Compound Information
Test on : RBC, Millipore
Compound Name
RBC : 1,3-Benzodioxole, 5-(2-nitroethenyl)-
Millipore : 1485-00-3
Inchikey
Same : KFLWBZPSJQPRDD-N
RBC : KFLWBZPSJQPRDD-UHFFFAOYSA-N
Millipore : KFLWBZPSJQPRDD-ONEGZZNKSA-N
ChemSpider
RBC : 85667
Millipore : 585303
Pubchem CID
RBC : 94945
Millipore : 672296
ChEMBL
RBC : -
Millipore : CHEMBL596380
| RBC | Millipore |
 |  |
|
DRx |
RBC |
Metz |
Millipore |
GPCR |
| bioactivity |
Kd (nM) |
Remain Activity (%) |
Ki (nM) |
Remain Activity (%) |
Inhibition (%) |
| active criteria |
<3000nM |
<50% |
<1000nM |
<50% |
>50% |
AGC
AGC - PDK1
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PDK1 | inactive (89.39%) | inactive (106%) |
AGC - Akt
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| AKT1 | inactive (102.54%) | inactive (100%) |
| AKT2 | inactive (90.77%) | inactive (111%) |
| AKT3 | inactive (95.55%) | inactive (125%) |
AGC - DMPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| DMPK1 | inactive (106.11%) | inactive (137%) |
| MRCKa | inactive (109.89%) | inactive (106%) |
| MRCKb | inactive (97.25%) | inactive (83%) |
| ROCK1 | inactive (109.87%) | inactive (109%) |
| ROCK2 | inactive (89.07%) | inactive (99%) |
AGC - GRK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| BARK1 | inactive (107.29%) | - |
| BARK2 | inactive (101.59%) | - |
| GPRK4 | inactive (101.84%) | - |
| GPRK5 | inactive (115.5%) | inactive (106%) |
| GPRK6 | inactive (99.33%) | inactive (105%) |
| GPRK7 | inactive (107.18%) | inactive (103%) |
AGC - RSK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MSK1 | inactive (103.35%) | inactive (125%) |
| MSK2 | inactive (85.3%) | inactive (90%) |
| p70S6K | inactive (101.72%) | inactive (137%) |
| p70S6Kb | inactive (98.85%) | - |
| RSK2 | inactive (93.08%) | inactive (118%) |
| RSK4 | inactive (111.19%) | inactive (128%) |
| RSK1 | inactive (95.75%) | inactive (105%) |
| RSK3 | inactive (93.78%) | inactive (137%) |
AGC - PKA
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PKACg | inactive (100.97%) | - |
| PRKX | inactive (95.62%) | inactive (102%) |
| PKACa | inactive (101.18%) | inactive (124%) |
AGC - PKC
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PKCa | inactive (120.64%) | inactive (111%) |
| PKCd | inactive (78.79%) | inactive (99%) |
| PKCe | inactive (92.69%) | inactive (81%) |
| PKCh | inactive (103.24%) | inactive (100%) |
| PKCg | inactive (103.78%) | inactive (103%) |
| PKCi | inactive (96.7%) | inactive (93%) |
| PKCt | inactive (111.29%) | inactive (95%) |
| PKCz | inactive (91.73%) | inactive (93%) |
| PKCb | inactive (101.91%) | - |
AGC - PKG
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PKG2 | inactive (94.68%) | - |
| PKG1 | inactive (72.62%) | - |
AGC - PKN
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PKN1 | inactive (91.58%) | - |
| PKN2 | inactive (82.22%) | inactive (102%) |
AGC - SGK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| SGK1 | inactive (96.07%) | inactive (76%) |
| SGK2 | inactive (102.23%) | inactive (89%) |
| SGK3 | inactive (92.77%) | inactive (110%) |
AGC - NDR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| NDR1 | inactive (103.1%) | - |
TK
TK - Abl
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ABL1 | inactive (99.97%) | inactive (96%) |
| ABL2 | inactive (96.01%) | inactive (104%) |
TK - Ack
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ACK | inactive (99.22%) | inactive (83%) |
TK - ALK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ALK | inactive (109.44%) | inactive (84%) |
| LTK | inactive (96.45%) | - |
TK - Axl
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| AXL | inactive (99.1%) | inactive (69%) |
| MER | inactive (77.62%) | inactive (106%) |
| TYRO3 | inactive (103.22%) | inactive (100%) |
TK - Src
