Showing entry for Combretastatin A4



                             
General Compound Information
BXGC IdBXGC0034941
Compound NameCombretastatin A4
Structure
FormulaC18H20O5
InchiKeyHVXBOLULGPECHP-WAYWQWQTSA-N
SMILESCOc1cc(/C=C\c2ccc(c(c2)O)OC)cc(c1OC)OC
InchiInChI=1S/C18H20O5/c1-20-15-8-7-12(9-14(15)19)5-6-13-10-16(21-2)18(23-4)17(11-13)22-3/h5-11,19H,1-4H3/b6-5-
IUPAC2-methoxy-5-[(Z)-2-(3,4,5-trimethoxyphenyl)ethenyl]phenol
Molecular Weight316.13
Pubchem Id5351344
Chembl IdCHEMBL67
Targets of Information Source
DrugBank n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
PDB 7BA
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - - - - -
Binding DB 50005480
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT005336 Tubulin polymerization-promoting protein reviewed Cellular structure TPPP - 2000 - -
reviewed BXGT005336 Tubulin polymerization-promoting protein reviewed Cellular structure TPPP - 32 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 530 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - >10000 - -
reviewed BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 - >10000 - -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - >10000 - -
reviewed BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC - >10000 - -
reviewed BXGT005891 Tubulin alpha-1A chain reviewed TUBA1A - 1200 - -
reviewed BXGT005891 Tubulin alpha-1A chain reviewed TUBA1A - 1000 - -
reviewed BXGT005891 Tubulin alpha-1A chain reviewed TUBA1A - 2100 - -
reviewed BXGT005891 Tubulin alpha-1A chain reviewed TUBA1A - 530 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 1200 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 1900 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 900 - -
reviewed BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 - 2030 - -
reviewed BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 - 180 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 1800 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 4900 - -
reviewed BXGT005891 Tubulin alpha-1A chain reviewed TUBA1A - 3900 - -
reviewed BXGT005892 Tubulin beta chain reviewed - - 1060 - -
reviewed BXGT005892 Tubulin beta chain reviewed - - 4000 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B - 2900 - -
reviewed BXGT016212 Tubulin beta-2B chain reviewed TUBB2B 180 - - -
reviewed BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 - 1200 - -
reviewed BXGT006741 ATP-dependent translocase ABCB1 reviewed Transporter ABCB1 - 12 - -
CHEMBL CHEMBL67
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 3200 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 3200 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 3200 nM
P04786 BXGT006262 DNA topoisomerase 1 reviewed - TOP1 IC50 '=' 7 ug.mL-1
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 97 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 97 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 97 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 97 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 97 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 97 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 97 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 97 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 97 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 97 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 97 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 97 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 97 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 97 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 97 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 88 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 88 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 88 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 94 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 94 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 94 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Control '=' 160 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1700 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1700 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1700 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 88 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 88 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 88 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 88 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 88 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 88 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 88 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 88 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 88 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 88 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 88 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 88 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 88 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 88 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 88 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 99 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 99 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 99 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 99 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 99 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 99 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 99 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 99 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 99 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 99 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 99 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 99 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 99 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 99 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 99 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2100 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2100 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2100 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 5800 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 5800 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 5800 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 5800 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 5800 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 5800 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 5800 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 5800 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 5800 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 5800 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 5800 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 5800 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 5800 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 5800 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 5800 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition - - -
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition - - -
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition - - -
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition - - -
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition - - -
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition - - -
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition - - -
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition - - -
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition - - -
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition - - -
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition - - -
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition - - -
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition - - -
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition - - -
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2200 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2200 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2200 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 40 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 40 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 40 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 40 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 40 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 40 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 40 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 40 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 40 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 40 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 40 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 40 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 40 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 40 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 40 um/min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 93 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 100 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1000 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 1000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1730 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1730 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1730 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1730 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1730 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1730 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1730 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1730 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1730 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1730 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1730 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1730 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1730 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1730 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1730 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1770 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 1770 nM
Q9UGI9 BXGT021682 5'-AMP-activated protein kinase subunit gamma-3 reviewed Enzyme modulator PRKAG3 Activity - - -
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Activity - - -
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Activity - - -
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Activity - - -
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Activity - - -
O43741 BXGT004620 5'-AMP-activated protein kinase subunit beta-2 reviewed Enzyme modulator PRKAB2 Activity - - -
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Activity - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1100 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1100 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1100 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 98 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 98 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 98 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 98 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 98 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 98 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 98 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 98 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 98 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 98 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 98 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 98 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 98 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 98 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 98 %
Q9NY65 BXGT021252 Tubulin alpha-8 chain reviewed Cellular structure TUBA8 Inhibition - - -
A6NHL2 BXGT001464 Tubulin alpha chain-like 3 reviewed - TUBAL3 Inhibition - - -
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition - - -
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition - - -
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition - - -
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition - - -
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition - - -
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 99 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 99 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 99 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1500 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1500 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1500 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1500 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1500 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1500 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1500 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1500 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1500 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1500 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1500 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1500 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1500 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1500 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1500 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1000 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1000 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1000 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1000 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1000 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1000 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1000 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1000 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1000 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1000 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1000 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1000 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1000 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1000 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1000 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2500 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2500 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2500 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 70 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 70 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 70 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 70 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 70 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 70 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 70 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 70 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 70 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 70 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 70 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 70 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 70 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 70 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 70 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 99000 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 99000 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 99000 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1900 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1900 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1770 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1770 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1770 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A FC '=' 6 -
