamylase inhibitor | CHEMBL2074 | Maltase-glucoamylase | "Maltase-glucoamylase, intestinal" | Homo sapiens | enzyme hydrolase | Small molecule | 1995 |
| P04746 | ACARBOSE | Pancreatic alpha-amylase inhibitor | CHEMBL2045 | Pancreatic alpha-amylase | Pancreatic alpha-amylase | Homo sapiens | enzyme hydrolase | Small molecule | 1995 |
| P08588 | ACEBUTOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| O00519 | ACETAMINOPHEN | Anandamide amidohydrolase inhibitor | CHEMBL2243 | Anandamide amidohydrolase | Fatty-acid amide hydrolase 1 | Homo sapiens | enzyme | Small molecule | 1968 |
| P21554 | ACETAMINOPHEN | Cannabinoid receptor 1 | Cannabinoid receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor cannabinoid receptor | Small molecule | 1968 | ||
| P23219 | ACETAMINOPHEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1968 |
| P35354 | ACETAMINOPHEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1968 |
| Q8NER1 | ACETAMINOPHEN | Vanilloid receptor opener | CHEMBL4794 | Vanilloid receptor | Transient receptor potential cation channel subfamily V member 1 | Homo sapiens | ion channel vgc trp | Small molecule | 1968 |
| O43570 | ACETAZOLAMIDE | Carbonic anhydrase XII inhibitor | CHEMBL3242 | Carbonic anhydrase XII | Carbonic anhydrase 12 | Homo sapiens | enzyme lyase | Small molecule | 1953 |
| P00915 | ACETAZOLAMIDE | Carbonic anhydrase I inhibitor | CHEMBL261 | Carbonic anhydrase I | Carbonic anhydrase 1 | Homo sapiens | enzyme lyase | Small molecule | 1953 |
| P00918 | ACETAZOLAMIDE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1953 |
| P22748 | ACETAZOLAMIDE | Carbonic anhydrase IV inhibitor | CHEMBL3729 | Carbonic anhydrase IV | Carbonic anhydrase 4 | Homo sapiens | enzyme lyase | Small molecule | 1953 |
| Q09428 | ACETOHEXAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1964 |
| Q14654 | ACETOHEXAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1964 |
| P18314 | ACETOHYDROXAMIC ACID | Urease subunit alpha | Urease subunit alpha | Enterobacter aerogenes | Hydrolase | Small molecule | 1983 | ||
| Q03282 | ACETOHYDROXAMIC ACID | Bacterial urease inhibitor | CHEMBL2364683 | Bacterial urease | Urease subunit gamma | Bacteria | enzyme hydrolase | Small molecule | 1983 |
| Q03283 | ACETOHYDROXAMIC ACID | Bacterial urease inhibitor | CHEMBL2364683 | Bacterial urease | Urease subunit beta | Bacteria | enzyme hydrolase | Small molecule | 1983 |
| Q03284 | ACETOHYDROXAMIC ACID | Bacterial urease inhibitor | CHEMBL2364683 | Bacterial urease | Urease subunit alpha | Bacteria | enzyme hydrolase | Small molecule | 1983 |
| P14416 | ACETOPHENAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1961 |
| P20309 | ACETYLCHOLINE | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1973 |
| P05023 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 0 |
| P05023 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 0 |
| P13637 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | enzyme hydrolase | Small molecule | 0 |
| P13637 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 0 |
| P50993 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | enzyme hydrolase | Small molecule | 0 |
| P50993 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 0 |
| Q13733 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | enzyme hydrolase | Small molecule | 0 |
| Q13733 | ACETYLDIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 0 |
| P10276 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1996 |
| P10826 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1996 |
| P13631 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1996 |
| P19793 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-alpha | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b1 | Small molecule | 1996 |
| P28702 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-beta | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b2 | Small molecule | 1996 |
| P48443 | ACITRETIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-gamma | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b3 | Small molecule | 1996 |
| P20309 | ACLIDINIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2012 |
| ACRISORCIN | Unknown | Small molecule | 1982 | ||||||
| P35367 | ACRIVASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1994 |
| P04293 | ACYCLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1982 |
| P09252 | ACYCLOVIR | DNA polymerase catalytic subunit | DNA polymerase catalytic subunit | Varicella-zoster virus (strain Dumas) | enzyme | Small molecule | 1982 | ||
| P01375 | ADALIMUMAB | TNF-alpha inhibitor | CHEMBL1825 | TNF-alpha | Tumor necrosis factor | Homo sapiens | secreted | Antibody | 2002 |
| P10276 | ADAPALENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1996 |
| P10826 | ADAPALENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1996 |
| P13631 | ADAPALENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1996 |
| P19793 | ADAPALENE | Retinoic acid receptor RXR-alpha | Retinoic acid receptor RXR-alpha | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b1 | Small molecule | 1996 | ||
| P28702 | ADAPALENE | Retinoic acid receptor RXR-beta | Retinoic acid receptor RXR-beta | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b2 | Small molecule | 1996 | ||
| P48443 | ADAPALENE | Retinoic acid receptor RXR-gamma | Retinoic acid receptor RXR-gamma | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b3 | Small molecule | 1996 | ||
| Q9IF40 | ADEFOVIR DIPIVOXIL | DNA polymerase/reverse transcriptase inhibitor | CHEMBL2362994 | DNA polymerase/reverse transcriptase | Protein P | Hepatitis B virus | enzyme transferase | Small molecule | 2002 |
| P0DMS8 | ADENOSINE | Adenosine receptor agonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A3 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1989 |
| P29274 | ADENOSINE | Adenosine receptor agonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1989 |
| P29275 | ADENOSINE | Adenosine receptor agonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2b | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1989 |
| P30542 | ADENOSINE | Adenosine receptor agonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A1 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1989 |
| P00533 | AFATINIB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2013 |
| P04626 | AFATINIB | Receptor protein-tyrosine kinase erbB-2 inhibitor | CHEMBL1824 | Receptor protein-tyrosine kinase erbB-2 | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2013 |
| Q15303 | AFATINIB | Receptor protein-tyrosine kinase erbB-4 inhibitor | CHEMBL3009 | Receptor protein-tyrosine kinase erbB-4 | Receptor tyrosine-protein kinase erbB-4 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2013 |
| P15692 | AFLIBERCEPT | Vascular endothelial growth factor A inhibitor | CHEMBL1783 | Vascular endothelial growth factor A | Vascular endothelial growth factor A | Homo sapiens | secreted | Protein | 2011 |
| P49763 | AFLIBERCEPT | Placenta growth factor inhibitor | CHEMBL1697671 | Placenta growth factor | Placenta growth factor | Homo sapiens | unclassified | Protein | 2011 |
| P49765 | AFLIBERCEPT | Vascular endothelial growth factor B | Vascular endothelial growth factor B | Homo sapiens | Unclassified | Protein | 2011 | ||
| AGALSIDASE BETA | Globotriosylceramide hydrolytic enzyme | CHEMBL2366040 | Globotriosylceramide | Homo sapiens | Enzyme | 2003 | |||
| P0AES4 | ALATROFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P0AES6 | ALATROFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P0AFI2 | ALATROFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P20083 | ALATROFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 1997 |
| C4PKY4 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 1 | Taeniidae | structural | Small molecule | 1996 |
| C4PKZ2 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 2 | Taeniidae | structural | Small molecule | 1996 |
| C4PKZ6 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 3 | Taeniidae | structural | Small molecule | 1996 |
| F1L4P8 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-1 chain | Nematoda | structural | Small molecule | 1996 |
| F1L7U3 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-2 chain | Nematoda | structural | Small molecule | 1996 |
| F1L8A5 | ALBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-4 chain | Nematoda | structural | Small molecule | 1996 |
| P43220 | ALBIGLUTIDE | Glucagon-like peptide 1 receptor agonist | CHEMBL1784 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon-like peptide receptor | Protein | 2014 |
| ALBUMIN HUMAN | Bilirubin chelating agent | CHEMBL2364174 | Bilirubin | Homo sapiens | Protein | 1997 | |||
| P07550 | ALBUTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1981 |
| P35367 | ALCAFTADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2010 |
| P04150 | ALCLOMETASONE DIPROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P06729 | ALEFACEPT | T-cell surface antigen CD2 inhibitor | CHEMBL2040 | T-cell surface antigen CD2 | T-cell surface antigen CD2 | Homo sapiens | surface antigen | Protein | 2003 |
| P31358 | ALEMTUZUMAB | CAMPATH-1 antigen inhibitor | CHEMBL1912 | CAMPATH-1 antigen | CAMPATH-1 antigen | Homo sapiens | surface antigen | Antibody | 2001 |
| P14324 | ALENDRONIC ACID | Farnesyl diphosphate synthase inhibitor | CHEMBL1782 | Farnesyl diphosphate synthase | Farnesyl pyrophosphate synthase | Homo sapiens | enzyme transferase | Small molecule | 1995 |
| P35372 | ALFENTANIL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1986 |
| P25100 | ALFUZOSIN | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2003 |
| P35348 | ALFUZOSIN | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2003 |
| P35368 | ALFUZOSIN | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2003 |
| ALGLUCERASE | Glucocerebroside hydrolytic enzyme | CHEMBL2364176 | Glucocerebroside | Homo sapiens | Enzyme | 1991 | |||
| ALGLUCOSIDASE ALFA | Starch hydrolytic enzyme | CHEMBL2364180 | Starch | Homo sapiens | Enzyme | 2006 | |||
| P00797 | ALISKIREN | Renin inhibitor | CHEMBL286 | Renin | Renin | Homo sapiens | enzyme protease aspartic aa a1a | Small molecule | 2007 |
| P10276 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1999 |
| P10826 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1999 |
| P13631 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1999 |
| P19793 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-alpha | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b1 | Small molecule | 1999 |
| P28702 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-beta | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b2 | Small molecule | 1999 |
| P48443 | ALITRETINOIN | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-gamma | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b3 | Small molecule | 1999 |
| ALKAVERVIR | Unknown | Small molecule | 1982 | ||||||
| P47989 | ALLOPURINOL | Xanthine dehydrogenase inhibitor | CHEMBL1929 | Xanthine dehydrogenase | Xanthine dehydrogenase/oxidase | Homo sapiens | enzyme reductase | Small molecule | 1966 |
| P28221 | ALMOTRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P28222 | ALMOTRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P30939 | ALMOTRIPTAN | Serotonin 1f (5-HT1f) receptor agonist | CHEMBL1805 | Serotonin 1f (5-HT1f) receptor | 5-hydroxytryptamine receptor 1F | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P27487 | ALOGLIPTIN | Dipeptidyl peptidase IV inhibitor | CHEMBL284 | Dipeptidyl peptidase IV | Dipeptidyl peptidase 4 | Homo sapiens | enzyme protease serine sc s9b | Small molecule | 2013 |
| P46098 | ALOSETRON | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 2000 |
| P14867 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P18507 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P31644 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P34903 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P47869 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q8N1C3 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q99928 | ALPRAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P34995 | ALPROSTADIL | Prostanoid EP1 receptor agonist | CHEMBL1811 | Prostanoid EP1 receptor | Prostaglandin E2 receptor EP1 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1981 |
| P43116 | ALPROSTADIL | Prostanoid EP2 receptor agonist | CHEMBL1881 | Prostanoid EP2 receptor | Prostaglandin E2 receptor EP2 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1981 |
| P08913 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P18089 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P18825 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P25100 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P35348 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P35368 | ALSEROXYLON | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P00747 | ALTEPLASE | Plasminogen activator | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Enzyme | 1996 |
| ALTRETAMINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1990 | |||
| ALUMINUM ACETATE | Unknown | Small molecule | 1976 | ||||||
| ALUMINUM HYDROXIDE | Unknown | Small molecule | 1983 | ||||||
| P35372 | ALVIMOPAN | Mu opioid receptor antagonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2008 |
| O15399 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| O60391 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| P06821 | AMANTADINE | Matrix protein 2 inhibitor | CHEMBL1932894 | Matrix protein 2 | Matrix protein 2 | Influenza A virus (strain A/Puerto Rico/8/1934 H1N1) | ion channel other misc m2-c | Small molecule | 1968 |
| Q05586 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| Q12879 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| Q13224 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| Q14957 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| Q8TCU5 | AMANTADINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1968 |
| P22303 | AMBENONIUM | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1956 |
| P24530 | AMBRISENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin B receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2007 |
| P25101 | AMBRISENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin-1 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2007 |
| P04150 | AMCINONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1979 |
| P0AD65 | AMDINOCILLIN | Bacterial penicillin-binding protein 2 inhibitor | CHEMBL2354313 | Bacterial penicillin-binding protein 2 | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| AMIFOSTINE | Reactive metabolite scavenging agent | Small molecule | 1995 | ||||||
| AMIKACIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1981 | ||
| P37088 | AMILORIDE | "Amiloride-sensitive sodium channel, ENaC blocker" | CHEMBL2107836 | "Amiloride-sensitive sodium channel, ENaC" | Amiloride-sensitive sodium channel subunit alpha | Homo sapiens | ion channel lgic enac | Small molecule | 1981 |
| P00747 | AMINOCAPROIC ACID | Plasminogen inhibitor | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 1964 |
| P00750 | AMINOCAPROIC ACID | Tissue-type plasminogen activator inhibitor | CHEMBL1873 | Tissue-type plasminogen activator | Tissue-type plasminogen activator | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 1964 |
| P05108 | AMINOGLUTETHIMIDE | Cytochrome P450 11A1 inhibitor | CHEMBL2033 | Cytochrome P450 11A1 | "Cholesterol side-chain cleavage enzyme, mitochondrial" | Homo sapiens | enzyme cytochrome p450 cyp_11 cyp_11a cyp_11a1 | Small molecule | 1980 |
| P11511 | AMINOGLUTETHIMIDE | Cytochrome P450 19A1 inhibitor | CHEMBL1978 | Cytochrome P450 19A1 | Aromatase | Homo sapiens | enzyme cytochrome p450 cyp_19 cyp_19a cyp_19a1 | Small molecule | 1980 |
| AMINOLEVULINIC ACID | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1999 | |||
| P23219 | AMINOSALICYLIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P35354 | AMINOSALICYLIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P08913 | AMIODARONE | Alpha-2A adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 | ||
| P35348 | AMIODARONE | Alpha-1A adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 | ||
| Q12809 | AMIODARONE | HERG blocker | CHEMBL240 | HERG | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1985 |
| Q14524 | AMIODARONE | Sodium channel protein type 5 subunit alpha | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 | ||
| Q96RP8 | AMIODARONE | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 7 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1985 | ||
| P23975 | AMITRIPTYLINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1961 |
| P28223 | AMITRIPTYLINE | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1961 | ||
| P28335 | AMITRIPTYLINE | 5-hydroxytryptamine receptor 2C | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1961 | ||
| P31645 | AMITRIPTYLINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1961 |
| P35367 | AMITRIPTYLINE | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1961 | ||
| P27815 | AMLEXANOX | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1996 |
| Q07343 | AMLEXANOX | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1996 |
| Q08493 | AMLEXANOX | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1996 |
| Q08499 | AMLEXANOX | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1996 |
| O60840 | AMLODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1992 |
| Q01668 | AMLODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1992 |
| Q13698 | AMLODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1992 |
| Q13936 | AMLODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1992 |
| AMMONIUM LACTATE | Unknown | Small molecule | 1985 | ||||||
| AMODIAQUINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 1982 | |||
| P14416 | AMOXAPINE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1980 |
| P21728 | AMOXAPINE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1980 |
| P21917 | AMOXAPINE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1980 |
| P21918 | AMOXAPINE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1980 |
| P23975 | AMOXAPINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1980 |
| P31645 | AMOXAPINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1980 |
| P35462 | AMOXAPINE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1980 |
| P02918 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P02919 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1974 |
| P08506 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P0AD65 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P0AD68 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1974 |
| P0AEB2 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P24228 | AMOXICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1974 |
| P23975 | AMPHETAMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| Q01959 | AMPHETAMINE | Dopamine transporter releasing agent | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| Q96RJ0 | AMPHETAMINE | Trace amine-associated receptor 1 | Trace amine-associated receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor trace amine receptor | Small molecule | 1955 | ||
| AMPHOTERICIN B | Ergosterol chelating agent | CHEMBL2364028 | Ergosterol | Candida albicans | Small molecule | 1964 | |||
| P02918 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1965 |
| P02919 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1965 |
| P08506 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1965 |
| P0AD65 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1965 |
| P0AD68 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1965 |
| P0AEB2 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1965 |
| P24228 | AMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1965 |
| Q72874 | AMPRENAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 1999 |
| AMYLASE | Starch hydrolytic enzyme | CHEMBL2364180 | Starch | Homo sapiens | Enzyme | 1996 | |||
| Q13370 | ANAGRELIDE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase B" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3b | Small molecule | 1997 |
| Q14432 | ANAGRELIDE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1997 |
| P14778 | ANAKINRA | Interleukin-1 receptor antagonist | CHEMBL1959 | Interleukin-1 receptor | Interleukin-1 receptor type 1 | Homo sapiens | membrane receptor | Protein | 2001 |
| P11511 | ANASTROZOLE | Cytochrome P450 19A1 inhibitor | CHEMBL1978 | Cytochrome P450 19A1 | Aromatase | Homo sapiens | enzyme cytochrome p450 cyp_19 cyp_19a cyp_19a1 | Small molecule | 1995 |
| O13428 | ANIDULAFUNGIN | "1,3-beta-glucan synthase inhibitor" | CHEMBL2364673 | "1,3-beta-glucan synthase" | "Beta-1,3-glucan synthase catalytic subunit 1" | Candida | enzyme transferase | Small molecule | 2006 |
| P35372 | ANILERIDINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1982 |
| P41145 | ANILERIDINE | Kappa opioid receptor agonist | CHEMBL237 | Kappa opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1982 |
| P38435 | ANISINDIONE | Vitamin K-dependent gamma-carboxylase inhibitor | CHEMBL2012 | Vitamin K-dependent gamma-carboxylase | Vitamin K-dependent gamma-carboxylase | Homo sapiens | enzyme lyase | Small molecule | 1957 |
| P08172 | ANISOTROPINE | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1962 | ||
| P11229 | ANISOTROPINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1962 |
| P20309 | ANISOTROPINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1962 |
| P35367 | ANTAZOLINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1994 |
| P00742 | APIXABAN | Coagulation factor X inhibitor | CHEMBL244 | Coagulation factor X | Coagulation factor X | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 2012 |
| P08913 | APOMORPHINE | Alpha-2A adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2004 | ||
| P14416 | APOMORPHINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2004 |
| P18089 | APOMORPHINE | Alpha-2B adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2004 | ||
| P18825 | APOMORPHINE | Alpha-2C adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2004 | ||
| P21917 | APOMORPHINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2004 |
| P21918 | APOMORPHINE | D(1B) dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2004 | ||
| P25100 | APOMORPHINE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2004 | ||
| P35462 | APOMORPHINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2004 |
| P08913 | APRACLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P18089 | APRACLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P18825 | APRACLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P27815 | APREMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 2014 |
| Q07343 | APREMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 2014 |
| Q08493 | APREMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 2014 |
| Q08499 | APREMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 2014 |
| P25103 | APREPITANT | Neurokinin 1 receptor antagonist | CHEMBL249 | Neurokinin 1 receptor | Substance-P receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide neurokinin receptor | Small molecule | 2003 |
| P00747 | APROTININ | Plasminogen inhibitor | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Unknown | 1993 |
| P03952 | APROTININ | Plasma kallikrein inhibitor | CHEMBL2000 | Plasma kallikrein | Plasma kallikrein | Homo sapiens | enzyme protease serine pas s1a | Unknown | 1993 |
| P01008 | ARDEPARIN SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 1997 |
| P07550 | ARFORMOTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2006 |
| P00734 | ARGATROBAN | Thrombin inhibitor | CHEMBL204 | Thrombin | Prothrombin | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 2000 |
| P08908 | ARIPIPRAZOLE | Serotonin 1a (5-HT1a) receptor partial agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| P14416 | ARIPIPRAZOLE | Dopamine D2 receptor partial agonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2002 |
| P18825 | ARIPIPRAZOLE | Alpha-2C adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2002 | ||
| P21917 | ARIPIPRAZOLE | D(4) dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2002 | ||
| P28223 | ARIPIPRAZOLE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| P28335 | ARIPIPRAZOLE | 5-hydroxytryptamine receptor 2C | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 | ||
| P35348 | ARIPIPRAZOLE | Alpha-1A adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2002 | ||
| P35368 | ARIPIPRAZOLE | Alpha-1B adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2002 | ||
| P35462 | ARIPIPRAZOLE | D(3) dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2002 | ||
| Q01959 | ARMODAFINIL | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2007 |
| Q16881 | ARSENIC TRIOXIDE | Thioredoxin reductase 1 inhibitor | CHEMBL1927 | Thioredoxin reductase 1 | "Thioredoxin reductase 1, cytoplasmic" | Homo sapiens | enzyme reductase | Small molecule | 2000 |
| ARTEMETHER | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 2009 | |||
| P35498 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| P35499 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q01118 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q14524 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q15858 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q99250 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9NY46 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UI33 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UQD0 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9Y5Y9 | ARTICAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| P14416 | ASENAPINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 0 |
| P28223 | ASENAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 0 |
| ASPARAGINASE | Asparagine hydrolytic enzyme | CHEMBL2364706 | Asparagine | Homo sapiens | Enzyme | 1994 | |||
| ASPARAGINASE ERWINIA CHRYSANTHEMI | Asparagine hydrolytic enzyme | CHEMBL2364706 | Asparagine | Homo sapiens | Enzyme | 2011 | |||
| P23219 | ASPIRIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P35354 | ASPIRIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P35367 | ASTEMIZOLE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1988 |
| Q72874 | ATAZANAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 2003 |
| P08588 | ATENOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1981 |
| P23975 | ATOMOXETINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2002 |
| P04035 | ATORVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1996 |
| Q02127 | ATOVAQUONE | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1992 | ||
| Q02768 | ATOVAQUONE | Cytochrome b inhibitor | CHEMBL1777 | Cytochrome b | Cytochrome b | Plasmodium falciparum | cytosolic other | Small molecule | 1992 |
| P02708 | ATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1983 |
| P07510 | ATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1983 |
| P11230 | ATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1983 |
| Q04844 | ATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1983 |
| Q07001 | ATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1983 |
| P08172 | ATROPINE | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 |
| P08173 | ATROPINE | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 | ||
| P08912 | ATROPINE | Muscarinic acetylcholine receptor M5 | Muscarinic acetylcholine receptor M5 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 | ||
| P11229 | ATROPINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 |
| P20309 | ATROPINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 |
| AURANOFIN | Unknown | Small molecule | 1985 | ||||||
| O76074 | AVANAFIL | Phosphodiesterase 5A inhibitor | CHEMBL1827 | Phosphodiesterase 5A | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 2011 |
| P05364 | AVIBACTAM | Beta-lactamase | Beta-lactamase | Enterobacter cloacae | enzyme | Small molecule | 2015 | ||
| P24735 | AVIBACTAM | Beta-lactamase | Beta-lactamase | Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 / 1C / PRS 101 / LMG 12228) | enzyme | Small molecule | 2015 | ||
| P62593 | AVIBACTAM | Bacterial beta-lactamase TEM inhibitor | CHEMBL2364670 | Bacterial beta-lactamase TEM | Beta-lactamase TEM | Bacteria | enzyme hydrolase | Small molecule | 2015 |
| Q9EXV5 | AVIBACTAM | Beta-lactamase | Beta-lactamase | Escherichia coli | unclassified | Small molecule | 2015 | ||
| P17948 | AXITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P35916 | AXITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P35968 | AXITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P26358 | AZACITIDINE | DNA (cytosine-5)-methyltransferase 1 inhibitor | CHEMBL1993 | DNA (cytosine-5)-methyltransferase 1 | DNA (cytosine-5)-methyltransferase 1 | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2004 |
| Q9Y6K1 | AZACITIDINE | DNA (cytosine-5)-methyltransferase 3A inhibitor | CHEMBL1992 | DNA (cytosine-5)-methyltransferase 3A | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator reader methyl-lysine pwwp | Small molecule | 2004 |
| Q9Y6K1 | AZACITIDINE | DNA (cytosine-5)-methyltransferase 3A inhibitor | CHEMBL1992 | DNA (cytosine-5)-methyltransferase 3A | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2004 |
| AZACITIDINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2004 | |||
| AZACITIDINE | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 2004 | |||
| P35367 | AZATADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1977 |
| P00492 | AZATHIOPRINE | Hypoxanthine-guanine phosphoribosyltransferase | Hypoxanthine-guanine phosphoribosyltransferase | Homo sapiens | enzyme | Small molecule | 1968 | ||
| P12268 | AZATHIOPRINE | Inosine-5'-monophosphate dehydrogenase 2 | Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 1968 | ||
| P20839 | AZATHIOPRINE | Inosine-5'-monophosphate dehydrogenase 1 | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1968 | ||
| Q06203 | AZATHIOPRINE | DNA inhibitor | CHEMBL2311221 | DNA | Amidophosphoribosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1968 |
| Q06203 | AZATHIOPRINE | Amidophosphoribosyltransferase inhibitor | CHEMBL2362992 | Amidophosphoribosyltransferase | Amidophosphoribosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1968 |
| AZATHIOPRINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1968 | |||
| AZELAIC ACID | Unknown | Small molecule | 1995 | ||||||
| P35367 | AZELASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1996 |
| P30556 | AZILSARTAN MEDOXOMIL | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 2011 |
| AZITHROMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1991 | ||
| Q07806 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | Penicillin-binding protein 1A | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| Q51504 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | Cell division protein | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| Q51505 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | Penicillin-binding protein 3A | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| Q9X6V3 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | Penicillin-binding protein 2 | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| Q9X6V7 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | D-ala-D-ala-carboxypeptidase | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| Q9X6W0 | AZLOCILLIN | Penicillin-binding protein inhibitor | CHEMBL2363020 | Penicillin-binding protein | Penicillin-binding protein | Pseudomonas aeruginosa | enzyme protease | Small molecule | 1982 |
| P02918 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1986 |
| P02919 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1986 |
| P08506 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1986 |
| P0AD65 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1986 |
| P0AD68 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1986 |
| P0AEB2 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1986 |
| P24228 | AZTREONAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1986 |
| P02918 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1980 |
| P02919 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1980 |
| P08506 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1980 |
| P0AD65 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1980 |
| P0AD68 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1980 |
| P0AEB2 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1980 |
| P24228 | BACAMPICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1980 |
| BACITRACIN | C55-isoprenyl pyrophosphate inhibitor | CHEMBL2364036 | C55-isoprenyl pyrophosphate | Bacteria | Protein | 1948 | |||
| O75899 | BACLOFEN | GABA-B receptor agonist | CHEMBL2111463 | GABA-B receptor | Gamma-aminobutyric acid type B receptor subunit 2 | Homo sapiens | membrane receptor 7tm3 smallmol neurotransmitter gaba-b receptor | Small molecule | 1977 |
| Q9UBS5 | BACLOFEN | GABA-B receptor agonist | CHEMBL2111463 | GABA-B receptor | Gamma-aminobutyric acid type B receptor subunit 1 | Homo sapiens | membrane receptor 7tm3 smallmol neurotransmitter gaba-b receptor | Small molecule | 1977 |
| P09917 | BALSALAZID | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 2000 |
| P23219 | BALSALAZID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 2000 |
| P35354 | BALSALAZID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 2000 |
| P37231 | BALSALAZID | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 2000 |
| P01589 | BASILIXIMAB | Interleukin-2 receptor inhibitor | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit alpha | Homo sapiens | membrane receptor | Antibody | 1998 |
| P03372 | BAZEDOXIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2009 |
| Q92731 | BAZEDOXIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 2009 |
| P09619 | BECAPLERMIN | Platelet-derived growth factor receptor agonist | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Protein | 1997 |
| P16234 | BECAPLERMIN | Platelet-derived growth factor receptor agonist | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Protein | 1997 |
| P04150 | BECLOMETHASONE DIPROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1976 |
| P9WPS1 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit c | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPU5 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit beta | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPU7 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit alpha | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPU9 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase gamma chain | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPV1 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase epsilon chain | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPV3 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit b-delta | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPV5 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit b | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P9WPV7 | BEDAQUILINE | ATP synthase inhibitor | CHEMBL2364166 | ATP synthase | ATP synthase subunit a | Mycobacterium tuberculosis | enzyme hydrolase | Small molecule | 2012 |
| P33681 | BELATACEPT | T-lymphocyte activation antigen CD80 inhibitor | CHEMBL2364157 | T-lymphocyte activation antigen CD80 | T-lymphocyte activation antigen CD80 | Homo sapiens | surface antigen | Protein | 2011 |
| P42081 | BELATACEPT | T-lymphocyte activation antigen CD86 inhibitor | CHEMBL2364156 | T-lymphocyte activation antigen CD86 | T-lymphocyte activation antigen CD86 | Homo sapiens | surface antigen | Protein | 2011 |
| Q9Y275 | BELIMUMAB | Tumor necrosis factor ligand superfamily member 13B inhibitor | CHEMBL2364158 | Tumor necrosis factor ligand superfamily member 13B | Tumor necrosis factor ligand superfamily member 13B | Homo sapiens | secreted | Antibody | 2011 |
| O15379 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 3 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2014 |
| P56524 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 4 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2014 |
| Q13547 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 1 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2014 |
| Q8WUI4 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 7 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2014 |
| Q92769 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 2 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2014 |
| Q969S8 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 10 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2014 |
| Q96DB2 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 11 | Homo sapiens | epigenetic regulator eraser hdac hdac class iv | Small molecule | 2014 |
| Q9BY41 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 8 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2014 |
| Q9UBN7 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 6 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2014 |
| Q9UKV0 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 9 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2014 |
| Q9UQL6 | BELINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 5 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2014 |
| P12821 | BENAZEPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1991 |
| BENDAMUSTINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2008 | |||
| P55017 | BENDROFLUMETHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1959 |
| P35498 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35499 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q01118 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q14524 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q15858 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q99250 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9NY46 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UI33 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UQD0 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | BENOXINATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| BENZONATATE | Slowly adapting pulmonary stretch receptor inhibitor | CHEMBL2364682 | Slowly adapting pulmonary stretch receptor | Homo sapiens | Small molecule | 1958 | |||
| P23975 | BENZPHETAMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 0 |
| Q05940 | BENZPHETAMINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 0 |
| P14416 | BENZQUINAMIDE | Dopamine D2 receptor modulator | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 |
| P55017 | BENZTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1960 |
| P08172 | BENZTROPINE | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 | ||
| P08173 | BENZTROPINE | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 | ||
| P08912 | BENZTROPINE | Muscarinic acetylcholine receptor M5 | Muscarinic acetylcholine receptor M5 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 | ||
| P11229 | BENZTROPINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 |
| P20309 | BENZTROPINE | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 | ||
| BENZYL ALCOHOL | Unknown | Small molecule | 2009 | ||||||
| BENZYL BENZOATE | Unknown | Small molecule | 1976 | ||||||
| P02918 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1947 |
| P02919 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1947 |
| P08506 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1947 |
| P0AD65 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1947 |
| P0AD68 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1947 |
| P0AEB2 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1947 |
| P24228 | BENZYLPENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1947 |
| P35367 | BEPOTASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2009 |
| O00305 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit beta-4 | Homo sapiens | auxiliary transport protein ca beta | Small molecule | 1990 |
| O00555 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent P/Q-type calcium channel subunit alpha-1A | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| O43497 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| O60359 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-3 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| O60840 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| O95180 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| P54284 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit beta-3 | Homo sapiens | auxiliary transport protein ca beta | Small molecule | 1990 |
| P54289 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 1990 |
| P62955 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-7 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q00975 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent N-type calcium channel subunit alpha-1B | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q01668 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q02641 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit beta-1 | Homo sapiens | auxiliary transport protein ca beta | Small molecule | 1990 |
| Q06432 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-1 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q08289 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit beta-2 | Homo sapiens | auxiliary transport protein ca beta | Small molecule | 1990 |
| Q13698 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q13936 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q15878 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent R-type calcium channel subunit alpha-1E | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q7Z3S7 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-4 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 1990 |
| Q8IZS8 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-3 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 1990 |
| Q8WXS5 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-8 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q9BXT2 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-6 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q9NY47 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-2 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 1990 |
| Q9P0X4 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q9UBN1 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-4 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q9UF02 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-5 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| Q9Y698 | BEPRIDIL | Voltage-gated calcium channel blocker | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel gamma-2 subunit | Homo sapiens | auxiliary transport protein ca gamma | Small molecule | 1990 |
| BERACTANT | Surfactant agent | Unknown | 1991 | ||||||
| P0AES4 | BESIFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 2009 |
| P0AES6 | BESIFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 2009 |
| P0AFI2 | BESIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 2009 |
| P20083 | BESIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 2009 |
| Q93088 | BETAINE | Betaine-homocysteine S-methyltransferase substrate | CHEMBL3391661 | Betaine-homocysteine S-methyltransferase | Betaine--homocysteine S-methyltransferase 1 | Homo sapiens | enzyme | Small molecule | 1996 |
| Q9H2M3 | BETAINE | Betaine-homocysteine S-methyltransferase substrate | CHEMBL3391661 | Betaine-homocysteine S-methyltransferase | S-methylmethionine--homocysteine S-methyltransferase BHMT2 | Homo sapiens | enzyme | Small molecule | 1996 |
| BETAINE | homocysteine | Homo sapiens | Small molecule | 1996 | |||||
| P04150 | BETAMETHASONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1961 |
| P04150 | BETAMETHASONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1965 |
| P04150 | BETAMETHASONE BENZOATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P04150 | BETAMETHASONE DIPROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1975 |
| P04150 | BETAMETHASONE PHOSPHORIC ACID | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1965 |
| P04150 | BETAMETHASONE VALERATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1967 |
| P08588 | BETAXOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P25021 | BETAZOLE | Histamine H2 receptor agonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| P08172 | BETHANECHOL | Muscarinic acetylcholine receptor M2 agonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1948 |
| P08173 | BETHANECHOL | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1948 | ||
| P20309 | BETHANECHOL | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1948 |
| P23975 | BETHANIDINE | Norepinephrine transporter substrate | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 |
| P15692 | BEVACIZUMAB | Vascular endothelial growth factor A inhibitor | CHEMBL1783 | Vascular endothelial growth factor A | Vascular endothelial growth factor A | Homo sapiens | secreted | Antibody | 2004 |
| P19793 | BEXAROTENE | Retinoid X receptor agonist | CHEMBL2363070 | Retinoid X receptor | Retinoic acid receptor RXR-alpha | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b1 | Small molecule | 1999 |
| P28702 | BEXAROTENE | Retinoid X receptor agonist | CHEMBL2363070 | Retinoid X receptor | Retinoic acid receptor RXR-beta | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b2 | Small molecule | 1999 |
| P48443 | BEXAROTENE | Retinoid X receptor agonist | CHEMBL2363070 | Retinoid X receptor | Retinoic acid receptor RXR-gamma | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b3 | Small molecule | 1999 |
| P10275 | BICALUTAMIDE | Androgen Receptor antagonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1995 |
| P43088 | BIMATOPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 2001 |
| P11229 | BIPERIDEN | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1959 |
| BISACODYL | Unknown | Small molecule | 2004 | ||||||
| P23219 | BISMUTH SUBSALICYLATE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1996 |
| P35354 | BISMUTH SUBSALICYLATE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1996 |
| P08588 | BISOPROLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1992 |
| P07550 | BITOLTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P00734 | BIVALIRUDIN | Thrombin inhibitor | CHEMBL204 | Thrombin | Prothrombin | Homo sapiens | enzyme protease serine pas s1a | Protein | 2000 |
| BLEOMYCIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1973 | |||
| P04234 | BLINATUMOMAB | T cell surface glycoprotein CD3 cross-linking agent | CHEMBL2364168 | T cell surface glycoprotein CD3 | T-cell surface glycoprotein CD3 delta chain | Homo sapiens | unclassified | Antibody | 2014 |
| P07766 | BLINATUMOMAB | T cell surface glycoprotein CD3 cross-linking agent | CHEMBL2364168 | T cell surface glycoprotein CD3 | T-cell surface glycoprotein CD3 epsilon chain | Homo sapiens | membrane receptor | Antibody | 2014 |
| P09693 | BLINATUMOMAB | T cell surface glycoprotein CD3 cross-linking agent | CHEMBL2364168 | T cell surface glycoprotein CD3 | T-cell surface glycoprotein CD3 gamma chain | Homo sapiens | unclassified | Antibody | 2014 |
| P15391 | BLINATUMOMAB | B-lymphocyte antigen CD19 cross-linking agent | CHEMBL3390821 | B-lymphocyte antigen CD19 | Homo sapiens | surface antigen | Antibody | 2014 | |
| A3EZI9 | BOCEPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | NS3 | Hepatitis C virus | enzyme protease serine pas s29 | Small molecule | 2011 |
| D2K2A8 | BOCEPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | Non-structural protein 4A | Hepatitis C virus | enzyme protease serine pas s29 reg | Small molecule | 2011 |
| P28074 | BORTEZOMIB | 26S proteosome inhibitor | CHEMBL2364701 | 26S proteosome | Proteasome subunit beta type-5 | Homo sapiens | enzyme protease threonine pbt t1a | Small molecule | 2003 |
| P24530 | BOSENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin B receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2001 |
| P25101 | BOSENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin-1 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2001 |
| P00519 | BOSUTINIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2010 |
| P07948 | BOSUTINIB | Tyrosine-protein kinase Lyn inhibitor | CHEMBL3905 | Tyrosine-protein kinase Lyn | Tyrosine-protein kinase Lyn | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2010 |
| P08631 | BOSUTINIB | Tyrosine-protein kinase HCK inhibitor | CHEMBL3234 | Tyrosine-protein kinase HCK | Tyrosine-protein kinase HCK | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2010 |
| P12931 | BOSUTINIB | Tyrosine-protein kinase SRC inhibitor | CHEMBL267 | Tyrosine-protein kinase SRC | Proto-oncogene tyrosine-protein kinase Src | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2010 |
| P60880 | BOTULINUM TOXIN TYPE A PURIFIED NEUROTOXIN COMPLEX | Synaptosomal-associated protein 25 inhibitor | CHEMBL2364159 | Synaptosomal-associated protein 25 | Synaptosomal-associated protein 25 | Homo sapiens | cytosolic other | Unknown | 1991 |
| P63027 | BOTULINUM TOXIN TYPE B | Vesicle-associated membrane protein 2 inhibitor | CHEMBL2364160 | Vesicle-associated membrane protein 2 | Vesicle-associated membrane protein 2 | Homo sapiens | ion channel other vesicle | Unknown | 2000 |
| P04350 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Antibody | 2011 |
| P07437 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Antibody | 2011 |
| P28908 | BRENTUXIMAB VEDOTIN | Tumor necrosis factor receptor superfamily member 8 inhibitor | CHEMBL2364161 | Tumor necrosis factor receptor superfamily member 8 | Tumor necrosis factor receptor superfamily member 8 | Homo sapiens | secreted | Antibody | 2011 |
| P68371 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Antibody | 2011 |
| Q13509 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Antibody | 2011 |
| Q13885 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Antibody | 2011 |
| Q3ZCM7 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Antibody | 2011 |
| Q9BUF5 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Antibody | 2011 |
| Q9BVA1 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Antibody | 2011 |
| Q9H4B7 | BRENTUXIMAB VEDOTIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Antibody | 2011 |
| P23975 | BRETYLIUM | Norepinephrine transporter substrate | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1986 |
| P08908 | BREXPIPRAZOLE | Serotonin 1a (5-HT1a) receptor partial agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2015 |
| P14416 | BREXPIPRAZOLE | Dopamine D2 receptor partial agonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2015 |
| P28223 | BREXPIPRAZOLE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2015 |
| P08913 | BRIMONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18089 | BRIMONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18825 | BRIMONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P00918 | BRINZOLAMIDE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1998 |
| P23219 | BROMFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 2005 |
| P35354 | BROMFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 2005 |
| P08908 | BROMOCRIPTINE | 5-hydroxytryptamine receptor 1A | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1978 | ||
| P08913 | BROMOCRIPTINE | Alpha-2A adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 | ||
| P14416 | BROMOCRIPTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1978 |
| P21728 | BROMOCRIPTINE | D(1A) dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1978 | ||
| P21917 | BROMOCRIPTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1978 |
| P25100 | BROMOCRIPTINE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 | ||
| P28221 | BROMOCRIPTINE | 5-hydroxytryptamine receptor 1D | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1978 | ||
| P35348 | BROMOCRIPTINE | Alpha-1A adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 | ||
| P35462 | BROMOCRIPTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1978 |
| P41595 | BROMOCRIPTINE | 5-hydroxytryptamine receptor 2B | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1978 | ||
| P35367 | BROMODIPHENHYDRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1954 |
| P35367 | BROMPHENIRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1957 |
| P35367 | BUCLIZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| P04150 | BUDESONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1994 |
| P05023 | BUMETANIDE | Sodium/potassium-transporting ATPase subunit alpha-1 | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 1983 | ||
| P05023 | BUMETANIDE | Sodium/potassium-transporting ATPase subunit alpha-1 | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1983 | ||
| P55011 | BUMETANIDE | Solute carrier family 12 member 2 | Solute carrier family 12 member 2 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1983 | ||
| Q13621 | BUMETANIDE | Sodium-(potassium)-chloride cotransporter 2 inhibitor | CHEMBL1874 | Sodium-(potassium)-chloride cotransporter 2 | Solute carrier family 12 member 1 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1983 |
| P35499 | BUPIVACAINE | Sodium channel protein type IV alpha subunit blocker | CHEMBL2072 | Sodium channel protein type IV alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1972 |
| P35372 | BUPRENORPHINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1981 |
| P41143 | BUPRENORPHINE | Delta-type opioid receptor | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1981 | ||
| P41145 | BUPRENORPHINE | Kappa opioid receptor agonist | CHEMBL237 | Kappa opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1981 |
| P23975 | BUPROPION | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1985 |
| Q01959 | BUPROPION | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1985 |
| P08908 | BUSPIRONE | Serotonin 1a (5-HT1a) receptor partial agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1986 |
| P14416 | BUSPIRONE | D(2) dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1986 | ||
| P21917 | BUSPIRONE | D(4) dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1986 | ||
| Q99720 | BUSPIRONE | Sigma non-opioid intracellular receptor 1 | Sigma non-opioid intracellular receptor 1 | Homo sapiens | membrane receptor | Small molecule | 1986 | ||
| BUSULFAN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1954 | |||
| P18505 | BUTABARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1939 |
| P28472 | BUTABARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1939 |
| P47870 | BUTABARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1939 |
| P18505 | BUTALBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1983 |
| P28472 | BUTALBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1983 |
| P47870 | BUTALBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1983 |
| Q4JEY0 | BUTENAFINE | Squalene monooxygenase inhibitor | CHEMBL2364679 | Squalene monooxygenase | Squalene epoxidase | Trichophyton | enzyme reductase | Small molecule | 1996 |
| P10613 | BUTOCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1985 |
| P35372 | BUTORPHANOL | Mu opioid receptor partial agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1978 |
| P41145 | BUTORPHANOL | Kappa opioid receptor partial agonist | CHEMBL237 | Kappa opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1978 |
| P04350 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 2010 |
| P07437 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 2010 |
| P68371 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 2010 |
| Q13509 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q13885 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 2010 |
| Q3ZCM7 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9BUF5 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9BVA1 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9H4B7 | CABAZITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 2010 |
| P08908 | CABERGOLINE | 5-hydroxytryptamine receptor 1A | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 | ||
| P08913 | CABERGOLINE | Alpha-2A adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 | ||
| P14416 | CABERGOLINE | Dopamine D2 receptor agonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 |
| P18825 | CABERGOLINE | Alpha-2C adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 | ||
| P21917 | CABERGOLINE | Dopamine receptor D4 | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 | ||
| P21918 | CABERGOLINE | Dopamine receptor D5 | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 | ||
| P28221 | CABERGOLINE | 5-hydroxytryptamine receptor 1D | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 | ||
| P28223 | CABERGOLINE | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 | ||
| P35462 | CABERGOLINE | Dopamine receptor D3 | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 | ||
| P07949 | CABOZANTINIB | Proto-oncogene tyrosine-protein kinase receptor Ret | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2012 | ||
| P08581 | CABOZANTINIB | Hepatocyte growth factor receptor inhibitor | CHEMBL3717 | Hepatocyte growth factor receptor | Hepatocyte growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk met | Small molecule | 2012 |
| P10721 | CABOZANTINIB | Mast/stem cell growth factor receptor Kit | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 | ||
| P35968 | CABOZANTINIB | Vascular endothelial growth factor receptor 2 inhibitor | CHEMBL279 | Vascular endothelial growth factor receptor 2 | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P36888 | CABOZANTINIB | Receptor-type tyrosine-protein kinase FLT3 | Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 | ||
| Q02763 | CABOZANTINIB | Angiopoietin-1 receptor | Angiopoietin-1 receptor | Homo sapiens | enzyme kinase protein kinase tk tie | Small molecule | 2012 | ||
| O15554 | CAFFEINE | Intermediate conductance calcium-activated potassium channel protein 4 | Intermediate conductance calcium-activated potassium channel protein 4 | Homo sapiens | ion channel vgc k ca act k | Small molecule | 1948 | ||
| P0DMS8 | CAFFEINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A3 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1948 |
| P29274 | CAFFEINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1948 |
| P29275 | CAFFEINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2b | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1948 |
| P30542 | CAFFEINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A1 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1948 |
| Q07343 | CAFFEINE | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1948 | ||
| P11473 | CALCIFEDIOL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 0 |
| P11473 | CALCIPOTRIENE | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1993 |
| P30988 | CALCITONIN HUMAN | Calcitonin receptor agonist | CHEMBL1832 | Calcitonin receptor | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 1986 |
| P30988 | CALCITONIN SALMON | Calcitonin receptor agonist | CHEMBL1832 | Calcitonin receptor | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 1978 |
| P30988 | CALCITONIN SALMON RECOMBINANT | Calcitonin receptor agonist | CHEMBL1832 | Calcitonin receptor | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 2005 |
| P11473 | CALCITRIOL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1978 |
| CALCIUM ACETATE | Phosphate chelating agent | CHEMBL2364184 | Phosphate | Homo sapiens | Small molecule | 1982 | |||
| CALFACTANT | Surfactant agent | Unknown | 1998 | ||||||
| P31639 | CANAGLIFLOZIN | Sodium/glucose cotransporter 2 inhibitor | CHEMBL3884 | Sodium/glucose cotransporter 2 | Sodium/glucose cotransporter 2 | Homo sapiens | transporter electrochemical slc slc05 | Small molecule | 2011 |
| P01584 | CANAKINUMAB | Interleukin-1 beta inhibitor | CHEMBL1909490 | Interleukin-1 beta | Interleukin-1 beta | Homo sapiens | secreted | Antibody | 2009 |
| P30556 | CANDESARTAN CILEXETIL | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1998 |
| CANDICIDIN | Cell membrane inhibitor | CHEMBL2364035 | Cell membrane | Candida albicans | Small molecule | 1982 | |||
| Q9H244 | CANGRELOR | Purinergic receptor P2Y12 antagonist | CHEMBL2001 | Purinergic receptor P2Y12 | P2Y purinoceptor 12 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor purine receptor | Small molecule | 2015 |