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| BLK | inactive (102.34%) | inactive (120%) |
| BRK | inactive (86.53%) | inactive (113%) |
| SRC | inactive (89.3%) | inactive (89%) |
| FGR | inactive (96.45%) | inactive (90%) |
| FRK | inactive (101.52%) | inactive (105%) |
| FYN | inactive (111.67%) | inactive (105%) |
| HCK | inactive (92.12%) | inactive (85%) |
| LCK | inactive (97.93%) | inactive (135%) |
| SRM | inactive (105.04%) | - |
| YES | inactive (107.99%) | inactive (118%) |
| LYN | inactive (96.61%) | inactive (90%) |
TK - Tec
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| BMX | inactive (77.6%) | inactive (98%) |
| BTK | inactive (92.53%) | inactive (96%) |
| ITK | inactive (102.53%) | inactive (105%) |
| TEC | inactive (133.68%) | - |
| TXK | inactive (101.88%) | inactive (76%) |
TK - PDGFR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| KIT | inactive (95.25%) | inactive (113%) |
| FLT3 | inactive (94.17%) | inactive (95%) |
| FMS | inactive (101.54%) | inactive (87%) |
| PDGFRb | inactive (110.33%) | inactive (94%) |
| PDGFRa | inactive (91.14%) | inactive (114%) |
TK - Csk
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CSK | inactive (101.25%) | inactive (112%) |
| CTK | inactive (90.84%) | - |
TK - DDR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| DDR2 | inactive (96.26%) | inactive (100%) |
TK - EGFR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| EGFR | inactive (96.58%) | inactive (132%) |
| ErbB2 | inactive (93.48%) | - |
| ErbB4 | inactive (81.69%) | inactive (86%) |
TK - Eph
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| EphA1 | inactive (98.79%) | inactive (95%) |
| EphA2 | inactive (103.34%) | inactive (106%) |
| EphA3 | inactive (104.43%) | inactive (115%) |
| EphA4 | inactive (97.57%) | inactive (112%) |
| EphA5 | inactive (94.99%) | inactive (103%) |
| EphA6 | inactive (99.06%) | - |
| EphA7 | inactive (86.78%) | inactive (95%) |
| EphA8 | inactive (91.61%) | inactive (100%) |
| EphB1 | inactive (96.39%) | inactive (115%) |
| EphB2 | inactive (98.1%) | inactive (116%) |
| EphB3 | inactive (97.85%) | inactive (117%) |
| EphB4 | inactive (87.47%) | inactive (114%) |
TK - FAK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| FAK | inactive (100.43%) | inactive (141%) |
| PYK2 | inactive (97.01%) | inactive (129%) |
TK - Fer
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| FER | inactive (88.02%) | inactive (114%) |
| FES | inactive (101.75%) | inactive (113%) |
TK - FGFR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| FGFR1 | inactive (88.59%) | inactive (115%) |
| FGFR2 | inactive (111.06%) | inactive (108%) |
| FGFR3 | inactive (96.9%) | inactive (104%) |
| FGFR4 | inactive (80.93%) | inactive (135%) |
TK - VEGFR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| FLT1 | inactive (89.78%) | inactive (97%) |
| FLT4 | inactive (94.91%) | inactive (88%) |
| KDR | inactive (104.09%) | inactive (101%) |
TK - InsR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| IGF1R | inactive (104.96%) | inactive (131%) |
| IRR | inactive (96.37%) | inactive (106%) |
| INSR | inactive (87.19%) | inactive (117%) |
TK - JakA
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| JAK1 | inactive (99.79%) | - |
| JAK2 | inactive (96.8%) | inactive (73%) |
| JAK3 | inactive (92.78%) | inactive (114%) |
| TYK2 | inactive (98.62%) | - |
TK - Musk
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MUSK | inactive (106.64%) | inactive (127%) |
TK - Ret
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| RET | inactive (91.36%) | inactive (96%) |
TK - Met
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| RON | inactive (101.22%) | inactive (100%) |
| MET | inactive (87.7%) | inactive (111%) |
TK - Sev
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ROS | inactive (101.15%) | inactive (95%) |