P02554 BXGT005892 Tubulin beta chain reviewed - FC '=' 6 -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1200 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1200 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1200 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 96 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 96 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 96 %
P04786 BXGT006262 DNA topoisomerase 1 reviewed - TOP1 IC50 '=' 6 ug.mL-1
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 100 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 100 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 100 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 100 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 100 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 100 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 100 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 100 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 100 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 100 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 100 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 100 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 100 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 100 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 100 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 600 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 600 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Inhibition - - -
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Inhibition - - -
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 97 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 96 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 530 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 530 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 530 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 87 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 87 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 87 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 87 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 87 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 87 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 87 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 87 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 87 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 87 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 87 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 87 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 87 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 87 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 87 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 4000 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 4000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity - - -
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity - - -
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity - - -
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity - - -
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity - - -
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity - - -
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity - - -
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity - - -
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity - - -
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity - - -
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity - - -
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity - - -
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity - - -
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity - - -
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity - - -
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 4920 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 4920 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 4920 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 4920 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 4920 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 4920 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 4920 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 4920 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 4920 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 4920 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 4920 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 4920 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 4920 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 4920 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 4920 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 93 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 93 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 93 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 93 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 93 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 93 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 93 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 93 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 93 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 93 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 93 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 93 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 93 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 93 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 93 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1200 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1200 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1200 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1200 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1200 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1200 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1200 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1200 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1200 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1200 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1200 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1200 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1200 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1200 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1200 nM
A6NNZ2 BXGT001465 Tubulin beta-8 chain-like protein LOC260334 reviewed - TUBB8B Inhibition '=' 99 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 99 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 99 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 99 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 99 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 99 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 99 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 99 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 99 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 99 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 82 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 82 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 82 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 82 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 82 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 82 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 82 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 82 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 82 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 82 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 82 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 82 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 82 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 82 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 82 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 95 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 95 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 95 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 4500 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 4500 nM
Q08493 BXGT012987 cAMP-specific 3',5'-cyclic phosphodiesterase 4C reviewed - PDE4C IC50 '>' 10000 nM
Q07343 BXGT012926 cAMP-specific 3',5'-cyclic phosphodiesterase 4B reviewed - PDE4B IC50 '>' 10000 nM
Q08499 BXGT012988 cAMP-specific 3',5'-cyclic phosphodiesterase 4D reviewed - PDE4D IC50 '>' 10000 nM
P27815 BXGT009208 cAMP-specific 3',5'-cyclic phosphodiesterase 4A reviewed - PDE4A IC50 '>' 10000 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition - - -
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition - - -
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition - - -
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 98 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 2200 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2200 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 2200 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 2200 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 2200 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 2200 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 2200 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 2200 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 2200 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 2200 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 2200 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 2200 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 2200 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2200 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 2200 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 84 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 84 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 84 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Ki '=' 120 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Ki '=' 120 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Ki '=' 120 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Ki '=' 120 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Ki '=' 120 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Ki '=' 120 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Ki '=' 120 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Ki '=' 120 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Ki '=' 120 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Ki '=' 120 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Ki '=' 120 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Ki '=' 120 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Ki '=' 120 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Ki '=' 120 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Ki '=' 120 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1700 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1700 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1700 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1700 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1700 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1700 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1700 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1700 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1700 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1700 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1700 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1700 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1700 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1700 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1700 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 88 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 88 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1400 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1400 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1400 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1400 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1400 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1400 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1400 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1400 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1400 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1400 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1400 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1400 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1400 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1400 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1400 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 5 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 91 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 91 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 91 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1000 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1000 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1000 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1200 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1900 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 88 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 5 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1200 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 86 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 86 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 86 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 86 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 86 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 86 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 86 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 86 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 86 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 