| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
7307 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
69 |
% |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
IC50 |
'=' |
12710 |
nM |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Tm |
'=' |
2 |
degrees C |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
31622 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
2807 |
nM |
| P51151 |
BXGT010837 |
Ras-related protein Rab-9A |
reviewed |
- |
RAB9A |
Potency |
'=' |
2818 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
25 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
35481 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
'=' |
4 |
uM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
19952 |
nM |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Tm |
'<' |
2 |
degrees C |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
6012 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
14125 |
nM |
| O75828 |
BXGT005154 |
Carbonyl reductase [NADPH] 3 |
reviewed |
- |
CBR3 |
Tm |
'<' |
2 |
degrees C |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
31622 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Activity |
- |
- |
- |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
10000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| Q13148 |
BXGT013318 |
TAR DNA-binding protein 43 |
reviewed |
- |
TARDBP |
Potency |
- |
3162 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
28183 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
45 |
% |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Activity |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
39810 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
- |
- |
- |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
Activity |
'=' |
10 |
% |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
3264 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
90 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
90 |
% |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
400 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
400 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
19952 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
EC50 |
'=' |
55941 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
EC50 |
'=' |
55941 |
nM |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
EC50 |
'=' |
55941 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
2238 |
nM |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
15848 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
7943 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Ki |
'=' |
12000 |
nM |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
26 |
% |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
12 |
% |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
34000 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
RBA |
'=' |
0 |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
15848 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
IC50 |
'=' |
1600000 |
nM |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Activity |
'=' |
9 |
% |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Ki |
'=' |
2030 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
'=' |
4 |
uM |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
2238 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
31622 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
31622 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
50118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
17782 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
31622 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Log IC50 |
'=' |
4 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
12589 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
2818 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
17782 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
23109 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
35481 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
33498 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
16360 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1258 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
2238 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
113000 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
10 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
12589 |
nM |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
0 |
% |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
100 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
100 |
% |
| P38398 |
BXGT010037 |
Breast cancer type 1 susceptibility protein |
reviewed |
Enzyme |
BRCA1 |
Potency |
- |
2511 |
nM |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
501 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Ratio IC50 |
'=' |
1400 |
- |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
80 |
% |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
96 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
96 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
30 |
ug.mL-1 |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
39810 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
178 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
28183 |
nM |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
8000 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
Activity |
- |
- |
- |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
84 |
% |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
52 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
74 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
74 |
% |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
IC50 |
- |
- |
- |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
15848 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
3 |
nM |
| P40763 |
BXGT010202 |
Signal transducer and activator of transcription 3 |
reviewed |
Nucleic acid binding |
STAT3 |
EC50 |
'>' |
55700 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
10000 |
nM |
| P02791 |
BXGT005965 |
Ferritin light chain |
reviewed |
- |
FTL |
Potency |
'=' |
31622 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
36100 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
31622 |
nM |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
12589 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
35481 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
10322 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
330 |
% |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
- |
- |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
-9 |
% |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
10000 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
10000 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
113 |
% |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
7079 |
nM |
| P42224 |
BXGT010286 |
Signal transducer and activator of transcription 1-alpha/beta |
reviewed |
Nucleic acid binding |
STAT1 |
EC50 |
'>' |
2060 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
6 |
% |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
100000 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'=' |
9900 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
98 |
% |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
127000 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'>' |
10000 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
- |
56234 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
9959 |
nM |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Activity |
- |
- |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
1900 |
nM |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'=' |
7078 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
2 |
% |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'>' |
10000 |
nM |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Inhibition |
- |
- |
- |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
371 |
nM |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Activity |
'=' |
55 |
% |
| P06401 |
BXGT006436 |
Progesterone receptor |
reviewed |
Nuclear receptor |
PGR |
Inhibition |
'>' |
90 |
% |