| P04818 | CAPECITABINE | Thymidylate synthase inhibitor | CHEMBL1952 | Thymidylate synthase | Thymidylate synthase | Homo sapiens | enzyme transferase | Small molecule | 1998 |
| CAPECITABINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1998 | |||
| CAPECITABINE | DNA inhibitor | CHEMBL2311221 | RNA | Homo sapiens | Small molecule | 1998 | |||
| CAPECITABINE | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 1998 | |||
| CAPREOMYCINE | 70S ribosome inhibitor | CHEMBL2363965 | 70S ribosome | 16S ribosomal RNA | Mycobacterium tuberculosis | Protein | 1971 | ||
| CAPREOMYCINE | 70S ribosome inhibitor | CHEMBL2363965 | 70S ribosome | 23S ribosomal RNA | Mycobacterium tuberculosis | Protein | 1971 | ||
| Q8NER1 | CAPSAICIN | Vanilloid receptor opener | CHEMBL4794 | Vanilloid receptor | Transient receptor potential cation channel subfamily V member 1 | Homo sapiens | ion channel vgc trp | Small molecule | 2009 |
| P12821 | CAPTOPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1981 |
| P20309 | CARBACHOL CHLORIDE | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1972 |
| P30926 | CARBAMAZEPINE | Neuronal acetylcholine receptor; alpha2/beta4 | Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1968 | ||
| P31645 | CARBAMAZEPINE | Sodium-dependent serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1968 | ||
| P35498 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| P35499 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q01118 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q14524 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q15822 | CARBAMAZEPINE | Neuronal acetylcholine receptor; alpha2/beta4 | Neuronal acetylcholine receptor subunit alpha-2 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1968 | ||
| Q15858 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q99250 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q9NY46 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q9UI33 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q9UQD0 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| Q9Y5Y9 | CARBAMAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1968 |
| P02918 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P02919 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1982 |
| P08506 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P0AD65 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P0AD68 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1982 |
| P0AEB2 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P24228 | CARBENICILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1982 |
| P02918 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1972 |
| P02919 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1972 |
| P08506 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1972 |
| P0AD65 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1972 |
| P0AD68 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1972 |
| P0AEB2 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1972 |
| P24228 | CARBENICILLIN INDANYL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1972 |
| P20711 | CARBIDOPA | DOPA decarboxylase inhibitor | CHEMBL1843 | DOPA decarboxylase | Aromatic-L-amino-acid decarboxylase | Homo sapiens | enzyme lyase | Small molecule | 1975 |
| P35367 | CARBINOXAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2003 |
| CARBOPLATIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1989 | |||
| P35408 | CARBOPROST | Prostaglandin E2 receptor EP4 subtype | Prostaglandin E2 receptor EP4 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1979 | ||
| P43088 | CARBOPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1979 |
| P43116 | CARBOPROST | Prostaglandin E2 receptor EP2 subtype | Prostaglandin E2 receptor EP2 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1979 | ||
| P28074 | CARFILZOMIB | 26S proteosome inhibitor | CHEMBL2364701 | 26S proteosome | Proteasome subunit beta type-5 | Homo sapiens | enzyme protease threonine pbt t1a | Protein | 2009 |
| P31327 | CARGLUMIC ACID | "Carbamoyl-phosphate synthase [ammonia], mitochondrial positive allosteric modulator" | CHEMBL2362990 | "Carbamoyl-phosphate synthase [ammonia], mitochondrial" | "Carbamoyl-phosphate synthase [ammonia], mitochondrial" | Homo sapiens | enzyme ligase | Small molecule | 2010 |
| CARISOPRODOL | Unknown | Small molecule | 1959 | ||||||
| P00390 | CARMUSTINE | Glutathione reductase inhibitor | CHEMBL2755 | Glutathione reductase | "Glutathione reductase, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1977 |
| CARMUSTINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1977 | |||
| CARMUSTINE | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 1977 | |||
| P14416 | CARPHENAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1982 |
| P28223 | CARPHENAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1982 |
| P28335 | CARPHENAZINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1982 |
| P35354 | CARPROFEN | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1987 |
| P07550 | CARTEOLOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1988 |
| P08588 | CARTEOLOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1988 |
| P13945 | CARTEOLOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1988 |
| P07550 | CARVEDILOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P08588 | CARVEDILOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P08908 | CARVEDILOL | 5-hydroxytryptamine receptor 1A | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1995 | ||
| P13945 | CARVEDILOL | Adrenergic receptor beta antagonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P25100 | CARVEDILOL | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P35348 | CARVEDILOL | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P35368 | CARVEDILOL | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1995 |
| P41595 | CARVEDILOL | 5-hydroxytryptamine receptor 2B | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1995 | ||
| O13428 | CASPOFUNGIN | "1,3-beta-glucan synthase inhibitor" | CHEMBL2364673 | "1,3-beta-glucan synthase" | "Beta-1,3-glucan synthase catalytic subunit 1" | Candida | enzyme transferase | Small molecule | 2001 |
| Q4WLT4 | CASPOFUNGIN | "1,3-beta-glucan synthase inhibitor" | CHEMBL2364674 | "1,3-beta-glucan synthase" | "1,3-beta-glucan synthase catalytic subunit FksP" | Aspergillus | enzyme transferase | Small molecule | 2001 |
| P02918 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1979 |
| P02919 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1979 |
| P08506 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1979 |
| P0AD65 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1979 |
| P0AD68 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1979 |
| P0AEB2 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1979 |
| P24228 | CEFACLOR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1979 |
| P02918 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P02919 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1978 |
| P08506 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P0AD65 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P0AD68 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1978 |
| P0AEB2 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P24228 | CEFADROXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1978 |
| P02918 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P02919 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1978 |
| P08506 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P0AD65 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P0AD68 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1978 |
| P0AEB2 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P24228 | CEFAMANDOLE NAFATE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1978 |
| P02918 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1973 |
| P02919 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1973 |
| P08506 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1973 |
| P0AD65 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1973 |
| P0AD68 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1973 |
| P0AEB2 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1973 |
| P24228 | CEFAZOLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1973 |
| P02918 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1997 |
| P02919 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1997 |
| P08506 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1997 |
| P0AD65 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1997 |
| P0AD68 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1997 |
| P0AEB2 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1997 |
| P24228 | CEFDINIR | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1997 |
| P02918 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 2001 |
| P02919 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 2001 |
| P08506 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 2001 |
| P0AD65 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 2001 |
| P0AD68 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 2001 |
| P0AEB2 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 2001 |
| P24228 | CEFDITOREN PIVOXIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 2001 |
| P02918 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1996 |
| P02919 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1996 |
| P08506 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1996 |
| P0AD65 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1996 |
| P0AD68 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1996 |
| P0AEB2 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1996 |
| P24228 | CEFEPIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1996 |
| P02918 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P02919 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1989 |
| P08506 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P0AD65 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P0AD68 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1989 |
| P0AEB2 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P10520 | CEFIXIME | Streptokinase A | Streptokinase A | Streptococcus pyogenes serotype M1 | unclassified | Small molecule | 1989 | ||
| P24228 | CEFIXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1989 |
| P02918 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1987 |
| P02919 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1987 |
| P08506 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1987 |
| P0AD65 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1987 |
| P0AD68 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1987 |
| P0AEB2 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1987 |
| P24228 | CEFMENOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1987 |
| P02918 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P02919 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1989 |
| P08506 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P0AD65 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P0AD68 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1989 |
| P0AEB2 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P24228 | CEFMETAZOLE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1989 |
| P02918 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P02919 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1984 |
| P08506 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P0AD65 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P0AD68 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1984 |
| P0AEB2 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P24228 | CEFONICID | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1984 |
| P02918 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P02919 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1982 |
| P08506 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P0AD65 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P0AD68 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1982 |
| P0AEB2 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P24228 | CEFOPERAZONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1982 |
| P02918 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P02919 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1984 |
| P08506 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P0AD65 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P0AD68 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1984 |
| P0AEB2 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P24228 | CEFORANIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1984 |
| P02918 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P02919 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1981 |
| P08506 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P0AD65 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P0AD68 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1981 |
| P0AEB2 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P24228 | CEFOTAXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1981 |
| P02918 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P02919 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1985 |
| P08506 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P0AD65 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P0AD68 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1985 |
| P0AEB2 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P24228 | CEFOTETAN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1985 |
| P02918 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1988 |
| P02919 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1988 |
| P08506 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1988 |
| P0AD65 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1988 |
| P0AD68 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1988 |
| P0AEB2 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1988 |
| P24228 | CEFOTIAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1988 |
| P02918 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P02919 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1978 |
| P08506 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P0AD65 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1978 |
| P0AD68 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1978 |
| P0AEB2 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1978 |
| P24228 | CEFOXITIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1978 |
| P02918 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P02919 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1989 |
| P08506 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P0AD65 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1989 |
| P0AD68 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1989 |
| P0AEB2 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1989 |
| P24228 | CEFPIRAMIDE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1989 |
| P02918 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1992 |
| P02919 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1992 |
| P08506 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1992 |
| P0AD65 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1992 |
| P0AD68 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1992 |
| P0AEB2 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1992 |
| P24228 | CEFPODOXIME PROXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1992 |
| P02918 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 0 |
| P02919 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 0 |
| P08506 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 0 |
| P0AD65 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 0 |
| P0AD68 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 0 |
| P0AEB2 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 0 |
| P24228 | CEFPROZIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 0 |
| P02918 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 2010 |
| P02919 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 2010 |
| P08506 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 2010 |
| P0AD65 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 2010 |
| P0AD68 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 2010 |
| P0AEB2 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 2010 |
| P24228 | CEFTAROLINE FOSAMIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 2010 |
| P02918 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P02919 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1985 |
| P08506 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P0AD65 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P0AD68 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1985 |
| P0AEB2 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P24228 | CEFTAZIDIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1985 |
| P02918 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1995 |
| P02919 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1995 |
| P08506 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1995 |
| P0AD65 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1995 |
| P0AD68 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1995 |
| P0AEB2 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1995 |
| P24228 | CEFTIBUTEN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1995 |
| P02918 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1983 |
| P02919 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1983 |
| P08506 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1983 |
| P0AD65 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1983 |
| P0AD68 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1983 |
| P0AEB2 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1983 |
| P24228 | CEFTIZOXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1983 |
| P02918 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 2014 |
| P02919 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 2014 |
| P08506 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 2014 |
| P0AD65 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 2014 |
| P0AD68 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 2014 |
| P0AEB2 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 2014 |
| P24228 | CEFTOLOZANE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 2014 |
| P02918 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P02919 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1984 |
| P08506 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P0AD65 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1984 |
| P0AD68 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1984 |
| P0AEB2 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1984 |
| P24228 | CEFTRIAXONE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1984 |
| P02918 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1983 |
| P02919 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1983 |
| P08506 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1983 |
| P0AD65 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1983 |
| P0AD68 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1983 |
| P0AEB2 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1983 |
| P24228 | CEFUROXIME | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1983 |
| P02918 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1987 |
| P02919 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1987 |
| P08506 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1987 |
| P0AD65 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1987 |
| P0AD68 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1987 |
| P0AEB2 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1987 |
| P24228 | CEFUROXIME AXETIL | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1987 |
| P35354 | CELECOXIB | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1998 |
| P02918 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1971 |
| P02919 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1971 |
| P08506 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1971 |
| P0AD65 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1971 |
| P0AD68 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1971 |
| P0AEB2 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1971 |
| P24228 | CEPHALEXIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1971 |
| P02918 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1970 |
| P02919 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1970 |
| P08506 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1970 |
| P0AD65 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1970 |
| P0AD68 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1970 |
| P0AEB2 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1970 |
| P24228 | CEPHALOGLYCIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1970 |
| P02918 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P02919 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1974 |
| P08506 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P0AD65 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P0AD68 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1974 |
| P0AEB2 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P24228 | CEPHALOTHIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1974 |
| P02918 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P02919 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1974 |
| P08506 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P0AD65 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P0AD68 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1974 |
| P0AEB2 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P24228 | CEPHAPIRIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1974 |
| P02918 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P02919 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1974 |
| P08506 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P0AD65 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1974 |
| P0AD68 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1974 |
| P0AEB2 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1974 |
| P24228 | CEPHRADINE | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1974 |
| Q9UM73 | CERITINIB | ALK tyrosine kinase receptor inhibitor | CHEMBL4247 | ALK tyrosine kinase receptor | ALK tyrosine kinase receptor | Homo sapiens | enzyme kinase protein kinase tkl stkr type1 | Small molecule | 2014 |
| P04035 | CERIVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1997 |
| P01375 | CERTOLIZUMAB PEGOL | TNF-alpha inhibitor | CHEMBL1825 | TNF-alpha | Tumor necrosis factor | Homo sapiens | secreted | Antibody | 2008 |
| P32238 | CERULETIDE | Cholecystokinin A receptor agonist | CHEMBL1901 | Cholecystokinin A receptor | Cholecystokinin receptor type A | Homo sapiens | membrane receptor 7tm1 peptide short peptide cholecystokinin receptor | Protein | 1982 |
| P35367 | CETIRIZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1995 |
| P30968 | CETRORELIX | Gonadotropin-releasing hormone receptor antagonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 2000 |
| P00533 | CETUXIMAB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Antibody | 2004 |
| CETYL ALCOHOL | Unknown | Small molecule | 1990 | ||||||
| P11229 | CEVIMELINE | Muscarinic acetylcholine receptor M1 agonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2000 |
| P20309 | CEVIMELINE | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2000 |
| Q96RI1 | CHENODIOL | Bile acid receptor FXR agonist | CHEMBL2047 | Bile acid receptor FXR | Bile acid receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1h nr1h4 | Small molecule | 1983 |
| CHLOPHEDIANOL | Unknown | Small molecule | 1982 | ||||||
| CHLORAMBUCIL | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1957 | |||
| CHLORAMPHENICOL | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1950 | ||
| CHLORAMPHENICOL PALMITATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1982 | ||
| CHLORAMPHENICOL SUCCINIC ACID | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1959 | ||
| P14867 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P18507 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P31644 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P34903 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P47869 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| Q8N1C3 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| Q99928 | CHLORDIAZEPOXIDE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| CHLORHEXIDINE | Cell membrane inhibitor | CHEMBL2364031 | Cell membrane | Bacteria | Small molecule | 1976 | |||
| CHLORMEZANONE | Unknown | Small molecule | 1960 | ||||||
| P13922 | CHLOROGUANIDE | Dihydrofolate reductase inhibitor | CHEMBL1939 | Dihydrofolate reductase | Bifunctional dihydrofolate reductase-thymidylate synthase | Plasmodium falciparum K1 | enzyme reductase | Small molecule | 2000 |
| P35498 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| P35499 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q01118 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q14524 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q15858 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q99250 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q9NY46 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q9UI33 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q9UQD0 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| Q9Y5Y9 | CHLOROPROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1955 |
| P69905 | CHLOROQUINE | Hemoglobin subunit alpha | Hemoglobin subunit alpha | Homo sapiens | secreted | Small molecule | 1949 | ||
| CHLOROQUINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 1949 | |||
| P55017 | CHLOROTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1958 |
| Q92731 | CHLOROTRIANISENE | Estrogen receptor beta modulator | CHEMBL242 | Estrogen receptor beta | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1982 |
| CHLOROXINE | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1976 | |||
| CHLORPHENESIN CARBAMATE | Unknown | Small molecule | 1965 | ||||||
| P35367 | CHLORPHENIRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1950 |
| P31645 | CHLORPHENTERMINE | Serotonin transporter substrate | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 |
| P14416 | CHLORPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1957 |
| P21917 | CHLORPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1957 |
| P25100 | CHLORPROMAZINE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1957 | ||
| P28223 | CHLORPROMAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1957 |
| P28335 | CHLORPROMAZINE | 5-hydroxytryptamine receptor 2C | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1957 | ||
| P35367 | CHLORPROMAZINE | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1957 | ||
| P35368 | CHLORPROMAZINE | Alpha-1B adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1957 | ||
| P35462 | CHLORPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1957 |
| Q9H3N8 | CHLORPROMAZINE | Histamine H4 receptor | Histamine H4 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1957 | ||
| Q09428 | CHLORPROPAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1958 |
| Q14654 | CHLORPROPAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1958 |
| P14416 | CHLORPROTHIXENE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P28223 | CHLORPROTHIXENE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1967 |
| P28335 | CHLORPROTHIXENE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1967 |
| P35462 | CHLORPROTHIXENE | Dopamine D3 receptor antagonist | CHEMBL234 | Dopamine D3 receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| CHLORTETRACYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1950 | ||
| P55017 | CHLORTHALIDONE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1960 |
| Q13621 | CHLORTHALIDONE | Solute carrier family 12 member 1 | Solute carrier family 12 member 1 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1960 | ||
| O15554 | CHLORZOXAZONE | Intermediate conductance calcium-activated potassium channel protein 4 opener | CHEMBL4305 | Intermediate conductance calcium-activated potassium channel protein 4 | Intermediate conductance calcium-activated potassium channel protein 4 | Homo sapiens | ion channel vgc k ca act k | Small molecule | 1958 |
| Q12791 | CHLORZOXAZONE | Calcium-activated potassium channel subunit alpha-1 | Calcium-activated potassium channel subunit alpha-1 | Homo sapiens | ion channel vgc k ca act k | Small molecule | 1958 | ||
| P11473 | CHOLECALCIFEROL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1999 |
| CHOLESTYRAMINE | Bile acids chelating agent | CHEMBL2364175 | Bile acids | Homo sapiens | Unknown | 1973 | |||
| CHOLIC ACID | Unknown | Small molecule | 2015 | ||||||
| P22888 | CHORIOGONADOTROPIN ALFA | Luteinizing hormone/Choriogonadotropin receptor agonist | CHEMBL1854 | Luteinizing hormone/Choriogonadotropin receptor | Lutropin-choriogonadotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Protein | 2000 |
| CHROMIC PHOSPHATE | Unknown | Small molecule | 1974 | ||||||
| CHYMOPAPAIN | Polypeptides proteolytic enzyme | CHEMBL2364181 | Polypeptides | Homo sapiens | Unknown | 1982 | |||
| CHYMOTRYPSIN | Polypeptides proteolytic enzyme | CHEMBL2364181 | Polypeptides | Homo sapiens | Unknown | 1959 | |||
| P04150 | CICLESONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 2006 |
| CICLOPIROX | Iron chelating agent | CHEMBL2363058 | Iron | Small molecule | 1982 | ||||
| CICLOPIROX | CHEMBL2363058 | Iron | Small molecule | 1982 | |||||
| CICLOPIROX | Aluminium chelating agent | CHEMBL2366381 | Aluminium | Small molecule | 1982 | ||||
| CICLOPIROX | CHEMBL2366381 | Aluminium | Small molecule | 1982 | |||||
| P04293 | CIDOFOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1996 |
| P07918 | CIDOFOVIR | DNA polymerase catalytic subunit | DNA polymerase catalytic subunit | Human herpesvirus 2 (strain 186) | Transferase | Small molecule | 1996 | ||
| P08546 | CIDOFOVIR | DNA polymerase catalytic subunit | DNA polymerase catalytic subunit | Human cytomegalovirus (strain AD169) | enzyme | Small molecule | 1996 | ||
| P16444 | CILASTATIN | Renal dipeptidase inhibitor | CHEMBL1989 | Renal dipeptidase | Dipeptidase 1 | Homo sapiens | enzyme protease metallo mj m19 | Small molecule | 1985 |
| P27815 | CILOSTAZOL | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1999 | ||
| Q14432 | CILOSTAZOL | Phosphodiesterase 3A inhibitor | CHEMBL241 | Phosphodiesterase 3A | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1999 |
| P25021 | CIMETIDINE | Histamine H2 receptor antagonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1977 |
| P41180 | CINACALCET | Calcium sensing receptor positive allosteric modulator | CHEMBL1878 | Calcium sensing receptor | Extracellular calcium-sensing receptor | Homo sapiens | membrane receptor 7tm3 ion calcium sensing receptor calcium sensing receptor | Small molecule | 2004 |
| P0AES4 | CINOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1980 |
| P0AES6 | CINOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1980 |
| P0AES4 | CIPROFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1987 |
| P0AES6 | CIPROFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1987 |
| P0C1U9 | CIPROFLOXACIN | DNA topoisomerase 4 subunit A | DNA topoisomerase 4 subunit A | Staphylococcus aureus | enzyme | Small molecule | 1987 | ||
| Q13639 | CISAPRIDE | Serotonin 4 (5-HT4) receptor agonist | CHEMBL1875 | Serotonin 4 (5-HT4) receptor | 5-hydroxytryptamine receptor 4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1993 |
| P02708 | CISATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1995 |
| P07510 | CISATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1995 |
| P11230 | CISATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1995 |
| Q04844 | CISATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1995 |
| Q07001 | CISATRACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1995 |
| CISPLATIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1978 | |||
| P31645 | CITALOPRAM | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1998 |
| CLADRIBINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1993 | |||
| CLARITHROMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1991 | ||
| P62593 | CLAVULANIC ACID | Bacterial beta-lactamase TEM inhibitor | CHEMBL2364670 | Bacterial beta-lactamase TEM | Beta-lactamase TEM | Bacteria | enzyme hydrolase | Small molecule | 1984 |
| P35367 | CLEMASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1977 |
| O60840 | CLEVIDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 2008 |
| Q01668 | CLEVIDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 2008 |
| Q13698 | CLEVIDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 2008 |
| Q13936 | CLEVIDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 2008 |
| P11229 | CLIDINIUM | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P20309 | CLIDINIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P0A7J6 | CLINDAMYCIN | 50S ribosomal protein L10 | 50S ribosomal protein L10 | Shigella flexneri | Unclassified | Small molecule | 1970 | ||
| CLINDAMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1970 | ||
| CLINDAMYCIN PALMITATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1986 | ||
| CLINDAMYCIN PHOSPHATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1972 | ||
| CLIOQUINOL | Zinc chelating agent | CHEMBL2363056 | Zinc | Small molecule | 1982 | ||||
| CLIOQUINOL | CHEMBL2363056 | Zinc | Small molecule | 1982 | |||||
| CLIOQUINOL | Copper chelating agent | CHEMBL2363057 | Copper | Small molecule | 1982 | ||||
| CLIOQUINOL | CHEMBL2363057 | Copper | Small molecule | 1982 | |||||
| CLIOQUINOL | Iron chelating agent | CHEMBL2363058 | Iron | Small molecule | 1982 | ||||
| CLIOQUINOL | CHEMBL2363058 | Iron | Small molecule | 1982 | |||||
| P14867 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| P18507 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| P31644 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| P34903 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| P47869 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| Q8N1C3 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| Q99928 | CLOBAZAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2005 |
| P04150 | CLOBETASOL PROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1985 |
| P04150 | CLOCORTOLONE PIVALATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1977 |
| P09884 | CLOFARABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| P09884 | CLOFARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| P23921 | CLOFARABINE | Ribonucleoside-diphosphate reductase RR1 inhibitor | CHEMBL2095215 | Ribonucleoside-diphosphate reductase RR1 | Ribonucleoside-diphosphate reductase large subunit | Homo sapiens | enzyme reductase | Small molecule | 2004 |
| P23921 | CLOFARABINE | DNA inhibitor | CHEMBL2311221 | DNA | Ribonucleoside-diphosphate reductase large subunit | Homo sapiens | enzyme reductase | Small molecule | 2004 |
| P27707 | CLOFARABINE | Deoxycytidine kinase | Deoxycytidine kinase | Homo sapiens | enzyme | Small molecule | 2004 | ||
| P28340 | CLOFARABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA polymerase delta catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| P28340 | CLOFARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase delta catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| Q07864 | CLOFARABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA polymerase epsilon catalytic subunit A | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| Q07864 | CLOFARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase epsilon catalytic subunit A | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| CLOFARABINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2004 | |||
| CLOFAZIMINE | DNA inhibitor | CHEMBL2366041 | DNA | Mycobacterium leprae | Small molecule | 1986 | |||
| Q07869 | CLOFIBRATE | Peroxisome proliferator-activated receptor alpha agonist | CHEMBL239 | Peroxisome proliferator-activated receptor alpha | Peroxisome proliferator-activated receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c1 | Small molecule | 1967 |
| P31645 | CLOMIPRAMINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1989 |
| P35367 | CLOMIPRAMINE | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1989 | ||
| P14867 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| P18507 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| P31644 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| P34903 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| P47869 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| Q8N1C3 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| Q99928 | CLONAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1975 |
| P08913 | CLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1974 |
| P18089 | CLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1974 |
| P18825 | CLONIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1974 |
| Q9H244 | CLOPIDOGREL | Purinergic receptor P2Y12 antagonist | CHEMBL2001 | Purinergic receptor P2Y12 | P2Y purinoceptor 12 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor purine receptor | Small molecule | 1997 |
| P14867 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P18507 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P31644 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P34903 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P47869 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| Q8N1C3 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| Q99928 | CLORAZEPIC ACID | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P10613 | CLOTRIMAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1975 |
| P72355 | CLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin-binding protein 4 | Staphylococcus | enzyme protease serine se s13 | Small molecule | 1974 |
| Q53707 | CLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | MecA PBP2' (penicillin binding protein 2') | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1974 |
| Q53725 | CLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | PASTA domain protein | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1974 |
| Q53729 | CLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin binding protein 2 | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1974 |
| Q9XDB3 | CLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin binding transpeptidase domain protein | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1974 |
| P14416 | CLOZAPINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1989 |
| P18089 | CLOZAPINE | Alpha-2B adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 | ||
| P20309 | CLOZAPINE | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1989 | ||
| P21728 | CLOZAPINE | D(1A) dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1989 | ||
| P21918 | CLOZAPINE | D(1B) dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1989 | ||
| P25100 | CLOZAPINE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 | ||
| P28223 | CLOZAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1989 |
| P34969 | CLOZAPINE | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1989 | ||
| P35367 | CLOZAPINE | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1989 | ||
| P41595 | CLOZAPINE | 5-hydroxytryptamine receptor 2B | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1989 | ||
| P08684 | COBICISTAT | Cytochrome P450 3A inhibitor | CHEMBL2364675 | Cytochrome P450 3A | Cytochrome P450 3A4 | Homo sapiens | enzyme cytochrome p450 cyp_3 cyp_3a cyp_3a4 | Small molecule | 2012 |
| P20815 | COBICISTAT | Cytochrome P450 3A inhibitor | CHEMBL2364675 | Cytochrome P450 3A | Cytochrome P450 3A5 | Homo sapiens | enzyme cytochrome p450 cyp_3 cyp_3a cyp_3a5 | Small molecule | 2012 |
| P24462 | COBICISTAT | Cytochrome P450 3A inhibitor | CHEMBL2364675 | Cytochrome P450 3A | Cytochrome P450 3A7 | Homo sapiens | enzyme reductase | Small molecule | 2012 |
| Q9HB55 | COBICISTAT | Cytochrome P450 3A inhibitor | CHEMBL2364675 | Cytochrome P450 3A | Cytochrome P450 3A43 | Homo sapiens | enzyme reductase | Small molecule | 2012 |
| P35372 | CODEINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1952 |
| P41143 | CODEINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1952 |
| P41145 | CODEINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1952 |
| P04350 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1961 |
| P07437 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1961 |
| P68371 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1961 |
| Q13509 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1961 |
| Q13885 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1961 |
| Q3ZCM7 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1961 |
| Q9BUF5 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1961 |
| Q9BVA1 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1961 |
| Q9H4B7 | COLCHICINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1961 |
| COLESEVELAM HYDROCHLORIDE | Bile acids chelating agent | CHEMBL2364175 | Bile acids | Homo sapiens | Small molecule | 2000 | |||
| COLESTIPOL HYDROCHLORIDE | Bile acids chelating agent | CHEMBL2364175 | Bile acids | Homo sapiens | Unknown | 1977 | |||
| COLISTIMETHATE SODIUM | Cell membrane inhibitor | CHEMBL2364031 | Cell membrane | Bacteria | Small molecule | 1970 | |||
| COLISTIN | Cell outer membrane inhibitor | CHEMBL2364032 | Cell outer membrane | Bacteria | Unknown | 1962 | |||
| A6NMZ7 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-6(VI) chain | Homo sapiens | structural | Enzyme | 2010 |
| A8TX70 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-5(VI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P02452 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(I) chain | Homo sapiens | structural | Enzyme | 2010 |
| P02458 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(II) chain | Homo sapiens | structural | Enzyme | 2010 |
| P02461 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(III) chain | Homo sapiens | structural | Enzyme | 2010 |
| P02462 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| P05997 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(V) chain | Homo sapiens | structural | Enzyme | 2010 |
| P08123 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(I) chain | Homo sapiens | structural | Enzyme | 2010 |
| P08572 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| P12107 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P12109 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(VI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P12110 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(VI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P12111 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(VI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P13942 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(XI) chain | Homo sapiens | structural | Enzyme | 2010 |
| P20908 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(V) chain | Homo sapiens | structural | Enzyme | 2010 |
| P25940 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(V) chain | Homo sapiens | structural | Enzyme | 2010 |
| P29400 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-5(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| P39059 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XV) chain | Homo sapiens | structural | Enzyme | 2010 |
| P39060 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XVIII) chain | Homo sapiens | structural | Enzyme | 2010 |
| P53420 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-4(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| Q01955 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| Q14031 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-6(IV) chain | Homo sapiens | structural | Enzyme | 2010 |
| Q17RW2 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXIV) chain | Homo sapiens | structural | Enzyme | 2010 |
| Q2UY09 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXVIII) chain | Homo sapiens | structural | Enzyme | 2010 |
| Q8IZC6 | COLLAGENASE CLOSTRIDIUM HISTOLYTICUM | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXVII) chain | Homo sapiens | structural | Enzyme | 2010 |
| P30518 | CONIVAPTAN | Vasopressin V2 receptor antagonist | CHEMBL1790 | Vasopressin V2 receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Small molecule | 2005 |
| P37288 | CONIVAPTAN | Vasopressin V1a receptor antagonist | CHEMBL1889 | Vasopressin V1a receptor | Vasopressin V1a receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Small molecule | 2005 |
| Q01718 | CORTICOTROPIN | Melanocortin receptor 2 agonist | CHEMBL1965 | Melanocortin receptor 2 | Adrenocorticotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide melanocortin receptor | Protein | 1950 |
| Q01718 | CORTICOTROPIN ZINC HYDROXIDE | Melanocortin receptor 2 agonist | CHEMBL1965 | Melanocortin receptor 2 | Adrenocorticotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide melanocortin receptor | Protein | 1955 |
| P04150 | CORTISONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1950 |
| Q01718 | COSYNTROPIN | Melanocortin receptor 2 agonist | CHEMBL1965 | Melanocortin receptor 2 | Adrenocorticotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide melanocortin receptor | Protein | 1970 |
| P08581 | CRIZOTINIB | Hepatocyte growth factor receptor inhibitor | CHEMBL3717 | Hepatocyte growth factor receptor | Hepatocyte growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk met | Small molecule | 2011 |
| Q9UM73 | CRIZOTINIB | ALK tyrosine kinase receptor inhibitor | CHEMBL4247 | ALK tyrosine kinase receptor | ALK tyrosine kinase receptor | Homo sapiens | enzyme kinase protein kinase tkl stkr type1 | Small molecule | 2011 |
| P13569 | CROFELEMER | Cystic fibrosis transmembrane conductance regulator inhibitor | CHEMBL4051 | Cystic fibrosis transmembrane conductance regulator | Cystic fibrosis transmembrane conductance regulator | Homo sapiens | ion channel other chloride cftr | Small molecule | 2012 |
| Q5XXA6 | CROFELEMER | Anoctamin-1 blocker | CHEMBL2046267 | Anoctamin-1 | Anoctamin-1 | Homo sapiens | ion channel other chloride ca act cl | Small molecule | 2012 |
| Q12791 | CROMOLYN | Calcium-activated potassium channel subunit alpha-1 | Calcium-activated potassium channel subunit alpha-1 | Homo sapiens | ion channel vgc k ca act k | Small molecule | 1982 | ||
| CROMOLYN | Unknown | Small molecule | 1982 | ||||||
| CROTAMITON | Unknown | Small molecule | 1949 | ||||||
| CRYPTENAMINE ACETATES | Unknown | Small molecule | 1982 | ||||||
| CRYPTENAMINE TANNATES | Unknown | Small molecule | 1982 | ||||||
| CRYSTAL VIOLET | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1982 | |||
| CUPRIC SULFATE | Unknown | Small molecule | 1987 | ||||||
| P02918 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1979 |
| P02919 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1979 |
| P08506 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1979 |
| P0AD65 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1979 |
| P0AD68 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1979 |
| P0AEB2 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1979 |
| P24228 | CYCLACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1979 |
| P35367 | CYCLIZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| P28223 | CYCLOBENZAPRINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1977 |
| P28335 | CYCLOBENZAPRINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1977 |
| P13922 | CYCLOGUANIL | Dihydrofolate reductase inhibitor | CHEMBL1939 | Dihydrofolate reductase | Bifunctional dihydrofolate reductase-thymidylate synthase | Plasmodium falciparum K1 | enzyme reductase | Small molecule | 0 |
| P20309 | CYCLOPENTOLATE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1974 |
| CYCLOPHOSPHAMIDE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1959 | |||
| A2VLV3 | CYCLOSERINE | D-alanine--D-alanine ligase | D-alanine--D-alanine ligase | Mycobacterium tuberculosis C | Unclassified | Small molecule | 1964 | ||
| P0A6J8 | CYCLOSERINE | D-alanine--D-alanine ligase A | D-alanine--D-alanine ligase A | Escherichia coli (strain K12) | Unclassified | Small molecule | 1964 | ||
| P9WP31 | CYCLOSERINE | D-alanylalanine synthetase inhibitor | CHEMBL2030 | D-alanylalanine synthetase | D-alanine--D-alanine ligase | Mycobacterium tuberculosis | enzyme ligase | Small molecule | 1964 |
| P9WQA9 | CYCLOSERINE | Alanine racemase inhibitor | CHEMBL2031 | Alanine racemase | Alanine racemase | Mycobacterium tuberculosis | enzyme isomerase | Small molecule | 1964 |
| Q9L888 | CYCLOSERINE | Alanine racemase | Alanine racemase | Mycobacterium avium | Isomerase | Small molecule | 1964 | ||
| P62937 | CYCLOSPORINE | Cyclophilin A modulator | CHEMBL1949 | Cyclophilin A | Peptidyl-prolyl cis-trans isomerase A | Homo sapiens | enzyme isomerase | Protein | 1983 |
| P62942 | CYCLOSPORINE | Peptidyl-prolyl cis-trans isomerase FKBP1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Protein | 1983 | ||
| Q02127 | CYCLOSPORINE | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | Homo sapiens | enzyme reductase | Protein | 1983 | ||
| P55017 | CYCLOTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1982 |
| P11229 | CYCRIMINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P08173 | CYPROHEPTADINE | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 | ||
| P08912 | CYPROHEPTADINE | Muscarinic acetylcholine receptor M5 | Muscarinic acetylcholine receptor M5 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 | ||
| P28223 | CYPROHEPTADINE | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1961 | ||
| P28335 | CYPROHEPTADINE | 5-hydroxytryptamine receptor 2C | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1961 | ||
| P35367 | CYPROHEPTADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1961 |
| P41595 | CYPROHEPTADINE | 5-hydroxytryptamine receptor 2B | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1961 | ||
| CYSTEAMINE | Cystine hydrolytic enzyme | CHEMBL2364039 | Cystine | Homo sapiens | Small molecule | 1994 | |||
| P09884 | CYTARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1969 |
| P28340 | CYTARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase delta catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1969 |
| Q07864 | CYTARABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase epsilon catalytic subunit A | Homo sapiens | enzyme transferase | Small molecule | 1969 |
| CYTARABINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1969 | |||
| CYTARABINE | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 1969 | |||
| P00734 | DABIGATRAN ETEXILATE | Thrombin inhibitor | CHEMBL204 | Thrombin | Prothrombin | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 2010 |
| P15056 | DABRAFENIB | Serine/threonine-protein kinase B-raf inhibitor | CHEMBL5145 | Serine/threonine-protein kinase B-raf | Serine/threonine-protein kinase B-raf | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2013 |
| DACARBAZINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1975 | |||
| P01589 | DACLIZUMAB | Interleukin-2 receptor inhibitor | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit alpha | Homo sapiens | membrane receptor | Antibody | 1997 |
| DACTINOMYCIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Protein | 1964 | |||
| DALBAVANCIN | Peptidoglycan inhibitor | CHEMBL3041361 | Peptidoglycan | Bacteria | Unknown | 2014 | |||
| O43525 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| O43526 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| O95259 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P16389 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P17658 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 6 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P22001 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P22459 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P22460 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P48547 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P51787 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| P56696 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q03721 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q09470 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q12809 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q14003 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q14721 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily B member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q16322 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 10 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q6PIU1 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily V member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q8NCM2 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q8TAE7 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q8TDN1 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q8TDN2 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily V member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q92953 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily B member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q96KK3 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q96L42 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 8 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q96PR1 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q96RP8 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 7 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9BQ31 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9H252 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 6 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9H3M0 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily F member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9NR82 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9NS40 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 7 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9NSA2 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9NZV8 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9UIX4 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9UJ96 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9UK17 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9ULD8 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9ULS6 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| Q9UQ05 | DALFAMPRIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2010 |
| DALFOPRISTIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1999 | ||
| P01008 | DALTEPARIN SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 1994 |
| P01008 | DANAPAROID SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Unknown | 1996 |
| P06401 | DANAZOL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1976 |
| P10275 | DANAZOL | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1976 |
| P30968 | DANAZOL | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Small molecule | 1976 | ||
| Q96P88 | DANAZOL | Putative gonadotropin-releasing hormone II receptor | Putative gonadotropin-releasing hormone II receptor | Homo sapiens | Unclassified | Small molecule | 1976 | ||
| P21817 | DANTROLENE | Ryanodine receptor 1 antagonist | CHEMBL1846 | Ryanodine receptor 1 | Ryanodine receptor 1 | Homo sapiens | ion channel lgic ryr | Small molecule | 1974 |
| Q15413 | DANTROLENE | Ryanodine receptor 3 antagonist | CHEMBL2062 | Ryanodine receptor 3 | Ryanodine receptor 3 | Homo sapiens | ion channel lgic ryr | Small molecule | 1974 |
| P31639 | DAPAGLIFLOZIN | Sodium/glucose cotransporter 2 inhibitor | CHEMBL3884 | Sodium/glucose cotransporter 2 | Sodium/glucose cotransporter 2 | Homo sapiens | transporter electrochemical slc slc05 | Small molecule | 2014 |
| P25100 | DAPIPRAZOLE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1990 | ||
| P35348 | DAPIPRAZOLE | Alpha-1a adrenergic receptor antagonist | CHEMBL229 | Alpha-1a adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1990 |
| P0C0X1 | DAPSONE | Dihydropteroate synthase 1 inhibitor | CHEMBL2362993 | Dihydropteroate synthase 1 | Dihydropteroate synthase 1 | Mycobacterium leprae (strain TN) | enzyme transferase | Small molecule | 1979 |
| DAPTOMYCIN | Cell membrane inhibitor | CHEMBL2364031 | Cell membrane | Bacteria | Small molecule | 2003 | |||
| P19235 | DARBEPOETIN ALFA | Erythropoietin receptor agonist | CHEMBL1817 | Erythropoietin receptor | Erythropoietin receptor | Homo sapiens | membrane receptor | Protein | 2001 |
| P08172 | DARIFENACIN | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| P20309 | DARIFENACIN | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| Q72874 | DARUNAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 2006 |
| Q8JXU8 | DASABUVIR | Hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor | CHEMBL5375 | Hepatitis C virus NS5B RNA-dependent RNA polymerase | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 2014 |
| P00519 | DASATINIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2006 |
| P06239 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Lck | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P06241 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Fyn | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P07947 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Yes | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P07948 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Lyn | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P08631 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase HCK | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P09619 | DASATINIB | Platelet-derived growth factor receptor beta inhibitor | CHEMBL1913 | Platelet-derived growth factor receptor beta | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P09769 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Fgr | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P10721 | DASATINIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P12931 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Proto-oncogene tyrosine-protein kinase Src | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P29317 | DASATINIB | Ephrin type-A receptor 2 inhibitor | CHEMBL2068 | Ephrin type-A receptor 2 | Ephrin type-A receptor 2 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2006 |
| P42685 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase FRK | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| P51451 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Blk | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2006 |
| Q9H3Y6 | DASATINIB | SRC inhibitor | CHEMBL2363074 | SRC | Tyrosine-protein kinase Srms | Homo sapiens | enzyme kinase protein kinase tk src srm | Small molecule | 2006 |
| P11388 | DAUNORUBICIN | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1979 |
| P11388 | DAUNORUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1979 |
| DAUNORUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1979 | |||
| P02708 | DECAMETHONIUM | Muscle-type nicotinic acetylcholine receptor partial agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 |
| P07510 | DECAMETHONIUM | Muscle-type nicotinic acetylcholine receptor partial agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1982 |
| P11230 | DECAMETHONIUM | Muscle-type nicotinic acetylcholine receptor partial agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 |
| Q04844 | DECAMETHONIUM | Muscle-type nicotinic acetylcholine receptor partial agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1982 |
| Q07001 | DECAMETHONIUM | Muscle-type nicotinic acetylcholine receptor partial agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1982 |
| P26358 | DECITABINE | DNA (cytosine-5)-methyltransferase 1 inhibitor | CHEMBL1993 | DNA (cytosine-5)-methyltransferase 1 | DNA (cytosine-5)-methyltransferase 1 | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2006 |
| P26358 | DECITABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA (cytosine-5)-methyltransferase 1 | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2006 |
