| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
16360 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
5040 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
35481 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
3040 |
nM |
| O35235 |
BXGT004518 |
Tumor necrosis factor ligand superfamily member 11 |
reviewed |
- |
Tnfsf11 |
Inhibition |
- |
- |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
39810 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Inhibition |
'=' |
17 |
% |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
12589 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'<' |
100000 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
15848 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'>' |
100000 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
12589 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
7 |
- |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
7 |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
15848 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
7 |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
1584 |
nM |
| P31639 |
BXGT009556 |
Sodium/glucose cotransporter 2 |
reviewed |
Transporter |
SLC5A2 |
Inhibition |
'=' |
75 |
% |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
31622 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
11220 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
31622 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
169 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
10000 |
nM |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
Activity |
- |
- |
- |
| P13866 |
BXGT007963 |
Sodium/glucose cotransporter 1 |
reviewed |
Transporter |
SLC5A1 |
Inhibition |
'<' |
25 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
3981 |
nM |
| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
7307 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
7307 |
nM |
| P62826 |
BXGT011463 |
GTP-binding nuclear protein Ran |
reviewed |
Enzyme modulator |
RAN |
Potency |
- |
7307 |
nM |
| P38398 |
BXGT010037 |
Breast cancer type 1 susceptibility protein |
reviewed |
Enzyme |
BRCA1 |
Potency |
- |
2238 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
12 |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
4 |
- |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
25118 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
Ratio IC50 |
'=' |
10 |
- |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Inhibition |
'=' |
10 |
% |
| P60568 |
BXGT011315 |
Interleukin-2 |
reviewed |
- |
IL2 |
Kd |
'=' |
5470 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
1 |
% |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Inhibition |
- |
- |
- |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Activity |
'=' |
57 |
% |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
7943 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5011 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
10 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
28183 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
2 |
- |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
- |
- |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
0 |
% |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
FC |
'=' |
1 |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
FC |
'=' |
1 |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
FC |
'=' |
1 |
- |
| Q04207 |
BXGT012755 |
Transcription factor p65 |
reviewed |
- |
Rela |
Inhibition |
- |
- |
- |
| P31750 |
BXGT009575 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
- |
Akt1 |
Inhibition |
- |
- |
- |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
4 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
114 |
% |
| Q9Z1B7 |
BXGT022403 |
Mitogen-activated protein kinase 13 |
reviewed |
- |
Mapk13 |
Inhibition |
- |
- |
- |
| Q9WUI1 |
BXGT021940 |
Mitogen-activated protein kinase 11 |
reviewed |
- |
Mapk11 |
Inhibition |
- |
- |
- |
| O08911 |
BXGT004043 |
Mitogen-activated protein kinase 12 |
reviewed |
- |
Mapk12 |
Inhibition |
- |
- |
- |
| P47811 |
BXGT010587 |
Mitogen-activated protein kinase 14 |
reviewed |
- |
Mapk14 |
Inhibition |
- |
- |
- |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
12 |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
3700 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
31622 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Inhibition |
- |
- |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
Inhibition |
- |
- |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Activity |
- |
- |
- |
| P23204 |
BXGT008836 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
- |
Ppara |
Activity |
- |
- |
- |
| P14916 |
BXGT008066 |
Urease subunit alpha |
reviewed |
- |
ureA |
IC50 |
'=' |
2003000 |
nM |
| P69996 |
BXGT011656 |
Urease subunit beta |
reviewed |
- |
ureB |
IC50 |
'=' |
2003000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
33 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
9 |
% |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Inhibition |
'>' |
90 |
% |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
1370 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
2 |
- |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
112201 |
nM |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Activity |
- |
- |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Inhibition |
'=' |
-1 |
% |