| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
8912 |
nM |
| Q57TT1 |
BXGT015153 |
Uncharacterized protein |
unreviewed |
- |
Tb927.8.6820 |
Potency |
- |
12589 |
nM |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
'>' |
50000 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
1995 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
631 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
580 |
nM |
| P03313 |
BXGT006046 |
Genome polyprotein |
reviewed |
- |
|
Inhibition |
- |
- |
- |
| Q194T1 |
BXGT013742 |
Neuraminidase |
unreviewed |
- |
NA |
Inhibition |
'=' |
3 |
% |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
354 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
17782 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'=' |
3200 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
10000 |
nM |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
112 |
% |
| P16581 |
BXGT008245 |
E-selectin |
reviewed |
- |
SELE |
IC50 |
'>' |
500000 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
15848 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
Potency |
'=' |
25118 |
nM |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'=' |
9800 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
12589 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
1000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
92 |
% |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
103 |
% |
| Q13093 |
BXGT013310 |
Platelet-activating factor acetylhydrolase |
reviewed |
Enzyme |
PLA2G7 |
Activity |
- |
- |
- |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
1000000 |
nM |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
Ki |
'=' |
9970 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
22387 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
19952 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
4216 |
nM |
| P10145 |
BXGT007542 |
Interleukin-8 |
reviewed |
Signaling |
CXCL8 |
Potency |
- |
47307 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
7780 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
7079 |
nM |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
Ki |
'=' |
7030 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
2250 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
22387 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
97 |
ug.mL-1 |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
Ki |
'=' |
4080 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
97 |
% |
| Q2PCB5 |
BXGT014154 |
Carbonic anhydrase |
unreviewed |
- |
ca |
Ki |
'=' |
4130 |
nM |
| P52020 |
BXGT010917 |
Squalene monooxygenase |
reviewed |
- |
Sqle |
IC50 |
'=' |
73000 |
nM |
| P22083 |
BXGT008727 |
Alpha-(1,3)-fucosyltransferase 4 |
reviewed |
Enzyme |
FUT4 |
IC50 |
'=' |
14000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
920 |
nM |
| Q194T1 |
BXGT013742 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
- |
- |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
10000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
67 |
% |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
4 |
% |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1995 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Inhibition |
- |
- |
- |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
14125 |
nM |
| Q72547 |
BXGT016709 |
Reverse transcriptase/RNaseH |
unreviewed |
- |
pol |
IC50 |
'>' |
100000 |
nM |
| P16109 |
BXGT008194 |
P-selectin |
reviewed |
- |
SELP |
IC50 |
'=' |
19100 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
63 |
% |
| P00883 |
BXGT005683 |
Fructose-bisphosphate aldolase A |
reviewed |
- |
ALDOA |
Potency |
'=' |
19952 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
15848 |
nM |
| P54300 |
BXGT011042 |
Autoinducer 2-binding periplasmic protein LuxP |
reviewed |
- |
luxP |
IC50 |
'=' |
50000 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'<' |
30 |
% |
| P12821 |
BXGT007849 |
Angiotensin-converting enzyme |
reviewed |
Enzyme |
ACE |
IC50 |
'=' |
7700000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
26608 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3981 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
6990 |
nM |
| P14151 |
BXGT007990 |
L-selectin |
reviewed |
- |
SELL |
IC50 |
'=' |
27600 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
50 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
50118 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
10000 |
nM |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ki |
'=' |
7490 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
25118 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
3539 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
281 |
nM |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
6070 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
4650 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
31 |
% |
| Q11130 |
BXGT013216 |
Alpha-(1,3)-fucosyltransferase 7 |
reviewed |
Enzyme |
FUT7 |
IC50 |
'=' |
60 |
nM |
| P78536 |
BXGT011847 |
Disintegrin and metalloproteinase domain-containing protein 17 |
reviewed |
- |
ADAM17 |
Inhibition |
'=' |
47 |
% |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
Ki |
'=' |
9860 |
nM |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
FC |
'=' |
1 |
- |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
0 |
pm/min/mg |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
10000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
1258 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
31622 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat |
'=' |
30 |
/s |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
1995 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
8912 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
2511 |
nM |
| P78536 |
BXGT011847 |
Disintegrin and metalloproteinase domain-containing protein 17 |
reviewed |
- |
ADAM17 |
Inhibition |
'=' |
38 |
% |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat/Km |
'=' |
0 |
/uM/s |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
31622 |
nM |
| P78536 |
BXGT011847 |
Disintegrin and metalloproteinase domain-containing protein 17 |
reviewed |
- |
ADAM17 |
Inhibition |
'=' |
43 |
% |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
0 |
- |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
Ki |
'=' |
6130 |
nM |
| Q72874 |
BXGT016711 |
Pol polyprotein |
unreviewed |
- |
pol |
IC50 |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
31622 |
nM |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
Activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
22387 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
91 |
% |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Km |
'=' |
176780 |
nM |