| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
39810 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
11000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
141 |
% |
| Q9UGP5 |
BXGT021689 |
DNA polymerase lambda |
reviewed |
Enzyme |
POLL |
Inhibition |
- |
- |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
31622 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
2818 |
nM |
| B2GV46 |
BXGT001957 |
Free fatty acid receptor 3 |
reviewed |
- |
Ffar3 |
EC50 |
- |
- |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
142 |
fmol |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
3 |
% |
| P04416 |
BXGT006211 |
Phospholipase A2, minor isoenzyme |
reviewed |
- |
|
K |
'=' |
1 |
10'4/M |
| P00592 |
BXGT005593 |
Phospholipase A2, major isoenzyme |
reviewed |
- |
PLA2G1B |
K |
'=' |
1 |
10'4/M |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
EC50 |
'=' |
316 |
nM |
| P05413 |
BXGT006355 |
Fatty acid-binding protein, heart |
reviewed |
- |
FABP3 |
IC50 |
'=' |
1000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
56234 |
nM |
| P51452 |
BXGT010849 |
Dual specificity protein phosphatase 3 |
reviewed |
- |
DUSP3 |
IC50 |
'>' |
100000 |
nM |
| P35610 |
BXGT009855 |
Sterol O-acyltransferase 1 |
reviewed |
Enzyme |
SOAT1 |
IC50 |
'>' |
1000000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
17782 |
nM |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'=' |
94000 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
31622 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Inhibition |
- |
- |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
48000 |
nM |
| P00761 |
BXGT005645 |
Trypsin |
reviewed |
- |
|
IC50 |
'>' |
200000 |
nM |
| O70536 |
BXGT005069 |
Sterol O-acyltransferase 1 |
reviewed |
- |
Soat1 |
IC50 |
'>' |
1000000 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
158 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
31622 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
177 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
85 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Potency |
- |
44668 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Regiospecificity |
- |
- |
- |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
26608 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
147 |
% |
| P13726 |
BXGT007950 |
Tissue factor |
reviewed |
Receptor |
F3 |
IC50 |
'=' |
41000 |
nM |
| P08709 |
BXGT006818 |
Coagulation factor VII |
reviewed |
Enzyme |
F7 |
IC50 |
'=' |
41000 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
31622 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
IC50 |
'=' |
65000 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
IC50 |
'=' |
1100 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
1800 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
8912 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
549 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
FC |
'=' |
2 |
- |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
170000 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Kd |
'=' |
4 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
1000 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
28183 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
44668 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Inhibition |
'=' |
81 |
% |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
IC50 |
'=' |
1000 |
nM |
| Q76JU9 |
BXGT016859 |
Free fatty acid receptor 1 |
reviewed |
- |
Ffar1 |
Activity |
'=' |
141 |
% |
| Q76JU9 |
BXGT016859 |
Free fatty acid receptor 1 |
reviewed |
- |
Ffar1 |
Activity |
'=' |
172 |
% |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
540 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
22387 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
IC50 |
'=' |
13600 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
26679 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
22 |
% |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
0 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
234 |
% |
| P35236 |
BXGT009802 |
Tyrosine-protein phosphatase non-receptor type 7 |
reviewed |
Enzyme |
PTPN7 |
IC50 |
'>' |
100000 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
Activity |
- |
- |
- |
| O14746 |
BXGT004091 |
Telomerase reverse transcriptase |
reviewed |
Enzyme |
TERT |
Activity |
'=' |
10 |
% |
| P05413 |
BXGT006355 |
Fatty acid-binding protein, heart |
reviewed |
- |
FABP3 |
Ki |
'=' |
9300 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
10 |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
35481 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
IC50 |
'=' |
6200 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Potency |
- |
28183 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
50118 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
56234 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
15848 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
28183 |
nM |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
Rmax |
'=' |
138 |
% |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
4800 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
IC50 |
'=' |
17700 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
13000 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
IC50 |
'=' |
10000 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Inhibition |
'=' |
85 |
% |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Ki |
'=' |
6800 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
13000 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Delta Tm |
'=' |
1 |
degrees C |