| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
112201 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
112201 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
20596 |
nM |
| Q9NZ08 |
BXGT021266 |
Endoplasmic reticulum aminopeptidase 1 |
reviewed |
Enzyme |
ERAP1 |
AC50 |
'=' |
12140 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
76 |
% |
| O15439 |
BXGT004169 |
Multidrug resistance-associated protein 4 |
reviewed |
Transporter |
ABCC4 |
Drug transport |
- |
- |
- |
| P35503 |
BXGT009840 |
UDP-glucuronosyltransferase 1-3 |
reviewed |
- |
UGT1A3 |
Activity |
'=' |
152 |
pm/min/mg |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
0 |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
25118 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
28183 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'=' |
58400 |
nM |
| Q00796 |
BXGT012549 |
Sorbitol dehydrogenase |
reviewed |
Enzyme |
SORD |
IC50 |
'=' |
120000 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
0 |
pm/min/mg |
| P0DTE4 |
BXGT022286 |
UDP-glucuronosyltransferase 2A1 |
reviewed |
- |
UGT2A1 |
Activity |
'=' |
600 |
pm/min/mg |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
50118 |
nM |
| P06280 |
BXGT006433 |
Alpha-galactosidase A |
reviewed |
- |
GLA |
Potency |
- |
35481 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'>' |
100000 |
nM |
| P06280 |
BXGT006433 |
Alpha-galactosidase A |
reviewed |
- |
GLA |
Potency |
'=' |
35481 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
39810 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
28183 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
56234 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
478 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
754 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
19952 |
nM |
| P80365 |
BXGT011895 |
Corticosteroid 11-beta-dehydrogenase isozyme 2 |
reviewed |
Enzyme |
HSD11B2 |
Inhibition |
- |
- |
- |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
56234 |
nM |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
236000 |
nM |
| P02791 |
BXGT005965 |
Ferritin light chain |
reviewed |
- |
FTL |
Potency |
'=' |
39810 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
39810 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
43000 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
100000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'>' |
500000 |
nM |
| P28845 |
BXGT009297 |
Corticosteroid 11-beta-dehydrogenase isozyme 1 |
reviewed |
- |
HSD11B1 |
Inhibition |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'>' |
100000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
0 |
pm/min/mg |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Kinact |
'=' |
0 |
uM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Kinact |
'>' |
100 |
uM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'<' |
30 |
% |
| P22513 |
BXGT008777 |
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal |
reviewed |
- |
|
IC50 |
'=' |
616580 |
nM |
| Q43570 |
BXGT014591 |
Zn finger protein |
unreviewed |
- |
NtBBF1.1 |
Ki |
'=' |
754 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'=' |
29000000 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Kinact |
'=' |
58 |
uM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
616595 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Kinact |
'=' |
0 |
uM |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
Potency |
'=' |
15848 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
28183 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'=' |
500 |
uM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
28183 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
'>' |
500000 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
31622 |
nM |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
72 |
pm/min/mg |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Inhibition |
'=' |
16 |
% |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
750 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
79432 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
11 |
pm/min/mg |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
170 |
pm/min/mg |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
665 |
pm/min/mg |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
IC50 |
'=' |
140000 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
501187 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
IC50 |
'=' |
420000 |
nM |
| P18405 |
BXGT008400 |
3-oxo-5-alpha-steroid 4-dehydrogenase 1 |
reviewed |
Enzyme |
SRD5A1 |
IC50 |
'>' |
20 |
ug.mL-1 |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
480 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
482 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
'=' |
30 |
% |
| O15438 |
BXGT004168 |
Canalicular multispecific organic anion transporter 2 |
reviewed |
Transporter |
ABCC3 |
Drug transport |
- |
- |
- |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
12589 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Drug transport |
- |
- |
- |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Drug transport |
- |
- |
- |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
22900 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'>' |
10000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
26 |
% |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Drug transport |
- |
- |
- |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Inhibition |
- |
- |
- |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
24 |
nM |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Activity |
- |
- |
- |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
467000 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
45 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'>' |
10000 |
nM |