TK - Syk
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| SYK | inactive (98.86%) | inactive (123%) |
| ZAP70 | inactive (112.16%) | inactive (111%) |
TK - Tie
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| TIE2 | inactive (99.06%) | inactive (80%) |
TK - Trk
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| TRKA | inactive (91.01%) | inactive (94%) |
| TRKB | inactive (98.59%) | inactive (120%) |
| TRKC | inactive (100.3%) | - |
TKL
TKL - STKR
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ALK1 | inactive (100.18%) | - |
| ALK2 | inactive (96.39%) | - |
| ALK4 | inactive (98.85%) | inactive (133%) |
| TGFbR1 | inactive (100.41%) | inactive (90%) |
| TGFbR2 | inactive (122.82%) | - |
TKL - RAF
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ARAF | inactive (94.4%) | - |
| BRAF | inactive (99.31%) | - |
| RAF1 | inactive (87.33%) | inactive (87%) |
TKL - IRAK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| IRAK1 | inactive (119.63%) | inactive (95%) |
| IRAK4 | inactive (98.56%) | inactive (116%) |
TKL - LISK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| LIMK1 | inactive (93.25%) | inactive (114%) |
TKL - LRRK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| LRRK2 | inactive (100.39%) | - |
TKL - MLK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MLK1 | inactive (89.83%) | inactive (100%) |
| MLK2 | inactive (95.62%) | - |
| MLK3 | inactive (96.04%) | - |
| TAK1 | inactive (100.9%) | inactive (92%) |
| ZAK | inactive (101.63%) | - |
TKL - RIPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| RIPK2 | inactive (94.71%) | inactive (100%) |
CAMK
CAMK - CAMKL
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| NuaK1 | inactive (91.65%) | inactive (107%) |
| BRSK1 | inactive (100.55%) | inactive (92%) |
| BRSK2 | inactive (102.19%) | inactive (113%) |
| CHK1 | inactive (98.29%) | inactive (85%) |
| LKB1 | inactive (91.56%) | inactive (105%) |
| MARK1 | inactive (111.72%) | inactive (91%) |
| MARK3 | inactive (86.87%) | - |
| MARK4 | inactive (112.18%) | - |
| MELK | inactive (95.92%) | inactive (78%) |
| PASK | inactive (83.52%) | inactive (107%) |
| QIK | inactive (97.51%) | - |
| NuaK2 | inactive (150.43%) | - |
| MARK2 | inactive (92.89%) | inactive (99%) |
| AMPKa1 | - | inactive (89%) |
| AMPKa2 | - | inactive (101%) |
| SIK | - | inactive (100%) |
CAMK - CAMK1
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CaMK1a | inactive (95.11%) | inactive (108%) |
| CaMK1b | inactive (92.42%) | - |
| CaMK1d | inactive (99.52%) | inactive (123%) |
| CaMK1g | inactive (96.98%) | - |
| CaMK4 | inactive (95.62%) | inactive (132%) |
CAMK - CAMK2
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CaMK2a | inactive (101.47%) | - |
| CaMK2b | inactive (90.85%) | inactive (90%) |
| CaMK2d | inactive (96.43%) | inactive (109%) |
| CaMK2g | inactive (94.32%) | inactive (107%) |
CAMK - RAD53
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CHK2 | inactive (96.08%) | inactive (85%) |
CAMK - DAPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| DAPK1 | inactive (108.98%) | inactive (85%) |
| DAPK2 | inactive (103.73%) | inactive (95%) |
| DRAK1 | inactive (115.7%) | inactive (119%) |
| DAPK3 | inactive (99.16%) | inactive (96%) |
CAMK - DCAMKL
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| DCLK2 | inactive (95.62%) | inactive (63%) |
CAMK - MAPKAPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MAPKAPK2 | inactive (98.97%) | inactive (84%) |
| MAPKAPK3 | inactive (93.52%) | inactive (93%) |
| MAPKAPK5 | inactive (93.74%) | inactive (85%) |
| MNK1 | inactive (93.51%) | - |
| MNK2 | inactive (90.2%) | inactive (116%) |
CAMK - MLCK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| smMLCK | inactive (105.86%) | inactive (89%) |
| skMLCK | inactive (100.38%) | - |