86 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 86 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 86 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 86 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 86 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 86 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 86 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 86 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 86 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 86 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 86 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 86 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 86 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 86 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 86 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 86 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 86 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 86 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 86 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 86 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 86 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 90 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 90 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 90 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 90 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 90 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 90 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 90 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 90 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 90 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 90 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 90 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 90 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 90 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 90 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 90 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 78 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 78 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 680 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 680 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 680 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 50 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 50 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 92 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 92 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 92 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 660 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 660 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 660 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 3900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2900 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2900 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2900 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 530000 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 530000 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 530000 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 530000 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 530000 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 530000 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 530000 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 530000 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 530000 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 530000 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 530000 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 530000 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 530000 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 530000 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 530000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 93 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 93 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 93 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 93 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 93 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 93 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 93 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 93 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 93 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 93 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 93 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 93 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 93 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 93 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 93 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q25270 BXGT013897 Beta-tubulin unreviewed - beta-tubulin IC50 '=' 1900 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 4000 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 4000 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 4000 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 530 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 98 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 98 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 98 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 2200 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 2200 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1100 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 1100 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Ki '=' 180 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 98 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 90 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 90 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 90 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 90 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 90 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 90 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 90 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 90 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 90 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 90 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 90 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 90 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 90 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 90 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 90 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 2500 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2500 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 2500 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 2500 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 2500 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 2500 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 2500 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 2500 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 2500 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 2500 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 2500 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 2500 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 2500 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2500 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 2500 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 300 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 300 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 300 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 300 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 300 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 300 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 300 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 300 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 300 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 300 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 300 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 300 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 300 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 300 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 300 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 10 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 10 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 10 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 10 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 10 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 10 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 10 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 10 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 10 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 10 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 10 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 10 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 10 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 10 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 10 um/min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 39 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 39 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 39 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 39 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 39 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 39 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 39 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 39 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 39 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 39 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 39 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 39 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 39 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 39 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 39 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 1 /min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 1 /min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 1 /min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 1 /min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 1 /min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 1 /min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 1 /min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 1 /min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 1 /min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 1 /min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 1 /min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 1 /min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 1 /min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 1 /min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 1 /min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 36 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 36 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 36 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 36 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 36 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 36 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 36 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 36 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 36 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 36 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 36 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 36 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 36 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 36 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 36 %
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC IC50 '>' 10000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 50 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 50 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 50 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 50 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 50 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 50 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 50 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 50 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 50 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 50 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 50 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 50 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 50 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 50 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 50 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 530 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 2100 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 1 /min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 1 /min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 1 /min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 1 /min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 1 /min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 1 /min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 1 /min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 1 /min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 1 /min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 1 /min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 1 /min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 1 /min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 1 /min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 1 /min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 1 /min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Ki '=' 3 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Ki '=' 3 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Ki '=' 3 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Ki '=' 3 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Ki '=' 3 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Ki '=' 3 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Ki '=' 3 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Ki '=' 3 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Ki '=' 3 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Ki '=' 3 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Ki '=' 3 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Ki '=' 3 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Ki '=' 3 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Ki '=' 3 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Ki '=' 3 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 89 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 89 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 89 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 89 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 89 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 89 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 89 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 89 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 89 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 89 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 89 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 89 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 89 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 89 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 89 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 810 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 810 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 810 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 810 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 810 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 810 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 810 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 810 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 810 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 810 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 810 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 810 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 810 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 810 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 810 nM
Q25270 BXGT013897 Beta-tubulin unreviewed - beta-tubulin IC50 '=' 2000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 30 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 30 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 30 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 30 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 30 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 30 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 30 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 30 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 30 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 30 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 30 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 30 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 30 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 30 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 30 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 94 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 94 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 94 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 94 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 94 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 94 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 94 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 94 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 94 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 94 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 94 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 94 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 94 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 94 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 94 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 92 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2030 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 12 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 12 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 12 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 12 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 12 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 12 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 12 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 12 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 12 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 12 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 12 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 12 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 12 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 12 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 12 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1080 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1080 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1080 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1080 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1080 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1080 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1080 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1080 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1080 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1080 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1080 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1080 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1080 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1080 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1080 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Control '=' 161 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1000 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 3900 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 3900 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 96 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 96 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 96 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 96 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 96 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 96 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 96 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 96 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 96 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 96 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 96 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 96 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 96 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 96 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 96 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 95 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 440 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 440 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 440 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 69 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 69 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 69 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 69 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 69 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 69 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 69 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 69 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 69 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 69 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 69 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 69 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 69 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 69 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 69 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 32 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 32 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 32 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 32 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 32 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 32 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 32 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 32 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 32 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 32 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 32 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 32 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 32 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 32 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 32 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 2100 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2100 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 2100 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 2100 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 2100 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 2100 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 2100 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 2100 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 2100 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 2100 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 2100 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 2100 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 2100 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2100 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 2100 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1200 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1100 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1100 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1100 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1100 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1100 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1100 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1100 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1100 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1100 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1100 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1100 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1100 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1100 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1100 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1100 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 97 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 97 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 97 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 92 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 92 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 92 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 92 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 92 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 92 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 92 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 92 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 92 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 92 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 92 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 92 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 92 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 92 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 92 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 81 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 81 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 81 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 81 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 81 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 81 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 81 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 81 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 81 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 81 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 81 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 81 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 81 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 81 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 81 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 53 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1300 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1300 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1300 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1300 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1300 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1300 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1300 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1300 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1300 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1300 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1300 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1300 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1300 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1300 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1300 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 500 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 500 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 500 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 500 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 500 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 500 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 500 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 500 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 500 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 500 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 500 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 500 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 500 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 500 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 500 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 180 nM
Q9WKE8 BXGT021921 Reverse transcriptase unreviewed - reverse IC50 - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2000 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 2000 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2000 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1320 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 1320 nM
O15244 BXGT004140 Solute carrier family 22 member 2 reviewed Transporter SLC22A2 Inhibition - - -
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A IC50 '=' 1060 nM
