Showing entry for Linonin



                             
General Compound Information
BXGC IdBXGC0003235
Compound NameLinonin
Structure
FormulaC26H30O8
InchiKeyKBDSLGBFQAGHBE-MSGMIQHVSA-N
SMILESCC1(C)O[C@H]2CC(=O)OC[C@@]22[C@H]1CC(=O)[C@]1(C)[C@@H]2CC[C@@]2(C)[C@@H](OC(=O)[C@H]3O[C@@]123)C1=COC=C1
InchiInChI=1S/C26H30O8/c1-22(2)15-9-16(27)24(4)14(25(15)12-31-18(28)10-17(25)33-22)5-7-23(3)19(13-6-8-30-11-13)32-21(29)20-26(23,24)34-20/h6,8,11,14-15,17,19-20H,5,7,9-10,12H2,1-4H3/t14-,15-,17-,19-,20+,23-,24-,25+,26+/m0/s1
IUPAC(1R,2R,7S,10R,13R,14R,16S,19R,20S)-19-(furan-3-yl)-9,9,13,20-tetramethyl-4,8,15,18-tetraoxahexacyclo[11.9.0.02,?.02,1?.01?,1?.01?,2?]docosane-5,12,17-trione
Molecular Weight470.52
Pubchem Id179651
Chembl IdCHEMBL517449
Targets of Information Source
DrugBank n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
PDB n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Binding DB n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
CHEMBL CHEMBL517449
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Kinact '=' 0 min-1
O42275 BXGT004559 Acetylcholinesterase reviewed - ache Inhibition '=' 0 %
Q9WKE8 BXGT021921 Reverse transcriptase unreviewed - reverse IC50 '=' 0 ug.mL-1
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '>' 100000 nM
Q9WKE8 BXGT021921 Reverse transcriptase unreviewed - reverse IC50 '=' 0 ug.mL-1
Q9WKE8 BXGT021921 Reverse transcriptase unreviewed - reverse IC50 '>' 200 ug.mL-1
P14679 BXGT008039 Tyrosinase reviewed Enzyme TYR Inhibition '=' 3 %
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Ki '=' 23200 nM
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 Inhibition '=' 92 %
P81908 BXGT011959 Cholinesterase reviewed - BCHE Inhibition '=' -14 %
Q9Y6L6 BXGT022334 Solute carrier organic anion transporter family member 1B1 reviewed Transporter SLCO1B1 Inhibition '=' 102 %
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF00054 Lemon Citrus limon Fruits
BXGF00055 Pummelo Citrus maxima Fruits
BXGF00056 Mandarin orange (Clementine, Tangerine) Citrus reticulata Fruits
BXGF00057 Sweet orange Citrus sinensis Fruits
BXGF00165 Common sage Salvia officinalis Herbs and Spices
BXGF00871 Citrus unshiu Citrus unshiu Medicinal Plant
BXGF00875 Glycosmis pseudoracemosa Glycosmis pseudoracemosa Medicinal Plant
BXGF01005 Dictamnus dasycarpus Dictamnus dasycarpus Medicinal Plant
BXGF01063 Corydalis persica Corydalis persica Others
BXGF01067 Salta triflora Salta triflora Others
BXGF01136 Inula grantioides Inula grantioides Medicinal Plant
BXGF01152 Vernonia chloropappa Vernonia chloropappa Others
BXGF01395 Juniperus horizontalis Juniperus horizontalis Medicinal Plant
BXGF01577 Strychnos spinosa Strychnos spinosa Medicinal Plant
BXGF01579 Esenbeckia hartmanii Esenbeckia hartmanii Others
BXGF01714 Amomum daniellii Amomum daniellii Others
BXGF01730 Aeollanthus buchnerianus Aeollanthus buchnerianus Others
BXGF01852 Plectranthus caninus Plectranthus caninus Medicinal Plant
BXGF01935 Lathyrus tingitanus Lathyrus tingitanus Human Edible Plant
BXGF01966 Chromolaena odorata Chromolaena odorata Medicinal Plant
BXGF01969 Echium plantagineum Echium plantagineum Medicinal Plant
BXGF01970 Rauvolfia salicifolia Rauvolfia salicifolia Others
BXGF01990 Balanophora japonica Balanophora japonica Medicinal Plant
BXGF02106 Citrus medica Citrus medica Medicinal Plant
BXGF02237 Citrus wilsonii Citrus wilsonii Medicinal Plant
BXGF02252 Leptospermum recurvum Leptospermum recurvum Others
BXGF02350 Cota tinctoria Cota tinctoria Medicinal Plant
BXGF02357 Euodia bodinieri Euodia bodinieri Others
BXGF02424 Pycnarrhena australiana Pycnarrhena australiana Others
BXGF02592 Ilex affinis Ilex affinis Human Edible Plant
BXGF02600 Berberis repens Berberis repens Others
BXGF02667 Anaxagorea clavata Anaxagorea clavata Others