CAMK - PHK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PHKg1 | inactive (93.92%) | - |
| PHKg2 | inactive (98.61%) | inactive (105%) |
CAMK - PIM
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PIM1 | inactive (104.15%) | inactive (79%) |
| PIM2 | inactive (93.63%) | inactive (134%) |
| PIM3 | inactive (83.96%) | inactive (101%) |
CAMK - PKD
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PKD1 | inactive (101.67%) | inactive (91%) |
| PKD3 | inactive (94.21%) | - |
| PKD2 | inactive (99.7%) | inactive (105%) |
CAMK - TSSK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| TSSK1 | inactive (109.06%) | inactive (96%) |
| TSSK2 | inactive (111.57%) | inactive (87%) |
CAMK - STK33
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| STK33 | inactive (94.22%) | inactive (93%) |
STE
STE - STE11
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MAP3K5 | inactive (105.06%) | inactive (109%) |
| MAP3K2 | inactive (76.88%) | - |
| MAP3K3 | inactive (89.5%) | - |
STE - STE-Unique
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| COT | inactive (97.88%) | - |
| NIK | inactive (106.13%) | - |
STE - STE20
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| GCK | inactive (102.42%) | inactive (92%) |
| HGK | inactive (89.84%) | - |
| KHS1 | inactive (105.53%) | - |
| LOK | inactive (91.9%) | inactive (104%) |
| MINK | inactive (105.79%) | inactive (97%) |
| MST1 | inactive (104.51%) | inactive (101%) |
| MST2 | inactive (106.92%) | inactive (104%) |
| MST3 | inactive (102.29%) | inactive (77%) |
| MST4 | inactive (103.11%) | - |
| OSR1 | inactive (92.23%) | - |
| PAK1 | inactive (96.85%) | - |
| PAK2 | inactive (73.25%) | inactive (111%) |
| PAK3 | inactive (101.38%) | inactive (112%) |
| PAK4 | inactive (88.71%) | inactive (91%) |
| PAK5 | inactive (97.58%) | inactive (103%) |
| PAK6 | inactive (104.9%) | inactive (105%) |
| SLK | inactive (103%) | - |
| YSK1 | inactive (96.68%) | - |
| STLK3 | inactive (89.29%) | - |
| TAO1 | inactive (93.35%) | inactive (101%) |
| TAO2 | inactive (92.04%) | inactive (107%) |
| TAO3 | inactive (101.32%) | inactive (90%) |
| MYO3B | inactive (92.91%) | - |
STE - STE7
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MAP2K1 | inactive (90.65%) | inactive (127%) |
| MAP2K2 | inactive (106.07%) | - |
| MAP2K6 | inactive (115.24%) | inactive (85%) |
| MAP2K7 | - | inactive (112%) |
Other
Other - Aur
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| AurA | inactive (96.16%) | inactive (99%) |
| AurB | inactive (94.61%) | inactive (108%) |
| AurC | inactive (83.7%) | inactive (102%) |
Other - CAMKK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CaMKK1 | inactive (105.48%) | - |
| CaMKK2 | inactive (96.94%) | - |
Other - Haspin
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| Haspin | inactive (99.33%) | inactive (128%) |
Other - IKK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| IKKa | inactive (115.4%) | inactive (91%) |
| IKKb | inactive (104.65%) | inactive (98%) |
| IKKe | inactive (103.75%) | - |
| TBK1 | inactive (94.04%) | inactive (87%) |
Other - NEK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| NEK1 | inactive (96.22%) | - |
| NEK11 | inactive (94.45%) | inactive (90%) |
| NEK2 | inactive (91.89%) | inactive (87%) |
| NEK4 | inactive (110.32%) | - |
| NEK6 | inactive (109.4%) | inactive (109%) |
| NEK7 | inactive (104.46%) | inactive (99%) |
| NEK9 | inactive (91.08%) | - |
| NEK3 | inactive (92.19%) | inactive (114%) |
Other - TOPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PBK | inactive (90.23%) | - |
Other - PLK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PLK1 | inactive (99.03%) | inactive (96%) |
| PLK2 | inactive (98.88%) | inactive (102%) |
| PLK3 | inactive (95.85%) | inactive (96%) |
Other - SgK496
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| SgK496 | inactive (89.48%) | - |
