| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
Ki |
'=' |
135 |
nM |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
Ki |
'=' |
135 |
nM |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Ki |
'=' |
135 |
nM |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
Ki |
'=' |
135 |
nM |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
Ki |
'=' |
135 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Ki |
'=' |
135 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Ki |
'=' |
135 |
nM |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
Ki |
'=' |
135 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Ki |
'=' |
135 |
nM |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Ki |
'=' |
135 |
nM |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Ki |
'=' |
135 |
nM |
| P42224 |
BXGT010286 |
Signal transducer and activator of transcription 1-alpha/beta |
reviewed |
Nucleic acid binding |
STAT1 |
Inhibition |
'=' |
-3 |
% |
| P40763 |
BXGT010202 |
Signal transducer and activator of transcription 3 |
reviewed |
Nucleic acid binding |
STAT3 |
Inhibition |
'=' |
5 |
% |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
Activity |
'=' |
40 |
% |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
Activity |
'=' |
40 |
% |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Activity |
'=' |
40 |
% |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
Activity |
'=' |
40 |
% |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
Activity |
'=' |
40 |
% |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Activity |
'=' |
40 |
% |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Activity |
'=' |
40 |
% |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
Activity |
'=' |
40 |
% |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Activity |
'=' |
40 |
% |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Activity |
'=' |
40 |
% |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Activity |
'=' |
40 |
% |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Inhibition |
'=' |
3 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'<' |
30 |
% |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
IC50 |
'=' |
375000 |
nM |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
IC50 |
'=' |
375000 |
nM |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
IC50 |
'=' |
375000 |
nM |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
IC50 |
'=' |
375000 |
nM |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
IC50 |
'=' |
375000 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
IC50 |
'=' |
375000 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
IC50 |
'=' |
375000 |
nM |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
IC50 |
'=' |
375000 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
IC50 |
'=' |
375000 |
nM |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
IC50 |
'=' |
375000 |
nM |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
IC50 |
'=' |
375000 |
nM |
| O60656 |
BXGT004889 |
UDP-glucuronosyltransferase 1-9 |
reviewed |
- |
UGT1A9 |
Activity |
'=' |
0 |
pm/min/mg |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
7 |
% |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
Inhibition |
- |
- |
- |
| Q13093 |
BXGT013310 |
Platelet-activating factor acetylhydrolase |
reviewed |
Enzyme |
PLA2G7 |
Activity |
- |
- |
- |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
87800 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
35481 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
1800 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
Inhibition |
'=' |
87 |
% |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
45800 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Km |
'=' |
1260 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
103 |
% |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
300 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
4 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
- |
- |
- |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
17782 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
58200 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
7900 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
3264 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
Inhibition |
'=' |
59 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
10 |
% |
| P51692 |
BXGT010885 |
Signal transducer and activator of transcription 5B |
reviewed |
Nucleic acid binding |
STAT5B |
Inhibition |
'=' |
-1 |
% |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Inhibition |
'=' |
12 |
% |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
31300 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
Inhibition |
'=' |
76 |
% |
| P19224 |
BXGT008468 |
UDP-glucuronosyltransferase 1-6 |
reviewed |
- |
UGT1A6 |
Activity |
'=' |
0 |
pm/min/mg |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
950 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
IC50 |
'>' |
200000 |
nM |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
IC50 |
'>' |
200000 |
nM |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
IC50 |
'>' |
200000 |
nM |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
IC50 |
'>' |
200000 |
nM |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
IC50 |
'>' |
200000 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
IC50 |
'>' |
200000 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
IC50 |
'>' |
200000 |
nM |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
IC50 |
'>' |
200000 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
IC50 |
'>' |
200000 |
nM |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
IC50 |
'>' |
200000 |
nM |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
IC50 |
'>' |
200000 |
nM |
| P03070 |
BXGT006016 |
Large T antigen |
reviewed |
- |
|
IC50 |
- |
14670 |
nM |
| O13383 |
BXGT004058 |
1,3-beta-D-glucan synthase catalytic subunit |
unreviewed |
- |
CaFKS1 |
IC50 |
'>' |
90000 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat |
'=' |
60 |
/s |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
105 |
% |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat/Km |
'=' |
48 |
/uM/s |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
12589 |
nM |
| O95398 |
BXGT005378 |
Rap guanine nucleotide exchange factor 3 |
reviewed |
Enzyme modulator |
RAPGEF3 |
Potency |
- |
31622 |
nM |
| Q8WZA2 |
BXGT019025 |
Rap guanine nucleotide exchange factor 4 |
reviewed |
Enzyme modulator |
RAPGEF4 |
Potency |
- |
39810 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
83 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
92900 |
nM |
| O43826 |
BXGT004629 |
Glucose-6-phosphate exchanger SLC37A4 |
reviewed |
Transporter |
SLC37A4 |
IC50 |
'=' |
226000 |
nM |
| O43826 |
BXGT004629 |
Glucose-6-phosphate exchanger SLC37A4 |
reviewed |
Transporter |
SLC37A4 |
Ki |
'=' |
260000 |
nM |
| P00690 |
BXGT005612 |
Pancreatic alpha-amylase |
reviewed |
- |
AMY2 |
Inhibition |
- |
- |
- |
| Q06124 |
BXGT012856 |
Tyrosine-protein phosphatase non-receptor type 11 |
reviewed |
- |
PTPN11 |
Inhibition |
'=' |
28 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
11100 |
nM |
| P29350 |
BXGT009335 |
Tyrosine-protein phosphatase non-receptor type 6 |
reviewed |
- |
PTPN6 |
Inhibition |
'=' |
32 |
% |
| P17706 |
BXGT008330 |
Tyrosine-protein phosphatase non-receptor type 2 |
reviewed |
- |
PTPN2 |
IC50 |
'=' |
77900 |
nM |
| P51452 |
BXGT010849 |
Dual specificity protein phosphatase 3 |
reviewed |
- |
DUSP3 |
Inhibition |
'=' |
30 |
% |
| P17706 |
BXGT008330 |
Tyrosine-protein phosphatase non-receptor type 2 |
reviewed |
- |
PTPN2 |
Inhibition |
'=' |
65 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Ki |
'=' |
15100 |
nM |