BXGF02804 Hernandia sonora Hernandia sonora Medicinal Plant
BXGF02838 Helianthus niveus Helianthus niveus Medicinal Plant
BXGF02978 Tetradium ruticarpum Tetradium ruticarpum Medicinal Plant
BXGF03038 Oricia suaveolens Oricia suaveolens Others
BXGF03144 Stenostomum lucidum Stenostomum lucidum Others
BXGF03147 Beyeria brevifolia Beyeria brevifolia Others
BXGF03227 Cynoglossum viridiflorum Cynoglossum viridiflorum Others
BXGF03327 Citrus trifoliata Citrus trifoliata Human Edible Plant
BXGF03421 Kaempferia pulchra Kaempferia pulchra Medicinal Plant
BXGF03427 Phellodendron chinense Phellodendron chinense Medicinal Plant
BXGF03534 Drosera peltata Drosera peltata Medicinal Plant
BXGF03625 Alchornea cordifolia Alchornea cordifolia Medicinal Plant
BXGF03706 Tetradium glabrifolium Tetradium glabrifolium Others
BXGF03712 Arnica nevadensis Arnica nevadensis Others
BXGF03745 Odixia angusta Odixia angusta Others
BXGF03760 Prunus laurocerasus Prunus laurocerasus Medicinal Plant
BXGF03812 Ficus formosana Ficus formosana Human Edible Plant
BXGF03828 Phellodendron amurense Phellodendron amurense Medicinal Plant
BXGF03843 Dipterocarpus alatus Dipterocarpus alatus Medicinal Plant
BXGF03864 Echinops amplexicaulis Echinops amplexicaulis Medicinal Plant
BXGF03873 Quercus aegilops Quercus aegilops Medicinal Plant
BXGF03883 Chloranthus tianmushanensis Chloranthus tianmushanensis Others
BXGF03897 Prosopis glandulosa Prosopis glandulosa Human Edible Plant
BXGF03916 Aria pallescens Aria pallescens Others
BXGF03926 Simira eliezeriana Simira eliezeriana Others
BXGF03939 Senecio squalidus Senecio squalidus Medicinal Plant
BXGF03951 Araujia sericifera Araujia sericifera Medicinal Plant
BXGF03966 Artemisia monogyna Artemisia monogyna Others
BXGF03986 Epaltes gariepina Epaltes gariepina Others
BXGF03991 Seriphidium cinum Seriphidium cinum Medicinal Plant
BXGF04002 Dendrosenecio kilimanjari Dendrosenecio kilimanjari Others
BXGF04009 Isodon kameba Isodon kameba Medicinal Plant
BXGF04016 Pterocarpus grandiflorus Pterocarpus grandiflorus Others
BXGF04030 Chromolaena pulchella Chromolaena pulchella Others
BXGF04041 Bursaria spinosa Bursaria spinosa Human Edible Plant
BXGF04054 Taxodium mucronatum Taxodium mucronatum Medicinal Plant
BXGF04066 Gardenia fosbergii Gardenia fosbergii Others
BXGF04073 Vitex madiensis Vitex madiensis Medicinal Plant
BXGF04144 Agnorhiza bolanderi Agnorhiza bolanderi Others
BXGF04256 Phellodendron chinese Phellodendron chinese Others
BXGF04371 Citrus yuko Citrus yuko Others
BXGF04708 Sesbania punicea Sesbania punicea Others
BXGF04928 Citrus grandis Citrus grandis Medicinal Plant
BXGF05111 Trifolium montanum Trifolium montanum Others
BXGF05188 Corynanthe pachyceras Corynanthe pachyceras Others
BXGF05356 Euodia officinalis Euodia officinalis Others
BXGF05431 Citrus natsudaidai Citrus natsudaidai Human Edible Plant
BXGF05455 Peucedanum oroselinum Peucedanum oroselinum Others
BXGF05463 Ageratina saltillensis Ageratina saltillensis Others
BXGF05470 Thalictrum lucidum Thalictrum lucidum Others
BXGF05471 Cynoglossum amabile Cynoglossum amabile Medicinal Plant
BXGF05506 Coptis chinensis Coptis chinensis Medicinal Plant
BXGF05704 Securidaca inappendiculata Securidaca inappendiculata Medicinal Plant
BXGF05746 Atalantia wightii Atalantia wightii Others
BXGF05797 Salvia polystachya Salvia polystachya Medicinal Plant
BXGF05819 Citrus aurantium Citrus aurantium Medicinal Plant
BXGF05843 Pteris prolifera Pteris prolifera Others
BXGF05939 Grewia villosa Grewia villosa Medicinal Plant
BXGF06002 Euodia ruticarpa Euodia ruticarpa Others
BXGF06044 Citrus junos Citrus junos Medicinal Plant
BXGF06143 Persicaria tinctoria Persicaria tinctoria Medicinal Plant
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease