| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
IC50 |
'=' |
31000 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Potency |
- |
35481 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
37933 |
nM |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'>' |
500000 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
35481 |
nM |
| Q9UGP5 |
BXGT021689 |
DNA polymerase lambda |
reviewed |
Enzyme |
POLL |
Inhibition |
- |
- |
- |
| P02692 |
BXGT005921 |
Fatty acid-binding protein, liver |
reviewed |
- |
Fabp1 |
Ki |
'=' |
2900 |
nM |
| P35610 |
BXGT009855 |
Sterol O-acyltransferase 1 |
reviewed |
Enzyme |
SOAT1 |
IC50 |
'>' |
1000000 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Inhibition |
'=' |
82 |
% |
| P00761 |
BXGT005645 |
Trypsin |
reviewed |
- |
|
IC50 |
'>' |
200000 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
32700 |
nM |
| P13726 |
BXGT007950 |
Tissue factor |
reviewed |
Receptor |
F3 |
IC50 |
'=' |
80000 |
nM |
| P08709 |
BXGT006818 |
Coagulation factor VII |
reviewed |
Enzyme |
F7 |
IC50 |
'=' |
80000 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
39810 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Inhibition |
- |
- |
- |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'>' |
500000 |
nM |
| Q13315 |
BXGT013339 |
Serine-protein kinase ATM |
reviewed |
Kinase |
ATM |
Potency |
'=' |
15848 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
15848 |
nM |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
19952 |
nM |
| O95398 |
BXGT005378 |
Rap guanine nucleotide exchange factor 3 |
reviewed |
Enzyme modulator |
RAPGEF3 |
Potency |
- |
5011 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
31622 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Ki |
'=' |
185 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Ki |
'=' |
1500 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
28183 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Ratio |
'=' |
2 |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
IC50 |
'=' |
4100 |
nM |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
5623 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Ki |
'=' |
22000 |
nM |
| O70536 |
BXGT005069 |
Sterol O-acyltransferase 1 |
reviewed |
- |
Soat1 |
IC50 |
'>' |
1000000 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'>' |
10 |
ug ml-1 |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
EC50 |
'=' |
10410 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
23778 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Inhibition |
'=' |
66 |
% |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Ratio |
'=' |
1 |
- |
| P07148 |
BXGT006559 |
Fatty acid-binding protein, liver |
reviewed |
- |
FABP1 |
Kd |
'=' |
200 |
nM |
| O14746 |
BXGT004091 |
Telomerase reverse transcriptase |
reviewed |
Enzyme |
TERT |
IC50 |
'=' |
8600 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Potency |
- |
37578 |
nM |
| Q01469 |
BXGT012590 |
Fatty acid-binding protein 5 |
reviewed |
- |
FABP5 |
Ki |
'=' |
248 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
IC50 |
'=' |
26100 |
nM |
| P02692 |
BXGT005921 |
Fatty acid-binding protein, liver |
reviewed |
- |
Fabp1 |
Ki |
'=' |
180 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
99 |
% |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
19 |
% |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
32196 |
nM |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Km |
'=' |
102000 |
nM |
| P05413 |
BXGT006355 |
Fatty acid-binding protein, heart |
reviewed |
- |
FABP3 |
Ki |
- |
- |
- |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
35481 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
14575 |
nM |
| P07148 |
BXGT006559 |
Fatty acid-binding protein, liver |
reviewed |
- |
FABP1 |
Kd |
'=' |
900 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
IC50 |
'=' |
600 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
IC50 |
'=' |
5300 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
79432 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
31622 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Potency |
- |
10621 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
35481 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
15848 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
3162 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
89125 |
nM |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
89125 |
nM |
| O00519 |
BXGT003934 |
Fatty-acid amide hydrolase 1 |
reviewed |
- |
FAAH |
Ki |
'=' |
6000 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
29855 |
nM |
| Q9WUD2 |
BXGT021939 |
Transient receptor potential cation channel subfamily V member 2 |
reviewed |
- |
Trpv2 |
IC50 |
'>' |
10000 |
nM |
| Q8WZA2 |
BXGT019025 |
Rap guanine nucleotide exchange factor 4 |
reviewed |
Enzyme modulator |
RAPGEF4 |
Potency |
- |
19952 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
3162 |
nM |
| P15090 |
BXGT008079 |
Fatty acid-binding protein, adipocyte |
reviewed |
- |
FABP4 |
Delta Tm |
'=' |
3 |
degrees C |