| Q9Y6K1 | DECITABINE | DNA (cytosine-5)-methyltransferase 3A inhibitor | CHEMBL1992 | DNA (cytosine-5)-methyltransferase 3A | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator reader methyl-lysine pwwp | Small molecule | 2006 |
| Q9Y6K1 | DECITABINE | DNA (cytosine-5)-methyltransferase 3A inhibitor | CHEMBL1992 | DNA (cytosine-5)-methyltransferase 3A | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2006 |
| Q9Y6K1 | DECITABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator reader methyl-lysine pwwp | Small molecule | 2006 |
| Q9Y6K1 | DECITABINE | DNA inhibitor | CHEMBL2311221 | DNA | DNA (cytosine-5)-methyltransferase 3A | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 2006 |
| DECITABINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2006 | |||
| DEFERASIROX | Iron chelating agent | CHEMBL2363058 | Iron | Small molecule | 2005 | ||||
| DEFERASIROX | CHEMBL2363058 | Iron | Small molecule | 2005 | |||||
| DEFERIPRONE | Unknown | Small molecule | 1999 | ||||||
| DEFEROXAMINE | Iron chelating agent | CHEMBL2363058 | Iron | Small molecule | 1968 | ||||
| DEFEROXAMINE | CHEMBL2363058 | Iron | Small molecule | 1968 | |||||
| P30968 | DEGARELIX | Gonadotropin-releasing hormone receptor antagonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 2008 |
| P03369 | DELAVIRDINE | Gag-Pol polyprotein | Gag-Pol polyprotein | Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) | Unclassified | Small molecule | 1997 | ||
| Q72547 | DELAVIRDINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1997 |
| P22303 | DEMECARIUM | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1959 |
| DEMECLOCYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1960 | ||
| P01589 | DENILEUKIN DIFTITOX | Interleukin-2 receptor binding agent | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit alpha | Homo sapiens | membrane receptor | Protein | 1999 |
| P13639 | DENILEUKIN DIFTITOX | Elongation factor 2 inhibitor | CHEMBL1795108 | Elongation factor 2 | Elongation factor 2 | Homo sapiens | unclassified | Protein | 1999 |
| P14784 | DENILEUKIN DIFTITOX | Interleukin-2 receptor binding agent | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit beta | Homo sapiens | membrane receptor | Protein | 1999 |
| O14788 | DENOSUMAB | Tumor necrosis factor ligand superfamily member 11 inhibitor | CHEMBL2364162 | Tumor necrosis factor ligand superfamily member 11 | Tumor necrosis factor ligand superfamily member 11 | Homo sapiens | secreted | Antibody | 2010 |
| DEOXYCHOLIC ACID | Cell membrane disrupting agent | CHEMBL3390826 | Cell membrane | Homo sapiens | Small molecule | 2015 | |||
| Q05940 | DESERPIDINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 1957 |
| O00591 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| O14649 | DESFLURANE | Potassium channel subfamily K member 3 opener | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1992 |
| O14764 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| O95069 | DESFLURANE | Potassium channel subfamily K member 2 opener | CHEMBL2321615 | Potassium channel subfamily K member 2 | Potassium channel subfamily K member 2 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1992 |
| P14867 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P18505 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P18507 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P23415 | DESFLURANE | Glycine receptor (alpha-1/beta) positive modulator | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 1992 |
| P28472 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P31644 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P34903 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P47869 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P47870 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P48169 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P57789 | DESFLURANE | Potassium channel subfamily K member 10 opener | CHEMBL2331041 | Potassium channel subfamily K member 10 | Potassium channel subfamily K member 10 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1992 |
| P78334 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| Q16445 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| Q7Z418 | DESFLURANE | Potassium channel subfamily K member 18 opener | CHEMBL2331042 | Potassium channel subfamily K member 18 | Potassium channel subfamily K member 18 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1992 |
| Q8N1C3 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| Q99928 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| Q9NPC2 | DESFLURANE | Potassium channel subfamily K member 9 opener | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1992 |
| Q9UN88 | DESFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P23975 | DESIPRAMINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1964 |
| P28223 | DESIPRAMINE | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1964 | ||
| P31645 | DESIPRAMINE | Sodium-dependent serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1964 | ||
| P35348 | DESIPRAMINE | Alpha-1A adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1964 | ||
| P35367 | DESIPRAMINE | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1964 | ||
| P00734 | DESIRUDIN | Thrombin inhibitor | CHEMBL204 | Thrombin | Prothrombin | Homo sapiens | enzyme protease serine pas s1a | Protein | 2003 |
| P05023 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P05023 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P13637 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P13637 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P50993 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P50993 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| Q13733 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| Q13733 | DESLANOSIDE | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P35367 | DESLORATADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2001 |
| P30518 | DESMOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1978 |
| P37288 | DESMOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1a receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1978 |
| P47901 | DESMOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1b receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1978 |
| P06401 | DESOGESTREL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1992 |
| P04150 | DESONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1972 |
| P04150 | DESOXIMETASONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1977 |
| P08235 | DESOXYCORTICOSTERONE ACETATE | Mineralocorticoid receptor agonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1939 |
| P08235 | DESOXYCORTICOSTERONE PIVALATE | Mineralocorticoid receptor agonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1982 |
| DESOXYRIBONUCLEASE | DNA hydrolytic enzyme | CHEMBL2311221 | DNA | Homo sapiens | Enzyme | 1964 | |||
| P23975 | DESVENLAFAXINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2008 |
| P31645 | DESVENLAFAXINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2008 |
| P04150 | DEXAMETHASONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1958 |
| P04150 | DEXAMETHASONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1973 |
| P04150 | DEXAMETHASONE PHOSPHORIC ACID | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1959 |
| P35367 | DEXBROMPHENIRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1963 |
| P35367 | DEXCHLORPHENIRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1981 |
| P20648 | DEXLANSOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 2009 |
| P20648 | DEXLANSOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 2009 |
| P08913 | DEXMEDETOMIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1999 |
| P18089 | DEXMEDETOMIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1999 |
| P18825 | DEXMEDETOMIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1999 |
| P23975 | DEXMETHYLPHENIDATE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2001 |
| Q01959 | DEXMETHYLPHENIDATE | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2001 |
| P23975 | DEXTROAMPHETAMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| Q01959 | DEXTROAMPHETAMINE | Dopamine transporter releasing agent | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| Q05940 | DEXTROAMPHETAMINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 1955 |
| P17787 | DEXTROMETHORPHAN | Neuronal acetylcholine receptor; alpha2/beta2 | Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 | ||
| P31645 | DEXTROMETHORPHAN | Sodium-dependent serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 | ||
| P32297 | DEXTROMETHORPHAN | Neuronal acetylcholine receptor; alpha3/beta2 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 | ||
| P43681 | DEXTROMETHORPHAN | Neuronal acetylcholine receptor; alpha4/beta2 | Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 | ||
| Q12879 | DEXTROMETHORPHAN | Glutamate [NMDA] receptor subunit epsilon 1 antagonist | CHEMBL1972 | Glutamate [NMDA] receptor subunit epsilon 1 | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1982 |
| Q15822 | DEXTROMETHORPHAN | Neuronal acetylcholine receptor; alpha2/beta2 | Neuronal acetylcholine receptor subunit alpha-2 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 | ||
| Q8TCU5 | DEXTROMETHORPHAN | "Glutamate receptor ionotropic, NMDA 3A" | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1982 | ||
| Q99720 | DEXTROMETHORPHAN | Sigma opioid receptor agonist | CHEMBL287 | Sigma opioid receptor | Sigma non-opioid intracellular receptor 1 | Homo sapiens | membrane receptor | Small molecule | 1982 |
| P10827 | DEXTROTHYROXINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a1 | Small molecule | 1967 |
| P10828 | DEXTROTHYROXINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a2 | Small molecule | 1967 |
| P35372 | DEZOCINE | Mu opioid receptor partial agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1989 |
| P41145 | DEZOCINE | Kappa opioid receptor antagonist | CHEMBL237 | Kappa opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1989 |
| P14867 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| P18507 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| P31644 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| P34903 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| P47869 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| Q8N1C3 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| Q99928 | DIAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1963 |
| P05023 | DIAZOXIDE | Sodium/potassium-transporting ATPase subunit alpha-1 | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 1973 | ||
| P05023 | DIAZOXIDE | Sodium/potassium-transporting ATPase subunit alpha-1 | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1973 | ||
| Q14654 | DIAZOXIDE | "Potassium channel, inwardly rectifying, subfamily J, member 11 opener" | CHEMBL1886 | "Potassium channel, inwardly rectifying, subfamily J, member 11" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1973 |
| Q15842 | DIAZOXIDE | "Potassium channel, inwardly rectifying, subfamily J, member 8 opener" | CHEMBL4770 | "Potassium channel, inwardly rectifying, subfamily J, member 8" | ATP-sensitive inward rectifier potassium channel 8 | Homo sapiens | ion channel vgc k kir | Small molecule | 1973 |
| Q14524 | DIBUCAINE | Sodium channel protein type V alpha subunit blocker | CHEMBL1980 | Sodium channel protein type V alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | DIBUCAINE | Sodium channel protein type X alpha subunit blocker | CHEMBL5451 | Sodium channel protein type X alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| O43570 | DICHLORPHENAMIDE | Carbonic anhydrase XII inhibitor | CHEMBL3242 | Carbonic anhydrase XII | Carbonic anhydrase 12 | Homo sapiens | enzyme lyase | Small molecule | 1958 |
| P00915 | DICHLORPHENAMIDE | Carbonic anhydrase I inhibitor | CHEMBL261 | Carbonic anhydrase I | Carbonic anhydrase 1 | Homo sapiens | enzyme lyase | Small molecule | 1958 |
| P00918 | DICHLORPHENAMIDE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1958 |
| P22748 | DICHLORPHENAMIDE | Carbonic anhydrase IV inhibitor | CHEMBL3729 | Carbonic anhydrase IV | Carbonic anhydrase 4 | Homo sapiens | enzyme lyase | Small molecule | 1958 |
| P43166 | DICHLORPHENAMIDE | Carbonic anhydrase 7 | Carbonic anhydrase 7 | Homo sapiens | enzyme lyase | Small molecule | 1958 | ||
| Q16790 | DICHLORPHENAMIDE | Carbonic anhydrase 9 | Carbonic anhydrase 9 | Homo sapiens | enzyme lyase | Small molecule | 1958 | ||
| Q9Y2D0 | DICHLORPHENAMIDE | "Carbonic anhydrase 5B, mitochondrial" | "Carbonic anhydrase 5B, mitochondrial" | Homo sapiens | enzyme lyase | Small molecule | 1958 | ||
| P23219 | DICLOFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1988 |
| P35354 | DICLOFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1988 |
| P10520 | DICLOXACILLIN | Streptokinase A | Streptokinase A | Streptococcus pyogenes serotype M1 | unclassified | Small molecule | 1968 | ||
| P72355 | DICLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin-binding protein 4 | Staphylococcus aureus | enzyme protease serine se s13 | Small molecule | 1968 |
| Q53707 | DICLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | MecA PBP2' (penicillin binding protein 2') | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1968 |
| Q53725 | DICLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | PASTA domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1968 |
| Q53729 | DICLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding protein 2 | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1968 |
| Q8XJ01 | DICLOXACILLIN | Penicillin-binding protein 1A | Penicillin-binding protein 1A | Clostridium perfringens (strain 13 / Type A) | Hydrolase | Small molecule | 1968 | ||
| Q9XDB3 | DICLOXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding transpeptidase domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1968 |
| Q9BQB6 | DICUMAROL | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor | CHEMBL1930 | Vitamin k epoxide reductase complex subunit 1 isoform 1 | Vitamin K epoxide reductase complex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1944 |
| P08172 | DICYCLOMINE | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1950 | ||
| P08173 | DICYCLOMINE | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1950 | ||
| P08912 | DICYCLOMINE | Muscarinic acetylcholine receptor M5 | Muscarinic acetylcholine receptor M5 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1950 | ||
| P11229 | DICYCLOMINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1950 |
| P20309 | DICYCLOMINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1950 |
| P03369 | DIDANOSINE | Gag-Pol polyprotein | Gag-Pol polyprotein | Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) | Unclassified | Small molecule | 1991 | ||
| Q72547 | DIDANOSINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1991 |
| Q72549 | DIDANOSINE | Reverse transcriptase/RNaseH | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | Transferase | Small molecule | 1991 | ||
| P03372 | DIENESTROL | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1947 |
| P06401 | DIENOGEST | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2010 | ||
| DIENOGEST | Unknown | Small molecule | 2010 | ||||||
| E1FVX6 | DIETHYLCARBAMAZINE | Nematode GABA-A receptor positive modulator | CHEMBL2364676 | Nematode GABA-A receptor | Uncharacterized protein | Onchocercidae | unclassified | Small molecule | 1950 |
| E1G1C3 | DIETHYLCARBAMAZINE | Nematode GABA-A receptor positive modulator | CHEMBL2364676 | Nematode GABA-A receptor | Uncharacterized protein | Onchocercidae | unclassified | Small molecule | 1950 |
| P23975 | DIETHYLPROPION | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1959 |
| Q01959 | DIETHYLPROPION | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1959 |
| P03372 | DIETHYLSTILBESTROL | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1973 |
| P03372 | DIETHYLSTILBESTROL DIPHOSPHATE | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1982 |
| Q92731 | DIETHYLSTILBESTROL DIPHOSPHATE | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1982 |
| P35372 | DIFENOXIN | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1978 |
| P04150 | DIFLORASONE DIACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1977 |
| P23219 | DIFLUNISAL | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P35354 | DIFLUNISAL | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P04150 | DIFLUPREDNATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 2008 |
| P05023 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P05023 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P13637 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P13637 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P50993 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P50993 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| Q13733 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| Q13733 | DIGITOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1982 |
| P05023 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | enzyme hydrolase | Small molecule | 1975 |
| P05023 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-1 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1975 |
| P13637 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | enzyme hydrolase | Small molecule | 1975 |
| P13637 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-3 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1975 |
| P50993 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | enzyme hydrolase | Small molecule | 1975 |
| P50993 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-2 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1975 |
| Q13733 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | enzyme hydrolase | Small molecule | 1975 |
| Q13733 | DIGOXIN | Sodium/potassium-transporting ATPase inhibitor | CHEMBL2095186 | Sodium/potassium-transporting ATPase | Sodium/potassium-transporting ATPase subunit alpha-4 | Homo sapiens | transporter ntpase p-type atpase na k atpase | Small molecule | 1975 |
| P35372 | DIHYDROCODEINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1983 |
| P28221 | DIHYDROERGOTAMINE | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1946 |
| O60840 | DILTIAZEM | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| Q01668 | DILTIAZEM | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| Q13698 | DILTIAZEM | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| Q13936 | DILTIAZEM | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| P20309 | DIMENHYDRINATE | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1972 | ||
| P35367 | DIMENHYDRINATE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1972 |
| DIMERCAPROL | Heavy metals chelating agent | CHEMBL2363053 | Heavy metals | Small molecule | 1946 | ||||
| DIMERCAPROL | CHEMBL2363053 | Heavy metals | Small molecule | 1946 | |||||
| Q14145 | DIMETHYL FUMARATE | Kelch-like ECH-associated protein 1 inhibitor | CHEMBL2069156 | Kelch-like ECH-associated protein 1 | Kelch-like ECH-associated protein 1 | Homo sapiens | unclassified | Small molecule | 2013 |
| DIMETHYL SULFOXIDE | Unknown | Small molecule | 1978 | ||||||
| P43088 | DINOPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1982 |
| P34995 | DINOPROSTONE | Prostaglandin E2 receptor agonist | CHEMBL2363068 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP1 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1977 |
| P35408 | DINOPROSTONE | Prostaglandin E2 receptor agonist | CHEMBL2363068 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP4 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1977 |
| P43115 | DINOPROSTONE | Prostaglandin E2 receptor agonist | CHEMBL2363068 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP3 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1977 |
| P43116 | DINOPROSTONE | Prostaglandin E2 receptor agonist | CHEMBL2363068 | Prostaglandin E2 receptor | Prostaglandin E2 receptor EP2 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1977 |
| DINUTUXIMAB | Disialoganglioside GD2 binding agent | CHEMBL3390823 | Disialoganglioside GD2 | Homo sapiens | Antibody | 2015 | |||
| P11229 | DIPHEMANIL | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P20309 | DIPHEMANIL | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P35367 | DIPHENHYDRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1946 |
| P11229 | DIPHENIDOL | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1967 |
| P35372 | DIPHENOXYLATE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1960 |
| P35367 | DIPHENYLPYRALINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| P07550 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P08588 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P08913 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P13945 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P18089 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P18825 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P25100 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P35348 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| P35368 | DIPIVEFRIN | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1980 |
| O00337 | DIPYRIDAMOLE | Sodium/nucleoside cotransporter 1 | Sodium/nucleoside cotransporter 1 | Homo sapiens | transporter electrochemical slc slc28 and slc29 slc28 | Small molecule | 1961 | ||
| O00408 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-dependent 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_2 pde_2a | Small molecule | 1961 |
| O43924 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6d | Small molecule | 1961 |
| O60658 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8a | Small molecule | 1961 |
| O76074 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 1961 |
| O76083 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A" | Homo sapiens | enzyme phosphodiesterase pde_9 pde_9a | Small molecule | 1961 |
| O95263 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8B" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8b | Small molecule | 1961 |
| P00813 | DIPYRIDAMOLE | Adenosine deaminase | Adenosine deaminase | Homo sapiens | enzyme hydrolase | Small molecule | 1961 | ||
| P16499 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6a | Small molecule | 1961 |
| P18545 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6g | Small molecule | 1961 |
| P27815 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1961 |
| P35913 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit beta" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6b | Small molecule | 1961 |
| P51160 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6c | Small molecule | 1961 |
| P54750 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1a | Small molecule | 1961 |
| Q01064 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1b | Small molecule | 1961 |
| Q07343 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1961 |
| Q08493 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1961 |
| Q08499 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1961 |
| Q13370 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-inhibited 3',5'-cyclic phosphodiesterase B" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3b | Small molecule | 1961 |
| Q13946 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7a | Small molecule | 1961 |
| Q13956 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6h | Small molecule | 1961 |
| Q14123 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1c | Small molecule | 1961 |
| Q14432 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1961 |
| Q99808 | DIPYRIDAMOLE | Equilibrative nucleoside transporter 1 inhibitor | CHEMBL1997 | Equilibrative nucleoside transporter 1 | Equilibrative nucleoside transporter 1 | Homo sapiens | transporter electrochemical slc slc28 and slc29 slc29 | Small molecule | 1961 |
| Q9NP56 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 7B" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7b | Small molecule | 1961 |
| Q9Y233 | DIPYRIDAMOLE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A" | Homo sapiens | enzyme phosphodiesterase pde_10 pde_10a | Small molecule | 1961 |
| DIRITHROMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1995 | ||
| O60939 | DISOPYRAMIDE | Sodium channel subunit beta-2 | Sodium channel subunit beta-2 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1977 | ||
| P35498 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| P35499 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| P48544 | DISOPYRAMIDE | G protein-activated inward rectifier potassium channel 4 | G protein-activated inward rectifier potassium channel 4 | Homo sapiens | ion channel vgc k kir | Small molecule | 1977 | ||
| Q01118 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q07699 | DISOPYRAMIDE | Sodium channel subunit beta-1 | Sodium channel subunit beta-1 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1977 | ||
| Q14524 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q15858 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q8IWT1 | DISOPYRAMIDE | Sodium channel subunit beta-4 | Sodium channel subunit beta-4 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1977 | ||
| Q99250 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q9NY46 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q9NY72 | DISOPYRAMIDE | Sodium channel subunit beta-3 | Sodium channel subunit beta-3 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1977 | ||
| Q9UI33 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q9UQD0 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| Q9Y5Y9 | DISOPYRAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1977 |
| P05091 | DISULFIRAM | Aldehyde dehydrogenase inhibitor | CHEMBL1935 | Aldehyde dehydrogenase | "Aldehyde dehydrogenase, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1951 |
| P07550 | DOBUTAMINE | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 |
| P08588 | DOBUTAMINE | Beta-1 adrenergic receptor agonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 |
| P04350 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1996 |
| P07437 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1996 |
| P68371 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1996 |
| Q13509 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1996 |
| Q13885 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1996 |
| Q3ZCM7 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1996 |
| Q9BUF5 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1996 |
| Q9BVA1 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1996 |
| Q9H4B7 | DOCETAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1996 |
| O09800 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein N | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P04288 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein M | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P04488 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein E | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P06477 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein H | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P06480 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein J | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P06484 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein G | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P06487 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein I | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P10185 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein L | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P10211 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein B | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P10228 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein C | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| P68331 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein K | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| Q69091 | DOCOSANOL | Envelope glycoprotein inhibitor | CHEMBL2364696 | Envelope glycoprotein | Envelope glycoprotein D | Human herpesvirus 1 | unclassified | Small molecule | 2000 |
| O95259 | DOFETILIDE | Potassium voltage-gated channel subfamily H member 1 | Potassium voltage-gated channel subfamily H member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1999 | ||
| Q12809 | DOFETILIDE | HERG blocker | CHEMBL240 | HERG | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1999 |
| P46098 | DOLASETRON | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 1997 |
| Q7ZJM1 | DOLUTEGRAVIR | Human immunodeficiency virus type 1 integrase inhibitor | CHEMBL3471 | Human immunodeficiency virus type 1 integrase | Integrase | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2013 |
| P22303 | DONEPEZIL | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1996 |
| P08588 | DOPAMINE | Beta-1 adrenergic receptor agonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1974 |
| P14416 | DOPAMINE | D(2) dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 | ||
| P21728 | DOPAMINE | D(1A) dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 | ||
| P21917 | DOPAMINE | D(4) dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 | ||
| P21918 | DOPAMINE | D(1B) dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 | ||
| P35462 | DOPAMINE | D(3) dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 | ||
| P02918 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 2007 |
| P02919 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 2007 |
| P08506 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 2007 |
| P0AD65 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 2007 |
| P0AD68 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 2007 |
| P0AEB2 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 2007 |
| P24228 | DORIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 2007 |
| P00918 | DORZOLAMIDE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1994 |
| P02708 | DOXACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1991 |
| P07510 | DOXACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1991 |
| P11230 | DOXACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1991 |
| Q04844 | DOXACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1991 |
| Q07001 | DOXACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1991 |
| O14649 | DOXAPRAM | Potassium channel subfamily K member 3 blocker | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1965 |
| Q9NPC2 | DOXAPRAM | Potassium channel subfamily K member 9 blocker | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1965 |
| P25100 | DOXAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1990 |
| P35348 | DOXAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1990 |
| P35368 | DOXAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1990 |
| P23975 | DOXEPIN | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1969 |
| P35367 | DOXEPIN | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1969 | ||
| P11473 | DOXERCALCIFEROL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1999 |
| P11388 | DOXORUBICIN | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1974 |
| P11388 | DOXORUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1974 |
| DOXORUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1974 | |||
| P03956 | DOXYCYCLINE | Matrix metalloproteinase-1 inhibitor | CHEMBL332 | Matrix metalloproteinase-1 | Interstitial collagenase | Homo sapiens | enzyme protease metallo mam m10a | Small molecule | 1967 |
| P09237 | DOXYCYCLINE | Matrix metalloproteinase 7 inhibitor | CHEMBL4073 | Matrix metalloproteinase 7 | Matrilysin | Homo sapiens | enzyme protease metallo mam m10a | Small molecule | 1967 |
| P0A7V8 | DOXYCYCLINE | 30S ribosomal protein S4 | 30S ribosomal protein S4 | Escherichia coli (strain K12) | cytosolic other | Small molecule | 1967 | ||
| P0A7X3 | DOXYCYCLINE | 30S ribosomal protein S9 | 30S ribosomal protein S9 | Escherichia coli (strain K12) | cytosolic other | Small molecule | 1967 | ||
| P22894 | DOXYCYCLINE | Matrix metalloproteinase 8 inhibitor | CHEMBL4588 | Matrix metalloproteinase 8 | Neutrophil collagenase | Homo sapiens | enzyme protease metallo mam m10a | Small molecule | 1967 |
| P45452 | DOXYCYCLINE | Matrix metalloproteinase 13 inhibitor | CHEMBL280 | Matrix metalloproteinase 13 | Collagenase 3 | Homo sapiens | enzyme protease metallo mam m10a | Small molecule | 1967 |
| P35367 | DOXYLAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1948 |
| P10275 | DROMOSTANOLONE PROPIONATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1982 |
| P21554 | DRONABINOL | Cannabinoid CB1 receptor agonist | CHEMBL218 | Cannabinoid CB1 receptor | Cannabinoid receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor cannabinoid receptor | Small molecule | 1985 |
| O60741 | DRONEDARONE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2009 | ||
| O60840 | DRONEDARONE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 2009 |
| P35498 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| P35499 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| P63252 | DRONEDARONE | Inward rectifier potassium channel 2 blocker | CHEMBL1914276 | Inward rectifier potassium channel 2 | Inward rectifier potassium channel 2 | Homo sapiens | ion channel vgc k kir | Small molecule | 2009 |
| Q01118 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q01668 | DRONEDARONE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 2009 |
| Q13698 | DRONEDARONE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 2009 |
| Q13936 | DRONEDARONE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 2009 |
| Q14524 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q15858 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q99250 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9NY46 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9P1Z3 | DRONEDARONE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2009 | ||
| Q9UI33 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9UL51 | DRONEDARONE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2009 | ||
| Q9UQD0 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9Y3Q4 | DRONEDARONE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker | CHEMBL1250417 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2009 |
| Q9Y5Y9 | DRONEDARONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| P14416 | DROPERIDOL | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1970 |
| P21917 | DROPERIDOL | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1970 |
| P28223 | DROPERIDOL | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1970 |
| P35462 | DROPERIDOL | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1970 |
| P06401 | DROSPIRENONE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2001 |
| P08235 | DROSPIRENONE | Mineralocorticoid receptor antagonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 2001 |
| P00451 | DROTRECOGIN ALFA (ACTIVATED) | Coagulation factor VIII inhibitor | CHEMBL3143 | Coagulation factor VIII | Coagulation factor VIII | Homo sapiens | secreted | Unknown | 2001 |
| P12259 | DROTRECOGIN ALFA (ACTIVATED) | Coagulation factor V inhibitor | CHEMBL3618 | Coagulation factor V | Coagulation factor V | Homo sapiens | secreted | Unknown | 2001 |
| P07550 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P08588 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P08913 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P13945 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P18089 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P18825 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P25100 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P35348 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P35368 | DROXIDOPA | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P43220 | DULAGLUTIDE | Glucagon-like peptide 1 receptor agonist | CHEMBL1784 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon-like peptide receptor | Protein | 2014 |
| P23975 | DULOXETINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2004 |
| P31645 | DULOXETINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2004 |
| P18405 | DUTASTERIDE | Steroid 5-alpha-reductase inhibitor | CHEMBL2363075 | Steroid 5-alpha-reductase | 3-oxo-5-alpha-steroid 4-dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 2001 |
| P31213 | DUTASTERIDE | Steroid 5-alpha-reductase inhibitor | CHEMBL2363075 | Steroid 5-alpha-reductase | 3-oxo-5-alpha-steroid 4-dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 2001 |
| Q9H8P0 | DUTASTERIDE | Steroid 5-alpha-reductase inhibitor | CHEMBL2363075 | Steroid 5-alpha-reductase | Polyprenol reductase | Homo sapiens | enzyme reductase | Small molecule | 2001 |
| P35498 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35499 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q01118 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q14524 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q15858 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q99250 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9NY46 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UI33 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UQD0 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | DYCLONINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P06401 | DYDROGESTERONE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1982 |
| P27815 | DYPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1951 |
| Q07343 | DYPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1951 |
| Q08493 | DYPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1951 |
| Q08499 | DYPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1951 |
| Q14432 | DYPHYLLINE | Phosphodiesterase 3A inhibitor | CHEMBL241 | Phosphodiesterase 3A | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1951 |
| P03952 | ECALLANTIDE | Plasma kallikrein inhibitor | CHEMBL2000 | Plasma kallikrein | Plasma kallikrein | Homo sapiens | enzyme protease serine pas s1a | Protein | 2009 |
| P22303 | ECHOTHIOPHATE | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1960 |
| P10613 | ECONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1982 |
| P01031 | ECULIZUMAB | Complement C5 inhibitor | CHEMBL2364163 | Complement C5 | Complement C5 | Homo sapiens | secreted | Antibody | 2007 |
| EDETATE CALCIUM DISODIUM | Unknown | Small molecule | 1953 | ||||||
| EDETATE DISODIUM | Calcium chelating agent | CHEMBL2364030 | Calcium | null | Small molecule | 1982 | |||
| EDETATE DISODIUM | CHEMBL2364030 | Calcium | Small molecule | 1982 | |||||
| P00742 | EDOXABAN | Coagulation factor X inhibitor | CHEMBL244 | Coagulation factor X | Coagulation factor X | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 2015 |
| P22303 | EDROPHONIUM | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1951 |
| P20701 | EFALIZUMAB | Integrin alpha-L/beta-2 (LFA-1) inhibitor | CHEMBL2364172 | Integrin alpha-L/beta-2 (LFA-1) | Integrin alpha-L | Homo sapiens | adhesion | Antibody | 2003 |
| P20701 | EFALIZUMAB | Integrin alpha-L/beta-2 (LFA-1) inhibitor | CHEMBL2364172 | Integrin alpha-L/beta-2 (LFA-1) | Integrin alpha-L | Homo sapiens | membrane receptor | Antibody | 2003 |
| P03369 | EFAVIRENZ | Gag-Pol polyprotein | Gag-Pol polyprotein | Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) | Unclassified | Small molecule | 1998 | ||
| Q72547 | EFAVIRENZ | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1998 |
| F2SHH3 | EFINACONAZOLE | Lanosterol 14-alpha demethylase inhibitor | CHEMBL3307221 | Lanosterol 14-alpha demethylase | Uncharacterized protein | Trichophyton rubrum (strain ATCC MYA-4607 / CBS 118892) (Athlete'sfoot fungus) | unclassified | Small molecule | 2014 |
| P11926 | EFLORNITHINE | Ornithine decarboxylase inhibitor | CHEMBL1869 | Ornithine decarboxylase | Ornithine decarboxylase | Homo sapiens | enzyme lyase | Small molecule | 1990 |
| Q9TZZ6 | EFLORNITHINE | Ornithine decarboxylase | Ornithine decarboxylase | Trypanosoma brucei gambiense | Lyase | Small molecule | 1990 | ||
| P28221 | ELETRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| P28222 | ELETRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| P30939 | ELETRIPTAN | Serotonin 1f (5-HT1f) receptor agonist | CHEMBL1805 | Serotonin 1f (5-HT1f) receptor | 5-hydroxytryptamine receptor 1F | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| Q16739 | ELIGLUSTAT | Ceramide glucosyltransferase inhibitor | CHEMBL2063 | Ceramide glucosyltransferase | Ceramide glucosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 2014 |
| ELOSULFASE ALFA | Keratan sulfate hydrolytic enzyme | CHEMBL3140341 | Keratan sulfate | Homo sapiens | Enzyme | 2014 | |||
| ELOSULFASE ALFA | Chondroitin-6-sulfate hydrolytic enzyme | CHEMBL3140342 | Chondroitin-6-sulfate | Homo sapiens | Enzyme | 2014 | |||
| P40238 | ELTROMBOPAG | Thrombopoietin receptor agonist | CHEMBL1864 | Thrombopoietin receptor | Thrombopoietin receptor | Homo sapiens | membrane receptor | Small molecule | 2008 |
| P35372 | ELUXADOLINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2015 |
| P41143 | ELUXADOLINE | Delta-type opioid receptor | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2015 | ||
| Q7ZJM1 | ELVITEGRAVIR | Human immunodeficiency virus type 1 integrase inhibitor | CHEMBL3471 | Human immunodeficiency virus type 1 integrase | Integrase | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2012 |
| P35367 | EMEDASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1997 |
| P31639 | EMPAGLIFLOZIN | Sodium/glucose cotransporter 2 inhibitor | CHEMBL3884 | Sodium/glucose cotransporter 2 | Sodium/glucose cotransporter 2 | Homo sapiens | transporter electrochemical slc slc05 | Small molecule | 2014 |
| Q72547 | EMTRICITABINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2003 |
| P12821 | ENALAPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1985 |
| P12821 | ENALAPRILAT | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1988 |
| P03372 | ENCLOMIPHENE | Estrogen receptor alpha modulator | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1967 |
| O00591 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| O14649 | ENFLURANE | Potassium channel subfamily K member 3 opener | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1972 |
| O14764 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| O95069 | ENFLURANE | Potassium channel subfamily K member 2 opener | CHEMBL2321615 | Potassium channel subfamily K member 2 | Potassium channel subfamily K member 2 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1972 |
| P03886 | ENFLURANE | NADH-ubiquinone oxidoreductase chain 1 | NADH-ubiquinone oxidoreductase chain 1 | Homo sapiens | enzyme reductase | Small molecule | 1972 | ||
| P14867 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P18505 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P18507 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P23415 | ENFLURANE | Glycine receptor (alpha-1/beta) positive modulator | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 1972 |
| P28472 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P30049 | ENFLURANE | "ATP synthase subunit delta, mitochondrial" | "ATP synthase subunit delta, mitochondrial" | Homo sapiens | Unclassified | Small molecule | 1972 | ||
| P31644 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P34903 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P42261 | ENFLURANE | Glutamate receptor 1 | Glutamate receptor 1 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 1972 | ||
| P47869 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P47870 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P48169 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P57789 | ENFLURANE | Potassium channel subfamily K member 10 opener | CHEMBL2331041 | Potassium channel subfamily K member 10 | Potassium channel subfamily K member 10 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1972 |
| P78334 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| P98194 | ENFLURANE | Calcium-transporting ATPase type 2C member 1 | Calcium-transporting ATPase type 2C member 1 | Homo sapiens | Hydrolase | Small molecule | 1972 | ||
| Q09470 | ENFLURANE | Potassium voltage-gated channel subfamily A member 1 | Potassium voltage-gated channel subfamily A member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1972 | ||
| Q16445 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| Q7Z418 | ENFLURANE | Potassium channel subfamily K member 18 opener | CHEMBL2331042 | Potassium channel subfamily K member 18 | Potassium channel subfamily K member 18 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1972 |
| Q8N1C3 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| Q99928 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| Q9NPC2 | ENFLURANE | Potassium channel subfamily K member 9 opener | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1972 |
| Q9UN88 | ENFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1972 |
| O40239 | ENFUVIRTIDE | Transmembrane glycoprotein gp41 inhibitor | CHEMBL2362987 | Transmembrane glycoprotein gp41 | Transmembrane glycoprotein gp41 | Human immunodeficiency virus | unclassified | Protein | 2003 |
| P22118 | ENOXACIN | DNA gyrase inhibitor | CHEMBL2311244 | DNA gyrase | DNA gyrase subunit B | Neisseria gonorrhoeae | enzyme isomerase | Small molecule | 1991 |
| P48371 | ENOXACIN | DNA gyrase inhibitor | CHEMBL2311244 | DNA gyrase | DNA gyrase subunit A | Neisseria gonorrhoeae | enzyme isomerase | Small molecule | 1991 |
| P48374 | ENOXACIN | Topoisomerase IV inhibitor | CHEMBL2363077 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Neisseria gonorrhoeae | enzyme isomerase | Small molecule | 1991 |
| Q5EP76 | ENOXACIN | Topoisomerase IV inhibitor | CHEMBL2363077 | Topoisomerase IV | TopB | Neisseria gonorrhoeae | enzyme isomerase | Small molecule | 1991 |
| P01008 | ENOXAPARIN SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 1993 |
| P21964 | ENTACAPONE | Catechol O-methyltransferase inhibitor | CHEMBL2023 | Catechol O-methyltransferase | Catechol O-methyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1999 |
| Q9IF40 | ENTECAVIR | DNA polymerase/reverse transcriptase inhibitor | CHEMBL2362994 | DNA polymerase/reverse transcriptase | Protein P | Hepatitis B virus | enzyme transferase | Small molecule | 2005 |
| P10275 | ENZALUTAMIDE | Androgen Receptor antagonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 2012 |
| P35367 | EPINASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2003 |
| P07550 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P08588 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P08913 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P13945 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P18089 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P18825 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P25100 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P35348 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P35368 | EPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1965 |
| P11388 | EPIRUBICIN | DNA topoisomerase 2-alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 0 | ||
| EPIRUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 0 | |||
| P08235 | EPLERENONE | Mineralocorticoid receptor antagonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 2002 |
| P19235 | EPOETIN ALFA | Erythropoietin receptor agonist | CHEMBL1817 | Erythropoietin receptor | Erythropoietin receptor | Homo sapiens | membrane receptor | Protein | 1989 |
| P34995 | EPOPROSTENOL | Prostaglandin E2 receptor EP1 subtype | Prostaglandin E2 receptor EP1 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1995 | ||
| P43119 | EPOPROSTENOL | Prostanoid IP receptor agonist | CHEMBL1995 | Prostanoid IP receptor | Prostacyclin receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1995 |
| P30556 | EPROSARTAN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1997 |
| P05106 | EPTIFIBATIDE | Integrin alpha-IIb/beta-3 inhibitor | CHEMBL2093869 | Integrin alpha-IIb/beta-3 | Integrin beta-3 | Homo sapiens | membrane receptor | Protein | 1998 |
| P08514 | EPTIFIBATIDE | Integrin alpha-IIb/beta-3 inhibitor | CHEMBL2093869 | Integrin alpha-IIb/beta-3 | Integrin alpha-IIb | Homo sapiens | membrane receptor | Protein | 1998 |
| P11473 | ERGOCALCIFEROL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1941 |
| P08908 | ERGOLOID | Serotonin 1a (5-HT1a) receptor agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1953 |
| P08913 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P14416 | ERGOLOID | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1953 |
| P18089 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P18825 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P21728 | ERGOLOID | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1953 |
| P21917 | ERGOLOID | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1953 |
| P21918 | ERGOLOID | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1953 |
| P25100 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P28222 | ERGOLOID | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1953 |
| P35348 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P35368 | ERGOLOID | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P35462 | ERGOLOID | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1953 |
| P08913 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P18089 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P18825 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P25100 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P28221 | ERGOTAMINE | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1948 |
| P35348 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P35368 | ERGOTAMINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1948 |
| P04350 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 2010 |
| P07437 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 2010 |
| P68371 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 2010 |
| Q13509 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q13885 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 2010 |
| Q3ZCM7 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9BUF5 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9BVA1 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 2010 |
| Q9H4B7 | ERIBULIN | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 2010 |
| P35498 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| P35499 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q01118 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q14524 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q15858 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q99250 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9NY46 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9UI33 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9UQD0 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9Y5Y9 | ERLOSAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| P00533 | ERLOTINIB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2004 |
| P02918 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 2001 |
| P02919 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 2001 |
| P08506 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 2001 |
| P0AD65 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 2001 |
| P0AD68 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 2001 |
| P0AEB2 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 2001 |
| P24228 | ERTAPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 2001 |
| ERYTHROMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1964 | ||
| ERYTHROMYCIN ESTOLATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1967 | ||
| ERYTHROMYCIN ETHYLSUCCINATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1965 | ||
| P31645 | ESCITALOPRAM | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2002 |
| P35498 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| P35499 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q01118 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q14524 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q15858 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q99250 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9NY46 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9UI33 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9UQD0 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| Q9Y5Y9 | ESLICARBAZEPINE ACETATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2009 |
| P07550 | ESMOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P08588 | ESMOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P20648 | ESOMEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 2001 |
| P20648 | ESOMEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 2001 |
| P14867 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| P18507 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| P31644 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| P34903 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| P47869 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| Q8N1C3 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| Q99928 | ESTAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1990 |
| P03372 | ESTRADIOL | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1975 |
| P03372 | ESTRADIOL ACETATE | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2003 |
| P03372 | ESTRADIOL CYPIONATE | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1979 |
| P03372 | ESTRADIOL VALERATE | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2010 |
| Q92731 | ESTRAMUSTINE PHOSPHATE | DNA inhibitor | CHEMBL2311221 | DNA | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1981 |
| Q92731 | ESTRAMUSTINE PHOSPHATE | Estrogen receptor beta | CHEMBL242 | Estrogen receptor beta | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1981 |
| ESTRAMUSTINE PHOSPHATE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1981 | |||
| P03372 | "ESTROGENS, CONJUGATED" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1942 |
| Q92731 | "ESTROGENS, CONJUGATED" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1942 |
| P03372 | "ESTROGENS, CONJUGATED SYNTHETIC A" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1999 |
| Q92731 | "ESTROGENS, CONJUGATED SYNTHETIC A" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1999 |
| P03372 | "ESTROGENS, ESTERIFIED" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1977 |
| Q92731 | "ESTROGENS, ESTERIFIED" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1977 |
| P03372 | ESTRONE | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1979 |
| Q92731 | ESTRONE | Estrogen receptor beta | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1979 | ||
| P03372 | ESTRONE SULFURIC ACID | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1977 |
| P14867 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P18507 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P31644 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P34903 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P47869 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q8N1C3 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| Q99928 | ESZOPICLONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2004 |
| P01375 | ETANERCEPT | TNF-alpha inhibitor | CHEMBL1825 | TNF-alpha | Tumor necrosis factor | Homo sapiens | secreted | Protein | 1998 |
| Q13621 | ETHACRYNIC ACID | Sodium-(potassium)-chloride cotransporter 2 inhibitor | CHEMBL1874 | Sodium-(potassium)-chloride cotransporter 2 | Solute carrier family 12 member 1 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1967 |
| P9WNL9 | ETHAMBUTOL | Arabinosyltransferase A inhibitor | CHEMBL1877 | Arabinosyltransferase A | Probable arabinosyltransferase A | Mycobacterium tuberculosis | enzyme transferase | Small molecule | 1967 |
| ETHANOLAMINE OLEATE | Calcium chelating agent | CHEMBL2364030 | Calcium | null | Small molecule | 1988 | |||
| ETHANOLAMINE OLEATE | CHEMBL2364030 | Calcium | Small molecule | 1988 | |||||
| O00591 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| O14764 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P14867 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P18505 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P18507 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P28472 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P31644 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P34903 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P47869 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P47870 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P48169 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| P78334 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| Q16445 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| Q8N1C3 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| Q99928 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| Q9UN88 | ETHCHLORVYNOL | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1961 |
| ETHINAMATE | Unknown | Small molecule | 1982 | ||||||
| P03372 | ETHINYL ESTRADIOL | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2001 |
| P9WGR1 | ETHIONAMIDE | Enoyl-[acyl-carrier-protein] reductase inhibitor | CHEMBL1849 | Enoyl-[acyl-carrier-protein] reductase | Enoyl-[acyl-carrier-protein] reductase [NADH] | Mycobacterium tuberculosis | enzyme reductase | Small molecule | 1965 |
| P11229 | ETHOPROPAZINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| O43497 | ETHOSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1960 |
| O95180 | ETHOSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1960 |
| Q9P0X4 | ETHOSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1960 |
| P35498 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| P35499 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q01118 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q14524 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q15858 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q99250 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9NY46 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9UI33 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9UQD0 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9Y5Y9 | ETHOTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| O43570 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 12 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P00915 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 1 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P00918 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P07451 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 3 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P22748 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 4 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P23280 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 6 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P35218 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | "Carbonic anhydrase 5A, mitochondrial" | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P43166 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 7 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| Q16790 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 9 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| Q8N1Q1 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 13 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| Q9ULX7 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | Carbonic anhydrase 14 | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| Q9Y2D0 | ETHOXZOLAMIDE | Carbonic anhydrase inhibitor | CHEMBL2095180 | Carbonic anhydrase | "Carbonic anhydrase 5B, mitochondrial" | Homo sapiens | enzyme lyase | Small molecule | 1982 |
| P10275 | ETHYLESTRENOL | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1964 |
| P06401 | ETHYNODIOL DIACETATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1966 |