P02554 BXGT005892 Tubulin beta chain reviewed - IC50 '=' 1060 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 84 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 84 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 84 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 84 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 84 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 84 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 84 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 84 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 84 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 84 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 84 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 84 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 84 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 84 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 84 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Ki '=' 2400 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Ki '=' 2400 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Ki '=' 2400 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 2000 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2000 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 2000 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 2000 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 2000 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 2000 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 2000 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 2000 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 2000 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 2000 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 2000 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 2000 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 2000 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2000 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 2000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 80 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 80 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 80 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 80 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 80 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 80 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 80 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 80 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 80 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 80 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 80 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 80 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 80 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 80 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 80 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1300 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1300 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1300 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 93 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 93 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition - - -
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition - - -
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 3981 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 3981 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 3981 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 3981 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 3981 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 3981 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 3981 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 3981 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 3981 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 3981 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 3981 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 3981 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 3981 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 3981 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 3981 nM
O15245 BXGT004141 Solute carrier family 22 member 1 reviewed Transporter SLC22A1 Inhibition - - -
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 80 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 80 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 900 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 900 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 35 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 35 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 35 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 35 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 35 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 35 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 35 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 35 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 35 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 35 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 35 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 35 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 35 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 35 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 35 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 89 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 89 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 89 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 89 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 89 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 89 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 89 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 89 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 89 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 89 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 89 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 89 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 89 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 89 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 89 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 920 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 920 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 920 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 920 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 920 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 920 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 920 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 920 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 920 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 920 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 920 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 920 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 920 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 920 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 920 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 4900 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 4900 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 93 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 93 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 93 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 93 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 93 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 93 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 93 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 93 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 93 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 93 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 93 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 93 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 93 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 93 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 93 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 2700 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 2700 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 2700 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 2700 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 2700 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 2700 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 2700 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 2700 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 2700 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 2700 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 2700 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 2700 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 2700 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 2700 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 2700 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 29 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 29 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 29 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 29 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 29 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 29 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 29 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 29 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 29 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 29 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 29 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 29 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 29 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 29 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 29 um/min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 23 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 23 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 23 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 23 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 23 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 23 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 23 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 23 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 23 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 23 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 23 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 23 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 23 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 23 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 23 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 960 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 960 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 960 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 960 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 960 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 960 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 960 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 960 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 960 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 960 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 960 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 960 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 960 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 960 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 960 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 99 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 99 %
A6NNZ2 BXGT001465 Tubulin beta-8 chain-like protein LOC260334 reviewed - TUBB8B Inhibition '=' 89 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 89 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 89 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 89 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 89 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 89 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 89 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 89 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 89 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 89 %
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 IC50 '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '>' 10000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 21 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 21 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 21 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 21 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 21 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 21 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 21 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 21 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 21 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 21 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 21 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 21 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 21 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 21 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 21 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A EC50 '=' 7 nM
P02554 BXGT005892 Tubulin beta chain reviewed - EC50 '=' 7 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1800 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1800 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1800 nM
P08183 BXGT006741 ATP-dependent translocase ABCB1 reviewed Transporter ABCB1 IC50 '=' 6 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 70 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 70 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 70 %
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 92 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 92 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 25 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 25 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 25 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 25 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 25 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 25 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 25 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 25 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 25 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 25 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 25 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 25 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 25 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 25 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 25 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 2 /min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 2 /min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 2 /min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 2 /min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 2 /min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 2 /min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 2 /min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 2 /min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 2 /min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 2 /min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 2 /min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 2 /min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 2 /min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 2 /min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 2 /min
