| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Activity |
- |
- |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Activity |
- |
- |
- |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Activity |
'=' |
15 |
% |
| P51151 |
BXGT010837 |
Ras-related protein Rab-9A |
reviewed |
- |
RAB9A |
Potency |
'=' |
3162 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Inhibition |
- |
- |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
Inhibition |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
39810 |
nM |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
5623 |
nM |
| H0W390 |
BXGT003577 |
Voltage-dependent L-type calcium channel subunit alpha |
unreviewed |
- |
CACNA1S |
Inhibition |
- |
- |
- |
| H0W4W8 |
BXGT003578 |
Voltage-dependent L-type calcium channel subunit alpha |
unreviewed |
- |
CACNA1F |
Inhibition |
- |
- |
- |
| H0VIT6 |
BXGT003575 |
Voltage-dependent L-type calcium channel subunit alpha |
unreviewed |
- |
CACNA1D |
Inhibition |
- |
- |
- |
| O35505 |
BXGT004533 |
Voltage-dependent L-type calcium channel subunit alpha-1C |
reviewed |
- |
CACNA1C |
Inhibition |
- |
- |
- |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
5623 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
1000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
25118 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
1901 |
nM |
| Q9UK17 |
BXGT021735 |
Potassium voltage-gated channel subfamily D member 3 |
reviewed |
Ion channel |
KCND3 |
Activity |
- |
- |
- |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
'=' |
2 |
uM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
39810 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
14 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
'=' |
2 |
uM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
80 |
nM |
| P22460 |
BXGT008774 |
Potassium voltage-gated channel subfamily A member 5 |
reviewed |
Ion channel |
KCNA5 |
IC50 |
'=' |
3400 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
14100 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
7943 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
7 |
- |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
2908 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
794 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
3162 |
nM |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
12589 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
7 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Inhibition |
'=' |
55 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
5 |
- |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
31622 |
nM |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'>' |
1000000 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
12 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
40 |
ug.mL-1 |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
251 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
26608 |
nM |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
10000 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
1258 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
'=' |
10000 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
49 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
14125 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'>' |
95 |
% |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
1258 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3548 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
25118 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
3 |
- |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
TIME |
'=' |
0 |
hr |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
12589 |
nM |
| P50750 |
BXGT010818 |
Cyclin-dependent kinase 9 |
reviewed |
Kinase |
CDK9 |
Ki |
'=' |
1258 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
11220 |
nM |
| Q9UK17 |
BXGT021735 |
Potassium voltage-gated channel subfamily D member 3 |
reviewed |
Ion channel |
KCND3 |
Activity |
'=' |
95 |
% |
| P15382 |
BXGT008116 |
Potassium voltage-gated channel subfamily E member 1 |
reviewed |
Ion channel |
KCNE1 |
IC50 |
'=' |
81400 |
nM |
| P51787 |
BXGT010889 |
Potassium voltage-gated channel subfamily KQT member 1 |
reviewed |
Ion channel |
KCNQ1 |
IC50 |
'=' |
81400 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
25118 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
86 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
2511 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
28183 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
63 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
25118 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
2511 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
80 |
nM |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
'=' |
32400 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
2 |
- |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
100000 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
2 |
- |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
1584 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| Q86831 |
BXGT017584 |
Polyprotein II |
unreviewed |
- |
|
Inhibition |
'=' |
48 |
% |
| P49336 |
BXGT010697 |
Cyclin-dependent kinase 8 |
reviewed |
Kinase |
CDK8 |
Ki |
'=' |
630 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Inhibition |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Inhibition |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
12589 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Inhibition |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| P15382 |
BXGT008116 |
Potassium voltage-gated channel subfamily E member 1 |
reviewed |
Ion channel |
KCNE1 |
Inhibition |
- |
- |
- |
| P51787 |
BXGT010889 |
Potassium voltage-gated channel subfamily KQT member 1 |
reviewed |
Ion channel |
KCNQ1 |
Inhibition |
- |
- |
- |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
22387 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
1000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
- |
- |
- |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
14125 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Ki |
'=' |
45 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
3548 |
nM |
| P22460 |
BXGT008774 |
Potassium voltage-gated channel subfamily A member 5 |
reviewed |
Ion channel |
KCNA5 |
Inhibition |
- |
- |
- |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Activity |
- |
- |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
7 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
10322 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
6 |
- |
| P38398 |
BXGT010037 |
Breast cancer type 1 susceptibility protein |
reviewed |
Enzyme |
BRCA1 |
Potency |
- |
17782 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
Inhibition |
'=' |
77 |
% |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
Inhibition |
- |
- |
- |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Ki |
'=' |
49 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Activity |
'>' |
90 |
% |
| P15382 |
BXGT008116 |
Potassium voltage-gated channel subfamily E member 1 |
reviewed |
Ion channel |
KCNE1 |
Activity |
'=' |
83 |
% |
| P51787 |
BXGT010889 |
Potassium voltage-gated channel subfamily KQT member 1 |
reviewed |
Ion channel |
KCNQ1 |
Activity |
'=' |
83 |
% |
| Q9UK17 |
BXGT021735 |
Potassium voltage-gated channel subfamily D member 3 |
reviewed |
Ion channel |
KCND3 |
TIME |
'=' |
0 |
hr |
| P22460 |
BXGT008774 |
Potassium voltage-gated channel subfamily A member 5 |
reviewed |
Ion channel |
KCNA5 |
IC50 |
'=' |
3200 |
nM |
| P22460 |
BXGT008774 |
Potassium voltage-gated channel subfamily A member 5 |
reviewed |
Ion channel |
KCNA5 |
Activity |
'=' |
94 |
% |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Inhibition |
- |
- |
- |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
123200 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
-2 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
-1 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23715 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Ratio IC50 |
'>' |
22 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
20 |
nM |
| Q9UK17 |
BXGT021735 |
Potassium voltage-gated channel subfamily D member 3 |
reviewed |
Ion channel |
KCND3 |
Inhibition |
- |
- |
- |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Inhibition |
- |
- |
- |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Inhibition |
- |
- |
- |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Inhibition |
- |
- |
- |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Activity |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
'=' |
59 |
nM |
| Q13148 |
BXGT013318 |
TAR DNA-binding protein 43 |
reviewed |
- |
TARDBP |
Potency |
- |
316 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
14 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ratio IC50 |
'>' |
5 |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
TDI |
- |
- |
- |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
TDI |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
121 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Ratio IC50 |
'=' |
75 |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
190 |
nM |
| Q9UK17 |
BXGT021735 |
Potassium voltage-gated channel subfamily D member 3 |
reviewed |
Ion channel |
KCND3 |
IC50 |
'=' |
9300 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Activity |
'=' |
90 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Inhibition |
- |
- |
- |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Inhibition |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Inhibition |
- |
- |
- |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Inhibition |
- |
- |
- |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Inhibition |
- |
- |
- |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Inhibition |
- |
- |
- |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
90 |
% |