| P35498 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| P35499 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q01118 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q14524 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q15858 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q99250 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q9NY46 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q9UI33 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q9UQD0 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| Q9Y5Y9 | ETIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1976 |
| ETIDRONIC ACID | ATP inhibitor | CHEMBL2366048 | ATP | Homo sapiens | Small molecule | 1977 | |||
| P35354 | ETODOLAC | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1991 |
| O00591 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| O14764 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P14867 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18505 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18507 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P31644 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P34903 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47869 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P48169 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P78334 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q16445 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q8N1C3 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q99928 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q9UN88 | ETOMIDATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P06401 | ETONOGESTREL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2001 |
| P11388 | ETOPOSIDE | DNA topoisomerase II inhibitor | CHEMBL2094255 | DNA topoisomerase II | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1983 |
| Q02880 | ETOPOSIDE | DNA topoisomerase II inhibitor | CHEMBL2094255 | DNA topoisomerase II | DNA topoisomerase 2-beta | Homo sapiens | enzyme isomerase | Small molecule | 1983 |
| P11388 | ETOPOSIDE PHOSPHATE | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1996 |
| Q72547 | ETRAVIRINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2008 |
| P10276 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1986 |
| P10826 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1986 |
| P13631 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1986 |
| P19793 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-alpha | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b1 | Small molecule | 1986 |
| P28702 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-beta | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b2 | Small molecule | 1986 |
| P48443 | ETRETINATE | Retinoid receptor agonist | CHEMBL2363071 | Retinoid receptor | Retinoic acid receptor RXR-gamma | Homo sapiens | transcription factor nuclear receptor nr2 nr2b nr2b3 | Small molecule | 1986 |
| P62942 | EVEROLIMUS | FK506-binding protein 1A inhibitor | CHEMBL1902 | FK506-binding protein 1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Small molecule | 2009 |
| P11511 | EXEMESTANE | Cytochrome P450 19A1 inhibitor | CHEMBL1978 | Cytochrome P450 19A1 | Aromatase | Homo sapiens | enzyme cytochrome p450 cyp_19 cyp_19a cyp_19a1 | Small molecule | 1999 |
| P43220 | EXENATIDE | Glucagon-like peptide 1 receptor agonist | CHEMBL1784 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon-like peptide receptor | Protein | 2005 |
| Q9UHC9 | EZETIMIBE | Niemann-Pick C1-like protein 1 inhibitor | CHEMBL2027 | Niemann-Pick C1-like protein 1 | Niemann-Pick C1-like protein 1 | Homo sapiens | membrane other | Small molecule | 2002 |
| O43525 | EZOGABINE | KCNQ (Kv7) potassium channel blocker | CHEMBL2363063 | KCNQ (Kv7) potassium channel | Potassium voltage-gated channel subfamily KQT member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2011 |
| O43526 | EZOGABINE | KCNQ (Kv7) potassium channel blocker | CHEMBL2363063 | KCNQ (Kv7) potassium channel | Potassium voltage-gated channel subfamily KQT member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2011 |
| P51787 | EZOGABINE | KCNQ (Kv7) potassium channel blocker | CHEMBL2363063 | KCNQ (Kv7) potassium channel | Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2011 |
| P56696 | EZOGABINE | KCNQ (Kv7) potassium channel blocker | CHEMBL2363063 | KCNQ (Kv7) potassium channel | Potassium voltage-gated channel subfamily KQT member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2011 |
| Q9NR82 | EZOGABINE | KCNQ (Kv7) potassium channel blocker | CHEMBL2363063 | KCNQ (Kv7) potassium channel | Potassium voltage-gated channel subfamily KQT member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 2011 |
| P04293 | FAMCICLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1994 |
| P25021 | FAMOTIDINE | Histamine H2 receptor antagonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1986 |
| P47989 | FEBUXOSTAT | Xanthine dehydrogenase inhibitor | CHEMBL1929 | Xanthine dehydrogenase | Xanthine dehydrogenase/oxidase | Homo sapiens | enzyme reductase | Small molecule | 2009 |
| O15399 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| O60391 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| Q05586 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| Q12879 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| Q13224 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| Q14957 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| Q8TCU5 | FELBAMATE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1993 |
| O60840 | FELODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1991 |
| P08235 | FELODIPINE | Mineralocorticoid receptor antagonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1991 |
| Q01668 | FELODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1991 |
| Q13698 | FELODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1991 |
| Q13936 | FELODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1991 |
| Q07869 | FENOFIBRATE | Peroxisome proliferator-activated receptor alpha agonist | CHEMBL239 | Peroxisome proliferator-activated receptor alpha | Peroxisome proliferator-activated receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c1 | Small molecule | 1993 |
| Q07869 | FENOFIBRIC ACID | Peroxisome proliferator-activated receptor alpha agonist | CHEMBL239 | Peroxisome proliferator-activated receptor alpha | Peroxisome proliferator-activated receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c1 | Small molecule | 2008 |
| P21728 | FENOLDOPAM | Dopamine D1 receptor agonist | CHEMBL2056 | Dopamine D1 receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P23219 | FENOPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P35354 | FENOPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P35372 | FENTANYL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1968 |
| FERRIC CITRATE | Phosphate chelating agent | CHEMBL2364184 | Phosphate | Homo sapiens | Small molecule | 2014 | |||
| FERUMOXYTOL | Unknown | Unknown | 2009 | ||||||
| P08172 | FESOTERODINE | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2008 |
| P20309 | FESOTERODINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2008 |
| P35367 | FEXOFENADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1996 |
| P02671 | "FIBRINOLYSIN, HUMAN" | Fibrinogen inhibitor | CHEMBL2364709 | Fibrinogen | Fibrinogen alpha chain | Homo sapiens | secreted | Unknown | 1964 |
| P02675 | "FIBRINOLYSIN, HUMAN" | Fibrinogen inhibitor | CHEMBL2364709 | Fibrinogen | Fibrinogen beta chain | Homo sapiens | secreted | Unknown | 1964 |
| P02679 | "FIBRINOLYSIN, HUMAN" | Fibrinogen inhibitor | CHEMBL2364709 | Fibrinogen | Fibrinogen gamma chain | Homo sapiens | secreted | Unknown | 1964 |
| Q182S6 | FIDAXOMICIN | DNA-directed RNA polymerase inhibitor | CHEMBL2363852 | DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit omega | Clostridium difficile | enzyme transferase | Small molecule | 2011 |
| Q18CF1 | FIDAXOMICIN | DNA-directed RNA polymerase inhibitor | CHEMBL2363852 | DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta | Clostridium difficile | enzyme transferase | Small molecule | 2011 |
| Q18CF3 | FIDAXOMICIN | DNA-directed RNA polymerase inhibitor | CHEMBL2363852 | DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta' | Clostridium difficile | enzyme transferase | Small molecule | 2011 |
| Q18CI5 | FIDAXOMICIN | DNA-directed RNA polymerase inhibitor | CHEMBL2363852 | DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit alpha | Clostridium difficile | enzyme transferase | Small molecule | 2011 |
| Q99062 | FILGRASTIM | Granulocyte colony stimulating factor receptor agonist | CHEMBL1996 | Granulocyte colony stimulating factor receptor | Granulocyte colony-stimulating factor receptor | Homo sapiens | membrane receptor | Protein | 1991 |
| P0A0K8 | FINAFLOXACIN | DNA gyrase inhibitor | CHEMBL3038482 | DNA gyrase | DNA gyrase subunit B | Staphylococcus aureus | enzyme | Small molecule | 2014 |
| P0C1S7 | FINAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL3038508 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Staphylococcus aureus | enzyme | Small molecule | 2014 |
| P0C1U9 | FINAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL3038508 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Staphylococcus aureus | enzyme | Small molecule | 2014 |
| P20831 | FINAFLOXACIN | DNA gyrase inhibitor | CHEMBL3038482 | DNA gyrase | DNA gyrase subunit A | Staphylococcus aureus | enzyme | Small molecule | 2014 |
| P48372 | FINAFLOXACIN | DNA gyrase inhibitor | CHEMBL3390828 | DNA gyrase | DNA gyrase subunit A | Pseudomonas aeruginosa | enzyme | Small molecule | 2014 |
| Q9HUJ8 | FINAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL3390827 | Topoisomerase IV | Pseudomonas aeruginosa | enzyme isomerase | Small molecule | 2014 | |
| Q9HUK1 | FINAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL3390827 | Topoisomerase IV | Pseudomonas aeruginosa | enzyme isomerase | Small molecule | 2014 | |
| Q9I7C2 | FINAFLOXACIN | DNA gyrase inhibitor | CHEMBL3390828 | DNA gyrase | DNA gyrase subunit B | Pseudomonas aeruginosa | enzyme | Small molecule | 2014 |
| P18405 | FINASTERIDE | 3-oxo-5-alpha-steroid 4-dehydrogenase 1 | 3-oxo-5-alpha-steroid 4-dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1992 | ||
| P31213 | FINASTERIDE | Steroid 5-alpha-reductase 2 inhibitor | CHEMBL1856 | Steroid 5-alpha-reductase 2 | 3-oxo-5-alpha-steroid 4-dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 1992 |
| O95136 | FINGOLIMOD | Sphingosine 1-phosphate receptor agonist | CHEMBL2363041 | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor 2 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor edg receptor | Small molecule | 2010 |
| O95977 | FINGOLIMOD | Sphingosine 1-phosphate receptor agonist | CHEMBL2363041 | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor 4 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor edg receptor | Small molecule | 2010 |
| P21453 | FINGOLIMOD | Sphingosine 1-phosphate receptor agonist | CHEMBL2363041 | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor edg receptor | Small molecule | 2010 |
| Q99500 | FINGOLIMOD | Sphingosine 1-phosphate receptor agonist | CHEMBL2363041 | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor 3 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor edg receptor | Small molecule | 2010 |
| Q9H228 | FINGOLIMOD | Sphingosine 1-phosphate receptor agonist | CHEMBL2363041 | Sphingosine 1-phosphate receptor | Sphingosine 1-phosphate receptor 5 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor edg receptor | Small molecule | 2010 |
| O60658 | FLAVOXATE | Phosphodiesterase 8 inhibitor | CHEMBL2363067 | Phosphodiesterase 8 | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8a | Small molecule | 1970 |
| O95263 | FLAVOXATE | Phosphodiesterase 8 inhibitor | CHEMBL2363067 | Phosphodiesterase 8 | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8B" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8b | Small molecule | 1970 |
| P27815 | FLAVOXATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1970 |
| Q07343 | FLAVOXATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1970 |
| Q08493 | FLAVOXATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1970 |
| Q08499 | FLAVOXATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1970 |
| Q13946 | FLAVOXATE | Phosphodiesterase 7 inhibitor | CHEMBL2111411 | Phosphodiesterase 7 | "High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7a | Small molecule | 1970 |
| Q9NP56 | FLAVOXATE | Phosphodiesterase 7 inhibitor | CHEMBL2111411 | Phosphodiesterase 7 | "cAMP-specific 3',5'-cyclic phosphodiesterase 7B" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7b | Small molecule | 1970 |
| Q14524 | FLECAINIDE | Sodium channel protein type V alpha subunit blocker | CHEMBL1980 | Sodium channel protein type V alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| P04818 | FLOXURIDINE | Thymidylate synthase inhibitor | CHEMBL1952 | Thymidylate synthase | Thymidylate synthase | Homo sapiens | enzyme transferase | Small molecule | 1970 |
| P10613 | FLUCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1990 |
| P0CS13 | FLUCYTOSINE | Thymidylate synthase inhibitor | CHEMBL4665 | Thymidylate synthase | Thymidylate synthase | Cryptococcus neoformans var. neoformans B-3501A | enzyme transferase | Small molecule | 1971 |
| P12461 | FLUCYTOSINE | Thymidylate synthase inhibitor | CHEMBL2364680 | Thymidylate synthase | Thymidylate synthase | Candida albicans | enzyme transferase | Small molecule | 1971 |
| P26358 | FLUCYTOSINE | DNA (cytosine-5)-methyltransferase 1 | DNA (cytosine-5)-methyltransferase 1 | Homo sapiens | epigenetic regulator writer dnmt | Small molecule | 1971 | ||
| P09884 | FLUDARABINE PHOSPHATE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1991 |
| P23921 | FLUDARABINE PHOSPHATE | Ribonucleoside-diphosphate reductase RR1 inhibitor | CHEMBL2095215 | Ribonucleoside-diphosphate reductase RR1 | Ribonucleoside-diphosphate reductase large subunit | Homo sapiens | enzyme reductase | Small molecule | 1991 |
| P28340 | FLUDARABINE PHOSPHATE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase delta catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1991 |
| Q07864 | FLUDARABINE PHOSPHATE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase epsilon catalytic subunit A | Homo sapiens | enzyme transferase | Small molecule | 1991 |
| P08235 | FLUDROCORTISONE ACETATE | Mineralocorticoid receptor agonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1955 |
| P14867 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| P18507 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| P31644 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| P34903 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| P47869 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| Q8N1C3 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| Q99928 | FLUMAZENIL | GABA-A receptor; anion channel allosteric antagonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1991 |
| P04150 | FLUMETHASONE PIVALATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P04150 | FLUNISOLIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1981 |
| P04150 | FLUOCINOLONE ACETONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1963 |
| P04150 | FLUOCINONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1971 |
| P04150 | FLUOROMETHOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1972 |
| P04150 | FLUOROMETHOLONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1986 |
| P04818 | FLUOROURACIL | Thymidylate synthase inhibitor | CHEMBL1952 | Thymidylate synthase | Thymidylate synthase | Homo sapiens | enzyme transferase | Small molecule | 1962 |
| FLUOROURACIL | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1962 | |||
| FLUOROURACIL | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 1962 | |||
| P31645 | FLUOXETINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1987 |
| P10275 | FLUOXYMESTERONE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1956 |
| P14416 | FLUPHENAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1959 |
| P25100 | FLUPHENAZINE | Alpha-1D adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1959 | ||
| P28223 | FLUPHENAZINE | 5-hydroxytryptamine receptor 2A | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1959 | ||
| P34969 | FLUPHENAZINE | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1959 | ||
| P35348 | FLUPHENAZINE | Alpha-1A adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1959 | ||
| P35462 | FLUPHENAZINE | D(3) dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1959 | ||
| P14416 | FLUPHENAZINE DECANOATE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1972 |
| P14416 | FLUPHENAZINE ENANTHATE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P04150 | FLUPREDNISOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P04150 | FLURANDRENOLIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1965 |
| P14867 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| P18507 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| P31644 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| P34903 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| P47869 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| Q8N1C3 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| Q99928 | FLURAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1970 |
| P23219 | FLURBIPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1986 |
| P35354 | FLURBIPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1986 |
| P10275 | FLUTAMIDE | Androgen Receptor antagonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1989 |
| P04150 | FLUTICASONE FUROATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 2007 |
| P04150 | FLUTICASONE PROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1990 |
| P06401 | FLUTICASONE PROPIONATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1990 |
| P04035 | FLUVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1993 |
| P31645 | FLUVOXAMINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1994 |
| P00325 | FOMEPIZOLE | Alcohol dehydrogenase class I inhibitor | CHEMBL2363044 | Alcohol dehydrogenase class I | Alcohol dehydrogenase 1B | Homo sapiens | enzyme reductase | Small molecule | 1997 |
| P00326 | FOMEPIZOLE | Alcohol dehydrogenase class I inhibitor | CHEMBL2363044 | Alcohol dehydrogenase class I | Alcohol dehydrogenase 1C | Homo sapiens | enzyme reductase | Small molecule | 1997 |
| P07327 | FOMEPIZOLE | Alcohol dehydrogenase class I inhibitor | CHEMBL2363044 | Alcohol dehydrogenase class I | Alcohol dehydrogenase 1A | Homo sapiens | enzyme reductase | Small molecule | 1997 |
| FOMIVIRSEN SODIUM | Major intermediate early region 2 mRNA antisense inhibitor | CHEMBL2364186 | Major intermediate early region 2 mRNA | Human cytomegalovirus | Oligonucleotide | 1998 | |||
| P01008 | FONDAPARINUX | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 2001 |
| P07550 | FORMOTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2001 |
| Q72874 | FOSAMPRENAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 2003 |
| P25103 | FOSAPREPITANT | Neurokinin 1 receptor antagonist | CHEMBL249 | Neurokinin 1 receptor | Substance-P receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide neurokinin receptor | Small molecule | 2008 |
| P04293 | FOSCARNET | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1991 |
| P0A749 | FOSFOMYCIN | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | CHEMBL1984 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase | UDP-N-acetylglucosamine 1-carboxyvinyltransferase | Escherichia coli K-12 | enzyme transferase | Small molecule | 1996 |
| P12821 | FOSINOPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1991 |
| P35498 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| P35499 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q01118 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q14524 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q15858 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q99250 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9NY46 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UI33 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UQD0 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9Y5Y9 | FOSPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| O14764 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P14867 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P18505 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P18507 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P28472 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P31644 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P34903 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P47869 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P47870 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| P48169 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| Q16445 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| Q8N1C3 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| Q99928 | FOSPROPOFOL | GABA-A receptor | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 2008 | ||
| FOSPROPOFOL | Unknown | Small molecule | 2008 | ||||||
| P28221 | FROVATRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P28222 | FROVATRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P03372 | FULVESTRANT | Estrogen receptor antagonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2002 |
| Q92731 | FULVESTRANT | Estrogen receptor antagonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 2002 |
| FURAZOLIDONE | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1958 | |||
| Q13621 | FUROSEMIDE | Sodium-(potassium)-chloride cotransporter 2 inhibitor | CHEMBL1874 | Sodium-(potassium)-chloride cotransporter 2 | Solute carrier family 12 member 1 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1966 |
| P54289 | GABAPENTIN | Voltage-gated calcium channel modulator | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 1993 |
| P54289 | GABAPENTIN ENACARBIL | Voltage-gated calcium channel modulator | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 2011 |
| GADOXETIC ACID | Unknown | Small molecule | 2008 | ||||||
| P22303 | GALANTAMINE | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 2001 |
| P02708 | GALLAMINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 |
| P07510 | GALLAMINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1982 |
| P11230 | GALLAMINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 |
| Q04844 | GALLAMINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1982 |
| Q07001 | GALLAMINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1982 |
| P31350 | GALLIUM NITRATE | Ribonucleoside-diphosphate reductase RR1 inhibitor | CHEMBL2095215 | Ribonucleoside-diphosphate reductase RR1 | Ribonucleoside-diphosphate reductase subunit M2 | Homo sapiens | enzyme | Small molecule | 1991 |
| P31350 | GALLIUM NITRATE | Hydroxyapatite chelating agent | CHEMBL2363055 | Hydroxyapatite | Ribonucleoside-diphosphate reductase subunit M2 | Homo sapiens | enzyme | Small molecule | 1991 |
| GALLIUM NITRATE | Hydroxyapatite chelating agent | CHEMBL2363055 | Hydroxyapatite | Homo sapiens | Small molecule | 1991 | |||
| GALSULFASE | Dermatan sulfate hydrolytic enzyme | CHEMBL2364179 | Dermatan sulfate | Homo sapiens | Enzyme | 2005 | |||
| P04293 | GANCICLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1989 |
| P30968 | GANIRELIX ACETATE | Gonadotropin-releasing hormone receptor antagonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1999 |
| P0A4L9 | GATIFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1999 |
| P72524 | GATIFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1999 |
| P72525 | GATIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1999 |
| Q59961 | GATIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1999 |
| P00533 | GEFITINIB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2003 |
| P04818 | GEMCITABINE | Thymidylate synthase | Thymidylate synthase | Homo sapiens | enzyme transferase | Small molecule | 1996 | ||
| P09884 | GEMCITABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1996 |
| P23921 | GEMCITABINE | Ribonucleoside-diphosphate reductase RR1 inhibitor | CHEMBL2095215 | Ribonucleoside-diphosphate reductase RR1 | Ribonucleoside-diphosphate reductase large subunit | Homo sapiens | enzyme reductase | Small molecule | 1996 |
| P28340 | GEMCITABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase delta catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 1996 |
| P30085 | GEMCITABINE | UMP-CMP kinase | UMP-CMP kinase | Homo sapiens | enzyme | Small molecule | 1996 | ||
| Q07864 | GEMCITABINE | DNA polymerase (alpha/delta/epsilon) inhibitor | CHEMBL2363042 | DNA polymerase (alpha/delta/epsilon) | DNA polymerase epsilon catalytic subunit A | Homo sapiens | enzyme transferase | Small molecule | 1996 |
| Q07869 | GEMFIBROZIL | Peroxisome proliferator-activated receptor alpha agonist | CHEMBL239 | Peroxisome proliferator-activated receptor alpha | Peroxisome proliferator-activated receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c1 | Small molecule | 1981 |
| P0A4L9 | GEMIFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 2003 |
| P72524 | GEMIFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 2003 |
| P72525 | GEMIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 2003 |
| Q59961 | GEMIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 2003 |
| P20138 | GEMTUZUMAB OZOGAMICIN | Myeloid cell surface antigen CD33 binding agent | CHEMBL1842 | Myeloid cell surface antigen CD33 | Myeloid cell surface antigen CD33 | Homo sapiens | surface antigen | Antibody | 2000 |
| P20138 | GEMTUZUMAB OZOGAMICIN | DNA inhibitor | CHEMBL2311221 | DNA | Myeloid cell surface antigen CD33 | Homo sapiens | surface antigen | Antibody | 2000 |
| GEMTUZUMAB OZOGAMICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Antibody | 2000 | |||
| GENTAMICIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1970 | ||
| GLATIRAMER ACETATE | Unknown | Small molecule | 1996 | ||||||
| O60706 | GLIMEPIRIDE | "Sulfonylurea receptor 2, Kir6.2" | ATP-binding cassette sub-family C member 9 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1995 | ||
| Q09428 | GLIMEPIRIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1995 |
| Q14654 | GLIMEPIRIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1995 |
| Q09428 | GLIPIZIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1984 |
| Q14654 | GLIPIZIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1984 |
| P47871 | GLUCAGON | Glucagon receptor agonist | CHEMBL1985 | Glucagon receptor | Glucagon receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon receptor | Protein | 1998 |
| P47871 | GLUCAGON HYDROCHLORIDE | Glucagon receptor agonist | CHEMBL1985 | Glucagon receptor | Glucagon receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon receptor | Protein | 1960 |
| P47871 | GLUCAGON HYDROCHLORIDE RECOMBINANT | Glucagon receptor agonist | CHEMBL1985 | Glucagon receptor | Glucagon receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon receptor | Protein | 1998 |
| GLUCARPIDASE | Methotrexate hydrolytic enzyme | CHEMBL2364710 | Methotrexate | Enzyme | 2012 | ||||
| GLUCARPIDASE | CHEMBL2364710 | Methotrexate | Enzyme | 2012 | |||||
| O00591 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| O14764 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P14867 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P18505 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P18507 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P28472 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P31644 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P34903 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P47869 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P47870 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P48169 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| P78334 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| Q16445 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| Q8N1C3 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| Q99928 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| Q9UN88 | GLUTETHIMIDE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1976 |
| Q09428 | GLYBURIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1984 |
| Q14654 | GLYBURIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1984 |
| GLYCEROL PHENYLBUTYRATE | Glutamine chelating agent | CHEMBL2366039 | Glutamine | Homo sapiens | Small molecule | 2013 | |||
| P08172 | GLYCOPYRROLATE | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 | ||
| P08173 | GLYCOPYRROLATE | Muscarinic acetylcholine receptor M4 | Muscarinic acetylcholine receptor M4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 | ||
| P08912 | GLYCOPYRROLATE | Muscarinic acetylcholine receptor M5 | Muscarinic acetylcholine receptor M5 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 | ||
| P11229 | GLYCOPYRROLATE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 |
| P20309 | GLYCOPYRROLATE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1961 |
| P01375 | GOLIMUMAB | TNF-alpha inhibitor | CHEMBL1825 | TNF-alpha | Tumor necrosis factor | Homo sapiens | secreted | Antibody | 2009 |
| P30968 | GONADORELIN | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1982 |
| P22888 | "GONADOTROPIN, CHORIONIC" | Luteinizing hormone/Choriogonadotropin receptor agonist | CHEMBL1854 | Luteinizing hormone/Choriogonadotropin receptor | Lutropin-choriogonadotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Protein | 1973 |
| P30968 | GOSERELIN | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1989 |
| GRAMICIDIN | Cell membrane inhibitor | CHEMBL2364031 | Cell membrane | Bacteria | Small molecule | 1968 | |||
| P46098 | GRANISETRON | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 1993 |
| P0A4L9 | GREPAFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1997 |
| P72524 | GREPAFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1997 |
| P72525 | GREPAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1997 |
| Q59961 | GREPAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1997 |
| F2SZD3 | GRISEOFULVIN | Tubulin inhibitor | CHEMBL2364703 | Tubulin | Tubulin beta chain | Trichophyton | structural | Small molecule | 1962 |
| GUAIFENESIN | Unknown | Small molecule | 2002 | ||||||
| P08913 | GUANABENZ | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P18089 | GUANABENZ | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P18825 | GUANABENZ | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P23975 | GUANADREL | Norepinephrine transporter substrate | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 |
| P23975 | GUANETHIDINE | Norepinephrine transporter substrate | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1960 |
| P08913 | GUANFACINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P18089 | GUANFACINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P18825 | GUANFACINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| O43525 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| O43526 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| O95259 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P16389 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P17658 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 6 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P22001 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P22459 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P22460 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P48547 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P51787 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P56696 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q03721 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q09470 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q12809 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q14003 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q14721 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily B member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q16322 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 10 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q6PIU1 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily V member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q8NCM2 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q8TAE7 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q8TDN1 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q8TDN2 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily V member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q92953 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily B member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q96KK3 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q96L42 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 8 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q96PR1 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily C member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q96RP8 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily A member 7 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9BQ31 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9H252 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 6 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9H3M0 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily F member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9NR82 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily KQT member 5 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9NS40 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 7 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9NSA2 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9NZV8 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9UIX4 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 1 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9UJ96 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily G member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9UK17 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily D member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9ULD8 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 3 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9ULS6 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily S member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| Q9UQ05 | GUANIDINE | Voltage-gated potassium channel blocker | CHEMBL2362996 | Voltage-gated potassium channel | Potassium voltage-gated channel subfamily H member 4 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1939 |
| P14867 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P18507 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P31644 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P34903 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P47869 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q8N1C3 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q99928 | HALAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P04150 | HALCINONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1974 |
| P04150 | HALOBETASOL PROPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1990 |
| HALOFANTRINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 1992 | |||
| P14416 | HALOPERIDOL | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P21917 | HALOPERIDOL | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P28223 | HALOPERIDOL | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1967 |
| P35462 | HALOPERIDOL | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P14416 | HALOPERIDOL DECANOATE | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1986 |
| P21917 | HALOPERIDOL DECANOATE | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1986 |
| P28223 | HALOPERIDOL DECANOATE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1986 |
| P35462 | HALOPERIDOL DECANOATE | D2-like dopamine receptor inverse agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1986 |
| HALOPROGIN | Cell membrane inhibitor | CHEMBL2364033 | Cell membrane | Trichophyton | Small molecule | 1982 | |||
| O00591 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| O14649 | HALOTHANE | Potassium channel subfamily K member 3 opener | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1958 |
| O14764 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| O95069 | HALOTHANE | Potassium channel subfamily K member 2 opener | CHEMBL2321615 | Potassium channel subfamily K member 2 | Potassium channel subfamily K member 2 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1958 |
| P14867 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P18505 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P18507 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P23415 | HALOTHANE | Glycine receptor (alpha-1/beta) positive modulator | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 1958 |
| P28472 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P31644 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P34903 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P47869 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P47870 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P48169 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P57789 | HALOTHANE | Potassium channel subfamily K member 10 opener | CHEMBL2331041 | Potassium channel subfamily K member 10 | Potassium channel subfamily K member 10 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1958 |
| P78334 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| Q16445 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| Q7Z418 | HALOTHANE | Potassium channel subfamily K member 18 opener | CHEMBL2331042 | Potassium channel subfamily K member 18 | Potassium channel subfamily K member 18 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1958 |
| Q8N1C3 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| Q99928 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| Q9NPC2 | HALOTHANE | Potassium channel subfamily K member 9 opener | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1958 |
| Q9UN88 | HALOTHANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1958 |
| P01008 | HEPARIN CALCIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 1982 |
| P01008 | HEPARIN SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 1939 |
| Q54618 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin binding protein 2B | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| Q75Y37 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin-binding protein 3 | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| Q75Y54 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin-binding protein 2X | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| Q75YD8 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin-binding protein 2A | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| Q75YK0 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin-binding protein 1B | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| Q9RET4 | HETACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362973 | Penicillin-binding protein | Penicillin-binding protein 1A | Streptococcus pneumoniae | enzyme protease | Small molecule | 1982 |
| P0AEK4 | HEXACHLOROPHENE | Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor | CHEMBL2364678 | Bacterial enoyl-[acyl-carrier-protein] reductase | Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Bacteria | enzyme reductase | Small molecule | 1949 |
| P22303 | HEXAFLUORENIUM | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1982 |
| P11229 | HEXOCYCLIUM | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P20309 | HEXOCYCLIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P35498 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35499 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q01118 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q14524 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q15858 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q99250 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9NY46 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UI33 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UQD0 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | HEXYLCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35367 | HISTAMINE | Histamine H1 receptor agonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1939 |
| P30968 | HISTRELIN | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1991 |
| HUMAN DNASE-1 | DNA hydrolytic enzyme | CHEMBL2311221 | DNA | Homo sapiens | Enzyme | 1993 | |||
| P23945 | HUMAN FSH | Follicle stimulating hormone receptor agonist | CHEMBL2024 | Follicle stimulating hormone receptor | Follicle-stimulating hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Protein | 1997 |
| P01589 | HUMAN INTERLEUKIN-2 | Interleukin-2 receptor agonist | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit alpha | Homo sapiens | membrane receptor | Protein | 1992 |
| P14784 | HUMAN INTERLEUKIN-2 | Interleukin-2 receptor agonist | CHEMBL2364167 | Interleukin-2 receptor | Interleukin-2 receptor subunit beta | Homo sapiens | membrane receptor | Protein | 1992 |
| P22888 | HUMAN LH | Luteinizing hormone/Choriogonadotropin receptor agonist | CHEMBL1854 | Luteinizing hormone/Choriogonadotropin receptor | Lutropin-choriogonadotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Unknown | 1975 |
| Q92736 | HYDRALAZINE | Ryanodine receptor 2 | Ryanodine receptor 2 | Homo sapiens | ion channel lgic ryr | Small molecule | 1953 | ||
| HYDRALAZINE | Unknown | Small molecule | 1953 | ||||||
| P55017 | HYDROCHLOROTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1959 |
| P35372 | HYDROCODONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1943 |
| P41143 | HYDROCODONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1943 |
| P41145 | HYDROCODONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1943 |
| P04150 | HYDROCORTAMATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1956 |
| P04150 | HYDROCORTISONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1952 |
| P04150 | HYDROCORTISONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1951 |
| P04150 | HYDROCORTISONE BUTYRATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P04150 | HYDROCORTISONE CYPIONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1955 |
| P04150 | HYDROCORTISONE HEMISUCCINATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1955 |
| P04150 | HYDROCORTISONE PHOSPHORIC ACID | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1960 |
| P04150 | HYDROCORTISONE PROBUTATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1997 |
| P04150 | HYDROCORTISONE VALERATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1978 |
| P55017 | HYDROFLUMETHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1959 |
| P35372 | HYDROMORPHONE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P07550 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P08588 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P08913 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P13945 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P18089 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P18825 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P25100 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P35348 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| P35368 | HYDROXYAMPHETAMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1969 |
| Q9NR96 | HYDROXYCHLOROQUINE | Toll-like receptor 9 antagonist | CHEMBL5804 | Toll-like receptor 9 | Toll-like receptor 9 | Homo sapiens | membrane receptor toll-like and il-1 | Small molecule | 1955 |
| Q9NYK1 | HYDROXYCHLOROQUINE | Toll-like receptor 7 antagonist | CHEMBL5936 | Toll-like receptor 7 | Toll-like receptor 7 | Homo sapiens | membrane receptor toll-like and il-1 | Small molecule | 1955 |
| HYDROXYCHLOROQUINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 1955 | |||
| P06401 | HYDROXYPROGESTERONE CAPROATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1975 |
| HYDROXYSTILBAMIDINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1953 | |||
| HYDROXYSTILBAMIDINE | RNA inhibitor | CHEMBL2311222 | RNA | Homo sapiens | Small molecule | 1953 | |||
| P31350 | HYDROXYUREA | Ribonucleoside-diphosphate reductase RR1 inhibitor | CHEMBL2095215 | Ribonucleoside-diphosphate reductase RR1 | Ribonucleoside-diphosphate reductase subunit M2 | Homo sapiens | enzyme | Small molecule | 1967 |
| P35367 | HYDROXYZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1956 |
| P14324 | IBANDRONIC ACID | Farnesyl diphosphate synthase inhibitor | CHEMBL1782 | Farnesyl diphosphate synthase | Farnesyl pyrophosphate synthase | Homo sapiens | enzyme transferase | Small molecule | 2003 |
| Q06187 | IBRUTINIB | Tyrosine-protein kinase BTK inhibitor | CHEMBL5251 | Tyrosine-protein kinase BTK | Tyrosine-protein kinase BTK | Homo sapiens | enzyme kinase protein kinase tk tec | Small molecule | 2013 |
| P23219 | IBUPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1974 |
| P35354 | IBUPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1974 |
| Q12809 | IBUTILIDE | HERG blocker | CHEMBL240 | HERG | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1995 |
| P30411 | ICATIBANT | Bradykinin B2 receptor antagonist | CHEMBL3157 | Bradykinin B2 receptor | B2 bradykinin receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide bradykinin receptor | Protein | 2011 |
| O75907 | ICOSAPENT ETHYL | Diacylglycerol O-acyltransferase 1 | Diacylglycerol O-acyltransferase 1 | Homo sapiens | enzyme | Small molecule | 2012 | ||
| ICOSAPENT ETHYL | Unknown | Small molecule | 2012 | ||||||
| P11388 | IDARUBICIN | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1990 |
| P11388 | IDARUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1990 |
| IDARUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1990 | |||
| O00329 | IDELALISIB | PI3-kinase p110-delta subunit inhibitor | CHEMBL3130 | PI3-kinase p110-delta subunit | "Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform" | Homo sapiens | enzyme | Small molecule | 2014 |
| IDOXURIDINE | DNA inhibitor | CHEMBL2366042 | DNA | Human herpesvirus 1 | Small molecule | 1963 | |||
| IDURSULFASE | Heparan sulfate hydrolytic enzyme | CHEMBL2364677 | Heparan sulfate | Homo sapiens | Enzyme | 2006 | |||
| IFOSFAMIDE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1988 | |||
| P14416 | ILOPERIDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2009 |
| P28223 | ILOPERIDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2009 |
| P43119 | ILOPROST | Prostanoid IP receptor agonist | CHEMBL1995 | Prostanoid IP receptor | Prostacyclin receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 2004 |
| P00519 | IMATINIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2001 |
| P09619 | IMATINIB | Platelet-derived growth factor receptor beta inhibitor | CHEMBL1913 | Platelet-derived growth factor receptor beta | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2001 |
| P10721 | IMATINIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2001 |
| IMIGLUCERASE | Glucocerebroside hydrolytic enzyme | CHEMBL2364176 | Glucocerebroside | Homo sapiens | Enzyme | 1994 | |||
| P02918 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P02919 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1985 |
| P08506 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P0AD65 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1985 |
| P0AD68 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1985 |
| P0AEB2 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1985 |
| P24228 | IMIPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1985 |
| P23975 | IMIPRAMINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1959 |
| P31645 | IMIPRAMINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1959 |
| Q9NYK1 | IMIQUIMOD | Toll-like receptor 7 agonist | CHEMBL5936 | Toll-like receptor 7 | Toll-like receptor 7 | Homo sapiens | membrane receptor toll-like and il-1 | Small molecule | 1997 |
| Q14432 | INAMRINONE | Phosphodiesterase 3A inhibitor | CHEMBL241 | Phosphodiesterase 3A | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1984 |
| P60880 | INCOBOTULINUMTOXINA | Synaptosomal-associated protein 25 inhibitor | CHEMBL2364159 | Synaptosomal-associated protein 25 | Synaptosomal-associated protein 25 | Homo sapiens | cytosolic other | Unknown | 2010 |
| P07550 | INDACATEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2011 |
| P55017 | INDAPAMIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1983 |
| P35498 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| P35499 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q01118 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q14524 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q15858 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q99250 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9NY46 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9UI33 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9UQD0 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9Y5Y9 | INDECAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q72874 | INDINAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 1996 |
| P23219 | INDOMETHACIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1965 |
| P35354 | INDOMETHACIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1965 |
| P01375 | INFLIXIMAB | TNF-alpha inhibitor | CHEMBL1825 | TNF-alpha | Tumor necrosis factor | Homo sapiens | secreted | Antibody | 1998 |
| INGENOL MEBUTATE | Unknown | Small molecule | 2010 | ||||||
| P06213 | INSULIN ASPART | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2000 |
| P06213 | INSULIN ASPART PROTAMINE RECOMBINANT | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2001 |
| P06213 | INSULIN DETEMIR | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2005 |
| P06213 | INSULIN GLARGINE | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2000 |
| P06213 | INSULIN GLULISINE | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2004 |
| P06213 | INSULIN HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN LISPRO | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1996 |
| P06213 | INSULIN LISPRO PROTAMINE RECOMBINANT | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1999 |
| P06213 | INSULIN PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1966 |
| P06213 | INSULIN PURIFIED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1980 |
| P06213 | INSULIN PURIFIED PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1979 |
| P06213 | INSULIN SUSP ISOPHANE BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN SUSP ISOPHANE BEEF/PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1966 |
| P06213 | INSULIN SUSP ISOPHANE PURIFIED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1980 |
| P06213 | INSULIN SUSP ISOPHANE PURIFIED PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1979 |
| P06213 | INSULIN SUSP ISOPHANE RECOMBINANT HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN SUSP ISOPHANE SEMISYNTHETIC PURIFIED HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1985 |
| P06213 | INSULIN SUSP PROTAMINE ZINC BEEF/PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1966 |
| P06213 | INSULIN SUSP PROTAMINE ZINC PURIFIED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1980 |
| P06213 | INSULIN SUSP PROTAMINE ZINC PURIFIED PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1979 |
| P06213 | INSULIN ZINC SUSP BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP EXTENDED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP EXTENDED PURIFIED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP EXTENDED RECOMBINANT HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1987 |
| P06213 | INSULIN ZINC SUSP PROMPT BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP PROMPT PURIFIED PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP PURIFIED BEEF | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1980 |
| P06213 | INSULIN ZINC SUSP PURIFIED BEEF/PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1982 |
| P06213 | INSULIN ZINC SUSP PURIFIED PORK | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1979 |
| P06213 | INSULIN ZINC SUSP RECOMBINANT HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1985 |
| P06213 | INSULIN ZINC SUSP SEMISYNTHETIC PURIFIED HUMAN | Insulin receptor agonist | CHEMBL1981 | Insulin receptor | Insulin receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 1983 |
| P17181 | INTERFERON ALFA-2A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1986 |
| P48551 | INTERFERON ALFA-2A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1986 |
| P17181 | INTERFERON ALFA-2B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1986 |
| P48551 | INTERFERON ALFA-2B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1986 |
| P17181 | INTERFERON ALFA-N3 | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1989 |
| P48551 | INTERFERON ALFA-N3 | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1989 |
| P17181 | INTERFERON ALFACON-1 | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1997 |
| P48551 | INTERFERON ALFACON-1 | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1997 |
| P17181 | INTERFERON BETA-1A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1996 |
| P48551 | INTERFERON BETA-1A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1996 |
| P17181 | INTERFERON BETA-1B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 1993 |
| P48551 | INTERFERON BETA-1B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 1993 |
| P15260 | INTERFERON GAMA-1B | Interferon gamma receptor agonist | CHEMBL2364171 | Interferon gamma receptor | Interferon gamma receptor 1 | Homo sapiens | membrane receptor | Protein | 1999 |
| P38484 | INTERFERON GAMA-1B | Interferon gamma receptor agonist | CHEMBL2364171 | Interferon gamma receptor | Interferon gamma receptor 2 | Homo sapiens | membrane receptor | Protein | 1999 |
| P16410 | IPILIMUMAB | Cytotoxic T-lymphocyte protein 4 inhibitor | CHEMBL2364164 | Cytotoxic T-lymphocyte protein 4 | Cytotoxic T-lymphocyte protein 4 | Homo sapiens | surface antigen | Antibody | 2011 |
| P20309 | IPRATROPIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1986 |
| P30556 | IRBESARTAN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1997 |
| P11387 | IRINOTECAN | DNA topoisomerase I inhibitor | CHEMBL1781 | DNA topoisomerase I | DNA topoisomerase 1 | Homo sapiens | enzyme isomerase | Small molecule | 1996 |
| Q969P6 | IRINOTECAN | "DNA topoisomerase I, mitochondrial" | "DNA topoisomerase I, mitochondrial" | Homo sapiens | enzyme isomerase | Small molecule | 1996 | ||
| A0A0A1P6P0 | ISAVUCONAZONIUM | Lanosterol 14-alpha demethylase inhibitor | CHEMBL3390825 | Lanosterol 14-alpha demethylase | Mucorales | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2015 | |
| A0A0D9MXW1 | ISAVUCONAZONIUM | Lanosterol 14-alpha demethylase inhibitor | CHEMBL3390824 | Lanosterol 14-alpha demethylase | Aspergillus | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2015 | |
| G4WW85 | ISAVUCONAZONIUM | Lanosterol 14-alpha demethylase inhibitor | CHEMBL3390824 | Lanosterol 14-alpha demethylase | Aspergillus | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2015 | |
| Q9P8R0 | ISAVUCONAZONIUM | Lanosterol 14-alpha demethylase inhibitor | CHEMBL3390824 | Lanosterol 14-alpha demethylase | Aspergillus | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2015 | |
| P21397 | ISOCARBOXAZID | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] A | Homo sapiens | enzyme reductase | Small molecule | 1959 |
| P27338 | ISOCARBOXAZID | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 1959 |
| P07550 | ISOETHARINE | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| O00591 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| O14649 | ISOFLURANE | Potassium channel subfamily K member 3 opener | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1979 |
| O14764 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| O95069 | ISOFLURANE | Potassium channel subfamily K member 2 opener | CHEMBL2321615 | Potassium channel subfamily K member 2 | Potassium channel subfamily K member 2 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1979 |
| P14867 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P18505 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P18507 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P23415 | ISOFLURANE | Glycine receptor (alpha-1/beta) positive modulator | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 1979 |
| P28472 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P31644 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P34903 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P47869 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P47870 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P48169 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P57789 | ISOFLURANE | Potassium channel subfamily K member 10 opener | CHEMBL2331041 | Potassium channel subfamily K member 10 | Potassium channel subfamily K member 10 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1979 |
| P78334 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| Q16445 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| Q7Z418 | ISOFLURANE | Potassium channel subfamily K member 18 opener | CHEMBL2331042 | Potassium channel subfamily K member 18 | Potassium channel subfamily K member 18 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1979 |
| Q8N1C3 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| Q99928 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| Q9NPC2 | ISOFLURANE | Potassium channel subfamily K member 9 opener | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1979 |
| Q9UN88 | ISOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1979 |
| P22303 | ISOFLUROPHATE | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1957 |
| P9WGR1 | ISONIAZID | Enoyl-[acyl-carrier-protein] reductase inhibitor | CHEMBL1849 | Enoyl-[acyl-carrier-protein] reductase | Enoyl-[acyl-carrier-protein] reductase [NADH] | Mycobacterium tuberculosis | enzyme reductase | Small molecule | 1952 |
| P11229 | ISOPROPAMIDE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1957 |
| P20309 | ISOPROPAMIDE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1957 |
| P07550 | ISOPROTERENOL | Adrenergic receptor beta agonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1956 |
| P08588 | ISOPROTERENOL | Adrenergic receptor beta agonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1956 |
| P13945 | ISOPROTERENOL | Adrenergic receptor beta agonist | CHEMBL2094118 | Adrenergic receptor beta | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1956 |
| ISOSORBIDE | Unknown | Small molecule | 1974 | ||||||
| O75343 | ISOSORBIDE DINITRATE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1986 |
| Q02153 | ISOSORBIDE DINITRATE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1986 |
| O75343 | ISOSORBIDE MONONITRATE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1991 |
| Q02153 | ISOSORBIDE MONONITRATE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1991 |
| P10276 | ISOTRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1982 |
| P10826 | ISOTRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1982 |
| P13631 | ISOTRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1982 |
| O60840 | ISRADIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q01668 | ISRADIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q13698 | ISRADIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| Q13936 | ISRADIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1990 |
| P10613 | ITRACONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1992 |
| O60741 | IVABRADINE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2015 | ||
| Q9P1Z3 | IVABRADINE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 3 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2015 | ||
| Q9UL51 | IVABRADINE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 2 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2015 | ||
| Q9Y3Q4 | IVABRADINE | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 blocker | CHEMBL1250417 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 | Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 | Homo sapiens | ion channel vgc c-gmp | Small molecule | 2015 |