Other - NAK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MPSK1 | inactive (105.83%) | - |
Other - TTK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| TTK | inactive (103.9%) | - |
Other - ULK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| ULK1 | inactive (82.85%) | - |
| ULK2 | inactive (103.94%) | inactive (102%) |
| ULK3 | inactive (65.36%) | inactive (111%) |
Other - WEE
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| Wee1 | inactive (87.11%) | - |
Other - WNK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| Wnk2 | inactive (99.74%) | inactive (109%) |
| Wnk3 | inactive (102.07%) | inactive (88%) |
Other - TLK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| TLK2 | inactive (77.87%) | inactive (99%) |
CK1
CK1
| Test Member No. in Family |
|---|
| Family | no. Member on 518kinase | RBC | Millipore |
|---|
| CK1 | 7 | 6 | 4 |
| VRK | 3 | 1 | 1 |
CK1 - CK1
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CK1d | inactive (102.25%) | inactive (98%) |
| CK1g1 | inactive (102.96%) | inactive (83%) |
| CK1g2 | inactive (102.42%) | inactive (89%) |
| CK1g3 | inactive (109.55%) | inactive (107%) |
| CK1a | inactive (102.2%) | - |
| CK1e | inactive (92.82%) | - |
CK1 - VRK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| VRK1 | inactive (103.4%) | - |
| VRK2 | - | inactive (101%) |
CMGC
CMGC
| Test Member No. in Family |
|---|
| Family | no. Member on 518kinase | RBC | Millipore |
|---|
| CK2 | 3 | 2 | 2 |
| CLK | 4 | 4 | 2 |
| DYRK | 10 | 9 | 4 |
| MAPK | 14 | 10 | 10 |
| GSK | 2 | 2 | 2 |
| SRPK | 3 | 3 | 3 |
CMGC - CK2
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CK2a1 | inactive (110.95%) | inactive (105%) |
| CK2a2 | inactive (91.15%) | inactive (134%) |
CMGC - CLK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| CLK1 | inactive (115.01%) | - |
| CLK2 | inactive (99.32%) | inactive (121%) |
| CLK3 | inactive (94.45%) | inactive (91%) |
| CLK4 | inactive (105.91%) | - |
CMGC - DYRK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| DYRK1A | inactive (82.92%) | - |
| DYRK1B | inactive (111.74%) | - |
| DYRK2 | inactive (100.25%) | inactive (101%) |
| DYRK3 | inactive (94.58%) | - |
| DYRK4 | inactive (84.94%) | - |
| HIPK1 | inactive (99.36%) | inactive (96%) |
| HIPK2 | inactive (90.09%) | inactive (93%) |
| HIPK3 | inactive (98.76%) | inactive (101%) |
| HIPK4 | inactive (92.54%) | - |
CMGC - MAPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| Erk1 | inactive (99.35%) | inactive (78%) |
| Erk2 | inactive (107.5%) | inactive (106%) |
| JNK3 | inactive (90.98%) | inactive (88%) |
| NLK | inactive (98.65%) | inactive (107%) |
| p38a | inactive (125.61%) | inactive (93%) |
| p38b | inactive (104.65%) | inactive (102%) |
| p38d | inactive (97.28%) | inactive (103%) |
| p38g | inactive (94.51%) | inactive (107%) |
| JNK1 | inactive (104.48%) | inactive (120%) |
| JNK2 | inactive (94.53%) | inactive (99%) |
CMGC - GSK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| GSK3A | inactive (93.77%) | inactive (125%) |
| GSK3B | inactive (105.37%) | inactive (108%) |
CMGC - SRPK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| MSSK1 | inactive (97.68%) | inactive (120%) |
| SRPK1 | inactive (101.52%) | inactive (111%) |
| SRPK2 | inactive (91.17%) | inactive (97%) |
Atypical
Atypical
| Test Member No. in Family |
|---|
| Family | no. Member on 518kinase | RBC | Millipore |
|---|
| PDHK | 5 | 1 | - |
| Alpha | 6 | - | 1 |
| PIKK | 6 | - | 1 |
Atypical - PDHK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| PDHK1 | inactive (89.39%) | - |
Atypical - Alpha
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| eEF2K | - | inactive (89%) |
Atypical - PIKK
| Bioactivity |
|---|
| Kinase | RBC | Millipore |
|---|
| FRAP | - | inactive (106%) |