| P13569 | IVACAFTOR | Cystic fibrosis transmembrane conductance regulator positive modulator | CHEMBL4051 | Cystic fibrosis transmembrane conductance regulator | Cystic fibrosis transmembrane conductance regulator | Homo sapiens | ion channel other chloride cftr | Small molecule | 2012 |
| P91730 | IVERMECTIN | Glutamate-gated chloride channel modulator | CHEMBL2363050 | Glutamate-gated chloride channel | Glutamate-gated chloride channel subunit beta | Strongyloides stercoralis | ion channel lgic | Unknown | 1996 |
| Q25634 | IVERMECTIN | Glutamate-gated chloride channel modulator | CHEMBL2363051 | Glutamate-gated chloride channel | Glutamate-gated chloride channel | Onchocerca volvulus | ion channel lgic | Unknown | 1996 |
| P04350 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 2007 |
| P07437 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 2007 |
| P68371 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 2007 |
| Q13509 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 2007 |
| Q13885 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 2007 |
| Q3ZCM7 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 2007 |
| Q9BUF5 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 2007 |
| Q9BVA1 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 2007 |
| Q9H4B7 | IXABEPILONE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 2007 |
| KANAMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1973 | ||
| O15399 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| O60391 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| Q05586 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| Q12879 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| Q13224 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| Q14957 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| Q8TCU5 | KETAMINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1970 |
| P05093 | KETOCONAZOLE | "Steroid 17-alpha-hydroxylase/17,20 lyase" | "Steroid 17-alpha-hydroxylase/17,20 lyase" | Homo sapiens | enzyme cytochrome p450 cyp_17 cyp_17a cyp_17a1 | Small molecule | 1981 | ||
| P10613 | KETOCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1981 |
| P15538 | KETOCONAZOLE | "Cytochrome P450 11B1, mitochondrial" | "Cytochrome P450 11B1, mitochondrial" | Homo sapiens | enzyme cytochrome p450 cyp_11 cyp_11b cyp_11b1 | Small molecule | 1981 | ||
| P23219 | KETOPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1986 |
| P35354 | KETOPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1986 |
| P23219 | KETOROLAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1989 |
| P35354 | KETOROLAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1989 |
| P35367 | KETOTIFEN | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1999 |
| P07550 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P08588 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P08913 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P13945 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P18089 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P18825 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P25100 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P35348 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| P35368 | LABETALOL | Adrenergic receptor antagonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1984 |
| LACTIC ACID | pH lowering agent | Small molecule | 2006 | ||||||
| LACTITOL | Colonic bacteria substrate | Small molecule | 1976 | ||||||
| Q72547 | LAMIVUDINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1995 |
| Q9IF40 | LAMIVUDINE | DNA polymerase/reverse transcriptase inhibitor | CHEMBL2362994 | DNA polymerase/reverse transcriptase | Protein P | Hepatitis B virus | enzyme transferase | Small molecule | 1995 |
| LAMIVUDINE | DNA inhibitor | CHEMBL2363046 | DNA | Human immunodeficiency virus 1 | Small molecule | 1995 | |||
| LAMIVUDINE | DNA inhibitor | CHEMBL2363047 | DNA | Human immunodeficiency virus 2 | Small molecule | 1995 | |||
| LAMIVUDINE | DNA inhibitor | CHEMBL2363048 | DNA | Hepatitis B virus | Small molecule | 1995 | |||
| P35498 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| P35499 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q01118 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q14524 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q15858 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q99250 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q9NY46 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q9UI33 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q9UQD0 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| Q9Y5Y9 | LAMOTRIGINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1994 |
| P30874 | LANREOTIDE | Somatostatin receptor 2 agonist | CHEMBL1804 | Somatostatin receptor 2 | Somatostatin receptor type 2 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2007 |
| P35346 | LANREOTIDE | Somatostatin receptor 5 agonist | CHEMBL1792 | Somatostatin receptor 5 | Somatostatin receptor type 5 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2007 |
| P20648 | LANSOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 1995 |
| P20648 | LANSOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 1995 |
| LANTHANUM CARBONATE | Phosphate chelating agent | CHEMBL2364184 | Phosphate | Homo sapiens | Small molecule | 2004 | |||
| P00533 | LAPATINIB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2007 |
| P04626 | LAPATINIB | Receptor protein-tyrosine kinase erbB-2 inhibitor | CHEMBL1824 | Receptor protein-tyrosine kinase erbB-2 | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2007 |
| LAPYRIUM | Unknown | Small molecule | 1982 | ||||||
| LARONIDASE | Dermatan sulfate hydrolytic enzyme | CHEMBL2364179 | Dermatan sulfate | Homo sapiens | Enzyme | 2003 | |||
| LARONIDASE | Heparan sulfate hydrolytic enzyme | CHEMBL2364677 | Heparan sulfate | Homo sapiens | Enzyme | 2003 | |||
| P43088 | LATANOPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1996 |
| Q5L478 | LEDIPASVIR | Nonstructural protein 5A inhibitor | CHEMBL3307224 | Nonstructural protein 5A | Nonstructural protein 5A | Hepatitis C virus | unclassified | Small molecule | 2014 |
| Q8JXU8 | LEDIPASVIR | Hepatitis C virus NS5B RNA-dependent RNA polymerase | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 2014 | ||
| Q02127 | LEFLUNOMIDE | Dihydroorotate dehydrogenase inhibitor | CHEMBL1966 | Dihydroorotate dehydrogenase | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1998 |
| Q96SW2 | LENALIDOMIDE | Protein cereblon | Protein cereblon | Homo sapiens | Unclassified | Small molecule | 2005 | ||
| LENALIDOMIDE | Unknown | Small molecule | 2005 | ||||||
| P07949 | LENVATINIB | Proto-oncogene tyrosine-protein kinase receptor Ret | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2015 | ||
| P10721 | LENVATINIB | Mast/stem cell growth factor receptor Kit | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2015 | ||
| P11362 | LENVATINIB | Fibroblast growth factor receptor 1 | Fibroblast growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2015 | ||
| P16234 | LENVATINIB | Platelet-derived growth factor receptor alpha | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2015 | ||
| P17948 | LENVATINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2015 |
| P35916 | LENVATINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2015 |
| P35968 | LENVATINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2015 |
| P00734 | LEPIRUDIN | Thrombin inhibitor | CHEMBL204 | Thrombin | Prothrombin | Homo sapiens | enzyme protease serine pas s1a | Protein | 1998 |
| P11511 | LETROZOLE | Cytochrome P450 19A1 inhibitor | CHEMBL1978 | Cytochrome P450 19A1 | Aromatase | Homo sapiens | enzyme cytochrome p450 cyp_19 cyp_19a cyp_19a1 | Small molecule | 1997 |
| P30968 | LEUPROLIDE | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1985 |
| P35372 | LEVALLORPHAN | Mu opioid receptor antagonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1982 |
| P41145 | LEVALLORPHAN | Kappa opioid receptor partial agonist | CHEMBL237 | Kappa opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1982 |
| O96760 | LEVAMISOLE | Nicotinic acetylcholine receptor alpha subunit agonist | CHEMBL1884 | Nicotinic acetylcholine receptor alpha subunit | Nicotinic acetylcholine receptor alpha subunit | Ascaris suum | ion channel lgic ach chrn alpha | Small molecule | 1990 |
| Q00975 | LEVETIRACETAM | Voltage-gated N-type calcium channel alpha-1B subunit blocker | CHEMBL4478 | Voltage-gated N-type calcium channel alpha-1B subunit | Voltage-dependent N-type calcium channel subunit alpha-1B | Homo sapiens | ion channel vgc vg ca | Small molecule | 1999 |
| Q7L0J3 | LEVETIRACETAM | Synaptic vesicle glycoprotein 2A modulator | CHEMBL1998 | Synaptic vesicle glycoprotein 2A | Synaptic vesicle glycoprotein 2A | Homo sapiens | transporter electrochemical vnt | Small molecule | 1999 |
| P08588 | LEVOBETAXOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2000 |
| P07550 | LEVOBUNOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P08588 | LEVOBUNOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P13945 | LEVOBUNOLOL | Beta-3 adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 | ||
| P35499 | LEVOBUPIVACAINE | Sodium channel protein type IV alpha subunit blocker | CHEMBL2072 | Sodium channel protein type IV alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1999 |
| P35367 | LEVOCABASTINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1993 |
| P08183 | LEVOCETIRIZINE | Multidrug resistance protein 1 | Multidrug resistance protein 1 | Homo sapiens | transporter ntpase atp binding cassette mdr | Small molecule | 2007 | ||
| P35367 | LEVOCETIRIZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 2007 |
| P35462 | LEVODOPA | Dopamine D3 receptor agonist | CHEMBL234 | Dopamine D3 receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1970 |
| P0A4L9 | LEVOFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1996 |
| P43700 | LEVOFLOXACIN | DNA gyrase subunit A | DNA gyrase subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1996 | ||
| P43702 | LEVOFLOXACIN | DNA topoisomerase 4 subunit A | DNA topoisomerase 4 subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1996 | ||
| P72524 | LEVOFLOXACIN | DNA gyrase inhibitor | CHEMBL2311225 | DNA gyrase | DNA gyrase subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1996 |
| P72525 | LEVOFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1996 |
| Q59961 | LEVOFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363033 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Streptococcus pneumoniae | enzyme isomerase | Small molecule | 1996 |
| LEVOLEUCOVORIN | Unknown | Small molecule | 2008 | ||||||
| LEVOMEFOLIC ACID | Unknown | Small molecule | 2010 | ||||||
| P14416 | LEVOMEPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1982 |
| P21917 | LEVOMEPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1982 |
| P35462 | LEVOMEPROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1982 |
| P35372 | LEVOMETHADYL ACETATE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1993 |
| P23975 | LEVOMILNACIPRAN | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2013 |
| P31645 | LEVOMILNACIPRAN | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2013 |
| P08913 | LEVONORDEFRIN | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1960 |
| P18089 | LEVONORDEFRIN | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1960 |
| P18825 | LEVONORDEFRIN | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1960 |
| P06401 | LEVONORGESTREL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1982 |
| LEVOPROPOXYPHENE | Unknown | Small molecule | 1962 | ||||||
| P35372 | LEVORPHANOL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1991 |
| P07550 | LEVOSALBUTAMOL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1999 |
| P10827 | LEVOTHYROXINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a1 | Small molecule | 2000 |
| P10828 | LEVOTHYROXINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a2 | Small molecule | 2000 |
| P35498 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| P35499 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q01118 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q14524 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q15858 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q99250 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q9NY46 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q9UI33 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q9UQD0 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| Q9Y5Y9 | LIDOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1948 |
| P25092 | LINACLOTIDE | Heat-stable enterotoxin receptor agonist | CHEMBL1795197 | Heat-stable enterotoxin receptor | Heat-stable enterotoxin receptor | Homo sapiens | enzyme lyase guanylate cyclase receptor guanylate cyclase | Protein | 2012 |
| P27487 | LINAGLIPTIN | Dipeptidyl peptidase IV inhibitor | CHEMBL284 | Dipeptidyl peptidase IV | Dipeptidyl peptidase 4 | Homo sapiens | enzyme protease serine sc s9b | Small molecule | 2011 |
| LINCOMYCIN | 70S ribosome inhibitor | CHEMBL2363853 | 70S ribosome | 23S ribosomal RNA | Streptococcus pneumoniae | Small molecule | 1964 | ||
| E0V9W2 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364025 | GABA-A receptor | "Gaba-gated chloride channel, putative" | Pediculus humanus | ion channel lgic | Small molecule | 1974 |
| E0VY07 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364025 | GABA-A receptor | "Gaba-gated chloride channel, putative" | Pediculus humanus | ion channel lgic | Small molecule | 1974 |
| E0W492 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364025 | GABA-A receptor | "Gaba-gated chloride channel, putative" | Pediculus humanus | ion channel lgic | Small molecule | 1974 |
| H9U2V9 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364024 | GABA-A receptor | GABA-gated chloride channel 1 | Sarcoptes scabiei | ion channel lgic | Small molecule | 1974 |
| H9U2W0 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364024 | GABA-A receptor | GABA-gated chloride channel 2 | Sarcoptes scabiei | ion channel lgic | Small molecule | 1974 |
| H9U2W1 | LINDANE | GABA-A receptor negative allosteric modulator | CHEMBL2364024 | GABA-A receptor | GABA-gated chloride channel 3 | Sarcoptes scabiei | ion channel lgic | Small molecule | 1974 |
| LINEZOLID | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 2000 | ||
| P10827 | LIOTHYRONINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a1 | Small molecule | 1956 |
| P10828 | LIOTHYRONINE | Thyroid hormone receptor agonist | CHEMBL2111462 | Thyroid hormone receptor | Thyroid hormone receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1a nr1a2 | Small molecule | 1956 |
| LIPASE | Fatty acids hydrolytic enzyme | CHEMBL2364711 | Fatty acids | Homo sapiens | Enzyme | 1996 | |||
| P43220 | LIRAGLUTIDE | Glucagon-like peptide 1 receptor agonist | CHEMBL1784 | Glucagon-like peptide 1 receptor | Glucagon-like peptide 1 receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon-like peptide receptor | Protein | 2010 |
| P23975 | LISDEXAMFETAMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2007 |
| Q01959 | LISDEXAMFETAMINE | Dopamine transporter releasing agent | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2007 |
| Q05940 | LISDEXAMFETAMINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 2007 |
| P12821 | LISINOPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1987 |
| P29218 | LITHIUM CARBONATE | Inositol-1(or 4)-monophosphatase 1 inhibitor | CHEMBL1786 | Inositol-1(or 4)-monophosphatase 1 | Inositol monophosphatase 1 | Homo sapiens | enzyme hydrolase | Small molecule | 1970 |
| P49840 | LITHIUM CARBONATE | Glycogen synthase kinase-3 inhibitor | CHEMBL2095188 | Glycogen synthase kinase-3 | Glycogen synthase kinase-3 alpha | Homo sapiens | enzyme kinase protein kinase cmgc gsk | Small molecule | 1970 |
| P49841 | LITHIUM CARBONATE | Glycogen synthase kinase-3 inhibitor | CHEMBL2095188 | Glycogen synthase kinase-3 | Glycogen synthase kinase-3 beta | Homo sapiens | enzyme kinase protein kinase cmgc gsk | Small molecule | 1970 |
| P29218 | LITHIUM CITRATE | Inositol-1(or 4)-monophosphatase 1 inhibitor | CHEMBL1786 | Inositol-1(or 4)-monophosphatase 1 | Inositol monophosphatase 1 | Homo sapiens | enzyme hydrolase | Small molecule | 1980 |
| P49840 | LITHIUM CITRATE | Glycogen synthase kinase-3 inhibitor | CHEMBL2095188 | Glycogen synthase kinase-3 | Glycogen synthase kinase-3 alpha | Homo sapiens | enzyme kinase protein kinase cmgc gsk | Small molecule | 1980 |
| P49841 | LITHIUM CITRATE | Glycogen synthase kinase-3 inhibitor | CHEMBL2095188 | Glycogen synthase kinase-3 | Glycogen synthase kinase-3 beta | Homo sapiens | enzyme kinase protein kinase cmgc gsk | Small molecule | 1980 |
| LODOXAMIDE | Unknown | Small molecule | 1993 | ||||||
| P0AES4 | LOMEFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1992 |
| P0AES6 | LOMEFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1992 |
| P55157 | LOMITAPIDE | Microsomal triglyceride transfer protein inhibitor | CHEMBL2364681 | Microsomal triglyceride transfer protein | Microsomal triglyceride transfer protein large subunit | Homo sapiens | cytosolic other | Small molecule | 2012 |
| LOMUSTINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1976 | |||
| P35372 | LOPERAMIDE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1976 |
| Q72874 | LOPINAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 2000 |
| P02918 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1991 |
| P02919 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1991 |
| P08506 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1991 |
| P0AD65 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1991 |
| P0AD68 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1991 |
| P0AEB2 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1991 |
| P24228 | LORACARBEF | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1991 |
| P35367 | LORATADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1993 |
| P14867 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| P18507 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| P31644 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| P34903 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| P47869 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| Q8N1C3 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| Q99928 | LORAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1977 |
| P28335 | LORCASERIN | Serotonin 2c (5-HT2c) receptor agonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2012 |
| P30556 | LOSARTAN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1995 |
| P04150 | LOTEPREDNOL ETABONATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1998 |
| P04035 | LOVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1987 |
| P14416 | LOXAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1975 |
| P21917 | LOXAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1975 |
| P28223 | LOXAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1975 |
| P28335 | LOXAPINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1975 |
| P35462 | LOXAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1975 |
| P51788 | LUBIPROSTONE | Chloride channel protein 2 opener | CHEMBL1628478 | Chloride channel protein 2 | Chloride channel protein 2 | Homo sapiens | ion channel other chloride clc | Small molecule | 2006 |
| LUCINACTANT | Surfactant agent | Unknown | 2012 | ||||||
| P10613 | LULICONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2013 |
| P13569 | LUMACAFTOR | Cystic fibrosis transmembrane conductance regulator stabiliser | CHEMBL4051 | Cystic fibrosis transmembrane conductance regulator | Cystic fibrosis transmembrane conductance regulator | Homo sapiens | ion channel other chloride cftr | Small molecule | 2015 |
| LUMEFANTRINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 2009 | |||
| P14416 | LURASIDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2010 |
| P28223 | LURASIDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2010 |
| P34969 | LURASIDONE | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2010 | ||
| P22888 | LUTROPIN ALFA | Luteinizing hormone/Choriogonadotropin receptor agonist | CHEMBL1854 | Luteinizing hormone/Choriogonadotropin receptor | Lutropin-choriogonadotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Protein | 2004 |
| P30518 | LYPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P37288 | LYPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1a receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P47901 | LYPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1b receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P24530 | MACITENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin B receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2010 |
| P25101 | MACITENTAN | "Endothelin receptor, ET-A/ET-B antagonist" | CHEMBL2096678 | "Endothelin receptor, ET-A/ET-B" | Endothelin-1 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide endothelin receptor | Small molecule | 2010 |
| P0AC13 | MAFENIDE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1969 |
| MAGNESIUM SULFATE ANHYDROUS | Unknown | Small molecule | 1981 | ||||||
| A2PZ98 | MALATHION | Acetylcholinesterase inhibitor | CHEMBL2362988 | Acetylcholinesterase | Acetylcholinesterase | Pediculus humanus capitis | enzyme hydrolase | Small molecule | 1982 |
| P23975 | MAPROTILINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1980 |
| P51681 | MARAVIROC | C-C chemokine receptor type 5 antagonist | CHEMBL274 | C-C chemokine receptor type 5 | C-C chemokine receptor type 5 | Homo sapiens | membrane receptor 7tm1 peptide chemokine receptor cc chemokine receptor | Small molecule | 2007 |
| P23975 | MAZINDOL | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1973 |
| P31645 | MAZINDOL | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1973 |
| Q01959 | MAZINDOL | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1973 |
| C4PKY4 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 1 | Taeniidae | structural | Small molecule | 1974 |
| C4PKZ2 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 2 | Taeniidae | structural | Small molecule | 1974 |
| C4PKZ6 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 3 | Taeniidae | structural | Small molecule | 1974 |
| F1L4P8 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-1 chain | Nematoda | structural | Small molecule | 1974 |
| F1L7U3 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-2 chain | Nematoda | structural | Small molecule | 1974 |
| F1L8A5 | MEBENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-4 chain | Nematoda | structural | Small molecule | 1974 |
| MEBUTAMATE | Unknown | Small molecule | 1982 | ||||||
| P30926 | MECAMYLAMINE | Neuronal acetylcholine receptor; alpha3/beta4 negative allosteric modulator | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1956 |
| P32297 | MECAMYLAMINE | Neuronal acetylcholine receptor; alpha3/beta4 negative allosteric modulator | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1956 |
| P08069 | MECASERMIN | Insulin-like growth factor I receptor agonist | CHEMBL1957 | Insulin-like growth factor I receptor | Insulin-like growth factor 1 receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2005 |
| P08069 | MECASERMIN RINFABATE | Insulin-like growth factor I receptor agonist | CHEMBL1957 | Insulin-like growth factor I receptor | Insulin-like growth factor 1 receptor | Homo sapiens | enzyme kinase protein kinase tk insr | Protein | 2005 |
| MECHLORETHAMINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1949 | |||
| P35367 | MECLIZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1957 |
| MECLOCYCLINE SULFOSALICYLATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1982 | ||
| P09917 | MECLOFENAMIC ACID | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 1980 |
| P23219 | MECLOFENAMIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1980 |
| P35354 | MECLOFENAMIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1980 |
| P06401 | MEDROXYPROGESTERONE ACETATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1959 |
| P04150 | MEDRYSONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1969 |
| P23219 | MEFENAMIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1967 |
| P35354 | MEFENAMIC ACID | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1967 |
| MEFLOQUINE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 1989 | |||
| P06401 | MEGESTROL ACETATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1971 |
| P35354 | MELOXICAM | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 2000 |
| MELPHALAN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1964 | |||
| O15399 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| O60391 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| Q05586 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| Q12879 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| Q13224 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| Q14957 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| Q8TCU5 | MEMANTINE | Glutamate [NMDA] receptor negative allosteric modulator | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 2003 |
| P22888 | MENOTROPINS | Luteinizing hormone/Choriogonadotropin receptor agonist | CHEMBL1854 | Luteinizing hormone/Choriogonadotropin receptor | Lutropin-choriogonadotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Unknown | 1975 |
| P23945 | MENOTROPINS | Follicle stimulating hormone receptor agonist | CHEMBL2024 | Follicle stimulating hormone receptor | Follicle-stimulating hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Unknown | 1975 |
| O75762 | MENTHOL | Transient receptor potential cation channel subfamily A member 1 opener | CHEMBL6007 | Transient receptor potential cation channel subfamily A member 1 | Transient receptor potential cation channel subfamily A member 1 | Homo sapiens | ion channel vgc trp | Small molecule | 2008 |
| Q7Z2W7 | MENTHOL | Transient receptor potential cation channel subfamily M member 8 opener | CHEMBL1075319 | Transient receptor potential cation channel subfamily M member 8 | Transient receptor potential cation channel subfamily M member 8 | Homo sapiens | ion channel vgc trp | Small molecule | 2008 |
| P11229 | MEPENZOLATE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1956 |
| P20309 | MEPENZOLATE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1956 |
| P35372 | MEPERIDINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1942 |
| P07550 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P08588 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P08913 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P13945 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P18089 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P18825 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P25100 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P35348 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P35368 | MEPHENTERMINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1951 |
| P35498 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| P35499 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q01118 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q14524 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q15858 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q99250 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q9NY46 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q9UI33 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q9UQD0 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| Q9Y5Y9 | MEPHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1946 |
| P35498 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| P35499 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q01118 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q14524 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q15858 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q99250 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q9NY46 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q9UI33 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q9UQD0 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| Q9Y5Y9 | MEPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1960 |
| P04150 | MEPREDNISONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| P14867 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P18505 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P28472 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P31644 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P34903 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P47869 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P47870 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P48169 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| Q16445 | MEPROBAMATE | GABA-A receptor; anion channel agonist | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1955 |
| P14679 | MEQUINOL | Tyrosinase inhibitor | CHEMBL1973 | Tyrosinase | Tyrosinase | Homo sapiens | enzyme reductase | Small molecule | 1999 |
| Q06203 | MERCAPTOPURINE | DNA inhibitor | CHEMBL2311221 | DNA | Amidophosphoribosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1953 |
| Q06203 | MERCAPTOPURINE | Amidophosphoribosyltransferase inhibitor | CHEMBL2362992 | Amidophosphoribosyltransferase | Amidophosphoribosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1953 |
| MERCAPTOPURINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1953 | |||
| P35498 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| P35499 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q01118 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q14524 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q15858 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q99250 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q9NY46 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q9UI33 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q9UQD0 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| Q9Y5Y9 | MERETHOXYLLINE PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 0 |
| P02918 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1996 |
| P02919 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1996 |
| P08506 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1996 |
| P0AD65 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1996 |
| P0AD68 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1996 |
| P0AEB2 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1996 |
| P24228 | MEROPENEM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1996 |
| P09917 | MESALAMINE | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 1987 |
| P23219 | MESALAMINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1987 |
| P35354 | MESALAMINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1987 |
| P37231 | MESALAMINE | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 1987 |
| P14416 | MESORIDAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1970 |
| P28223 | MESORIDAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1970 |
| P03372 | MESTRANOL | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1961 |
| P07550 | METAPROTERENOL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1973 |
| P25100 | METARAMINOL | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1954 |
| P35348 | METARAMINOL | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1954 |
| P35368 | METARAMINOL | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1954 |
| METAXALONE | Unknown | Small molecule | 1962 | ||||||
| O00217 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 8, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O00483 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | Cytochrome c oxidase subunit NDUFA4 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O14561 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "Acyl carrier protein, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O15239 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43181 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 4, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43674 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 5, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43676 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 3 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43677 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 subunit C1, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43678 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 2 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O43920 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] iron-sulfur protein 5 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O75251 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 7, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O75306 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 2, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O75380 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 6, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O75438 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O75489 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] iron-sulfur protein 3, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95139 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 6 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95167 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 3 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95168 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 4 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95169 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 8, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95178 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 2, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95182 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 7 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95298 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 subunit C2 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O95299 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 10, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| O96000 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 10 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03886 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 1 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03891 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 2 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03897 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 3 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03901 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 4L | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03905 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 4 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03915 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 5 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P03923 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH-ubiquinone oxidoreductase chain 6 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P17568 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 7 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P19404 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] flavoprotein 2, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P28331 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH-ubiquinone oxidoreductase 75 kDa subunit, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P43304 | METFORMIN | Mitochondrial glycerol-3-phosphate dehydrogenase inhibitor | CHEMBL3391681 | Mitochondrial glycerol-3-phosphate dehydrogenase | "Glycerol-3-phosphate dehydrogenase, mitochondrial" | Homo sapiens | enzyme | Small molecule | 1995 |
| P49821 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] flavoprotein 1, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P51970 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 8 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P56181 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] flavoprotein 3, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P56556 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 6 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q16718 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 5 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q16795 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 9, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q86Y39 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 11 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q8N183 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "Mimitin, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9BU61 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex assembly factor 3 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9NRX3 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 4-like 2 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9NX14 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 11, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9P032 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex assembly factor 4 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9P0J0 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9UI09 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 12 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9Y375 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | "Complex I intermediate-associated protein 30, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| Q9Y6M9 | METFORMIN | Mitochondrial complex I (NADH dehydrogenase) inhibitor | CHEMBL2363065 | Mitochondrial complex I (NADH dehydrogenase) | NADH dehydrogenase [ubiquinone] 1 beta subcomplex subunit 9 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P20309 | METHACHOLINE | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1986 |
| METHACYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1982 | ||
| P35372 | METHADONE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1947 |
| P23975 | METHAMPHETAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1943 |
| P31645 | METHAMPHETAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1943 |
| Q01959 | METHAMPHETAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1943 |
| P25021 | METHANTHELINE | Histamine H2 receptor antagonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1951 |
| P18505 | METHARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | METHARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | METHARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P00915 | METHAZOLAMIDE | Carbonic anhydrase I inhibitor | CHEMBL261 | Carbonic anhydrase I | Carbonic anhydrase 1 | Homo sapiens | enzyme lyase | Small molecule | 1959 |
| P00918 | METHAZOLAMIDE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1959 |
| P22748 | METHAZOLAMIDE | Carbonic anhydrase IV inhibitor | CHEMBL3729 | Carbonic anhydrase IV | Carbonic anhydrase 4 | Homo sapiens | enzyme lyase | Small molecule | 1959 |
| P43166 | METHAZOLAMIDE | Carbonic anhydrase VII inhibitor | CHEMBL2326 | Carbonic anhydrase VII | Carbonic anhydrase 7 | Homo sapiens | enzyme lyase | Small molecule | 1959 |
| P35367 | METHDILAZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| METHENAMINE | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1967 | |||
| P72355 | METHICILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin-binding protein 4 | Staphylococcus | enzyme protease serine se s13 | Small molecule | 1982 |
| Q53707 | METHICILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | MecA PBP2' (penicillin binding protein 2') | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1982 |
| Q53725 | METHICILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | PASTA domain protein | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1982 |
| Q53729 | METHICILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin binding protein 2 | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1982 |
| Q9XDB3 | METHICILLIN | Penicillin-binding protein inhibitor | CHEMBL2363021 | Penicillin-binding protein | Penicillin binding transpeptidase domain protein | Staphylococcus | enzyme protease serine unclassified | Small molecule | 1982 |
| P07202 | METHIMAZOLE | Thyroid peroxidase inhibitor | CHEMBL1839 | Thyroid peroxidase | Thyroid peroxidase | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P11229 | METHIXENE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P28335 | METHIXENE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1982 |
| P00915 | METHOCARBAMOL | Carbonic anhydrase I inhibitor | CHEMBL261 | Carbonic anhydrase I | Carbonic anhydrase 1 | Homo sapiens | enzyme lyase | Small molecule | 1957 |
| P18505 | METHOHEXITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P28472 | METHOHEXITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P47870 | METHOHEXITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1960 |
| P00374 | METHOTREXATE | Dihydrofolate reductase inhibitor | CHEMBL202 | Dihydrofolate reductase | Dihydrofolate reductase | Homo sapiens | enzyme reductase | Small molecule | 1953 |
| P25100 | METHOXAMINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P35348 | METHOXAMINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P35368 | METHOXAMINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| METHOXSALEN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1954 | |||
| O00591 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| O14764 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P14867 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P18505 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P18507 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P23415 | METHOXYFLURANE | Glycine receptor (alpha-1/beta) agonist | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 0 |
| P28472 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P31644 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P34903 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P47869 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P47870 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P48169 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P78334 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| Q16445 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| Q8N1C3 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| Q99928 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| Q9UN88 | METHOXYFLURANE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 0 |
| P11229 | METHSCOPOLAMINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1953 |
| P20309 | METHSCOPOLAMINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1953 |
| O43497 | METHSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1957 |
| O95180 | METHSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1957 |
| Q9P0X4 | METHSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1957 |
| P55017 | METHYCLOTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1960 |
| METHYL AMINOLEVULINATE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2004 | |||
| METHYL SALICYLATE | Unknown | Small molecule | 2008 | ||||||
| P08913 | METHYLDOPA | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P18089 | METHYLDOPA | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P18825 | METHYLDOPA | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P08913 | METHYLDOPATE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P18089 | METHYLDOPATE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P18825 | METHYLDOPATE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1962 |
| P21728 | METHYLERGONOVINE | Dopamine D1 receptor antagonist | CHEMBL2056 | Dopamine D1 receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1946 |
| P41595 | METHYLERGONOVINE | Serotonin 2b (5-HT2b) receptor partial agonist | CHEMBL1833 | Serotonin 2b (5-HT2b) receptor | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1946 |
| METHYLHOMATROPINE | Unknown | Small molecule | 1943 | ||||||
| P35372 | METHYLNALTREXONE | Mu opioid receptor antagonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2008 |
| P23975 | METHYLPHENIDATE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| Q01959 | METHYLPHENIDATE | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1955 |
| P04150 | METHYLPREDNISOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1957 |
| P04150 | METHYLPREDNISOLONE HEMISUCCINATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1959 |
| P35367 | METHYLPROMAZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1982 |
| P10275 | METHYLTESTOSTERONE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1973 |
| O00591 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| O14764 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P14867 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18505 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18507 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P31644 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P34903 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47869 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P48169 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P78334 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q16445 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q8N1C3 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q99928 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q9UN88 | METHYPRYLON | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P08908 | METHYSERGIDE | Serotonin 1a (5-HT1a) receptor partial agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1962 |
| P28335 | METHYSERGIDE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1962 |
| P41595 | METHYSERGIDE | Serotonin 2b (5-HT2b) receptor antagonist | CHEMBL1833 | Serotonin 2b (5-HT2b) receptor | 5-hydroxytryptamine receptor 2B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1962 |
| P07550 | METIPRANOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 |
| P08588 | METIPRANOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 |
| P14416 | METOCLOPRAMIDE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1979 |
| P46098 | METOCLOPRAMIDE | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 1979 |
| Q13639 | METOCLOPRAMIDE | Serotonin 4 (5-HT4) receptor agonist | CHEMBL1875 | Serotonin 4 (5-HT4) receptor | 5-hydroxytryptamine receptor 4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1979 |
| P02708 | METOCURINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 |
| P07510 | METOCURINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1982 |
| P11230 | METOCURINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 |
| Q04844 | METOCURINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1982 |
| Q07001 | METOCURINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1982 |
| P55017 | METOLAZONE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1973 |
| P08588 | METOPROLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 |
| P48357 | METRELEPTIN | Leptin receptor agonist | CHEMBL5913 | Leptin receptor | Leptin receptor | Homo sapiens | unclassified | Protein | 2014 |
| METRONIDAZOLE | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1963 | |||
| P07101 | METYROSINE | Tyrosine 3-hydroxylase inhibitor | CHEMBL1969 | Tyrosine 3-hydroxylase | Tyrosine 3-monooxygenase | Homo sapiens | enzyme reductase | Small molecule | 1979 |
| P35498 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| P35499 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q01118 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q14524 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q15858 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q99250 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q9NY46 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q9UI33 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q9UQD0 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| Q9Y5Y9 | MEXILETINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1985 |
| P02918 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P02919 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1981 |
| P08506 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P0AD65 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P0AD68 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1981 |
| P0AEB2 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P24228 | MEZLOCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1981 |
| O43497 | MIBEFRADIL | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1997 |
| O95180 | MIBEFRADIL | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1997 |
| Q9P0X4 | MIBEFRADIL | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1997 |
| O13428 | MICAFUNGIN | "1,3-beta-glucan synthase inhibitor" | CHEMBL2364673 | "1,3-beta-glucan synthase" | "Beta-1,3-glucan synthase catalytic subunit 1" | Candida | enzyme transferase | Small molecule | 2005 |
| P10613 | MICONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1974 |
| P14867 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P18507 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P31644 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P34903 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P47869 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| Q8N1C3 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| Q99928 | MIDAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P25100 | MIDODRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P35348 | MIDODRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P35368 | MIDODRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P04150 | MIFEPRISTONE | Glucocorticoid receptor antagonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 2000 |
| P06401 | MIFEPRISTONE | Progesterone receptor antagonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2000 |
| O43451 | MIGLITOL | Maltase-glucoamylase inhibitor | CHEMBL2074 | Maltase-glucoamylase | "Maltase-glucoamylase, intestinal" | Homo sapiens | enzyme hydrolase | Small molecule | 1996 |
| P10253 | MIGLITOL | Lysosomal alpha-glucosidase inhibitor | CHEMBL2608 | Lysosomal alpha-glucosidase | Lysosomal alpha-glucosidase | Homo sapiens | enzyme hydrolase | Small molecule | 1996 |
| Q16739 | MIGLUSTAT | Ceramide glucosyltransferase inhibitor | CHEMBL2063 | Ceramide glucosyltransferase | Ceramide glucosyltransferase | Homo sapiens | enzyme transferase | Small molecule | 2003 |
| P23975 | MILNACIPRAN | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2009 |
| P31645 | MILNACIPRAN | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2009 |
| Q14432 | MILRINONE | Phosphodiesterase 3A inhibitor | CHEMBL241 | Phosphodiesterase 3A | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1987 |
| MILTEFOSINE | Unknown | Small molecule | 2014 | ||||||
| MINOCYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1971 | ||
| O60706 | MINOXIDIL | "Sulfonylurea receptor 2, Kir6.2 opener" | CHEMBL2095198 | "Sulfonylurea receptor 2, Kir6.2" | ATP-binding cassette sub-family C member 9 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1979 |
| MIPOMERSEN | Apo-B 100 mRNA antisense inhibitor | CHEMBL2364185 | Apo-B 100 mRNA | Apo-B 100 mRNA | Homo sapiens | Oligonucleotide | 2013 | ||
| P13945 | MIRABEGRON | Beta-3 adrenergic receptor agonist | CHEMBL246 | Beta-3 adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2012 |
| P08913 | MIRTAZAPINE | Adrenergic receptor alpha-2 antagonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18089 | MIRTAZAPINE | Adrenergic receptor alpha-2 antagonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18825 | MIRTAZAPINE | Adrenergic receptor alpha-2 antagonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P28223 | MIRTAZAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 |
| P28335 | MIRTAZAPINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 |
| P43115 | MISOPROSTOL | Prostanoid EP3 receptor agonist | CHEMBL3710 | Prostanoid EP3 receptor | Prostaglandin E2 receptor EP3 subtype | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 1988 |
| MITOMYCIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1981 | |||
| P05108 | MITOTANE | Cytochrome P450 11A1 inhibitor | CHEMBL2033 | Cytochrome P450 11A1 | "Cholesterol side-chain cleavage enzyme, mitochondrial" | Homo sapiens | enzyme cytochrome p450 cyp_11 cyp_11a cyp_11a1 | Small molecule | 1970 |
| P15538 | MITOTANE | Cytochrome P450 11B1 inhibitor | CHEMBL1908 | Cytochrome P450 11B1 | "Cytochrome P450 11B1, mitochondrial" | Homo sapiens | enzyme cytochrome p450 cyp_11 cyp_11b cyp_11b1 | Small molecule | 1970 |
| P06241 | MITOXANTRONE | Tyrosine-protein kinase Fyn | Tyrosine-protein kinase Fyn | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 1987 | ||
| P11388 | MITOXANTRONE | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1987 |
| P11388 | MITOXANTRONE | DNA inhibitor | CHEMBL2311221 | DNA | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1987 |
| MITOXANTRONE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1987 | |||
| P02708 | MIVACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1992 |
| P07510 | MIVACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1992 |
| P11230 | MIVACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1992 |
| Q04844 | MIVACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1992 |
| Q07001 | MIVACURIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1992 |
| Q01959 | MODAFINIL | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1998 |
| P12821 | MOEXIPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1995 |
| P14416 | MOLINDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1974 |
| P28223 | MOLINDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1974 |
| P04150 | MOMETASONE FUROATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1987 |
| P14679 | MONOBENZONE | Tyrosinase inhibitor | CHEMBL1973 | Tyrosinase | Tyrosinase | Homo sapiens | enzyme reductase | Small molecule | 1952 |
| MONOCTANOIN | Unknown | Small molecule | 1985 | ||||||
| Q9Y271 | MONTELUKAST | Cysteinyl leukotriene receptor 1 antagonist | CHEMBL1798 | Cysteinyl leukotriene receptor 1 | Cysteinyl leukotriene receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor leukotriene receptor | Small molecule | 1998 |
| P35498 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| P35499 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q01118 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q14524 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q15858 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q99250 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q9NY46 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q9UI33 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q9UQD0 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| Q9Y5Y9 | MORICIZINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1990 |
| P35372 | MORPHINE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P02918 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P02919 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1982 |
| P08506 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P0AD65 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1982 |
| P0AD68 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1982 |
| P0AEB2 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1982 |
| P24228 | MOXALACTAM | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1982 |
| P0AES4 | MOXIFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1999 |
| P0AES6 | MOXIFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1999 |
| P0AFI2 | MOXIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 1999 |
| P20083 | MOXIFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 1999 |
| P43700 | MOXIFLOXACIN | DNA gyrase subunit A | DNA gyrase subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1999 | ||
| P43702 | MOXIFLOXACIN | DNA topoisomerase 4 subunit A | DNA topoisomerase 4 subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1999 | ||
| P41972 | MUPIROCIN | Isoleucyl-tRNA synthetase inhibitor | CHEMBL1982 | Isoleucyl-tRNA synthetase | Isoleucine--tRNA ligase | Staphylococcus aureus | enzyme ligase | Small molecule | 1987 |
| Q99YW3 | MUPIROCIN | Isoleucyl-tRNA synthetase inhibitor | CHEMBL2364671 | Isoleucyl-tRNA synthetase | Isoleucine--tRNA ligase | Streptococcus pyogenes | enzyme ligase | Small molecule | 1987 |
| P07766 | MUROMONAB-CD3 | T cell surface glycoprotein CD3 inhibitor | CHEMBL2364168 | T cell surface glycoprotein CD3 | T-cell surface glycoprotein CD3 epsilon chain | Homo sapiens | membrane receptor | Antibody | 1986 |
| P12268 | MYCOPHENOLATE MOFETIL | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P20839 | MYCOPHENOLATE MOFETIL | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1995 |
| P12268 | MYCOPHENOLIC ACID | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 2004 |
| P20839 | MYCOPHENOLIC ACID | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 2004 |
| P21554 | NABILONE | Cannabinoid CB1 receptor agonist | CHEMBL218 | Cannabinoid CB1 receptor | Cannabinoid receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor cannabinoid receptor | Small molecule | 1985 |
| P35354 | NABUMETONE | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1991 |
| P07550 | NADOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P08588 | NADOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P30968 | NAFARELIN | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 1990 |
| P72355 | NAFCILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin-binding protein 4 | Staphylococcus aureus | enzyme protease serine se s13 | Small molecule | 1965 |
| Q53707 | NAFCILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | MecA PBP2' (penicillin binding protein 2') | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1965 |
| Q53725 | NAFCILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | PASTA domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1965 |
| Q53729 | NAFCILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding protein 2 | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1965 |
| Q9XDB3 | NAFCILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding transpeptidase domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1965 |
| Q4JEY0 | NAFTIFINE | Squalene monooxygenase inhibitor | CHEMBL2364679 | Squalene monooxygenase | Squalene epoxidase | Trichophyton | enzyme reductase | Small molecule | 1988 |
| P35372 | NALBUPHINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1979 |
| P41143 | NALBUPHINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1979 |
| P41145 | NALBUPHINE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1979 |
| P0AES4 | NALIDIXIC ACID | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1964 |
| P0AES6 | NALIDIXIC ACID | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1964 |
| P35372 | NALMEFENE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1995 |
| P41143 | NALMEFENE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1995 |
| P41145 | NALMEFENE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1995 |
| P35372 | NALOXEGOL | Mu opioid receptor antagonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2014 |
| P35372 | NALOXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1971 |
| P41143 | NALOXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1971 |
| P41145 | NALOXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1971 |
| P35372 | NALTREXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P41143 | NALTREXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P41145 | NALTREXONE | Opioid receptors; mu/kappa/delta antagonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P10275 | NANDROLONE DECANOATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1983 |
| P10275 | NANDROLONE PHENPROPIONATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1959 |
| P08913 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P18089 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P18825 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P25100 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P35348 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P35368 | NAPHAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1971 |
| P23219 | NAPROXEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P35354 | NAPROXEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P28221 | NARATRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1998 |
| P28222 | NARATRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1998 |
| P13612 | NATALIZUMAB | Integrin alpha-4/beta-1 inhibitor | CHEMBL1907599 | Integrin alpha-4/beta-1 | Integrin alpha-4 | Homo sapiens | membrane receptor | Antibody | 2004 |
| P13612 | NATALIZUMAB | Integrin alpha-4/beta-7 inhibitor | CHEMBL2095184 | Integrin alpha-4/beta-7 | Integrin alpha-4 | Homo sapiens | membrane receptor | Antibody | 2004 |
| NATAMYCIN | Ergosterol chelating agent | CHEMBL2364028 | Ergosterol | Candida albicans | Small molecule | 1978 | |||
| Q09428 | NATEGLINIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 2000 |
| Q14654 | NATEGLINIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 2000 |
| P07550 | NEBIVOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2007 |
| P08588 | NEBIVOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2007 |
| NEDOCROMIL | Unknown | Small molecule | 1992 | ||||||
| P23975 | NEFAZODONE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1994 |
| P28223 | NEFAZODONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1994 |
| P28335 | NEFAZODONE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1994 |
| P31645 | NEFAZODONE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1994 |
| P09884 | NELARABINE | DNA polymerase alpha catalytic subunit | DNA polymerase alpha catalytic subunit | Homo sapiens | enzyme transferase | Small molecule | 2005 | ||
| P27707 | NELARABINE | Deoxycytidine kinase | Deoxycytidine kinase | Homo sapiens | enzyme | Small molecule | 2005 | ||
| P60891 | NELARABINE | Ribose-phosphate pyrophosphokinase 1 | Ribose-phosphate pyrophosphokinase 1 | Homo sapiens | enzyme | Small molecule | 2005 | ||
| NELARABINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2005 | |||
| Q72874 | NELFINAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 1997 |
| NEOMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1957 | ||
| P22303 | NEOSTIGMINE | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 2013 |
| P23219 | NEPAFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 2005 |
| P35354 | NEPAFENAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 2005 |
| P16066 | NESIRITIDE | Atrial natriuretic peptide receptor A agonist | CHEMBL1988 | Atrial natriuretic peptide receptor A | Atrial natriuretic peptide receptor 1 | Homo sapiens | enzyme lyase guanylate cyclase receptor guanylate cyclase | Protein | 2001 |
| NETILMICIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1983 | ||
| P25103 | NETUPITANT | Neurokinin 1 receptor antagonist | CHEMBL249 | Neurokinin 1 receptor | Substance-P receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide neurokinin receptor | Small molecule | 2014 |
| Q72547 | NEVIRAPINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1996 |
| O60840 | NICARDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| Q01668 | NICARDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| Q13698 | NICARDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| Q13936 | NICARDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| NICLOSAMIDE | DNA inhibitor | CHEMBL2366043 | DNA | Schistosoma mansoni | Small molecule | 1982 | |||
| NICLOSAMIDE | DNA inhibitor | CHEMBL2366044 | DNA | Taenia | Small molecule | 1982 | |||
| P17787 | NICOTINE | Neuronal acetylcholine receptor; alpha4/beta2 agonist | CHEMBL1907589 | Neuronal acetylcholine receptor; alpha4/beta2 | Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1984 |
| P43681 | NICOTINE | Neuronal acetylcholine receptor; alpha4/beta2 agonist | CHEMBL1907589 | Neuronal acetylcholine receptor; alpha4/beta2 | Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1984 |
| O60840 | NIFEDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q01668 | NIFEDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q13698 | NIFEDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q13936 | NIFEDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| P00519 | NILOTINIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2007 |
| P10275 | NILUTAMIDE | Androgen Receptor antagonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1996 |
| O60840 | NIMODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| P08235 | NIMODIPINE | Mineralocorticoid receptor antagonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1988 |
| Q01668 | NIMODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| Q13698 | NIMODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| Q13936 | NIMODIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1988 |
| P09619 | NINTEDANIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2014 |
| P11362 | NINTEDANIB | Fibroblast growth factor receptor inhibitor | CHEMBL2095217 | Fibroblast growth factor receptor | Fibroblast growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2014 |
| P16234 | NINTEDANIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2014 |
| P17948 | NINTEDANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2014 |
| P21802 | NINTEDANIB | Fibroblast growth factor receptor inhibitor | CHEMBL2095217 | Fibroblast growth factor receptor | Fibroblast growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2014 |
| P22455 | NINTEDANIB | Fibroblast growth factor receptor inhibitor | CHEMBL2095217 | Fibroblast growth factor receptor | Fibroblast growth factor receptor 4 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2014 |
| P22607 | NINTEDANIB | Fibroblast growth factor receptor inhibitor | CHEMBL2095217 | Fibroblast growth factor receptor | Fibroblast growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2014 |
| P35916 | NINTEDANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2014 |
| P35968 | NINTEDANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2014 |
| O60840 | NISOLDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1995 |
| Q01668 | NISOLDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1995 |
| Q13698 | NISOLDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1995 |
| Q13936 | NISOLDIPINE | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1995 |
| Q24982 | NITAZOXANIDE | Pyruvate:ferredoxin oxidoreductase inhibitor | CHEMBL2364027 | Pyruvate:ferredoxin oxidoreductase | Pyruvate:ferredoxin oxidoreductase | Giardia intestinalis | enzyme reductase | Small molecule | 2002 |
| Q968X7 | NITAZOXANIDE | Pyruvate:ferredoxin oxidoreductase inhibitor | CHEMBL2364026 | Pyruvate:ferredoxin oxidoreductase | Pyruvate dehydrogenase [NADP(+)] | Cryptosporidium parvum | enzyme reductase | Small molecule | 2002 |
| P32754 | NITISINONE | 4-hydroxyphenylpyruvate dioxygenase inhibitor | CHEMBL1861 | 4-hydroxyphenylpyruvate dioxygenase | 4-hydroxyphenylpyruvate dioxygenase | Homo sapiens | enzyme reductase | Small molecule | 2002 |
| O75343 | NITRIC OXIDE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1999 |
| Q02153 | NITRIC OXIDE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1999 |
| NITROFURANTOIN | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1953 | |||
| NITROFURAZONE | DNA inhibitor | CHEMBL2364041 | DNA | Bacteria | Small molecule | 1945 | |||
| O75343 | NITROGLYCERIN | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1981 |
| Q02153 | NITROGLYCERIN | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1981 |
| O75343 | NITROPRUSSIDE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1981 |
| Q02153 | NITROPRUSSIDE | Soluble guanylate cyclase activator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 1981 |
| Q15116 | NIVOLUMAB | Programmed cell death protein 1 inhibitor | CHEMBL3307223 | Programmed cell death protein 1 | Programmed cell death protein 1 | Homo sapiens | surface antigen | Antibody | 2015 |
| P25021 | NIZATIDINE | Histamine H2 receptor antagonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1988 |
| NORDIHYDROGUAIARETIC ACID | Unknown | Small molecule | 1992 | ||||||
| P06401 | NORELGESTROMIN | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2001 |
| P07550 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P08588 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P08913 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P13945 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P18089 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P18825 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P25100 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P35348 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P35368 | NOREPINEPHRINE | Adrenergic receptor agonist | CHEMBL2331074 | Adrenergic receptor | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1950 |
| P06401 | NORETHINDRONE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1962 |
| P06401 | NORETHINDRONE ACETATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1973 |
| P06401 | NORETHYNODREL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1961 |
| P0AES4 | NORFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1986 |
| P0AES6 | NORFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1986 |
| P0AFI2 | NORFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 1986 |
| P20083 | NORFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 1986 |
| P43700 | NORFLOXACIN | DNA gyrase subunit A | DNA gyrase subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1986 | ||
| P43702 | NORFLOXACIN | DNA topoisomerase 4 subunit A | DNA topoisomerase 4 subunit A | Haemophilus influenzae (strain ATCC 51907 / DSM 11121 / KW20 / Rd) | Isomerase | Small molecule | 1986 | ||
| P72525 | NORFLOXACIN | DNA topoisomerase 4 subunit A | DNA topoisomerase 4 subunit A | Streptococcus pneumoniae serotype 4 (strain ATCC BAA-334 / TIGR4) | enzyme isomerase | Small molecule | 1986 | ||
| P06401 | NORGESTIMATE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1989 |
| P06401 | NORGESTREL | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1968 |
| P23975 | NORTRIPTYLINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1964 |
| P31645 | NORTRIPTYLINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1964 |
| Q5HK03 | NOVOBIOCIN | DNA gyrase inhibitor | CHEMBL2331040 | DNA gyrase | DNA gyrase subunit B | Staphylococcus epidermidis | enzyme isomerase | Small molecule | 0 |
| Q5HK04 | NOVOBIOCIN | DNA gyrase inhibitor | CHEMBL2331040 | DNA gyrase | DNA gyrase subunit A | Staphylococcus epidermidis | enzyme isomerase | Small molecule | 0 |
| NYSTATIN | Ergosterol chelating agent | CHEMBL2364028 | Ergosterol | Candida albicans | Small molecule | 1964 | |||
| P11836 | OBINUTUZUMAB | B-lymphocyte antigen CD20 inhibitor | CHEMBL2058 | B-lymphocyte antigen CD20 | B-lymphocyte antigen CD20 | Homo sapiens | ion channel other misc cd20 | Antibody | 2013 |
| A4D0S4 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit beta-4 | Homo sapiens | structural | Unknown | 2010 |
| A6NMZ7 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-6(VI) chain | Homo sapiens | structural | Unknown | 2010 |
| A8TX70 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-5(VI) chain | Homo sapiens | structural | Unknown | 2010 |
| O15230 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit alpha-5 | Homo sapiens | structural | Unknown | 2010 |
| P02452 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(I) chain | Homo sapiens | structural | Unknown | 2010 |
| P02458 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(II) chain | Homo sapiens | structural | Unknown | 2010 |
| P02461 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(III) chain | Homo sapiens | structural | Unknown | 2010 |
| P02462 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| P02751 | OCRIPLASMIN | Fibronectin proteolytic enzyme | CHEMBL3810 | Fibronectin | Fibronectin | Homo sapiens | adhesion | Unknown | 2010 |
| P05997 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(V) chain | Homo sapiens | structural | Unknown | 2010 |
| P07942 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit beta-1 | Homo sapiens | structural | Unknown | 2010 |
| P08123 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(I) chain | Homo sapiens | structural | Unknown | 2010 |
| P08572 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| P11047 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit gamma-1 | Homo sapiens | structural | Unknown | 2010 |
| P12107 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XI) chain | Homo sapiens | structural | Unknown | 2010 |
| P12109 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(VI) chain | Homo sapiens | structural | Unknown | 2010 |
| P12110 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(VI) chain | Homo sapiens | structural | Unknown | 2010 |
| P12111 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(VI) chain | Homo sapiens | structural | Unknown | 2010 |
| P13942 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-2(XI) chain | Homo sapiens | structural | Unknown | 2010 |
| P20908 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(V) chain | Homo sapiens | structural | Unknown | 2010 |
| P24043 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit alpha-2 | Homo sapiens | structural | Unknown | 2010 |
| P25391 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit alpha-1 | Homo sapiens | structural | Unknown | 2010 |
| P25940 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(V) chain | Homo sapiens | structural | Unknown | 2010 |
| P29400 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-5(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| P39059 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XV) chain | Homo sapiens | structural | Unknown | 2010 |
| P39060 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XVIII) chain | Homo sapiens | structural | Unknown | 2010 |
| P53420 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-4(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| P55268 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit beta-2 | Homo sapiens | structural | Unknown | 2010 |
| Q01955 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-3(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| Q13751 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit beta-3 | Homo sapiens | structural | Unknown | 2010 |
| Q13753 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit gamma-2 | Homo sapiens | structural | Unknown | 2010 |
| Q14031 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-6(IV) chain | Homo sapiens | structural | Unknown | 2010 |
| Q16363 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit alpha-4 | Homo sapiens | structural | Unknown | 2010 |
| Q16787 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit alpha-3 | Homo sapiens | structural | Unknown | 2010 |
| Q17RW2 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXIV) chain | Homo sapiens | structural | Unknown | 2010 |
| Q2UY09 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXVIII) chain | Homo sapiens | structural | Unknown | 2010 |
| Q8IZC6 | OCRIPLASMIN | Collagen hydrolytic enzyme | CHEMBL2364188 | Collagen | Collagen alpha-1(XXVII) chain | Homo sapiens | structural | Unknown | 2010 |
| Q9Y6N6 | OCRIPLASMIN | Laminin hydrolytic enzyme | CHEMBL2364187 | Laminin | Laminin subunit gamma-3 | Homo sapiens | structural | Unknown | 2010 |
| P30872 | OCTREOTIDE | Somatostatin receptor agonist | CHEMBL2111436 | Somatostatin receptor | Somatostatin receptor type 1 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 1988 |
| P30874 | OCTREOTIDE | Somatostatin receptor agonist | CHEMBL2111436 | Somatostatin receptor | Somatostatin receptor type 2 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 1988 |
| P31391 | OCTREOTIDE | Somatostatin receptor agonist | CHEMBL2111436 | Somatostatin receptor | Somatostatin receptor type 4 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 1988 |
| P32745 | OCTREOTIDE | Somatostatin receptor agonist | CHEMBL2111436 | Somatostatin receptor | Somatostatin receptor type 3 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 1988 |
| P35346 | OCTREOTIDE | Somatostatin receptor agonist | CHEMBL2111436 | Somatostatin receptor | Somatostatin receptor type 5 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 1988 |
| P11836 | OFATUMUMAB | B-lymphocyte antigen CD20 inhibitor | CHEMBL2058 | B-lymphocyte antigen CD20 | B-lymphocyte antigen CD20 | Homo sapiens | ion channel other misc cd20 | Antibody | 2009 |
| P0AES4 | OFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1990 |
| P0AES6 | OFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1990 |
| P10520 | OFLOXACIN | Streptokinase A | Streptokinase A | Streptococcus pyogenes serotype M1 | unclassified | Small molecule | 1990 | ||
| P14416 | OLANZAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 |
| P21917 | OLANZAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 |
| P28223 | OLANZAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 |
| P28335 | OLANZAPINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1996 |
| P35462 | OLANZAPINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1996 |
| P09874 | OLAPARIB | "PARP 1, 2 & 3 inhibitor" | CHEMBL3390820 | "PARP 1, 2 and 3" | Poly [ADP-ribose] polymerase 1 | Homo sapiens | enzyme | Small molecule | 2014 |
| Q9UGN5 | OLAPARIB | "PARP 1, 2 & 3 inhibitor" | CHEMBL3390820 | "PARP 1, 2 and 3" | Poly [ADP-ribose] polymerase 2 | Homo sapiens | enzyme | Small molecule | 2014 |
| Q9Y6F1 | OLAPARIB | "PARP 1, 2 & 3 inhibitor" | CHEMBL3390820 | "PARP 1, 2 and 3" | Poly [ADP-ribose] polymerase 3 | Homo sapiens | enzyme | Small molecule | 2014 |
| P30556 | OLMESARTAN MEDOXOMIL | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 2002 |
| P07550 | OLODATEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2014 |
| P35367 | OLOPATADINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1996 |
| P09917 | OLSALAZINE | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 1990 |
| P23219 | OLSALAZINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1990 |
| P35354 | OLSALAZINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1990 |
| P37231 | OLSALAZINE | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 1990 |
| OMACETAXINE MEPESUCCINATE | Protein synthesis inhibitor | Small molecule | 2009 | ||||||
| P01854 | OMALIZUMAB | Ig epsilon chain C region inhibitor | CHEMBL1834 | Ig epsilon chain C region | Ig epsilon chain C region | Homo sapiens | secreted | Antibody | 2003 |
| Q5L478 | OMBITASVIR | Nonstructural protein 5A inhibitor | CHEMBL3307224 | Nonstructural protein 5A | Nonstructural protein 5A | Hepatitis C virus | unclassified | Small molecule | 2014 |
| Q8JXU8 | OMBITASVIR | Hepatitis C virus NS5B RNA-dependent RNA polymerase | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 2014 | ||
| OMEGA-3-ACID ETHYL ESTERS | Unknown | Small molecule | 2004 | ||||||
| P20648 | OMEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 1989 |
| P20648 | OMEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 1989 |
| P46098 | ONDANSETRON | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 1991 |
| Q14626 | OPRELVEKIN | Interleukin 11 receptor alpha agonist | CHEMBL2050 | Interleukin 11 receptor alpha | Interleukin-11 receptor subunit alpha | Homo sapiens | membrane receptor | Protein | 1997 |
| ORITAVANCIN | Peptidoglycan inhibitor | CHEMBL3041361 | Peptidoglycan | Bacteria | Unknown | 2014 | |||
| P07098 | ORLISTAT | Gastric lipase inhibitor | CHEMBL1796 | Gastric lipase | Gastric triacylglycerol lipase | Homo sapiens | enzyme hydrolase | Small molecule | 1999 |
| P16233 | ORLISTAT | Pancreatic lipase inhibitor | CHEMBL1812 | Pancreatic lipase | Pancreatic triacylglycerol lipase | Homo sapiens | enzyme hydrolase | Small molecule | 1999 |
| P49327 | ORLISTAT | Fatty acid synthase inhibitor | CHEMBL4158 | Fatty acid synthase | Fatty acid synthase | Homo sapiens | enzyme transferase | Small molecule | 1999 |
| O15399 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2D" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| O60391 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| P23975 | ORPHENADRINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1957 |
| P35367 | ORPHENADRINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1957 |
| P35498 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| P35499 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q01118 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q05586 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 1" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| Q12879 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| Q13224 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2B" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| Q14524 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q14957 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 2C" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| Q15858 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q8TCU5 | ORPHENADRINE | Glutamate [NMDA] receptor antagonist | CHEMBL2094124 | Glutamate [NMDA] receptor | "Glutamate receptor ionotropic, NMDA 3A" | Homo sapiens | ion channel lgic glut nmda | Small molecule | 1957 |
| Q99250 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9NY46 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9UI33 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9UQD0 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| Q9Y5Y9 | ORPHENADRINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1957 |
| P03468 | OSELTAMIVIR | Neuraminidase inhibitor | CHEMBL2051 | Neuraminidase | Neuraminidase | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | enzyme hydrolase | Small molecule | 1999 |
| P03474 | OSELTAMIVIR | Neuraminidase inhibitor | CHEMBL3377 | Neuraminidase | Neuraminidase | Influenza B virus (strain B/Lee/1940) | enzyme hydrolase | Small molecule | 1999 |
| P03372 | OSPEMIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2013 |
| Q92731 | OSPEMIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 2013 |
| P72355 | OXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin-binding protein 4 | Staphylococcus aureus | enzyme protease serine se s13 | Small molecule | 1971 |
| Q53707 | OXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | MecA PBP2' (penicillin binding protein 2') | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1971 |
| Q53725 | OXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | PASTA domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1971 |
| Q53729 | OXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding protein 2 | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1971 |
| Q9XDB3 | OXACILLIN | Penicillin-binding protein inhibitor | CHEMBL2362972 | Penicillin-binding protein | Penicillin binding transpeptidase domain protein | Staphylococcus aureus | enzyme protease serine unclassified | Small molecule | 1971 |
| OXALIPLATIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2002 | |||
| OXAMNIQUINE | DNA inhibitor | CHEMBL2366043 | DNA | Schistosoma mansoni | Small molecule | 1980 | |||
| P10275 | OXANDROLONE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1964 |
| P23219 | OXAPROZIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1992 |
| P35354 | OXAPROZIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1992 |
| P14867 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| P18507 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| P31644 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| P34903 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| P47869 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| Q8N1C3 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| Q99928 | OXAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1965 |
| P35498 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| P35499 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q01118 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q14524 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q15858 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q99250 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9NY46 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UI33 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UQD0 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9Y5Y9 | OXCARBAZEPINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| P10613 | OXICONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1988 |
| P00390 | OXIGLUTATIONE | Glutathione reductase | CHEMBL2755 | Glutathione reductase | "Glutathione reductase, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 2008 |
| P07550 | OXPRENOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1983 |
| P08588 | OXPRENOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1983 |
| O75899 | OXYBATE | GABA-B receptor agonist | CHEMBL2111463 | GABA-B receptor | Gamma-aminobutyric acid type B receptor subunit 2 | Homo sapiens | membrane receptor 7tm3 smallmol neurotransmitter gaba-b receptor | Small molecule | 2002 |
| Q9UBS5 | OXYBATE | GABA-B receptor agonist | CHEMBL2111463 | GABA-B receptor | Gamma-aminobutyric acid type B receptor subunit 1 | Homo sapiens | membrane receptor 7tm3 smallmol neurotransmitter gaba-b receptor | Small molecule | 2002 |
| P08172 | OXYBUTYNIN | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1975 |
| P20309 | OXYBUTYNIN | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1975 |
| P35372 | OXYCODONE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1950 |
| P08913 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P18089 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P18825 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P25100 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P35348 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P35368 | OXYMETAZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| P10275 | OXYMETHOLONE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1972 |
| P35372 | OXYMORPHONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1959 |
| P41143 | OXYMORPHONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1959 |
| P41145 | OXYMORPHONE | Opioid receptors; mu/kappa/delta agonist | CHEMBL2095181 | Opioid receptors; mu/kappa/delta | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1959 |
| P23219 | OXYPHENBUTAZONE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1960 |
| P35354 | OXYPHENBUTAZONE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1960 |
| P11229 | OXYPHENCYCLIMINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P20309 | OXYPHENCYCLIMINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P11229 | OXYPHENONIUM | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| P20309 | OXYPHENONIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1982 |
| OXYTETRACYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1964 | ||
| P30559 | OXYTOCIN | Oxytocin receptor agonist | CHEMBL2049 | Oxytocin receptor | Oxytocin receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1980 |
| P04350 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1992 |
| P07437 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1992 |
| P68371 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1992 |
| Q13509 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1992 |
| Q13885 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1992 |
| Q3ZCM7 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1992 |
| Q9BUF5 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1992 |
| Q9BVA1 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1992 |
| Q9H4B7 | PACLITAXEL | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1992 |
| P11802 | PALBOCICLIB | CDK4/cyclin D1 inhibitor | CHEMBL1907601 | Cyclin-dependent kinase 4/cyclin D1 | Cyclin-dependent kinase 4 | Homo sapiens | enzyme kinase protein kinase cmgc | Small molecule | 2015 |
| P24385 | PALBOCICLIB | CDK4/cyclin D1 inhibitor | CHEMBL2111455 | CDK6/cyclin D1 | G1/S-specific cyclin-D1 | Homo sapiens | cytosolic other | Small molecule | 2015 |
| P24385 | PALBOCICLIB | CDK6/cyclin D1 inhibitor | CHEMBL2111455 | CDK6/cyclin D1 | G1/S-specific cyclin-D1 | Homo sapiens | cytosolic other | Small molecule | 2015 |
| Q00534 | PALBOCICLIB | CDK4/cyclin D1 inhibitor | CHEMBL2111455 | CDK6/cyclin D1 | Cyclin-dependent kinase 6 | Homo sapiens | enzyme kinase protein kinase cmgc | Small molecule | 2015 |
| Q00534 | PALBOCICLIB | CDK6/cyclin D1 inhibitor | CHEMBL2111455 | CDK6/cyclin D1 | Cyclin-dependent kinase 6 | Homo sapiens | enzyme kinase protein kinase cmgc | Small molecule | 2015 |
| P21802 | PALIFERMIN | Fibroblast growth factor receptor 2 agonist | CHEMBL4142 | Fibroblast growth factor receptor 2 | Fibroblast growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Protein | 2005 |
| P14416 | PALIPERIDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2006 |
| P28223 | PALIPERIDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2006 |
| P03420 | PALIVIZUMAB | Fusion glycoprotein F0 | Fusion glycoprotein F0 | Human respiratory syncytial virus A (strain A2) | Unclassified | Antibody | 1998 | ||
| Q89535 | PALIVIZUMAB | Fusion glycoprotein F0 inhibitor | CHEMBL2364165 | Fusion glycoprotein F0 | Fusion glycoprotein F0 | Human respiratory syncytial virus | unclassified | Antibody | 1998 |
| P46098 | PALONOSETRON | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 2003 |
| P14324 | PAMIDRONIC ACID | Farnesyl diphosphate synthase inhibitor | CHEMBL1782 | Farnesyl diphosphate synthase | Farnesyl pyrophosphate synthase | Homo sapiens | enzyme transferase | Small molecule | 1991 |
| PANCRELIPASE | Starch hydrolytic enzyme | CHEMBL2364180 | Starch | Homo sapiens | Enzyme | 1996 | |||
| PANCRELIPASE | Polypeptides hydrolytic enzyme | CHEMBL2364181 | Polypeptides | Homo sapiens | Enzyme | 1996 | |||
| PANCRELIPASE | Fatty acids hydrolytic enzyme | CHEMBL2364711 | Fatty acids | Homo sapiens | Enzyme | 1996 | |||
| P02708 | PANCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1972 |
| P07510 | PANCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1972 |
| P11230 | PANCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1972 |
| Q04844 | PANCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1972 |
| Q07001 | PANCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1972 |
| P00533 | PANITUMUMAB | Epidermal growth factor receptor erbB1 inhibitor | CHEMBL203 | Epidermal growth factor receptor erbB1 | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Antibody | 2006 |
| O15379 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 3 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2015 |
| P56524 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 4 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2015 |
| Q13547 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 1 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2015 |
| Q8WUI4 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 7 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2015 |
| Q92769 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 2 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2015 |
| Q969S8 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 10 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2015 |
| Q96DB2 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 11 | Homo sapiens | epigenetic regulator eraser hdac hdac class iv | Small molecule | 2015 |
| Q9BY41 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 8 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2015 |
| Q9UBN7 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 6 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2015 |
| Q9UKV0 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 9 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2015 |
| Q9UQL6 | PANOBINOSTAT | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 5 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2015 |
| P20648 | PANTOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 2000 |
| P20648 | PANTOPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 2000 |
| O43497 | PARAMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1949 |
| O95180 | PARAMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1949 |
| Q9P0X4 | PARAMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1949 |
| P04150 | PARAMETHASONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1982 |
| Q03431 | PARATHYROID HORMONE | Parathyroid hormone receptor agonist | CHEMBL1793 | Parathyroid hormone receptor | Parathyroid hormone/parathyroid hormone-related peptide receptor | Homo sapiens | membrane receptor 7tm2 peptide parathyroid hormone receptor parathyroid hormone receptor | Protein | 2015 |
| P21397 | PARGYLINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] A | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P27338 | PARGYLINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P11473 | PARICALCITOL | Vitamin D receptor agonist | CHEMBL1977 | Vitamin D receptor | Vitamin D3 receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1i nr1i1 | Small molecule | 1998 |
| A3EZI9 | PARITAPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | NS3 | Hepatitis C virus | enzyme protease serine pas s29 | Small molecule | 2014 |
| D2K2A8 | PARITAPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | Non-structural protein 4A | Hepatitis C virus | enzyme protease serine pas s29 reg | Small molecule | 2014 |
| PAROMOMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1969 | ||
| P31645 | PAROXETINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1992 |
| P30872 | PASIREOTIDE | Somatostatin receptor 1 agonist | CHEMBL1917 | Somatostatin receptor 1 | Somatostatin receptor type 1 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2012 |
| P30874 | PASIREOTIDE | Somatostatin receptor 2 agonist | CHEMBL1804 | Somatostatin receptor 2 | Somatostatin receptor type 2 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2012 |
| P32745 | PASIREOTIDE | Somatostatin receptor 3 agonist | CHEMBL2028 | Somatostatin receptor 3 | Somatostatin receptor type 3 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2012 |
| P35346 | PASIREOTIDE | Somatostatin receptor 5 agonist | CHEMBL1792 | Somatostatin receptor 5 | Somatostatin receptor type 5 | Homo sapiens | membrane receptor 7tm1 peptide short peptide somatostatin receptor | Protein | 2012 |
| P06239 | PAZOPANIB | Tyrosine-protein kinase LCK inhibitor | CHEMBL258 | Tyrosine-protein kinase LCK | Tyrosine-protein kinase Lck | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2009 |
| P07333 | PAZOPANIB | Macrophage colony stimulating factor receptor inhibitor | CHEMBL1844 | Macrophage colony stimulating factor receptor | Macrophage colony-stimulating factor 1 receptor | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2009 |
| P09619 | PAZOPANIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2009 |
| P10721 | PAZOPANIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2009 |
| P11362 | PAZOPANIB | Fibroblast growth factor receptor 1 inhibitor | CHEMBL3650 | Fibroblast growth factor receptor 1 | Fibroblast growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2009 |
| P16234 | PAZOPANIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2009 |
| P17948 | PAZOPANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2009 |
| P22607 | PAZOPANIB | Fibroblast growth factor receptor 3 inhibitor | CHEMBL2742 | Fibroblast growth factor receptor 3 | Fibroblast growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2009 |
| P35916 | PAZOPANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2009 |
| P35968 | PAZOPANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2009 |
| Q08881 | PAZOPANIB | Tyrosine-protein kinase ITK/TSK inhibitor | CHEMBL2959 | Tyrosine-protein kinase ITK/TSK | Tyrosine-protein kinase ITK/TSK | Homo sapiens | enzyme kinase protein kinase tk tec | Small molecule | 2009 |
| PEGADEMASE BOVINE | 2'-deoxyadenosine hydrolytic enzyme | CHEMBL2364177 | 2'-deoxyadenosine | Homo sapiens | Enzyme | 1990 | |||
| PEGADEMASE BOVINE | Adenosine hydrolytic enzyme | CHEMBL2364178 | Adenosine | Homo sapiens | Enzyme | 1990 | |||
| P15692 | PEGAPTANIB SODIUM | Vascular endothelial growth factor A antagonist | CHEMBL1783 | Vascular endothelial growth factor A | Vascular endothelial growth factor A | Homo sapiens | secreted | Unknown | 2004 |
| PEGASPARGASE | Asparagine hydrolytic enzyme | CHEMBL2364706 | Asparagine | Homo sapiens | Enzyme | 1994 | |||
| Q99062 | PEGFILGRASTIM | Granulocyte colony stimulating factor receptor agonist | CHEMBL1996 | Granulocyte colony stimulating factor receptor | Granulocyte colony-stimulating factor receptor | Homo sapiens | membrane receptor | Protein | 2002 |
| P19235 | PEGINESATIDE ACETATE | Erythropoietin receptor agonist | CHEMBL1817 | Erythropoietin receptor | Erythropoietin receptor | Homo sapiens | membrane receptor | Protein | 2012 |
| P17181 | PEGINTERFERON ALFA-2A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 2002 |
| P48551 | PEGINTERFERON ALFA-2A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 2002 |
| P17181 | PEGINTERFERON ALFA-2B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 2001 |
| P48551 | PEGINTERFERON ALFA-2B | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 2001 |
| P17181 | PEGINTERFERON BETA-1A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 1 | Homo sapiens | membrane receptor | Protein | 2014 |
| P48551 | PEGINTERFERON BETA-1A | Interferon alpha/beta receptor agonist | CHEMBL2364170 | Interferon alpha/beta receptor | Interferon alpha/beta receptor 2 | Homo sapiens | membrane receptor | Protein | 2014 |
| PEGLOTICASE | Uric acid oxidative enzyme | CHEMBL2364183 | Uric acid | Homo sapiens | Enzyme | 2010 | |||
| P10912 | PEGVISOMANT | Growth hormone receptor antagonist | CHEMBL1976 | Growth hormone receptor | Growth hormone receptor | Homo sapiens | membrane receptor | Protein | 2003 |
| Q15116 | PEMBROLIZUMAB | Programmed cell death protein 1 inhibitor | CHEMBL3307223 | Programmed cell death protein 1 | Programmed cell death protein 1 | Homo sapiens | surface antigen | Antibody | 2014 |
| P00374 | PEMETREXED | Dihydrofolate reductase inhibitor | CHEMBL202 | Dihydrofolate reductase | Dihydrofolate reductase | Homo sapiens | enzyme reductase | Small molecule | 2004 |
| P04818 | PEMETREXED | Thymidylate synthase inhibitor | CHEMBL1952 | Thymidylate synthase | Thymidylate synthase | Homo sapiens | enzyme transferase | Small molecule | 2004 |
| P22102 | PEMETREXED | GAR transformylase inhibitor | CHEMBL3972 | GAR transformylase | Trifunctional purine biosynthetic protein adenosine-3 | Homo sapiens | enzyme ligase | Small molecule | 2004 |
| PEMIROLAST | Unknown | Small molecule | 1999 | ||||||
| PEMOLINE | Unknown | Small molecule | 1975 | ||||||
| P07550 | PENBUTOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P08588 | PENBUTOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P04293 | PENCICLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1996 |
| PENICILLAMINE | Copper chelating agent | CHEMBL2363057 | Copper | Small molecule | 1970 | ||||
| PENICILLAMINE | CHEMBL2363057 | Copper | Small molecule | 1970 | |||||
| P02918 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1958 |
| P02919 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1958 |
| P08506 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1958 |
| P0AD65 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1958 |
| P0AD68 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1958 |
| P0AEB2 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1958 |
| P24228 | PENICILLIN V | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1958 |
| PENTAMIDINE | DNA inhibitor | CHEMBL2366046 | DNA | Pneumocystis jirovecii | Small molecule | 1984 | |||
| PENTAMIDINE | Kinetoplast DNA inhibitor | CHEMBL2366047 | Kinetoplast DNA | Trypanosoma brucei | Small molecule | 1984 | |||
| Q99720 | PENTAZOCINE | Sigma opioid receptor modulator | CHEMBL287 | Sigma opioid receptor | Sigma non-opioid intracellular receptor 1 | Homo sapiens | membrane receptor | Small molecule | 1967 |
| PENTETIC ACID | Radioactive metals chelating agent | CHEMBL2366037 | Radioactive metals | Small molecule | 2004 | ||||
| PENTETIC ACID | CHEMBL2366037 | Radioactive metals | Small molecule | 2004 | |||||
| P18505 | PENTOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1973 |
| P28472 | PENTOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1973 |
| P47870 | PENTOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1973 |
| P30926 | PENTOLINIUM | Neuronal acetylcholine receptor; alpha3/beta4 antagonist | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 |
| P32297 | PENTOLINIUM | Neuronal acetylcholine receptor; alpha3/beta4 antagonist | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 |
| PENTOSAN POLYSULFATE SODIUM | Unknown | Small molecule | 1996 | ||||||
| P00813 | PENTOSTATIN | Adenosine deaminase inhibitor | CHEMBL1910 | Adenosine deaminase | Adenosine deaminase | Homo sapiens | enzyme hydrolase | Small molecule | 1991 |
| O00408 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-dependent 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_2 pde_2a | Small molecule | 1984 |
| O43924 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6d | Small molecule | 1984 |
| O60658 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8a | Small molecule | 1984 |
| O76074 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 1984 |
| O76083 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A" | Homo sapiens | enzyme phosphodiesterase pde_9 pde_9a | Small molecule | 1984 |
| O95263 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8B" | Homo sapiens | enzyme phosphodiesterase pde_8 pde_8b | Small molecule | 1984 |
| P16499 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6a | Small molecule | 1984 |
| P18545 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6g | Small molecule | 1984 |
| P27815 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1984 |
| P29274 | PENTOXIFYLLINE | Adenosine A2 receptor antagonist | CHEMBL2094257 | Adenosine A2 receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1984 |
| P29275 | PENTOXIFYLLINE | Adenosine A2 receptor antagonist | CHEMBL2094257 | Adenosine A2 receptor | Adenosine receptor A2b | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1984 |
| P35913 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Rod cGMP-specific 3',5'-cyclic phosphodiesterase subunit beta" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6b | Small molecule | 1984 |
| P51160 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha'" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6c | Small molecule | 1984 |
| P54750 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1A" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1a | Small molecule | 1984 |
| Q01064 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1b | Small molecule | 1984 |
| Q07343 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1984 |
| Q08493 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1984 |
| Q08499 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1984 |
| Q13370 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-inhibited 3',5'-cyclic phosphodiesterase B" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3b | Small molecule | 1984 |
| Q13946 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "High affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7a | Small molecule | 1984 |
| Q13956 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Retinal cone rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit gamma" | Homo sapiens | enzyme phosphodiesterase pde_6 pde_6h | Small molecule | 1984 |
| Q14123 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C" | Homo sapiens | enzyme phosphodiesterase pde_1 pde_1c | Small molecule | 1984 |
| Q14432 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1984 |
| Q9NP56 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP-specific 3',5'-cyclic phosphodiesterase 7B" | Homo sapiens | enzyme phosphodiesterase pde_7 pde_7b | Small molecule | 1984 |
| Q9Y233 | PENTOXIFYLLINE | "3',5'-cyclic phosphodiesterase inhibitor" | CHEMBL2363066 | "3',5'-cyclic phosphodiesterase" | "cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A" | Homo sapiens | enzyme phosphodiesterase pde_10 pde_10a | Small molecule | 1984 |
| P03468 | PERAMIVIR | Neuraminidase inhibitor | CHEMBL2051 | Neuraminidase | Neuraminidase | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | enzyme hydrolase | Small molecule | 2014 |
| P03474 | PERAMIVIR | Neuraminidase inhibitor | CHEMBL3377 | Neuraminidase | Neuraminidase | Influenza B virus (strain B/Lee/1940) | enzyme hydrolase | Small molecule | 2014 |
| P42261 | PERAMPANEL | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 1 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 2012 |
| P42262 | PERAMPANEL | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 2 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 2012 |
| P42263 | PERAMPANEL | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 3 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 2012 |
| P48058 | PERAMPANEL | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 4 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 2012 |
| P14416 | PERGOLIDE | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1988 |
| P21728 | PERGOLIDE | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1988 |
| P21917 | PERGOLIDE | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1988 |
| P21918 | PERGOLIDE | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1988 |
| P35462 | PERGOLIDE | Dopamine receptor agonist | CHEMBL2096905 | Dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1988 |
| P12821 | PERINDOPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1993 |
| Q2VKV7 | PERMETHRIN | Voltage-sensitive sodium channel blocker | CHEMBL2362985 | Voltage-sensitive sodium channel | Sodium channel protein | Sarcoptes scabiei type hominis | ion channel vgc vg na | Small molecule | 1986 |
| P14416 | PERPHENAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1957 |
| P04626 | PERTUZUMAB | Receptor protein-tyrosine kinase erbB-2 inhibitor | CHEMBL1824 | Receptor protein-tyrosine kinase erbB-2 | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Antibody | 2012 |
| P35498 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| P35499 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q01118 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q14524 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q15858 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q99250 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q9NY46 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q9UI33 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q9UQD0 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| Q9Y5Y9 | PHENACEMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1951 |
| P35498 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| P35499 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q01118 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q14524 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q15858 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q99250 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q9NY46 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q9UI33 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q9UQD0 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| Q9Y5Y9 | PHENAZOPYRIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1987 |
| P23975 | PHENDIMETRAZINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1976 |
| Q01959 | PHENDIMETRAZINE | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1976 |
| P21397 | PHENELZINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] A | Homo sapiens | enzyme reductase | Small molecule | 1961 |
| P27338 | PHENELZINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 1961 |
| Q9BQB6 | PHENINDIONE | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor | CHEMBL1930 | Vitamin k epoxide reductase complex subunit 1 isoform 1 | Vitamin K epoxide reductase complex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P35367 | PHENIRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1994 |
| P23975 | PHENMETRAZINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 |
| Q01959 | PHENMETRAZINE | Dopamine transporter inhibitor | CHEMBL238 | Dopamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1982 |
| P08913 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P18089 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P18825 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P25100 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P35348 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| P35368 | PHENOXYBENZAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1953 |
| Q9BQB6 | PHENPROCOUMON | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor | CHEMBL1930 | Vitamin k epoxide reductase complex subunit 1 isoform 1 | Vitamin K epoxide reductase complex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1957 |
| O43497 | PHENSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| O95180 | PHENSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| Q9P0X4 | PHENSUXIMIDE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1982 |
| P23975 | PHENTERMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1959 |
| P08913 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P18089 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P18825 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P25100 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P35348 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P35368 | PHENTOLAMINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| PHENYL AMINOSALICYLATE | Unknown | Small molecule | 1982 | ||||||
| PHENYLBUTANOIC ACID | Glutamine chelating agent | CHEMBL2366039 | Glutamine | Homo sapiens | Small molecule | 1996 | |||
| P23219 | PHENYLBUTAZONE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1980 |
| P35354 | PHENYLBUTAZONE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1980 |
| P25100 | PHENYLEPHRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P35348 | PHENYLEPHRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P35368 | PHENYLEPHRINE | Adrenergic receptor alpha-1 agonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1952 |
| P23975 | PHENYLPROPANOLAMINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1958 |
| P35348 | PHENYLPROPANOLAMINE | Alpha-1a adrenergic receptor agonist | CHEMBL229 | Alpha-1a adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1958 |
| P35498 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| P35499 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q01118 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q14524 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q15858 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q99250 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9NY46 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9UI33 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9UQD0 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9Y5Y9 | PHENYTOIN | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| P11229 | PILOCARPINE | Muscarinic acetylcholine receptor M1 agonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1974 |
| P20309 | PILOCARPINE | Muscarinic acetylcholine receptor M3 agonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1974 |
| P62942 | PIMECROLIMUS | FK506-binding protein 1A inhibitor | CHEMBL1902 | FK506-binding protein 1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Small molecule | 2001 |
| P14416 | PIMOZIDE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1984 |
| P21728 | PIMOZIDE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(1A) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1984 |
| P21917 | PIMOZIDE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1984 |
| P21918 | PIMOZIDE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(1B) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1984 |
| P28223 | PIMOZIDE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1984 |
| P35462 | PIMOZIDE | Dopamine receptor antagonist | CHEMBL2096905 | Dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1984 |
| O60706 | PINACIDIL | "Sulfonylurea receptor 2, Kir6.2 opener" | CHEMBL2095198 | "Sulfonylurea receptor 2, Kir6.2" | ATP-binding cassette sub-family C member 9 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1989 |
| P07550 | PINDOLOL | Beta-2 adrenergic receptor partial agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P08588 | PINDOLOL | Beta-1 adrenergic receptor partial agonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P37231 | PIOGLITAZONE | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 1999 |
| P02708 | PIPECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1990 |
| P07510 | PIPECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1990 |
| P11230 | PIPECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1990 |
| Q04844 | PIPECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1990 |
| Q07001 | PIPECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1990 |
| PIPERACETAZINE | Unknown | Small molecule | 1969 | ||||||
| P02918 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P02919 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1981 |
| P08506 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P0AD65 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1981 |
| P0AD68 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1981 |
| P0AEB2 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1981 |
| P24228 | PIPERACILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1981 |
| E1FVX6 | PIPERAZINE CITRATE | Nematode GABA-A receptor positive modulator | CHEMBL2364676 | Nematode GABA-A receptor | Uncharacterized protein | Onchocercidae | unclassified | Small molecule | 1954 |
| E1G1C3 | PIPERAZINE CITRATE | Nematode GABA-A receptor positive modulator | CHEMBL2364676 | Nematode GABA-A receptor | Uncharacterized protein | Onchocercidae | unclassified | Small molecule | 1954 |
| E0V9R7 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VAD1 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VBK5 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VCA5 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VCW8 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | Putative uncharacterized protein | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VCW9 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VDM3 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VDR0 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VED4 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VGV6 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VHL8 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VHZ1 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VJJ0 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VM29 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VMV6 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VMV7 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VMW9 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VQ45 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VQ46 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VQ47 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VRD2 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VSD4 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VSD5 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VUR0 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VUR1 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VV39 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VV52 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VV70 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VV72 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VXT9 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0VZW4 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0W115 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0W2B1 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0W389 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | "Cytochrome P-450, putative" | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| E0W4F7 | PIPERONYL BUTOXIDE | Cytochrome P450 inhibitor | CHEMBL2364702 | Cytochrome P450 | NADH-Ubiquinone oxidoreductase 39kDa subunit | Pediculus humanus capitis | enzyme reductase | Small molecule | 2000 |
| PIPOBROMAN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1966 | |||
| P07550 | PIRBUTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1986 |
| PIRFENIDONE | Unknown | Small molecule | 2011 | ||||||
| P23219 | PIROXICAM | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P35354 | PIROXICAM | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1982 |
| P04035 | PITAVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 2009 |
| P61073 | PLERIXAFOR | C-X-C chemokine receptor type 4 partial agonist | CHEMBL2107 | C-X-C chemokine receptor type 4 | C-X-C chemokine receptor type 4 | Homo sapiens | membrane receptor 7tm1 peptide chemokine receptor cxc chemokine receptor | Small molecule | 2008 |
| PLICAMYCIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1970 | |||
| P11388 | PODOFILOX | DNA topoisomerase 2-alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1990 | ||
| PODOFILOX | Unknown | Small molecule | 1990 | ||||||
| POLIDOCANOL | Unknown | Small molecule | 2010 | ||||||
| P03372 | POLYESTRADIOL PHOSPHATE | Estrogen receptor alpha agonist | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1957 |
| POLYMYXIN B | Cell outer membrane inhibitor | CHEMBL2364032 | Cell outer membrane | Bacteria | Protein | 1957 | |||
| P55017 | POLYTHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1961 |
| Q96SW2 | POMALIDOMIDE | Protein cereblon | Protein cereblon | Homo sapiens | Unclassified | Small molecule | 2013 | ||
| POMALIDOMIDE | Unknown | Small molecule | 2013 | ||||||
| P00519 | PONATINIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2012 |
| P00519 | PONATINIB | Bcr/Abl fusion protein inhibitor | CHEMBL2096618 | Bcr/Abl fusion protein | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2012 |
| P07948 | PONATINIB | Tyrosine-protein kinase Lyn | Tyrosine-protein kinase Lyn | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2012 | ||
| P10721 | PONATINIB | Mast/stem cell growth factor receptor Kit | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 | ||
| P11274 | PONATINIB | Bcr/Abl fusion protein inhibitor | CHEMBL2096618 | Bcr/Abl fusion protein | Breakpoint cluster region protein | Homo sapiens | cytosolic other | Small molecule | 2012 |
| P11274 | PONATINIB | Bcr/Abl fusion protein inhibitor | CHEMBL2096618 | Bcr/Abl fusion protein | Breakpoint cluster region protein | Homo sapiens | enzyme kinase protein kinase atypical bcr | Small molecule | 2012 |
| P11274 | PONATINIB | Breakpoint cluster region protein inhibitor | CHEMBL5146 | Breakpoint cluster region protein | Breakpoint cluster region protein | Homo sapiens | cytosolic other | Small molecule | 2012 |
| P11274 | PONATINIB | Breakpoint cluster region protein inhibitor | CHEMBL5146 | Breakpoint cluster region protein | Breakpoint cluster region protein | Homo sapiens | enzyme kinase protein kinase atypical bcr | Small molecule | 2012 |
| P11362 | PONATINIB | Fibroblast growth factor receptor 1 | Fibroblast growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2012 | ||
| P16234 | PONATINIB | Platelet-derived growth factor receptor alpha | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 | ||
| P35968 | PONATINIB | Vascular endothelial growth factor receptor 2 | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 | ||
| P41240 | PONATINIB | Tyrosine-protein kinase CSK | Tyrosine-protein kinase CSK | Homo sapiens | enzyme kinase protein kinase tk csk | Small molecule | 2012 | ||
| PORACTANT ALFA | Surfactant agent | Unknown | 1999 | ||||||
| PORFIMER SODIUM | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1995 | |||
| P10613 | POSACONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2006 |
| POTASSIUM IODIDE | Unknown | Small molecule | 1979 | ||||||
| POTASSIUM SULFATE | Unknown | Small molecule | 2010 | ||||||
| P00374 | PRALATREXATE | Dihydrofolate reductase inhibitor | CHEMBL202 | Dihydrofolate reductase | Dihydrofolate reductase | Homo sapiens | enzyme reductase | Small molecule | 2009 |
| P22303 | PRALIDOXIME | Acetylcholinesterase activator | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1964 |
| P14416 | PRAMIPEXOLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P21917 | PRAMIPEXOLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P35462 | PRAMIPEXOLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P30988 | PRAMLINTIDE ACETATE | "Amylin receptor AMY1, CALCR/RAMP1 agonist" | CHEMBL2111189 | "Amylin receptor AMY1, CALCR/RAMP1" | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 2005 |
| P30988 | PRAMLINTIDE ACETATE | Amylin receptor AMY3; CALCR/RAMP3 agonist | CHEMBL2111190 | Amylin receptor AMY3; CALCR/RAMP3 | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 2005 |
| P30988 | PRAMLINTIDE ACETATE | Amylin receptor AMY2; CALCR/RAMP2 agonist | CHEMBL2364173 | Amylin receptor AMY2; CALCR/RAMP2 | Calcitonin receptor | Homo sapiens | membrane receptor 7tm2 peptide calcitonin-like calcitonin receptor | Protein | 2005 |
| PRAMOXINE | Unknown | Small molecule | 1976 | ||||||
| Q9H244 | PRASUGREL | Purinergic receptor P2Y12 antagonist | CHEMBL2001 | Purinergic receptor P2Y12 | P2Y purinoceptor 12 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor purine receptor | Small molecule | 2009 |
| P04035 | PRAVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1991 |
| P14867 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18507 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P31644 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P34903 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47869 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q8N1C3 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q99928 | PRAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q95US7 | PRAZIQUANTEL | Voltage-activated calcium channel beta 1 subunit blocker | CHEMBL2363079 | Voltage-activated calcium channel beta 1 subunit | High voltage-activated calcium channel beta subunit CavB1 | Schistosoma mansoni | auxiliary transport protein ca beta | Small molecule | 1982 |
| Q962H3 | PRAZIQUANTEL | Voltage-activated calcium channel beta 2 subunit blocker | CHEMBL2363080 | Voltage-activated calcium channel beta 2 subunit | High voltage-activated calcium channel beta subunit CavB2 | Schistosoma mansoni | auxiliary transport protein ca beta | Small molecule | 1982 |
| P25100 | PRAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1976 |
| P35348 | PRAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1976 |
| P35368 | PRAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1976 |
| P04150 | PREDNICARBATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1991 |
| P04150 | PREDNISOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1955 |
| P04150 | PREDNISOLONE ACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1955 |
| P04150 | PREDNISOLONE PHOSPHORIC ACID | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1973 |
| P04150 | PREDNISOLONE TEBUTATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1956 |
| P04150 | PREDNISONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1955 |
| P54289 | PREGABALIN | Voltage-gated calcium channel modulator | CHEMBL2363032 | Voltage-gated calcium channel | Voltage-dependent calcium channel subunit alpha-2/delta-1 | Homo sapiens | auxiliary transport protein ca alpha2delta | Small molecule | 2004 |
| P35498 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| P35499 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q01118 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q14524 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q15858 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q99250 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q9NY46 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q9UI33 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q9UQD0 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| Q9Y5Y9 | PRILOCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1965 |
| PRIMAQUINE | Unknown | Small molecule | 1952 | ||||||
| P18505 | PRIMIDONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1954 |
| P28472 | PRIMIDONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1954 |
| P35498 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| P35499 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| P47870 | PRIMIDONE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1954 |
| Q01118 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q14524 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q15858 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q99250 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9NY46 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9UI33 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9UQD0 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9Y5Y9 | PRIMIDONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q4U2R8 | PROBENECID | Solute carrier family 22 member 6 inhibitor | CHEMBL1641347 | Solute carrier family 22 member 6 | Solute carrier family 22 member 6 | Homo sapiens | transporter electrochemical slc slc22 | Small molecule | 1951 |
| Q8TCC7 | PROBENECID | Solute carrier family 22 member 8 inhibitor | CHEMBL1641348 | Solute carrier family 22 member 8 | Solute carrier family 22 member 8 | Homo sapiens | transporter electrochemical slc slc22 | Small molecule | 1951 |
| Q9NSA0 | PROBENECID | Solute carrier family 22 member 11 inhibitor | CHEMBL2073677 | Solute carrier family 22 member 11 | Solute carrier family 22 member 11 | Homo sapiens | transporter electrochemical slc slc22 | Small molecule | 1951 |
| O95477 | PROBUCOL | ATP-binding cassette sub-family A member 1 inhibitor | CHEMBL2362986 | ATP-binding cassette sub-family A member 1 | ATP-binding cassette sub-family A member 1 | Homo sapiens | transporter ntpase atp binding cassette abca | Small molecule | 1977 |
| O60939 | PROCAINAMIDE | Sodium channel subunit beta-2 | Sodium channel subunit beta-2 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1950 | ||
| P35498 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| P35499 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q01118 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q07699 | PROCAINAMIDE | Sodium channel subunit beta-1 | Sodium channel subunit beta-1 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1950 | ||
| Q14524 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q15858 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q8IWT1 | PROCAINAMIDE | Sodium channel subunit beta-4 | Sodium channel subunit beta-4 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1950 | ||
| Q99250 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9NY46 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9NY72 | PROCAINAMIDE | Sodium channel subunit beta-3 | Sodium channel subunit beta-3 | Homo sapiens | auxiliary transport protein na beta | Small molecule | 1950 | ||
| Q9UI33 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9UQD0 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9Y5Y9 | PROCAINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| P35498 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| P35499 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q01118 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q14524 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q15858 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q99250 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9NY46 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9UI33 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9UQD0 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| Q9Y5Y9 | PROCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1954 |
| PROCAINE BENZYLPENICILLIN | Unknown | Small molecule | 1948 | ||||||
| PROCARBAZINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1969 | |||
| P14416 | PROCHLORPERAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1956 |
| P35462 | PROCHLORPERAZINE | D(3) dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1956 | ||
| P11229 | PROCYCLIDINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1955 |
| P06401 | PROGESTERONE | Progesterone receptor agonist | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 1976 |
| P14416 | PROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1956 |
| P21917 | PROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1956 |
| P28223 | PROMAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1956 |
| P35462 | PROMAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1956 |
| P35367 | PROMETHAZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1951 |
| P07550 | PROPAFENONE | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 |
| P08588 | PROPAFENONE | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1989 |
| P35498 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| P35499 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q01118 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q14524 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q15858 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q99250 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9NY46 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9UI33 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9UQD0 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| Q9Y5Y9 | PROPAFENONE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1989 |
| P08172 | PROPANTHELINE | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1953 |
| P11229 | PROPANTHELINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1953 |
| P20309 | PROPANTHELINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1953 |
| P35498 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| P35499 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q01118 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q14524 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q15858 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q99250 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9NY46 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9UI33 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9UQD0 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| Q9Y5Y9 | PROPARACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1953 |
| P35367 | PROPIOMAZINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1960 |
| O00591 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| O14764 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P14867 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P18505 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P18507 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P28472 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P31644 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P34903 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P47869 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P47870 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P48169 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P78334 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| Q16445 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| Q8N1C3 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| Q99928 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| Q9UN88 | PROPOFOL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1989 |
| P35498 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35499 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q01118 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q14524 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q15858 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q99250 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9NY46 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UI33 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UQD0 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | PROPOXYCAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35372 | PROPOXYPHENE | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1957 |
| P41143 | PROPOXYPHENE | Delta-type opioid receptor | Delta-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1957 | ||
| P41145 | PROPOXYPHENE | Kappa-type opioid receptor | Kappa-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1957 | ||
| P07550 | PROPRANOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1967 |
| P08588 | PROPRANOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1967 |
| P13945 | PROPRANOLOL | Beta-3 adrenergic receptor | Beta-3 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1967 | ||
| P07202 | PROPYLTHIOURACIL | Thyroid peroxidase inhibitor | CHEMBL1839 | Thyroid peroxidase | Thyroid peroxidase | Homo sapiens | enzyme reductase | Small molecule | 1947 |
| P49895 | PROPYLTHIOURACIL | Type I iodothyronine deiodinase (Type-I 5'deiodinase) (DIOI) (Type 1 DI) (5DI) inhibitor | CHEMBL2019 | Type I iodothyronine deiodinase (Type-I 5'-deiodinase) (DIOI) (Type 1 DI) (5DI) | Type I iodothyronine deiodinase | Homo sapiens | enzyme reductase | Small molecule | 1947 |
| PROTAMINE SULFATE | Heparin inhibitor | CHEMBL2364712 | Heparin | Homo sapiens | Protein | 1969 | |||
| PROTEASE | Polypeptides hydrolytic enzyme | CHEMBL2364181 | Polypeptides | Homo sapiens | Enzyme | 1996 | |||
| P34981 | PROTIRELIN | Thyrotropin-releasing hormone receptor agonist | CHEMBL1810 | Thyrotropin-releasing hormone receptor | Thyrotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide neuropeptide receptor | Protein | 1976 |
| P07550 | PROTOKYLOL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1982 |
| P23975 | PROTRIPTYLINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1967 |
| P31645 | PROTRIPTYLINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1967 |
| PRUSSIAN BLUE INSOLUBLE | Radioactive metals chelating agent | CHEMBL2366037 | Radioactive metals | Small molecule | 2003 | ||||
| PRUSSIAN BLUE INSOLUBLE | CHEMBL2366037 | Radioactive metals | Small molecule | 2003 | |||||
| P23975 | PSEUDOEPHEDRINE | Norepinephrine transporter releasing agent | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1963 |
| P95029 | PYRAZINAMIDE | Fatty acid synthase inhibitor | CHEMBL2011 | Fatty acid synthase | 3-oxoacyl-ACP synthase | Mycobacterium tuberculosis | enzyme transferase | Small molecule | 1971 |
| P9WH43 | PYRAZINAMIDE | 70S ribosome inhibitor | CHEMBL2363965 | 70S ribosome | 30S ribosomal protein S1 | Mycobacterium tuberculosis | cytosolic other | Small molecule | 1971 |
| Q86DI9 | PYRETHRINS | Voltage-sensitive sodium channel alpha-subunit blocker | CHEMBL2362984 | Voltage-sensitive sodium channel alpha-subunit | Sodium channel protein | Pediculus humanus | ion channel vgc vg na | Small molecule | 2000 |
| P22303 | PYRIDOSTIGMINE | Acetylcholinesterase inhibitor | CHEMBL220 | Acetylcholinesterase | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1955 |
| P35367 | PYRILAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1973 |
| P13922 | PYRIMETHAMINE | Dihydrofolate reductase inhibitor | CHEMBL1939 | Dihydrofolate reductase | Bifunctional dihydrofolate reductase-thymidylate synthase | Plasmodium falciparum K1 | enzyme reductase | Small molecule | 1953 |
| PYRITHIONE | Unknown | Small molecule | 1986 | ||||||
| PYRVINIUM | Unknown | Small molecule | 1982 | ||||||
| P14867 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P18507 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P31644 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P34903 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P47869 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| Q8N1C3 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| Q99928 | QUAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1985 |
| P14416 | QUETIAPINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P28223 | QUETIAPINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1997 |
| P28335 | QUETIAPINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1997 |
| P12821 | QUINAPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1991 |
| P03372 | QUINESTROL | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1982 |
| Q92731 | QUINESTROL | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1982 |
| P55017 | QUINETHAZONE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1963 |
| P10635 | QUINIDINE | Cytochrome P450 2D6 | Cytochrome P450 2D6 | Homo sapiens | enzyme cytochrome p450 cyp_2 cyp_2d cyp_2d6 | Small molecule | 1950 | ||
| P35498 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| P35499 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q01118 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q14524 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q15858 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q99250 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9NY46 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9UI33 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9UQD0 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| Q9Y5Y9 | QUINIDINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1950 |
| P35498 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| P35499 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q01118 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q14524 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q15858 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q99250 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9NY46 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UI33 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9UQD0 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| Q9Y5Y9 | QUINIDINE POLYGALACTURONATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1982 |
| QUININE | Ferriprotoporphyrin IX inhibitor | CHEMBL613897 | Ferriprotoporphyrin IX | Plasmodium falciparum | Small molecule | 2005 | |||
| QUINUPRISTIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 1999 | ||
| P20648 | RABEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | enzyme hydrolase | Small molecule | 1999 |
| P20648 | RABEPRAZOLE | Potassium-transporting ATPase inhibitor | CHEMBL2095173 | Potassium-transporting ATPase | Potassium-transporting ATPase alpha chain 1 | Homo sapiens | transporter ntpase p-type atpase h k atpase | Small molecule | 1999 |
| RADIUM DICHLORIDE | Radiotherapy agent | Small molecule | 2013 | ||||||
| P03372 | RALOXIFENE | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1997 | ||
| Q92731 | RALOXIFENE | Estrogen receptor beta modulator | CHEMBL242 | Estrogen receptor beta | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1997 |
| P03367 | RALTEGRAVIR | Gag-Pol polyprotein | Gag-Pol polyprotein | Human immunodeficiency virus type 1 group M subtype B (isolate BRU/LAI) | Unclassified | Small molecule | 2007 | ||
| Q7ZJM1 | RALTEGRAVIR | Human immunodeficiency virus type 1 integrase inhibitor | CHEMBL3471 | Human immunodeficiency virus type 1 integrase | Integrase | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2007 |
| P48039 | RAMELTEON | Melatonin receptor agonist | CHEMBL2094268 | Melatonin receptor | Melatonin receptor type 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine-derivative melatonin receptor | Small molecule | 2005 |
| P49286 | RAMELTEON | Melatonin receptor agonist | CHEMBL2094268 | Melatonin receptor | Melatonin receptor type 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine-derivative melatonin receptor | Small molecule | 2005 |
| P12821 | RAMIPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1991 |
| P35968 | RAMUCIRUMAB | Vascular endothelial growth factor receptor 2 inhibitor | CHEMBL279 | Vascular endothelial growth factor receptor 2 | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Antibody | 2014 |
| P15692 | RANIBIZUMAB | Vascular endothelial growth factor A inhibitor | CHEMBL1783 | Vascular endothelial growth factor A | Vascular endothelial growth factor A | Homo sapiens | secreted | Antibody | 2006 |
| P25021 | RANITIDINE | Histamine H2 receptor antagonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1983 |
| P35499 | RANOLAZINE | Sodium channel protein type IV alpha subunit blocker | CHEMBL2072 | Sodium channel protein type IV alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2006 |
| Q14524 | RANOLAZINE | Sodium channel protein type V alpha subunit blocker | CHEMBL1980 | Sodium channel protein type V alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2006 |
| P02708 | RAPACURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1999 |
| P07510 | RAPACURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1999 |
| P11230 | RAPACURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1999 |
| Q04844 | RAPACURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1999 |
| Q07001 | RAPACURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1999 |
| P27338 | RASAGILINE | Monoamine oxidase B inhibitor | CHEMBL2039 | Monoamine oxidase B | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 2006 |
| RASBURICASE | Uric acid oxidative enzyme | CHEMBL2364183 | Uric acid | Homo sapiens | Enzyme | 2002 | |||
| P08913 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P18089 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P18825 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P25100 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P35348 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P35368 | RAUWOLFIA SERPENTINA | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 0 |
| P13423 | RAXIBACUMAB | Protective antigen binding agent | CHEMBL5352 | Protective antigen | Protective antigen | Bacillus anthracis | unclassified | Antibody | 2012 |
| P29274 | REGADENOSON | Adenosine A2a receptor agonist | CHEMBL251 | Adenosine A2a receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 2008 |
| P00519 | REGORAFENIB | Tyrosine-protein kinase ABL inhibitor | CHEMBL1862 | Tyrosine-protein kinase ABL | Tyrosine-protein kinase ABL1 | Homo sapiens | enzyme kinase protein kinase tk abl | Small molecule | 2012 |
| P04049 | REGORAFENIB | Serine/threonine-protein kinase RAF inhibitor | CHEMBL1906 | Serine/threonine-protein kinase RAF | RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2012 |
| P07949 | REGORAFENIB | Tyrosine-protein kinase receptor RET inhibitor | CHEMBL2041 | Tyrosine-protein kinase receptor RET | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2012 |
| P09619 | REGORAFENIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 |
| P10721 | REGORAFENIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 |
| P11362 | REGORAFENIB | Fibroblast growth factor receptor 1 inhibitor | CHEMBL3650 | Fibroblast growth factor receptor 1 | Fibroblast growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2012 |
| P15056 | REGORAFENIB | Serine/threonine-protein kinase B-raf inhibitor | CHEMBL5145 | Serine/threonine-protein kinase B-raf | Serine/threonine-protein kinase B-raf | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2012 |
| P16234 | REGORAFENIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2012 |
| P17948 | REGORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P21802 | REGORAFENIB | Fibroblast growth factor receptor 2 inhibitor | CHEMBL4142 | Fibroblast growth factor receptor 2 | Fibroblast growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk fgfr | Small molecule | 2012 |
| P35916 | REGORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P35968 | REGORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2012 |
| P42685 | REGORAFENIB | Tyrosine-protein kinase FRK inhibitor | CHEMBL4223 | Tyrosine-protein kinase FRK | Tyrosine-protein kinase FRK | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2012 |
| Q02763 | REGORAFENIB | Tyrosine-protein kinase TIE-2 inhibitor | CHEMBL4128 | Tyrosine-protein kinase TIE-2 | Angiopoietin-1 receptor | Homo sapiens | enzyme kinase protein kinase tk tie | Small molecule | 2012 |
| Q15759 | REGORAFENIB | MAP kinase p38 beta inhibitor | CHEMBL3961 | MAP kinase p38 beta | Mitogen-activated protein kinase 11 | Homo sapiens | enzyme kinase protein kinase cmgc mapk p38 | Small molecule | 2012 |
| Q16832 | REGORAFENIB | Discoidin domain-containing receptor 2 inhibitor | CHEMBL5122 | Discoidin domain-containing receptor 2 | Discoidin domain-containing receptor 2 | Homo sapiens | enzyme kinase protein kinase tk ddr | Small molecule | 2012 |
| P35372 | REMIFENTANIL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1996 |
| Q09428 | REPAGLINIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1997 |
| Q14654 | REPAGLINIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1997 |
| Q05940 | RESCINNAMINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 1956 |
| Q05940 | RESERPINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 1960 |
| Q2FW06 | RETAPAMULIN | 70S ribosome inhibitor | CHEMBL2364096 | 70S ribosome | 50S ribosomal protein L3 | Staphylococcus aureus | cytosolic other | Small molecule | 2007 |
| Q9A1X4 | RETAPAMULIN | 70S ribosome inhibitor | CHEMBL2364103 | 70S ribosome | 50S ribosomal protein L3 | Streptococcus pyogenes | cytosolic other | Small molecule | 2007 |
| P00747 | RETEPLASE | Plasminogen activator | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Enzyme | 1996 |
| P20839 | RIBAVIRIN | Inosine-5'-monophosphate dehydrogenase 1 inhibitor | CHEMBL1822 | Inosine-5'-monophosphate dehydrogenase 1 | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1985 |
| Q8JXU8 | RIBAVIRIN | RNA inhibitor | CHEMBL2363073 | RNA | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 1985 |
| Q8JXU8 | RIBAVIRIN | Hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor | CHEMBL5375 | Hepatitis C virus NS5B RNA-dependent RNA polymerase | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 1985 |
| RIBAVIRIN | RNA inhibitor | CHEMBL2363073 | RNA | Hepatitis C virus | Small molecule | 1985 | |||
| RIBOFLAVIN 5'-PHOSPHATE | Unknown | Small molecule | 1985 | ||||||
| P0A8T7 | RIFABUTIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta' | Bacteria | enzyme transferase | Small molecule | 1992 |
| P0A8V2 | RIFABUTIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta | Bacteria | enzyme transferase | Small molecule | 1992 |
| P0A8T7 | RIFAMPICIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta' | Bacteria | enzyme transferase | Small molecule | 1971 |
| P0A8V2 | RIFAMPICIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta | Bacteria | enzyme transferase | Small molecule | 1971 |
| P0A8T7 | RIFAPENTINE | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta' | Bacteria | enzyme transferase | Small molecule | 1998 |
| P0A8V2 | RIFAPENTINE | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta | Bacteria | enzyme transferase | Small molecule | 1998 |
| P0A8T7 | RIFAXIMIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta' | Bacteria | enzyme transferase | Small molecule | 2004 |
| P0A8V2 | RIFAXIMIN | Bacterial DNA-directed RNA polymerase inhibitor | CHEMBL2364672 | Bacterial DNA-directed RNA polymerase | DNA-directed RNA polymerase subunit beta | Bacteria | enzyme transferase | Small molecule | 2004 |
| P01584 | RILONACEPT | Interleukin-1 beta inhibitor | CHEMBL1909490 | Interleukin-1 beta | Interleukin-1 beta | Homo sapiens | secreted | Protein | 2008 |
| Q72547 | RILPIVIRINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2011 |
| P35498 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| P35499 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q01118 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q14524 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q15858 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q99250 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q9NY46 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q9UI33 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q9UQD0 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| Q9Y5Y9 | RILUZOLE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1995 |
| P63231 | RIMANTADINE | Influenza virus A matrix protein M2 inhibitor | CHEMBL2052 | Influenza virus A matrix protein M2 | Matrix protein 2 | Influenza A virus (A/Udorn/307/1972(H3N2)) | ion channel other misc m2-c | Small molecule | 1993 |
| P04150 | RIMEXOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1994 |
| O75343 | RIOCIGUAT | Soluble guanylate cyclase positive allosteric modulator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 2013 |
| P33402 | RIOCIGUAT | Soluble guanylate cyclase positive allosteric modulator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit alpha-2 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 2013 |
| Q02108 | RIOCIGUAT | Soluble guanylate cyclase positive allosteric modulator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit alpha-3 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 2013 |
| Q02153 | RIOCIGUAT | Soluble guanylate cyclase positive allosteric modulator | CHEMBL2111348 | Soluble guanylate cyclase | Guanylate cyclase soluble subunit beta-1 | Homo sapiens | enzyme lyase guanylate cyclase soluble guanylate cyclase | Small molecule | 2013 |
| P14324 | RISEDRONIC ACID | Farnesyl diphosphate synthase inhibitor | CHEMBL1782 | Farnesyl diphosphate synthase | Farnesyl pyrophosphate synthase | Homo sapiens | enzyme transferase | Small molecule | 1998 |
| P14416 | RISPERIDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1993 |
| P28221 | RISPERIDONE | 5-hydroxytryptamine receptor 1D | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1993 | ||
| P28222 | RISPERIDONE | 5-hydroxytryptamine receptor 1B | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1993 | ||
| P28223 | RISPERIDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1993 |
| P28335 | RISPERIDONE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1993 |
| P07550 | RITODRINE | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1991 |
| Q72874 | RITONAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 1996 |
| P11836 | RITUXIMAB | B-lymphocyte antigen CD20 inhibitor | CHEMBL2058 | B-lymphocyte antigen CD20 | B-lymphocyte antigen CD20 | Homo sapiens | ion channel other misc cd20 | Antibody | 1997 |
| P00742 | RIVAROXABAN | Coagulation factor X inhibitor | CHEMBL244 | Coagulation factor X | Coagulation factor X | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 2011 |
| P06276 | RIVASTIGMINE | Cholinesterases; ACHE & BCHE inhibitor | CHEMBL2095233 | Cholinesterases; ACHE & BCHE | Cholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 2000 |
| P22303 | RIVASTIGMINE | Cholinesterases; ACHE & BCHE inhibitor | CHEMBL2095233 | Cholinesterases; ACHE & BCHE | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 2000 |
| P28221 | RIZATRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1998 |
| P28222 | RIZATRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1998 |
| P02708 | ROCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1994 |
| P07510 | ROCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1994 |
| P11230 | ROCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1994 |
| Q04844 | ROCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1994 |
| Q07001 | ROCURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1994 |
| P35354 | ROFECOXIB | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1999 |
| P27815 | ROFLUMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 2011 |
| Q07343 | ROFLUMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 2011 |
| Q08493 | ROFLUMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 2011 |
| Q08499 | ROFLUMILAST | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 2011 |
| O15379 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 3 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2009 |
| P56524 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 4 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2009 |
| Q13547 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 1 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2009 |
| Q8WUI4 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 7 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2009 |
| Q92769 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 2 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2009 |
| Q969S8 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 10 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2009 |
| Q96DB2 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 11 | Homo sapiens | epigenetic regulator eraser hdac hdac class iv | Small molecule | 2009 |
| Q9BY41 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 8 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2009 |
| Q9UBN7 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 6 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2009 |
| Q9UKV0 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 9 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2009 |
| Q9UQL6 | ROMIDEPSIN | Histone deacetylase inhibitor | CHEMBL2093865 | Histone deacetylase | Histone deacetylase 5 | Homo sapiens | epigenetic regulator eraser hdac hdac class iia | Small molecule | 2009 |
| P40238 | ROMIPLOSTIM | Thrombopoietin receptor agonist | CHEMBL1864 | Thrombopoietin receptor | Thrombopoietin receptor | Homo sapiens | membrane receptor | Protein | 2008 |
| P14416 | ROPINIROLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P21917 | ROPINIROLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P35462 | ROPINIROLE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1997 |
| P35498 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| P35499 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q01118 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q14524 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q15858 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q99250 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9NY46 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UI33 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UQD0 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9Y5Y9 | ROPIVACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| P37231 | ROSIGLITAZONE | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 1999 |
| P04035 | ROSUVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 2003 |
| P14416 | ROTIGOTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2007 |
| P21917 | ROTIGOTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2007 |
| P35462 | ROTIGOTINE | D2-like dopamine receptor agonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2007 |
| P35498 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| P35499 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q01118 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q14524 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q15858 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q99250 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9NY46 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9UI33 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9UQD0 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| Q9Y5Y9 | RUFINAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2008 |
| O60674 | RUXOLITINIB | Tyrosine-protein kinase JAK2 inhibitor | CHEMBL2971 | Tyrosine-protein kinase JAK2 | Tyrosine-protein kinase JAK2 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2011 |
| O60674 | RUXOLITINIB | Tyrosine-protein kinase JAK2 inhibitor | CHEMBL2971 | Tyrosine-protein kinase JAK2 | Tyrosine-protein kinase JAK2 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2011 |
| P23458 | RUXOLITINIB | Tyrosine-protein kinase JAK1 inhibitor | CHEMBL2835 | Tyrosine-protein kinase JAK1 | Tyrosine-protein kinase JAK1 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2011 |
| P23458 | RUXOLITINIB | Tyrosine-protein kinase JAK1 inhibitor | CHEMBL2835 | Tyrosine-protein kinase JAK1 | Tyrosine-protein kinase JAK1 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2011 |
| SACROSIDASE | Sucrose hydrolytic enzyme | CHEMBL2364182 | Sucrose | Homo sapiens | Enzyme | 1998 | |||
| P08473 | SACUBITRIL | Neprilysin inhibitor | CHEMBL1944 | Neprilysin | Neprilysin | Homo sapiens | enzyme protease metallo mae m13 | Small molecule | 2015 |
| P07550 | SALMETEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1994 |
| SAMARIUM(II) LEXIDRONAM | Unknown | Small molecule | 1997 | ||||||
| P00439 | SAPROPTERIN | Phenylalanine-4-hydroxylase activator | CHEMBL3076 | Phenylalanine-4-hydroxylase | Phenylalanine-4-hydroxylase | Homo sapiens | enzyme reductase | Small molecule | 2007 |
| Q72874 | SAQUINAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 1995 |
| P30556 | SARALASIN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Protein | 1982 |
| P15509 | SARGRAMOSTIM | Granulocyte-macrophage colony-stimulating factor receptor agonist | CHEMBL2364169 | Granulocyte-macrophage colony-stimulating factor receptor | Granulocyte-macrophage colony-stimulating factor receptor subunit alpha | Homo sapiens | membrane receptor | Protein | 1991 |
| P27487 | SAXAGLIPTIN | Dipeptidyl peptidase IV inhibitor | CHEMBL284 | Dipeptidyl peptidase IV | Dipeptidyl peptidase 4 | Homo sapiens | enzyme protease serine sc s9b | Small molecule | 2009 |
| P11229 | SCOPOLAMINE | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1979 |
| P18505 | SECOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1950 |
| P28472 | SECOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1950 |
| P47870 | SECOBARBITAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1950 |
| P47872 | SECRETIN | Secretin receptor agonist | CHEMBL1925 | Secretin receptor | Secretin receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like secretin receptor | Protein | 2002 |
| P47872 | SECRETIN SYNTHETIC HUMAN | Secretin receptor agonist | CHEMBL1925 | Secretin receptor | Secretin receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like secretin receptor | Protein | 2004 |
| P47872 | SECRETIN SYNTHETIC PORCINE | Secretin receptor agonist | CHEMBL1925 | Secretin receptor | Secretin receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like secretin receptor | Protein | 2002 |
| Q16552 | SECUKINUMAB | Interleukin 17A inhibitor | CHEMBL3390822 | Interleukin 17A | Homo sapiens | secreted | Antibody | 2015 | |
| P27338 | SELEGILINE | Monoamine oxidase B inhibitor | CHEMBL2039 | Monoamine oxidase B | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 1989 |
| SELENIUM SULFIDE | Unknown | Small molecule | 1951 | ||||||
| Q01718 | SERACTIDE ACETATE | Melanocortin receptor 2 agonist | CHEMBL1965 | Melanocortin receptor 2 | Adrenocorticotropic hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide melanocortin receptor | Protein | 1978 |
| Q02643 | SERMORELIN ACETATE | Growth hormone-releasing hormone receptor agonist | CHEMBL2032 | Growth hormone-releasing hormone receptor | Growth hormone-releasing hormone receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like growth hormone-releasing hormone receptor | Protein | 1990 |
| P10613 | SERTACONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2003 |
| P31645 | SERTRALINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1991 |
| SEVELAMER | Unknown | Small molecule | 2007 | ||||||
| SEVELAMER HYDROCHLORIDE | Phosphate chelating agent | CHEMBL2364184 | Phosphate | Homo sapiens | Small molecule | 1998 | |||
| O00591 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| O14649 | SEVOFLURANE | Potassium channel subfamily K member 3 opener | CHEMBL2321613 | Potassium channel subfamily K member 3 | Potassium channel subfamily K member 3 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1995 |
| O14764 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| O95069 | SEVOFLURANE | Potassium channel subfamily K member 2 opener | CHEMBL2321615 | Potassium channel subfamily K member 2 | Potassium channel subfamily K member 2 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1995 |
| P14867 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P18505 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P18507 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P23415 | SEVOFLURANE | Glycine receptor (alpha-1/beta) positive modulator | CHEMBL2363052 | Glycine receptor (alpha-1/beta) | Glycine receptor subunit alpha-1 | Homo sapiens | ion channel lgic gly | Small molecule | 1995 |
| P28472 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P31644 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P34903 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P47869 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P47870 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P48169 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P57789 | SEVOFLURANE | Potassium channel subfamily K member 10 opener | CHEMBL2331041 | Potassium channel subfamily K member 10 | Potassium channel subfamily K member 10 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1995 |
| P78334 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| Q16445 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| Q7Z418 | SEVOFLURANE | Potassium channel subfamily K member 18 opener | CHEMBL2331042 | Potassium channel subfamily K member 18 | Potassium channel subfamily K member 18 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1995 |
| Q8N1C3 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| Q99928 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| Q9NPC2 | SEVOFLURANE | Potassium channel subfamily K member 9 opener | CHEMBL2321614 | Potassium channel subfamily K member 9 | Potassium channel subfamily K member 9 | Homo sapiens | ion channel vgc k k2p | Small molecule | 1995 |
| Q9UN88 | SEVOFLURANE | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1995 |
| P23975 | SIBUTRAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1997 |
| P31645 | SIBUTRAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1997 |
| Q01959 | SIBUTRAMINE | Monoamine transporter inhibitor | CHEMBL2363064 | Monoamine transporter | Sodium-dependent dopamine transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1997 |
| O76074 | SILDENAFIL | Phosphodiesterase 5A inhibitor | CHEMBL1827 | Phosphodiesterase 5A | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 1998 |
| P35348 | SILODOSIN | Alpha-1a adrenergic receptor antagonist | CHEMBL229 | Alpha-1a adrenergic receptor | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2008 |
| P05231 | SILTUXIMAB | Interleukin-6 inhibitor | CHEMBL1795129 | Interleukin-6 | Interleukin-6 | Homo sapiens | secreted | Antibody | 2014 |
| A3EZI9 | SIMEPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | NS3 | Hepatitis C virus | enzyme protease serine pas s29 | Small molecule | 2013 |
| D2K2A8 | SIMEPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | Non-structural protein 4A | Hepatitis C virus | enzyme protease serine pas s29 reg | Small molecule | 2013 |
| SIMETHICONE | Antifoaming agent | Small molecule | 1996 | ||||||
| P04035 | SIMVASTATIN | HMG-CoA reductase inhibitor | CHEMBL402 | HMG-CoA reductase | 3-hydroxy-3-methylglutaryl-coenzyme A reductase | Homo sapiens | enzyme reductase | Small molecule | 1991 |
| SINECATECHINS | Unknown | Unknown | 2006 | ||||||
| P62942 | SIROLIMUS | FK506-binding protein 1A inhibitor | CHEMBL1902 | FK506-binding protein 1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Small molecule | 1999 |
| P27487 | SITAGLIPTIN | Dipeptidyl peptidase IV inhibitor | CHEMBL284 | Dipeptidyl peptidase IV | Dipeptidyl peptidase 4 | Homo sapiens | enzyme protease serine sc s9b | Small molecule | 2006 |
| SODIUM BENZOATE | Unknown | Small molecule | 1987 | ||||||
| SODIUM PHENYLACETATE | Glutamine chelating agent | CHEMBL2366039 | Glutamine | Homo sapiens | Small molecule | 1987 | |||
| SODIUM PHOSPHATE | Unknown | Small molecule | 1957 | ||||||
| Q8JXU8 | SOFOSBUVIR | Hepatitis C virus NS5B RNA-dependent RNA polymerase inhibitor | CHEMBL5375 | Hepatitis C virus NS5B RNA-dependent RNA polymerase | NS5B protein | Hepatitis C virus | enzyme transferase | Small molecule | 2013 |
| P08172 | SOLIFENACIN | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| P20309 | SOLIFENACIN | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| P10912 | SOMATREM | Growth hormone receptor agonist | CHEMBL1976 | Growth hormone receptor | Growth hormone receptor | Homo sapiens | membrane receptor | Protein | 1985 |
| P10912 | SOMATROPIN | Growth hormone receptor agonist | CHEMBL1976 | Growth hormone receptor | Growth hormone receptor | Homo sapiens | membrane receptor | Protein | 1976 |
| P04049 | SORAFENIB | Serine/threonine-protein kinase RAF inhibitor | CHEMBL1906 | Serine/threonine-protein kinase RAF | RAF proto-oncogene serine/threonine-protein kinase | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2005 |
| P07949 | SORAFENIB | Tyrosine-protein kinase receptor RET inhibitor | CHEMBL2041 | Tyrosine-protein kinase receptor RET | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2005 |
| P09619 | SORAFENIB | Platelet-derived growth factor receptor beta inhibitor | CHEMBL1913 | Platelet-derived growth factor receptor beta | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2005 |
| P10721 | SORAFENIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2005 |
| P15056 | SORAFENIB | Serine/threonine-protein kinase B-raf inhibitor | CHEMBL5145 | Serine/threonine-protein kinase B-raf | Serine/threonine-protein kinase B-raf | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2005 |
| P17948 | SORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2005 |
| P35916 | SORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2005 |
| P35968 | SORAFENIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2005 |
| P36888 | SORAFENIB | Tyrosine-protein kinase receptor FLT3 inhibitor | CHEMBL1974 | Tyrosine-protein kinase receptor FLT3 | Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2005 |
| P07550 | SOTALOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1992 |
| P08588 | SOTALOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1992 |
| Q12809 | SOTALOL | HERG blocker | CHEMBL240 | HERG | Potassium voltage-gated channel subfamily H member 2 | Homo sapiens | ion channel vgc k vg k | Small molecule | 1992 |
| P0AES4 | SPARFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1996 |
| P0AES6 | SPARFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1996 |
| P0AFI2 | SPARFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 1996 |
| P20083 | SPARFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 1996 |
| SPECTINOMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1971 | ||
| E0VB18 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "Acetylcholine receptor protein alpha 1, 2, 3, 4 invertebrate, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| E0VB20 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "Acetylcholine receptor protein alpha 1, 2, 3, 4 invertebrate, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| E0VDF4 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "Acetylcholine receptor protein alpha 1, 2, 3, 4 invertebrate, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| E0VDF5 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "Acetylcholine receptor protein subunit alpha-L1, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| E0VDF7 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "Acetylcholine receptor protein alpha 1, 2, 3, 4 invertebrate, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| E0VP62 | SPINOSAD | Nicotinic acetylcholine receptor agonist | CHEMBL2364023 | Nicotinic acetylcholine receptor | "DrosGluCl, putative" | Pediculus humanus capitis | ion channel lgic | Small molecule | 2011 |
| P12821 | SPIRAPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1994 |
| P08235 | SPIRONOLACTONE | Mineralocorticoid receptor antagonist | CHEMBL1994 | Mineralocorticoid receptor | Mineralocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c2 | Small molecule | 1960 |
| P10275 | STANOZOLOL | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1962 |
| Q72547 | STAVUDINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1994 |
| P00747 | STREPTOKINASE | Plasminogen activator | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Enzyme | 1997 |
| STREPTOMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1946 | ||
| STREPTOZOTOCIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1982 | |||
| STRONTIUM CHLORIDE | Unknown | Small molecule | 1993 | ||||||
| SUCCIMER | Lead chelating agent | CHEMBL2364029 | Lead | null | Small molecule | 1991 | |||
| SUCCIMER | CHEMBL2364029 | Lead | Small molecule | 1991 | |||||
| SUCROFERRIC OXYHYDROXIDE | Phosphate chelating agent | CHEMBL2364184 | Phosphate | Homo sapiens | Unknown | 2013 | |||
| P35372 | SUFENTANIL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1984 |
| P62593 | SULBACTAM | Bacterial beta-lactamase TEM inhibitor | CHEMBL2364670 | Bacterial beta-lactamase TEM | Beta-lactamase TEM | Bacteria | enzyme hydrolase | Small molecule | 1986 |
| P10613 | SULCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1985 |
| SULFABENZAMIDE | Unknown | Small molecule | 1945 | ||||||
| P0AC13 | SULFACETAMIDE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1945 |
| Q25704 | SULFACYTINE | Dihydropteroate synthetase inhibitor | CHEMBL2013 | Dihydropteroate synthetase | "7,8-dihydro-6-hydroxymethylpterin pyrophosphokinase-dihydropteroate synthase" | Plasmodium falciparum | enzyme transferase | Small molecule | 1975 |
| P0AC13 | SULFADIAZINE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1941 |
| Q25704 | SULFADOXINE | Dihydropteroate synthetase inhibitor | CHEMBL2013 | Dihydropteroate synthetase | "7,8-dihydro-6-hydroxymethylpterin pyrophosphokinase-dihydropteroate synthase" | Plasmodium falciparum | enzyme transferase | Small molecule | 1981 |
| P0AC13 | SULFALENE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 0 |
| P0AC13 | SULFAMERAZINE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1982 |
| P0AC13 | SULFAMETER | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1966 |
| P0AC13 | SULFAMETHAZINE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1949 |
| P0AC13 | SULFAMETHIZOLE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1953 |
| P0AC13 | SULFAMETHOXAZOLE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1973 |
| P0AC13 | SULFANILAMIDE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1985 |
| P0AC13 | SULFAPHENAZOLE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1982 |
| P0AC13 | SULFAPYRIDINE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1939 |
| P09917 | SULFASALAZINE | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P23219 | SULFASALAZINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P35354 | SULFASALAZINE | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1950 |
| P0AC13 | SULFATHIAZOLE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1945 |
| Q96S37 | SULFINPYRAZONE | Solute carrier family 22 member 12 inhibitor | CHEMBL6120 | Solute carrier family 22 member 12 | Solute carrier family 22 member 12 | Homo sapiens | transporter electrochemical slc slc22 | Small molecule | 1959 |
| P0AC13 | SULFISOXAZOLE | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1971 |
| P0AC13 | SULFISOXAZOLE ACETYL | Bacterial dihydropteroate synthase inhibitor | CHEMBL2364668 | Bacterial dihydropteroate synthase | Dihydropteroate synthase | Bacteria | enzyme transferase | Small molecule | 1953 |
| P0C0X1 | SULFOXONE | Dihydropteroate synthase 1 inhibitor | CHEMBL2362993 | Dihydropteroate synthase 1 | Dihydropteroate synthase 1 | Mycobacterium leprae (strain TN) | enzyme transferase | Small molecule | 1982 |
| P23219 | SULINDAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1978 |
| P35354 | SULINDAC | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1978 |
| P28221 | SUMATRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1992 |
| P28222 | SUMATRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1992 |
| P07333 | SUNITINIB | Macrophage colony stimulating factor receptor inhibitor | CHEMBL1844 | Macrophage colony stimulating factor receptor | Macrophage colony-stimulating factor 1 receptor | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P07949 | SUNITINIB | Tyrosine-protein kinase receptor RET inhibitor | CHEMBL2041 | Tyrosine-protein kinase receptor RET | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2006 |
| P09619 | SUNITINIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor beta | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P10721 | SUNITINIB | Stem cell growth factor receptor inhibitor | CHEMBL1936 | Stem cell growth factor receptor | Mast/stem cell growth factor receptor Kit | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P16234 | SUNITINIB | Platelet-derived growth factor receptor inhibitor | CHEMBL2095189 | Platelet-derived growth factor receptor | Platelet-derived growth factor receptor alpha | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P17948 | SUNITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2006 |
| P35916 | SUNITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2006 |
| P35968 | SUNITINIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2006 |
| P36888 | SUNITINIB | Tyrosine-protein kinase receptor FLT3 inhibitor | CHEMBL1974 | Tyrosine-protein kinase receptor FLT3 | Receptor-type tyrosine-protein kinase FLT3 | Homo sapiens | enzyme kinase protein kinase tk pdgfr | Small molecule | 2006 |
| P23219 | SUPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1988 |
| P35354 | SUPROFEN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1988 |
| O43613 | SUVOREXANT | Orexin receptor antagonist | CHEMBL3307226 | Orexin receptor | Orexin receptor type 1 | Homo sapiens | membrane receptor 7tm1 peptide short peptide orexin receptor | Small molecule | 2014 |
| O43614 | SUVOREXANT | Orexin receptor antagonist | CHEMBL3307226 | Orexin receptor | Orexin receptor type 2 | Homo sapiens | membrane receptor 7tm1 peptide short peptide orexin receptor | Small molecule | 2014 |
| P02708 | SUXAMETHONIUM | Muscle-type nicotinic acetylcholine receptor agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1952 |
| P07510 | SUXAMETHONIUM | Muscle-type nicotinic acetylcholine receptor agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1952 |
| P11230 | SUXAMETHONIUM | Muscle-type nicotinic acetylcholine receptor agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1952 |
| Q04844 | SUXAMETHONIUM | Muscle-type nicotinic acetylcholine receptor agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1952 |
| Q07001 | SUXAMETHONIUM | Muscle-type nicotinic acetylcholine receptor agonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1952 |
| P03372 | "SYNTHETIC CONJUGATED ESTROGENS, B" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 2004 |
| Q92731 | "SYNTHETIC CONJUGATED ESTROGENS, B" | Estrogen receptor agonist | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 2004 |
| P0DJD9 | Sucralfate | Glycoproteins cross-linking agent | CHEMBL2363054 | Glycoproteins | Pepsin A-5 | Homo sapiens | enzyme protease aspartic aa a1a | Unknown | 1981 |
| P0DJD9 | Sucralfate | Pepsin A inhibitor | CHEMBL3295 | Pepsin A | Pepsin A-5 | Homo sapiens | enzyme protease aspartic aa a1a | Unknown | 1981 |
| Sucralfate | Glycoproteins cross-linking agent | CHEMBL2363054 | Glycoproteins | Homo sapiens | Unknown | 1981 | |||
| P06276 | TACRINE | Cholinesterases; ACHE & BCHE inhibitor | CHEMBL2095233 | Cholinesterases; ACHE & BCHE | Cholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1993 |
| P22303 | TACRINE | Cholinesterases; ACHE & BCHE inhibitor | CHEMBL2095233 | Cholinesterases; ACHE & BCHE | Acetylcholinesterase | Homo sapiens | enzyme hydrolase | Small molecule | 1993 |
| P62942 | TACROLIMUS | FK506-binding protein 1A inhibitor | CHEMBL1902 | FK506-binding protein 1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Small molecule | 1994 |
| O76074 | TADALAFIL | Phosphodiesterase 5A inhibitor | CHEMBL1827 | Phosphodiesterase 5A | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 2003 |
| P43088 | TAFLUPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 2012 |
| P18505 | TALBUTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | TALBUTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | TALBUTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| TALIGLUCERASE ALFA | Glucocerebroside hydrolytic enzyme | CHEMBL2364176 | Glucocerebroside | Homo sapiens | Enzyme | 2012 | |||
| P03372 | TAMOXIFEN | Estrogen receptor alpha modulator | CHEMBL206 | Estrogen receptor alpha | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1977 |
| P25100 | TAMSULOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1997 |
| P35348 | TAMSULOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1997 |
| P35368 | TAMSULOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1997 |
| P23975 | TAPENTADOL | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2008 |
| P35372 | TAPENTADOL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 2008 |
| P48039 | TASIMELTEON | Melatonin receptor agonist | CHEMBL2094268 | Melatonin receptor | Melatonin receptor type 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine-derivative melatonin receptor | Small molecule | 2014 |
| P49286 | TASIMELTEON | Melatonin receptor agonist | CHEMBL2094268 | Melatonin receptor | Melatonin receptor type 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine-derivative melatonin receptor | Small molecule | 2014 |
| F2SF18 | TAVABOROLE | Leucine-tRNA ligase inhibitor | CHEMBL3307222 | Leucine-tRNA ligase | Leucine-tRNA ligase | Trichophyton rubrum (strain ATCC MYA-4607 / CBS 118892) (Athlete'sfoot fungus) | unclassified | Small molecule | 2014 |
| P10276 | TAZAROTENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1997 |
| P10826 | TAZAROTENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1997 |
| P13631 | TAZAROTENE | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1997 |
| P62593 | TAZOBACTAM | Bacterial beta-lactamase TEM inhibitor | CHEMBL2364670 | Bacterial beta-lactamase TEM | Beta-lactamase TEM | Bacteria | enzyme hydrolase | Small molecule | 1993 |
| TEDIZOLID PHOSPHATE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 2014 | ||
| O95838 | TEDUGLUTIDE | Glucagon-like peptide 2 receptor agonist | CHEMBL5844 | Glucagon-like peptide 2 receptor | Glucagon-like peptide 2 receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like glucagon-like peptide receptor | Protein | 2012 |
| Q13639 | TEGASEROD | Serotonin 4 (5-HT4) receptor partial agonist | CHEMBL1875 | Serotonin 4 (5-HT4) receptor | 5-hydroxytryptamine receptor 4 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2002 |
| A3EZI9 | TELAPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | NS3 | Hepatitis C virus | enzyme protease serine pas s29 | Protein | 2011 |
| D2K2A8 | TELAPREVIR | "Hepatitis C virus serine protease, NS3/NS4A inhibitor" | CHEMBL2095231 | "Hepatitis C virus serine protease, NS3/NS4A" | Non-structural protein 4A | Hepatitis C virus | enzyme protease serine pas s29 reg | Protein | 2011 |
| TELAVANCIN | Cell outer membrane inhibitor | CHEMBL2364032 | Cell outer membrane | Bacteria | Small molecule | 2009 | |||
| Q67889 | TELBIVUDINE | Protein P | Protein P | Hepatitis B virus | Unclassified | Small molecule | 2006 | ||
| Q9IF40 | TELBIVUDINE | DNA polymerase/reverse transcriptase inhibitor | CHEMBL2362994 | DNA polymerase/reverse transcriptase | Protein P | Hepatitis B virus | enzyme transferase | Small molecule | 2006 |
| TELITHROMYCIN | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 23S ribosomal RNA | Bacteria | Small molecule | 2004 | ||
| P30556 | TELMISARTAN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1998 |
| P14867 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P18507 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P31644 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P34903 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| P47869 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q8N1C3 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| Q99928 | TEMAZEPAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1981 |
| TEMOZOLOMIDE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1999 | |||
| P62942 | TEMSIROLIMUS | FK506-binding protein 1A inhibitor | CHEMBL1902 | FK506-binding protein 1A | Peptidyl-prolyl cis-trans isomerase FKBP1A | Homo sapiens | enzyme isomerase | Small molecule | 2007 |
| P00747 | TENECTEPLASE | Plasminogen activator | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Enzyme | 2000 |
| P11388 | TENIPOSIDE | DNA topoisomerase II inhibitor | CHEMBL2094255 | DNA topoisomerase II | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1992 |
| Q02880 | TENIPOSIDE | DNA topoisomerase II inhibitor | CHEMBL2094255 | DNA topoisomerase II | DNA topoisomerase 2-beta | Homo sapiens | enzyme isomerase | Small molecule | 1992 |
| Q72547 | TENOFOVIR DISOPROXIL | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 2001 |
| P25100 | TERAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P35348 | TERAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| P35368 | TERAZOSIN | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1987 |
| Q4JEY0 | TERBINAFINE | Squalene monooxygenase inhibitor | CHEMBL2364679 | Squalene monooxygenase | Squalene epoxidase | Trichophyton | enzyme reductase | Small molecule | 1992 |
| P07550 | TERBUTALINE | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1974 |
| P10613 | TERCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1987 |
| Q02127 | TERIFLUNOMIDE | Dihydroorotate dehydrogenase inhibitor | CHEMBL1966 | Dihydroorotate dehydrogenase | "Dihydroorotate dehydrogenase (quinone), mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 2012 |
| Q03431 | TERIPARATIDE | Parathyroid hormone receptor agonist | CHEMBL1793 | Parathyroid hormone receptor | Parathyroid hormone/parathyroid hormone-related peptide receptor | Homo sapiens | membrane receptor 7tm2 peptide parathyroid hormone receptor parathyroid hormone receptor | Protein | 2002 |
| Q03431 | TERIPARATIDE ACETATE | Parathyroid hormone receptor agonist | CHEMBL1793 | Parathyroid hormone receptor | Parathyroid hormone/parathyroid hormone-related peptide receptor | Homo sapiens | membrane receptor 7tm2 peptide parathyroid hormone receptor parathyroid hormone receptor | Protein | 1987 |
| Q02643 | TESAMORELIN | Growth hormone-releasing hormone receptor agonist | CHEMBL2032 | Growth hormone-releasing hormone receptor | Growth hormone-releasing hormone receptor | Homo sapiens | membrane receptor 7tm2 peptide glucagon-like growth hormone-releasing hormone receptor | Protein | 2010 |
| P11511 | TESTOLACTONE | Cytochrome P450 19A1 inhibitor | CHEMBL1978 | Cytochrome P450 19A1 | Aromatase | Homo sapiens | enzyme cytochrome p450 cyp_19 cyp_19a cyp_19a1 | Small molecule | 1969 |
| P10275 | TESTOSTERONE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1972 |
| P10275 | TESTOSTERONE CYPIONATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1978 |
| P10275 | TESTOSTERONE ENANTHATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1953 |
| P10275 | TESTOSTERONE PROPIONATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 1974 |
| P10275 | TESTOSTERONE UNDECANOATE | Androgen Receptor agonist | CHEMBL1871 | Androgen Receptor | Androgen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c4 | Small molecule | 2014 |
| Q05940 | TETRABENAZINE | Synaptic vesicular amine transporter inhibitor | CHEMBL1893 | Synaptic vesicular amine transporter | Synaptic vesicular amine transporter | Homo sapiens | transporter electrochemical slc slc18 | Small molecule | 2008 |
| P35498 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| P35499 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q01118 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q14524 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q15858 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q99250 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q9NY46 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q9UI33 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q9UQD0 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| Q9Y5Y9 | TETRACAINE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2005 |
| TETRACYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 1953 | ||
| TETRADECYL SULFURIC ACID | Unknown | Small molecule | 1946 | ||||||
| P08913 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P18089 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P18825 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P25100 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P35348 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P35368 | TETRAHYDROZOLINE | Adrenergic receptor alpha agonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| Q96SW2 | THALIDOMIDE | Protein cereblon | Protein cereblon | Homo sapiens | Unclassified | Small molecule | 1998 | ||
| THALIDOMIDE | Unknown | Small molecule | 1998 | ||||||
| P0DMS8 | THEOPHYLLINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A3 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1940 |
| P27815 | THEOPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1940 |
| P29274 | THEOPHYLLINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1940 |
| P29275 | THEOPHYLLINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2b | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1940 |
| P30542 | THEOPHYLLINE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A1 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1940 |
| Q07343 | THEOPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1940 |
| Q08493 | THEOPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1940 |
| Q08499 | THEOPHYLLINE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1940 |
| Q13370 | THEOPHYLLINE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase B" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3b | Small molecule | 1940 |
| Q14432 | THEOPHYLLINE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1940 |
| P0DMS8 | THEOPHYLLINE GLYCINATE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A3 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1982 |
| P27815 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4A" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4a | Small molecule | 1982 |
| P29274 | THEOPHYLLINE GLYCINATE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2a | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1982 |
| P29275 | THEOPHYLLINE GLYCINATE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A2b | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1982 |
| P30542 | THEOPHYLLINE GLYCINATE | Adenosine receptor antagonist | CHEMBL2111329 | Adenosine receptor | Adenosine receptor A1 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor adenosine receptor | Small molecule | 1982 |
| Q07343 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4B" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4b | Small molecule | 1982 |
| Q08493 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4C" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4c | Small molecule | 1982 |
| Q08499 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 4 inhibitor | CHEMBL2093863 | Phosphodiesterase 4 | "cAMP-specific 3',5'-cyclic phosphodiesterase 4D" | Homo sapiens | enzyme phosphodiesterase pde_4 pde_4d | Small molecule | 1982 |
| Q13370 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase B" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3b | Small molecule | 1982 |
| Q14432 | THEOPHYLLINE GLYCINATE | Phosphodiesterase 3 inhibitor | CHEMBL2094125 | Phosphodiesterase 3 | "cGMP-inhibited 3',5'-cyclic phosphodiesterase A" | Homo sapiens | enzyme phosphodiesterase pde_3 pde_3a | Small molecule | 1982 |
| C4PKY4 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 1 | Taeniidae | structural | Small molecule | 1967 |
| C4PKZ2 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 2 | Taeniidae | structural | Small molecule | 1967 |
| C4PKZ6 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364704 | Tubulin | Beta-tubulin isoform 3 | Taeniidae | structural | Small molecule | 1967 |
| F1L4P8 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-1 chain | Nematoda | structural | Small molecule | 1967 |
| F1L7U3 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-2 chain | Nematoda | structural | Small molecule | 1967 |
| F1L8A5 | THIABENDAZOLE | Tubulin inhibitor | CHEMBL2364705 | Tubulin | Tubulin beta-4 chain | Nematoda | structural | Small molecule | 1967 |
| P18505 | THIAMYLAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | THIAMYLAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | THIAMYLAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P14416 | THIETHYLPERAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1961 |
| P12268 | THIOGUANINE | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 1966 |
| P12268 | THIOGUANINE | DNA inhibitor | CHEMBL2311221 | DNA | Inosine-5'-monophosphate dehydrogenase 2 | Homo sapiens | enzyme reductase | Small molecule | 1966 |
| P20839 | THIOGUANINE | Inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitor | CHEMBL2111369 | Inosine-5'-monophosphate dehydrogenase (IMPDH) | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1966 |
| P20839 | THIOGUANINE | DNA inhibitor | CHEMBL2311221 | DNA | Inosine-5'-monophosphate dehydrogenase 1 | Homo sapiens | enzyme reductase | Small molecule | 1966 |
| THIOGUANINE | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1966 | |||
| P18505 | THIOPENTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | THIOPENTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | THIOPENTAL | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P14416 | THIORIDAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1962 |
| P21917 | THIORIDAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1962 |
| P28223 | THIORIDAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1962 |
| P28335 | THIORIDAZINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1962 |
| P35462 | THIORIDAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1962 |
| THIOTEPA | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1959 | |||
| P14416 | THIOTHIXENE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1967 |
| P28223 | THIOTHIXENE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1967 |
| THYROGLOBULIN | Iodine storage agent | Unknown | 1982 | ||||||
| P16473 | THYROTROPIN | Thyroid stimulating hormone receptor agonist | CHEMBL1963 | Thyroid stimulating hormone receptor | Thyrotropin receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Unknown | 1953 |
| P16473 | THYROTROPIN ALFA | Thyroid stimulating hormone receptor agonist | CHEMBL1963 | Thyroid stimulating hormone receptor | Thyrotropin receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Protein | 1998 |
| P30531 | TIAGABINE | GABA transporter 1 inhibitor | CHEMBL1903 | GABA transporter 1 | Sodium- and chloride-dependent GABA transporter 1 | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1997 |
| Q9H244 | TICAGRELOR | Purinergic receptor P2Y12 negative allosteric modulator | CHEMBL2001 | Purinergic receptor P2Y12 | P2Y purinoceptor 12 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor purine receptor | Small molecule | 2011 |
| P02918 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1A | Bacteria | enzyme protease serine unclassified | Small molecule | 1976 |
| P02919 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 1B | Bacteria | enzyme protease | Small molecule | 1976 |
| P08506 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacC | Bacteria | enzyme protease serine se s11 | Small molecule | 1976 |
| P0AD65 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Penicillin-binding protein 2 | Bacteria | enzyme protease serine unclassified | Small molecule | 1976 |
| P0AD68 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | Peptidoglycan synthase FtsI | Bacteria | enzyme protease | Small molecule | 1976 |
| P0AEB2 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacA | Bacteria | enzyme protease serine se s11 | Small molecule | 1976 |
| P24228 | TICARCILLIN | Bacterial penicillin-binding protein inhibitor | CHEMBL2354204 | Bacterial penicillin-binding protein | D-alanyl-D-alanine carboxypeptidase DacB | Bacteria | enzyme protease serine se s13 | Small molecule | 1976 |
| Q9H244 | TICLOPIDINE | Purinergic receptor P2Y12 antagonist | CHEMBL2001 | Purinergic receptor P2Y12 | P2Y purinoceptor 12 | Homo sapiens | membrane receptor 7tm1 smallmol nucleotide-like receptor purine receptor | Small molecule | 1991 |
| TIGECYCLINE | Bacterial 70S ribosome inhibitor | CHEMBL2363135 | Bacterial 70S ribosome | 16S ribosomal RNA | Bacteria | Small molecule | 2005 | ||
| TILUDRONIC ACID | ATP inhibitor | CHEMBL2366048 | ATP | Homo sapiens | Small molecule | 1997 | |||
| P07550 | TIMOLOL | Beta-2 adrenergic receptor antagonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 |
| P08588 | TIMOLOL | Beta-1 adrenergic receptor antagonist | CHEMBL213 | Beta-1 adrenergic receptor | Beta-1 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1978 |
| TINIDAZOLE | DNA inhibitor | CHEMBL2366045 | DNA | Trichomonas | Small molecule | 2004 | |||
| P01008 | TINZAPARIN SODIUM | Antithrombin-III activator | CHEMBL1950 | Antithrombin-III | Antithrombin-III | Homo sapiens | secreted | Oligosaccharide | 2000 |
| P10613 | TIOCONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 1983 |
| TIOPRONIN | Reducing agent | Small molecule | 1988 | ||||||
| P20309 | TIOTROPIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 0 |
| Q72874 | TIPRANAVIR | Human immunodeficiency virus type 1 protease inhibitor | CHEMBL243 | Human immunodeficiency virus type 1 protease | Pol polyprotein | Human immunodeficiency virus 1 | enzyme protease aspartic aa a2a | Small molecule | 2005 |
| P05106 | TIROFIBAN | Integrin alpha-IIb/beta-3 inhibitor | CHEMBL2093869 | Integrin alpha-IIb/beta-3 | Integrin beta-3 | Homo sapiens | membrane receptor | Small molecule | 1998 |
| P08514 | TIROFIBAN | Integrin alpha-IIb/beta-3 inhibitor | CHEMBL2093869 | Integrin alpha-IIb/beta-3 | Integrin alpha-IIb | Homo sapiens | membrane receptor | Small molecule | 1998 |
| P08913 | TIZANIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18089 | TIZANIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| P18825 | TIZANIDINE | Adrenergic receptor alpha-2 agonist | CHEMBL2095158 | Adrenergic receptor alpha-2 | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1996 |
| TOBRAMYCIN | 70S ribosome inhibitor | CHEMBL2364022 | 70S ribosome | 23S ribosomal RNA | Pseudomonas aeruginosa | Small molecule | 1975 | ||
| P35498 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| P35499 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q01118 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q14524 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q15858 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q99250 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q9NY46 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q9UI33 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q9UQD0 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| Q9Y5Y9 | TOCAINIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1984 |
| P08887 | TOCILIZUMAB | Interleukin-6 receptor alpha subunit inhibitor | CHEMBL2364155 | Interleukin-6 receptor alpha subunit | Interleukin-6 receptor subunit alpha | Homo sapiens | secreted | Antibody | 2005 |
| P40189 | TOCILIZUMAB | Interleukin-6 receptor | Interleukin-6 receptor subunit beta | Homo sapiens | membrane receptor | Antibody | 2005 | ||
| O60674 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK2 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2012 |
| O60674 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK2 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2012 |
| P23458 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK1 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2012 |
| P23458 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK1 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2012 |
| P29597 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2012 |
| P29597 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Non-receptor tyrosine-protein kinase TYK2 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2012 |
| P52333 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK3 | Homo sapiens | enzyme kinase protein kinase tk jaka | Small molecule | 2012 |
| P52333 | TOFACITINIB | Janus Kinase (JAK) inhibitor | CHEMBL2363062 | Janus Kinase (JAK) | Tyrosine-protein kinase JAK3 | Homo sapiens | enzyme kinase protein kinase tk jakb | Small molecule | 2012 |
| Q09428 | TOLAZAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1966 |
| Q14654 | TOLAZAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1966 |
| P08913 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P18089 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P18825 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-2C adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P25021 | TOLAZOLINE | Histamine H2 receptor agonist | CHEMBL1941 | Histamine H2 receptor | Histamine H2 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1985 |
| P25100 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P35348 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| P35367 | TOLAZOLINE | Histamine H1 receptor agonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1985 |
| P35368 | TOLAZOLINE | Adrenergic receptor alpha antagonist | CHEMBL2095203 | Adrenergic receptor alpha | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1985 |
| Q09428 | TOLBUTAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-binding cassette sub-family C member 8 | Homo sapiens | transporter ntpase atp binding cassette mrp | Small molecule | 1961 |
| Q14654 | TOLBUTAMIDE | "Sulfonylurea receptor 1, Kir6.2 blocker" | CHEMBL2096972 | "Sulfonylurea receptor 1, Kir6.2" | ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens | ion channel vgc k kir | Small molecule | 1961 |
| P21964 | TOLCAPONE | Catechol O-methyltransferase inhibitor | CHEMBL2023 | Catechol O-methyltransferase | Catechol O-methyltransferase | Homo sapiens | enzyme transferase | Small molecule | 1998 |
| P23219 | TOLMETIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 1 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P35354 | TOLMETIN | Cyclooxygenase inhibitor | CHEMBL2094253 | Cyclooxygenase | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 1976 |
| P08172 | TOLTERODINE | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1998 |
| P20309 | TOLTERODINE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1998 |
| P30518 | TOLVAPTAN | Vasopressin V2 receptor antagonist | CHEMBL1790 | Vasopressin V2 receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Small molecule | 2009 |
| O00591 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| O14764 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P00918 | TOPIRAMATE | Carbonic anhydrase II inhibitor | CHEMBL205 | Carbonic anhydrase II | Carbonic anhydrase 2 | Homo sapiens | enzyme lyase | Small molecule | 1996 |
| P14867 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P18505 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P18507 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P22748 | TOPIRAMATE | Carbonic anhydrase IV inhibitor | CHEMBL3729 | Carbonic anhydrase IV | Carbonic anhydrase 4 | Homo sapiens | enzyme lyase | Small molecule | 1996 |
| P28472 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P31644 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P34903 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P35498 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| P35499 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| P39086 | TOPIRAMATE | Glutamate receptor ionotropic kainate antagonist | CHEMBL2109241 | Glutamate receptor ionotropic kainate | "Glutamate receptor ionotropic, kainate 1" | Homo sapiens | ion channel lgic glut kainate | Small molecule | 1996 |
| P42261 | TOPIRAMATE | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 1 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 1996 |
| P42262 | TOPIRAMATE | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 2 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 1996 |
| P42263 | TOPIRAMATE | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 3 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 1996 |
| P47869 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P47870 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P48058 | TOPIRAMATE | Glutamate receptor ionotropic AMPA antagonist | CHEMBL2096670 | Glutamate receptor ionotropic AMPA | Glutamate receptor 4 | Homo sapiens | ion channel lgic glut ampa | Small molecule | 1996 |
| P48169 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| P78334 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| Q01118 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q13002 | TOPIRAMATE | Glutamate receptor ionotropic kainate antagonist | CHEMBL2109241 | Glutamate receptor ionotropic kainate | "Glutamate receptor ionotropic, kainate 2" | Homo sapiens | ion channel lgic glut kainate | Small molecule | 1996 |
| Q13003 | TOPIRAMATE | Glutamate receptor ionotropic kainate antagonist | CHEMBL2109241 | Glutamate receptor ionotropic kainate | "Glutamate receptor ionotropic, kainate 3" | Homo sapiens | ion channel lgic glut kainate | Small molecule | 1996 |
| Q14524 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q15858 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q16099 | TOPIRAMATE | Glutamate receptor ionotropic kainate antagonist | CHEMBL2109241 | Glutamate receptor ionotropic kainate | "Glutamate receptor ionotropic, kainate 4" | Homo sapiens | ion channel lgic glut kainate | Small molecule | 1996 |
| Q16445 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| Q16478 | TOPIRAMATE | Glutamate receptor ionotropic kainate antagonist | CHEMBL2109241 | Glutamate receptor ionotropic kainate | "Glutamate receptor ionotropic, kainate 5" | Homo sapiens | ion channel lgic glut kainate | Small molecule | 1996 |
| Q8N1C3 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| Q99250 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q99928 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| Q9NY46 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UI33 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9UN88 | TOPIRAMATE | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1996 |
| Q9UQD0 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q9Y5Y9 | TOPIRAMATE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 1996 |
| Q969P6 | TOPOTECAN | "DNA topoisomerase I, mitochondrial inhibitor" | CHEMBL2362989 | "DNA topoisomerase I, mitochondrial" | "DNA topoisomerase I, mitochondrial" | Homo sapiens | enzyme isomerase | Small molecule | 1996 |
| P03372 | TOREMIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a1 | Small molecule | 1997 |
| Q92731 | TOREMIFENE | Estrogen receptor modulator | CHEMBL2093866 | Estrogen receptor | Estrogen receptor beta | Homo sapiens | transcription factor nuclear receptor nr3 nr3a nr3a2 | Small molecule | 1997 |
| Q13621 | TORSEMIDE | Sodium-(potassium)-chloride cotransporter 2 inhibitor | CHEMBL1874 | Sodium-(potassium)-chloride cotransporter 2 | Solute carrier family 12 member 1 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1993 |
| P11836 | TOSITUMOMAB | B-lymphocyte antigen CD20 inhibitor | CHEMBL2058 | B-lymphocyte antigen CD20 | B-lymphocyte antigen CD20 | Homo sapiens | ion channel other misc cd20 | Antibody | 2003 |
| P35372 | TRAMADOL | Mu opioid receptor agonist | CHEMBL233 | Mu opioid receptor | Mu-type opioid receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide opioid receptor | Small molecule | 1995 |
| P36507 | TRAMETINIB | Dual specificity mitogen-activated protein kinase kinase 2 inhibitor | CHEMBL2964 | Dual specificity mitogen-activated protein kinase kinase 2 | Dual specificity mitogen-activated protein kinase kinase 2 | Homo sapiens | enzyme kinase protein kinase ste ste7 | Small molecule | 2013 |
| Q02750 | TRAMETINIB | Dual specificity mitogen-activated protein kinase kinase 1 inhibitor | CHEMBL3587 | Dual specificity mitogen-activated protein kinase kinase 1 | Dual specificity mitogen-activated protein kinase kinase 1 | Homo sapiens | enzyme kinase protein kinase ste ste7 | Small molecule | 2013 |
| P12821 | TRANDOLAPRIL | Angiotensin-converting enzyme inhibitor | CHEMBL1808 | Angiotensin-converting enzyme | Angiotensin-converting enzyme | Homo sapiens | enzyme protease metallo mae m2 | Small molecule | 1996 |
| P00747 | TRANEXAMIC ACID | Plasminogen inhibitor | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Small molecule | 1986 |
| P21397 | TRANYLCYPROMINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] A | Homo sapiens | enzyme reductase | Small molecule | 1961 |
| P27338 | TRANYLCYPROMINE | Monoamine oxidase inhibitor | CHEMBL2095205 | Monoamine oxidase | Amine oxidase [flavin-containing] B | Homo sapiens | enzyme reductase | Small molecule | 1961 |
| P04626 | TRASTUZUMAB | Receptor protein-tyrosine kinase erbB-2 inhibitor | CHEMBL1824 | Receptor protein-tyrosine kinase erbB-2 | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Antibody | 1998 |
| P04350 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Antibody | 2013 |
| P04626 | TRASTUZUMAB EMTANSINE | Receptor protein-tyrosine kinase erbB-2 inhibitor | CHEMBL1824 | Receptor protein-tyrosine kinase erbB-2 | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Antibody | 2013 |
| P07437 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Antibody | 2013 |
| P68371 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Antibody | 2013 |
| Q13509 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Antibody | 2013 |
| Q13885 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Antibody | 2013 |
| Q3ZCM7 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Antibody | 2013 |
| Q9BUF5 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Antibody | 2013 |
| Q9BVA1 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Antibody | 2013 |
| Q9H4B7 | TRASTUZUMAB EMTANSINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Antibody | 2013 |
| P43088 | TRAVOPROST | Prostanoid FP receptor agonist | CHEMBL1987 | Prostanoid FP receptor | Prostaglandin F2-alpha receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 2001 |
| P28223 | TRAZODONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1981 |
| P28335 | TRAZODONE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1981 |
| P31645 | TRAZODONE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1981 |
| P43119 | TREPROSTINIL | Prostanoid IP receptor agonist | CHEMBL1995 | Prostanoid IP receptor | Prostacyclin receptor | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor prostanoid receptor | Small molecule | 2002 |
| P10276 | TRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor alpha | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b1 | Small molecule | 1971 |
| P10826 | TRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor beta | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b2 | Small molecule | 1971 |
| P13631 | TRETINOIN | Retinoic acid receptor agonist | CHEMBL2363069 | Retinoic acid receptor | Retinoic acid receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1b nr1b3 | Small molecule | 1971 |
| P04150 | TRIAMCINOLONE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1957 |
| P04150 | TRIAMCINOLONE ACETONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1960 |
| P04150 | TRIAMCINOLONE DIACETATE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1959 |
| P04150 | TRIAMCINOLONE HEXACETONIDE | Glucocorticoid receptor agonist | CHEMBL2034 | Glucocorticoid receptor | Glucocorticoid receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c1 | Small molecule | 1969 |
| P37088 | TRIAMTERENE | "Amiloride-sensitive sodium channel, ENaC blocker" | CHEMBL2107836 | "Amiloride-sensitive sodium channel, ENaC" | Amiloride-sensitive sodium channel subunit alpha | Homo sapiens | ion channel lgic enac | Small molecule | 1964 |
| P14867 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18507 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P31644 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P34903 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47869 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q8N1C3 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q99928 | TRIAZOLAM | GABA-A receptor; anion channel positive allosteric modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P55017 | TRICHLORMETHIAZIDE | Thiazide-sensitive sodium-chloride cotransporter inhibitor | CHEMBL1876 | Thiazide-sensitive sodium-chloride cotransporter | Solute carrier family 12 member 3 | Homo sapiens | transporter electrochemical slc slc12 | Small molecule | 1960 |
| O00591 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit pi | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| O14764 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit delta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P14867 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18505 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P18507 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P28472 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P31644 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-5 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P34903 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47869 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P47870 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P48169 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-4 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P78334 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit epsilon | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q16445 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit alpha-6 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q8N1C3 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q99928 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit gamma-3 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| Q9UN88 | TRICLOFOS | GABA-A receptor; anion channel positive modulator | CHEMBL2093872 | GABA-A receptor; anion channel | Gamma-aminobutyric acid receptor subunit theta | Homo sapiens | ion channel lgic gabaa | Small molecule | 1982 |
| P0AEK4 | TRICLOSAN | Bacterial enoyl-[acyl-carrier-protein] reductase inhibitor | CHEMBL2364678 | Bacterial enoyl-[acyl-carrier-protein] reductase | Enoyl-[acyl-carrier-protein] reductase [NADH] FabI | Bacteria | enzyme reductase | Small molecule | 1997 |
| P11229 | TRIDIHEXETHYL | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 |
| P20309 | TRIDIHEXETHYL | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1954 |
| TRIENTINE | Copper chelating agent | CHEMBL2363057 | Copper | Small molecule | 1985 | ||||
| TRIENTINE | CHEMBL2363057 | Copper | Small molecule | 1985 | |||||
| P14416 | TRIFLUOPERAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1959 |
| P21917 | TRIFLUOPERAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(4) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1959 |
| P28223 | TRIFLUOPERAZINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1959 |
| P28335 | TRIFLUOPERAZINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1959 |
| P35462 | TRIFLUOPERAZINE | D2-like dopamine receptor antagonist | CHEMBL2331075 | D2-like dopamine receptor | D(3) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1959 |
| P14416 | TRIFLUPROMAZINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1957 |
| TRIFLURIDINE | DNA inhibitor | CHEMBL2366042 | DNA | Human herpesvirus 1 | Small molecule | 1980 | |||
| P11229 | TRIHEXYPHENIDYL | Muscarinic acetylcholine receptor M1 antagonist | CHEMBL216 | Muscarinic acetylcholine receptor M1 | Muscarinic acetylcholine receptor M1 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1949 |
| P26439 | TRILOSTANE | 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type II inhibitor | CHEMBL3670 | 3-beta-hydroxysteroid dehydrogenase/delta 5-->4-isomerase type II | 3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 2 | Homo sapiens | enzyme reductase | Small molecule | 1984 |
| O43497 | TRIMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1946 |
| O95180 | TRIMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1946 |
| Q9P0X4 | TRIMETHADIONE | Voltage-gated T-type calcium channel blocker | CHEMBL2362995 | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1946 |
| P30926 | TRIMETHAPHAN | Neuronal acetylcholine receptor; alpha3/beta4 antagonist | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1982 |
| P32297 | TRIMETHAPHAN | Neuronal acetylcholine receptor; alpha3/beta4 antagonist | CHEMBL1907594 | Neuronal acetylcholine receptor; alpha3/beta4 | Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1982 |
| TRIMETHOBENZAMIDE | Unknown | Small molecule | 1974 | ||||||
| P0ABQ4 | TRIMETHOPRIM | Bacterial dihydrofolate reductase inhibitor | CHEMBL2364669 | Bacterial dihydrofolate reductase | Dihydrofolate reductase | Bacteria | enzyme reductase | Small molecule | 1973 |
| P16184 | TRIMETREXATE | Dihydrofolate reductase inhibitor | CHEMBL1926 | Dihydrofolate reductase | Dihydrofolate reductase | Pneumocystis carinii | enzyme reductase | Small molecule | 1993 |
| P14416 | TRIMIPRAMINE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 1979 |
| P23975 | TRIMIPRAMINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1979 |
| P25100 | TRIMIPRAMINE | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1D adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P28223 | TRIMIPRAMINE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1979 |
| P28335 | TRIMIPRAMINE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1979 |
| P35348 | TRIMIPRAMINE | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1A adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| P35367 | TRIMIPRAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1979 |
| P35368 | TRIMIPRAMINE | Adrenergic receptor alpha-1 antagonist | CHEMBL2094251 | Adrenergic receptor alpha-1 | Alpha-1B adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 1979 |
| TRIOXSALEN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1964 | |||
| P35367 | TRIPELENNAMINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1948 |
| P35367 | TRIPROLIDINE | Histamine H1 receptor antagonist | CHEMBL231 | Histamine H1 receptor | Histamine H1 receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor histamine receptor | Small molecule | 1983 |
| P30968 | TRIPTORELIN | Gonadotropin-releasing hormone receptor agonist | CHEMBL1855 | Gonadotropin-releasing hormone receptor | Gonadotropin-releasing hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide gnrh receptor | Protein | 2000 |
| P37231 | TROGLITAZONE | Peroxisome proliferator-activated receptor gamma agonist | CHEMBL235 | Peroxisome proliferator-activated receptor gamma | Peroxisome proliferator-activated receptor gamma | Homo sapiens | transcription factor nuclear receptor nr1 nr1c nr1c3 | Small molecule | 1997 |
| TROLEANDOMYCIN | 70S ribosome inhibitor | CHEMBL2363853 | 70S ribosome | 23S ribosomal RNA | Streptococcus pneumoniae | Small molecule | 1969 | ||
| TROMETHAMINE | Unknown | Small molecule | 1965 | ||||||
| P20309 | TROPICAMIDE | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 1960 |
| P08172 | TROSPIUM | Muscarinic acetylcholine receptor M2 antagonist | CHEMBL211 | Muscarinic acetylcholine receptor M2 | Muscarinic acetylcholine receptor M2 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| P20309 | TROSPIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2004 |
| P0AES4 | TROVAFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit A | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P0AES6 | TROVAFLOXACIN | Bacterial DNA gyrase inhibitor | CHEMBL2311224 | Bacterial DNA gyrase | DNA gyrase subunit B | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P0AFI2 | TROVAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit A | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P20083 | TROVAFLOXACIN | Topoisomerase IV inhibitor | CHEMBL2363076 | Topoisomerase IV | DNA topoisomerase 4 subunit B | Bacteria | enzyme isomerase | Small molecule | 1997 |
| P02708 | TUBOCURARINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1945 |
| P07510 | TUBOCURARINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1945 |
| P11230 | TUBOCURARINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1945 |
| Q04844 | TUBOCURARINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1945 |
| Q07001 | TUBOCURARINE | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1945 |
| TYLOXAPOL | Surfactant agent | Unknown | 1990 | ||||||
| P06401 | ULIPRISTAL ACETATE | Progesterone receptor modulator | CHEMBL208 | Progesterone receptor | Progesterone receptor | Homo sapiens | transcription factor nuclear receptor nr3 nr3c nr3c3 | Small molecule | 2010 |
| P20309 | UMECLIDINIUM | Muscarinic acetylcholine receptor M3 antagonist | CHEMBL245 | Muscarinic acetylcholine receptor M3 | Muscarinic acetylcholine receptor M3 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor acetylcholine receptor | Small molecule | 2013 |
| UNOPROSTONE ISOPROPYL | Unknown | Small molecule | 2000 | ||||||
| URACIL MUSTARD | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1962 | |||
| P23945 | UROFOLLITROPIN | Follicle stimulating hormone receptor agonist | CHEMBL2024 | Follicle stimulating hormone receptor | Follicle-stimulating hormone receptor | Homo sapiens | membrane receptor 7tm1 peptide glycohormone receptor glycohormone receptor | Unknown | 1986 |
| P00747 | UROKINASE | Plasminogen activator | CHEMBL1801 | Plasminogen | Plasminogen | Homo sapiens | enzyme protease serine pas s1a | Enzyme | 2007 |
| Q96RI1 | URSODIOL | Bile acid receptor FXR agonist | CHEMBL2047 | Bile acid receptor FXR | Bile acid receptor | Homo sapiens | transcription factor nuclear receptor nr1 nr1h nr1h4 | Small molecule | 1987 |
| P29460 | USTEKINUMAB | Interleukin-12 inhibitor | CHEMBL2364153 | Interleukin-12 | Interleukin-12 subunit beta | Homo sapiens | secreted | Antibody | 2009 |
| P29460 | USTEKINUMAB | Interleukin-23 inhibitor | CHEMBL2364154 | Interleukin-23 | Interleukin-12 subunit beta | Homo sapiens | secreted | Antibody | 2009 |
| P04293 | VALACYCLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1995 |
| Q9QNF7 | VALACYCLOVIR | Thymidine kinase | Thymidine kinase | Human herpesvirus 1 | enzyme | Small molecule | 1995 | ||
| P35354 | VALDECOXIB | Cyclooxygenase-2 inhibitor | CHEMBL230 | Cyclooxygenase-2 | Prostaglandin G/H synthase 2 | Homo sapiens | enzyme reductase | Small molecule | 2001 |
| P04293 | VALGANCICLOVIR | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 2001 |
| P51649 | VALPROIC ACID | Succinate semialdehyde dehydrogenase inhibitor | CHEMBL1911 | Succinate semialdehyde dehydrogenase | "Succinate-semialdehyde dehydrogenase, mitochondrial" | Homo sapiens | enzyme reductase | Small molecule | 1978 |
| P80404 | VALPROIC ACID | "4-aminobutyrate aminotransferase, mitochondrial" | "4-aminobutyrate aminotransferase, mitochondrial" | Homo sapiens | enzyme transferase | Small molecule | 1978 | ||
| P11388 | VALRUBICIN | DNA topoisomerase II alpha inhibitor | CHEMBL1806 | DNA topoisomerase II alpha | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1998 |
| P11388 | VALRUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | DNA topoisomerase 2-alpha | Homo sapiens | enzyme isomerase | Small molecule | 1998 |
| VALRUBICIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 1998 | |||
| P30556 | VALSARTAN | Type-1 angiotensin II receptor antagonist | CHEMBL227 | Type-1 angiotensin II receptor | Type-1 angiotensin II receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide angiotensin receptor | Small molecule | 1996 |
| VANCOMYCIN | Peptidoglycan inhibitor | CHEMBL3041361 | Peptidoglycan | Bacteria | Small molecule | 1964 | |||
| O15197 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-B receptor 6 | Homo sapiens | unclassified | Small molecule | 2011 |
| P00533 | VANDETANIB | Epidermal growth factor receptor inhibitor | CHEMBL2363049 | Epidermal growth factor receptor | Epidermal growth factor receptor | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2011 |
| P04626 | VANDETANIB | Epidermal growth factor receptor inhibitor | CHEMBL2363049 | Epidermal growth factor receptor | Receptor tyrosine-protein kinase erbB-2 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2011 |
| P07949 | VANDETANIB | Tyrosine-protein kinase receptor RET inhibitor | CHEMBL2041 | Tyrosine-protein kinase receptor RET | Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens | enzyme kinase protein kinase tk ret | Small molecule | 2011 |
| P12931 | VANDETANIB | Tyrosine-protein kinase SRC inhibitor | CHEMBL267 | Tyrosine-protein kinase SRC | Proto-oncogene tyrosine-protein kinase Src | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2011 |
| P17948 | VANDETANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 1 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2011 |
| P21709 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 1 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P21860 | VANDETANIB | Epidermal growth factor receptor inhibitor | CHEMBL2363049 | Epidermal growth factor receptor | Receptor tyrosine-protein kinase erbB-3 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2011 |
| P29317 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 2 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P29320 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 3 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P29322 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 8 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P29323 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-B receptor 2 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P35916 | VANDETANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 3 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2011 |
| P35968 | VANDETANIB | Vascular endothelial growth factor receptor inhibitor | CHEMBL2095227 | Vascular endothelial growth factor receptor | Vascular endothelial growth factor receptor 2 | Homo sapiens | enzyme kinase protein kinase tk vegfr | Small molecule | 2011 |
| P54753 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-B receptor 3 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P54756 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 5 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P54760 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-B receptor 4 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P54762 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-B receptor 1 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| P54764 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 4 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| Q02763 | VANDETANIB | Tyrosine-protein kinase TIE-2 inhibitor | CHEMBL4128 | Tyrosine-protein kinase TIE-2 | Angiopoietin-1 receptor | Homo sapiens | enzyme kinase protein kinase tk tie | Small molecule | 2011 |
| Q13882 | VANDETANIB | Tyrosine-protein kinase BRK inhibitor | CHEMBL4601 | Tyrosine-protein kinase BRK | Protein-tyrosine kinase 6 | Homo sapiens | enzyme kinase protein kinase tk src | Small molecule | 2011 |
| Q15303 | VANDETANIB | Epidermal growth factor receptor inhibitor | CHEMBL2363049 | Epidermal growth factor receptor | Receptor tyrosine-protein kinase erbB-4 | Homo sapiens | enzyme kinase protein kinase tk egfr | Small molecule | 2011 |
| Q15375 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 7 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| Q5JZY3 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 10 | Homo sapiens | enzyme kinase | Small molecule | 2011 |
| Q9UF33 | VANDETANIB | Ephrin receptor inhibitor | CHEMBL2363043 | Ephrin receptor | Ephrin type-A receptor 6 | Homo sapiens | enzyme kinase protein kinase tk eph | Small molecule | 2011 |
| O76074 | VARDENAFIL | Phosphodiesterase 5A inhibitor | CHEMBL1827 | Phosphodiesterase 5A | "cGMP-specific 3',5'-cyclic phosphodiesterase" | Homo sapiens | enzyme phosphodiesterase pde_5 pde_5a | Small molecule | 2003 |
| P17787 | VARENICLINE | Neuronal acetylcholine receptor; alpha4/beta2 agonist | CHEMBL1907589 | Neuronal acetylcholine receptor; alpha4/beta2 | Neuronal acetylcholine receptor subunit beta-2 | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 2006 |
| P43681 | VARENICLINE | Neuronal acetylcholine receptor; alpha4/beta2 agonist | CHEMBL1907589 | Neuronal acetylcholine receptor; alpha4/beta2 | Neuronal acetylcholine receptor subunit alpha-4 | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 2006 |
| P30518 | VASOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 2014 |
| P37288 | VASOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1a receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 2014 |
| P47901 | VASOPRESSIN | Vasopressin receptor agonist | CHEMBL2363078 | Vasopressin receptor | Vasopressin V1b receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 2014 |
| P30518 | VASOPRESSIN TANNATE | Vasopressin V2 receptor agonist | CHEMBL1790 | Vasopressin V2 receptor | Vasopressin V2 receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P37288 | VASOPRESSIN TANNATE | Vasopressin V1a receptor agonist | CHEMBL1889 | Vasopressin V1a receptor | Vasopressin V1a receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P47901 | VASOPRESSIN TANNATE | Vasopressin V1b receptor agonist | CHEMBL1921 | Vasopressin V1b receptor | Vasopressin V1b receptor | Homo sapiens | membrane receptor 7tm1 peptide short peptide vasopressin and oxytocin receptor | Protein | 1982 |
| P02708 | VECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit alpha | Homo sapiens | ion channel lgic ach chrn alpha | Small molecule | 1984 |
| P07510 | VECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit gamma | Homo sapiens | ion channel lgic ach chrn gamma | Small molecule | 1984 |
| P11230 | VECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit beta | Homo sapiens | ion channel lgic ach chrn beta | Small molecule | 1984 |
| Q04844 | VECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit epsilon | Homo sapiens | ion channel lgic ach chrn epsilon | Small molecule | 1984 |
| Q07001 | VECURONIUM | Muscle-type nicotinic acetylcholine receptor antagonist | CHEMBL2362997 | Muscle-type nicotinic acetylcholine receptor | Acetylcholine receptor subunit delta | Homo sapiens | ion channel lgic ach chrn delta | Small molecule | 1984 |
| P13612 | VEDOLIZUMAB | Integrin alpha-4/beta-7 inhibitor | CHEMBL2095184 | Integrin alpha-4/beta-7 | Integrin alpha-4 | Homo sapiens | membrane receptor | Antibody | 2014 |
| P26010 | VEDOLIZUMAB | Integrin alpha-4/beta-7 inhibitor | CHEMBL2095184 | Integrin alpha-4/beta-7 | Integrin beta-7 | Homo sapiens | membrane receptor | Antibody | 2014 |
| VELAGLUCERASE ALFA | Glucocerebroside hydrolytic enzyme | CHEMBL2364176 | Glucocerebroside | Homo sapiens | Enzyme | 2010 | |||
| P15056 | VEMURAFENIB | Serine/threonine-protein kinase B-raf inhibitor | CHEMBL5145 | Serine/threonine-protein kinase B-raf | Serine/threonine-protein kinase B-raf | Homo sapiens | enzyme kinase protein kinase tkl raf | Small molecule | 2011 |
| P23975 | VENLAFAXINE | Norepinephrine transporter inhibitor | CHEMBL222 | Norepinephrine transporter | Sodium-dependent noradrenaline transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1993 |
| P31645 | VENLAFAXINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 1993 |
| O43497 | VERAPAMIL | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1G | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 | ||
| O60840 | VERAPAMIL | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1F | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| O95180 | VERAPAMIL | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1H | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 | ||
| Q01668 | VERAPAMIL | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1D | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q13698 | VERAPAMIL | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1S | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q13936 | VERAPAMIL | Voltage-gated L-type calcium channel blocker | CHEMBL2095229 | Voltage-gated L-type calcium channel | Voltage-dependent L-type calcium channel subunit alpha-1C | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 |
| Q9P0X4 | VERAPAMIL | Voltage-gated T-type calcium channel | Voltage-dependent T-type calcium channel subunit alpha-1I | Homo sapiens | ion channel vgc vg ca | Small molecule | 1981 | ||
| VERATRUM VIRIDE | Unknown | Small molecule | 1982 | ||||||
| VERTEPORFIN | DNA inhibitor | CHEMBL2311221 | DNA | Homo sapiens | Small molecule | 2000 | |||
| P04293 | VIDARABINE | Human herpesvirus 1 DNA polymerase inhibitor | CHEMBL1872 | Human herpesvirus 1 DNA polymerase | DNA polymerase catalytic subunit | Herpes simplex virus (type 1 / strain 17) | enzyme transferase | Small molecule | 1976 |
| P80404 | VIGABATRIN | Gamma-amino-N-butyrate transaminase inhibitor | CHEMBL2044 | Gamma-amino-N-butyrate transaminase | "4-aminobutyrate aminotransferase, mitochondrial" | Homo sapiens | enzyme transferase | Small molecule | 2009 |
| P07550 | VILANTEROL | Beta-2 adrenergic receptor agonist | CHEMBL210 | Beta-2 adrenergic receptor | Beta-2 adrenergic receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor adrenergic receptor | Small molecule | 2013 |
| P08908 | VILAZODONE | Serotonin 1a (5-HT1a) receptor partial agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2011 |
| P31645 | VILAZODONE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2011 |
| P04350 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1965 |
| P07437 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1965 |
| P68371 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1965 |
| Q13509 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1965 |
| Q13885 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1965 |
| Q3ZCM7 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1965 |
| Q9BUF5 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1965 |
| Q9BVA1 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1965 |
| Q9H4B7 | VINBLASTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1965 |
| P04350 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1963 |
| P07437 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1963 |
| P68371 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1963 |
| Q13509 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1963 |
| Q13885 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1963 |
| Q3ZCM7 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1963 |
| Q9BUF5 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1963 |
| Q9BVA1 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1963 |
| Q9H4B7 | VINCRISTINE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1963 |
| P04350 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4A chain | Homo sapiens | structural | Small molecule | 1994 |
| P07437 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta chain | Homo sapiens | structural | Small molecule | 1994 |
| P68371 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-4B chain | Homo sapiens | structural | Small molecule | 1994 |
| Q13509 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-3 chain | Homo sapiens | structural | Small molecule | 1994 |
| Q13885 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2A chain | Homo sapiens | structural | Small molecule | 1994 |
| Q3ZCM7 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-8 chain | Homo sapiens | structural | Small molecule | 1994 |
| Q9BUF5 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-6 chain | Homo sapiens | structural | Small molecule | 1994 |
| Q9BVA1 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-2B chain | Homo sapiens | structural | Small molecule | 1994 |
| Q9H4B7 | VINORELBINE BASE | Tubulin inhibitor | CHEMBL2095182 | Tubulin | Tubulin beta-1 chain | Homo sapiens | structural | Small molecule | 1994 |
| VIOMYCIN | 70S ribosome inhibitor | CHEMBL2363965 | 70S ribosome | 16S ribosomal RNA | Mycobacterium tuberculosis | Protein | 1982 | ||
| VIOMYCIN | 70S ribosome inhibitor | CHEMBL2363965 | 70S ribosome | 23S ribosomal RNA | Mycobacterium tuberculosis | Protein | 1982 | ||
| Q99835 | VISMODEGIB | Smoothened homolog inhibitor | CHEMBL5971 | Smoothened homolog | Smoothened homolog | Homo sapiens | membrane receptor 7tmfz smoothened | Small molecule | 2012 |
| P25116 | VORAPAXAR | Proteinase-activated receptor 1 antagonist | CHEMBL3974 | Proteinase-activated receptor 1 | Proteinase-activated receptor 1 | Homo sapiens | membrane receptor 7tm1 peptide protease-activated receptor protease-activated receptor | Small molecule | 2014 |
| P10613 | VORICONAZOLE | Cytochrome P450 51 inhibitor | CHEMBL1780 | Cytochrome P450 51 | Lanosterol 14-alpha demethylase | Candida albicans (strain SC5314 / ATCC MYA-2876) (Yeast) | enzyme cytochrome p450 cyp_51 cyp_51a cyp_51a1 | Small molecule | 2002 |
| O15379 | VORINOSTAT | Histone deacetylase 3 inhibitor | CHEMBL1829 | Histone deacetylase 3 | Histone deacetylase 3 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2006 |
| Q13547 | VORINOSTAT | Histone deacetylase 1 inhibitor | CHEMBL325 | Histone deacetylase 1 | Histone deacetylase 1 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2006 |
| Q92769 | VORINOSTAT | Histone deacetylase 2 inhibitor | CHEMBL1937 | Histone deacetylase 2 | Histone deacetylase 2 | Homo sapiens | epigenetic regulator eraser hdac hdac class i | Small molecule | 2006 |
| Q9UBN7 | VORINOSTAT | Histone deacetylase 6 inhibitor | CHEMBL1865 | Histone deacetylase 6 | Histone deacetylase 6 | Homo sapiens | epigenetic regulator eraser hdac hdac class iib | Small molecule | 2006 |
| P08908 | VORTIOXETINE | Serotonin 1a (5-HT1a) receptor agonist | CHEMBL214 | Serotonin 1a (5-HT1a) receptor | 5-hydroxytryptamine receptor 1A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2013 |
| P28221 | VORTIOXETINE | 5-hydroxytryptamine receptor 1D | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2013 | ||
| P28222 | VORTIOXETINE | 5-hydroxytryptamine receptor 1B | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2013 | ||
| P31645 | VORTIOXETINE | Serotonin transporter inhibitor | CHEMBL228 | Serotonin transporter | Sodium-dependent serotonin transporter | Homo sapiens | transporter electrochemical slc slc06 | Small molecule | 2013 |
| P34969 | VORTIOXETINE | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2013 | ||
| P46098 | VORTIOXETINE | Serotonin 3a (5-HT3a) receptor antagonist | CHEMBL1899 | Serotonin 3a (5-HT3a) receptor | 5-hydroxytryptamine receptor 3A | Homo sapiens | ion channel lgic 5ht3 | Small molecule | 2013 |
| Q9BQB6 | WARFARIN | Vitamin k epoxide reductase complex subunit 1 isoform 1 inhibitor | CHEMBL1930 | Vitamin k epoxide reductase complex subunit 1 isoform 1 | Vitamin K epoxide reductase complex subunit 1 | Homo sapiens | enzyme reductase | Small molecule | 1954 |
| YTTERBIUM PENTETATE | Radioactive metals chelating agent | CHEMBL2366037 | Radioactive metals | Small molecule | 1976 | ||||
| YTTERBIUM PENTETATE | CHEMBL2366037 | Radioactive metals | Small molecule | 1976 | |||||
| P11836 | YTTRIUM Y 90 IBRITUMOMAB TIUXETAN | B-lymphocyte antigen CD20 binding agent | CHEMBL2058 | B-lymphocyte antigen CD20 | B-lymphocyte antigen CD20 | Homo sapiens | ion channel other misc cd20 | Antibody | 2002 |
| Q9Y271 | ZAFIRLUKAST | Cysteinyl leukotriene receptor 1 antagonist | CHEMBL1798 | Cysteinyl leukotriene receptor 1 | Cysteinyl leukotriene receptor 1 | Homo sapiens | membrane receptor 7tm1 smallmol lipid-like ligand receptor leukotriene receptor | Small molecule | 1996 |
| Q72547 | ZALCITABINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1992 |
| P18505 | ZALEPLON | GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator | CHEMBL2111392 | GABA A receptor alpha-1/beta-1/gamma-2 | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1999 |
| P18507 | ZALEPLON | GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator | CHEMBL2111392 | GABA A receptor alpha-1/beta-1/gamma-2 | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1999 |
| P47870 | ZALEPLON | GABA-A receptor alpha-1/beta-2/gamma-2 | Gamma-aminobutyric acid receptor subunit beta-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1999 | ||
| P03468 | ZANAMIVIR | Neuraminidase inhibitor | CHEMBL2051 | Neuraminidase | Neuraminidase | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) | enzyme hydrolase | Small molecule | 1999 |
| P03474 | ZANAMIVIR | Neuraminidase inhibitor | CHEMBL3377 | Neuraminidase | Neuraminidase | Influenza B virus (strain B/Lee/1940) | enzyme hydrolase | Small molecule | 1999 |
| Q00975 | ZICONOTIDE ACETATE | Voltage-gated N-type calcium channel alpha-1B subunit blocker | CHEMBL4478 | Voltage-gated N-type calcium channel alpha-1B subunit | Voltage-dependent N-type calcium channel subunit alpha-1B | Homo sapiens | ion channel vgc vg ca | Protein | 2004 |
| P03362 | ZIDOVUDINE | Gag-Pro-Pol polyprotein | Gag-Pro-Pol polyprotein | Human T-cell leukemia virus 1 (strain Japan ATK-1 subtype A) | Unclassified | Small molecule | 1987 | ||
| P03369 | ZIDOVUDINE | Gag-Pol polyprotein | Gag-Pol polyprotein | Human immunodeficiency virus type 1 group M subtype B (isolate ARV2/SF2) | Unclassified | Small molecule | 1987 | ||
| Q72547 | ZIDOVUDINE | Human immunodeficiency virus type 1 reverse transcriptase inhibitor | CHEMBL247 | Human immunodeficiency virus type 1 reverse transcriptase | Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | enzyme hydrolase | Small molecule | 1987 |
| P09917 | ZILEUTON | Arachidonate 5-lipoxygenase inhibitor | CHEMBL215 | Arachidonate 5-lipoxygenase | Arachidonate 5-lipoxygenase | Homo sapiens | enzyme reductase | Small molecule | 1996 |
| P14416 | ZIPRASIDONE | Dopamine D2 receptor antagonist | CHEMBL217 | Dopamine D2 receptor | D(2) dopamine receptor | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor dopamine receptor | Small molecule | 2001 |
| P28223 | ZIPRASIDONE | Serotonin 2a (5-HT2a) receptor antagonist | CHEMBL224 | Serotonin 2a (5-HT2a) receptor | 5-hydroxytryptamine receptor 2A | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P28335 | ZIPRASIDONE | Serotonin 2c (5-HT2c) receptor antagonist | CHEMBL225 | Serotonin 2c (5-HT2c) receptor | 5-hydroxytryptamine receptor 2C | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 2001 |
| P14324 | ZOLEDRONIC ACID | Farnesyl diphosphate synthase inhibitor | CHEMBL1782 | Farnesyl diphosphate synthase | Farnesyl pyrophosphate synthase | Homo sapiens | enzyme transferase | Small molecule | 2001 |
| P28221 | ZOLMITRIPTAN | Serotonin 1d (5-HT1d) receptor agonist | CHEMBL1983 | Serotonin 1d (5-HT1d) receptor | 5-hydroxytryptamine receptor 1D | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1997 |
| P28222 | ZOLMITRIPTAN | Serotonin 1b (5-HT1b) receptor agonist | CHEMBL1898 | Serotonin 1b (5-HT1b) receptor | 5-hydroxytryptamine receptor 1B | Homo sapiens | membrane receptor 7tm1 smallmol monoamine receptor serotonin receptor | Small molecule | 1997 |
| P18505 | ZOLPIDEM | GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator | CHEMBL2111392 | GABA A receptor alpha-1/beta-1/gamma-2 | Gamma-aminobutyric acid receptor subunit beta-1 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P18507 | ZOLPIDEM | GABA A receptor alpha-1/beta-1/gamma-2 positive allosteric modulator | CHEMBL2111392 | GABA A receptor alpha-1/beta-1/gamma-2 | Gamma-aminobutyric acid receptor subunit gamma-2 | Homo sapiens | ion channel lgic gabaa | Small molecule | 1992 |
| P35498 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 1 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| P35499 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 4 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q01118 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 7 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q14524 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 5 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q15858 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 9 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q99250 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 2 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9NY46 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 3 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UI33 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 11 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9UQD0 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 8 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |
| Q9Y5Y9 | ZONISAMIDE | Sodium channel alpha subunit blocker | CHEMBL2331043 | Sodium channel alpha subunit | Sodium channel protein type 10 subunit alpha | Homo sapiens | ion channel vgc vg na | Small molecule | 2000 |