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 35 %
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 35 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 35 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 13 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 13 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 13 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 13 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 13 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 13 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 13 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 13 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 13 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 13 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 13 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 13 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 13 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 13 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 13 um/min
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Activity - - -
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - Activity - - -
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Activity - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 - - -
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 43 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 43 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 43 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 43 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 43 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 43 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 43 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 43 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 43 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 43 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 43 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 43 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 43 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 43 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 43 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 1 /min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 1 /min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 1 /min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 1 /min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 1 /min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 1 /min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 1 /min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 1 /min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 1 /min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 1 /min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 1 /min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 1 /min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 1 /min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 1 /min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 1 /min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 91 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 91 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 91 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 91 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 91 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 91 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 91 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 91 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 91 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 91 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 91 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 91 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 91 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 91 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 91 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 11 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 11 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 11 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 11 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 11 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 11 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 11 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 11 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 11 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 11 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 11 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 11 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 11 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 11 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 11 um/min
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 66 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 66 %
Q8TCC7 BXGT018794 Solute carrier family 22 member 8 reviewed Transporter SLC22A8 IC50 '=' 16390 nM
O15245 BXGT004141 Solute carrier family 22 member 1 reviewed Transporter SLC22A1 IC50 '>' 200000 nM
P08183 BXGT006741 ATP-dependent translocase ABCB1 reviewed Transporter ABCB1 IC50 '=' 11 nM
O15244 BXGT004140 Solute carrier family 22 member 2 reviewed Transporter SLC22A2 Drug uptake - - -
O94956 BXGT005343 Solute carrier organic anion transporter family member 2B1 reviewed Transporter SLCO2B1 Inhibition - - -
Q8TCC7 BXGT018794 Solute carrier family 22 member 8 reviewed Transporter SLC22A8 Inhibition - - -
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 9000 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 9000 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 9000 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 9000 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 9000 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 9000 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 9000 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 9000 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 9000 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 9000 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 9000 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 9000 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 9000 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 9000 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 9000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1800 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1800 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1800 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1800 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1800 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1800 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1800 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1800 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1800 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1800 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1800 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1800 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1800 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1800 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1800 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 EC50 '=' 9 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B EC50 '=' 9 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A EC50 '=' 9 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E EC50 '=' 9 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C EC50 '=' 9 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B EC50 '=' 9 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB EC50 '=' 9 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 EC50 '=' 9 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A EC50 '=' 9 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A EC50 '=' 9 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 EC50 '=' 9 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A EC50 '=' 9 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C EC50 '=' 9 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 EC50 '=' 9 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B EC50 '=' 9 nM
O15245 BXGT004141 Solute carrier family 22 member 1 reviewed Transporter SLC22A1 Drug uptake - - -
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 IC50 '>' 10000 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 65 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 65 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 65 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 65 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 65 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 65 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 65 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 65 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 65 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 65 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 65 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 65 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 65 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 65 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 65 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 10 um/min
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 10 um/min
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 10 um/min
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 10 um/min
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 10 um/min
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 10 um/min
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 10 um/min
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 10 um/min
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 10 um/min
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 10 um/min
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 10 um/min
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 10 um/min
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 10 um/min
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 10 um/min
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 10 um/min
O15244 BXGT004140 Solute carrier family 22 member 2 reviewed Transporter SLC22A2 IC50 '=' 61940 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 87 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 87 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Inhibition '=' 95 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 95 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Inhibition '=' 95 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Inhibition '=' 95 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Inhibition '=' 95 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Inhibition '=' 95 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Inhibition '=' 95 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Inhibition '=' 95 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Inhibition '=' 95 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Inhibition '=' 95 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Inhibition '=' 95 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Inhibition '=' 95 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Inhibition '=' 95 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Inhibition '=' 95 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Inhibition '=' 95 %
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB IC50 - - -
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1800 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1800 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 Activity '=' 20 %
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B Activity '=' 20 %
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A Activity '=' 20 %
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E Activity '=' 20 %
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C Activity '=' 20 %
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B Activity '=' 20 %
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB Activity '=' 20 %
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 Activity '=' 20 %
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A Activity '=' 20 %
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A Activity '=' 20 %
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 Activity '=' 20 %
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A Activity '=' 20 %
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C Activity '=' 20 %
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 Activity '=' 20 %
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B Activity '=' 20 %
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 TIME '=' 0 hr
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B TIME '=' 0 hr
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A TIME '=' 0 hr
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E TIME '=' 0 hr
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C TIME '=' 0 hr
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B TIME '=' 0 hr
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB TIME '=' 0 hr
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 TIME '=' 0 hr
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A TIME '=' 0 hr
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A TIME '=' 0 hr
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 TIME '=' 0 hr
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A TIME '=' 0 hr
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C TIME '=' 0 hr
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 TIME '=' 0 hr
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B TIME '=' 0 hr
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 650 nM
Q862L2 BXGT017582 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 650 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 650 nM
Q4U2R8 BXGT014891 Solute carrier family 22 member 6 reviewed Transporter SLC22A6 Drug uptake - - -
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 Inhibition - - -
Q4U2R8 BXGT014891 Solute carrier family 22 member 6 reviewed Transporter SLC22A6 IC50 '=' 41360 nM
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 IC50 '=' 194540 nM
Q9BUF5 BXGT020135 Tubulin beta-6 chain reviewed Cellular structure TUBB6 IC50 '=' 1020 nM
Q9BVA1 BXGT020142 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1020 nM
Q13885 BXGT013400 Tubulin beta-2A chain reviewed Cellular structure TUBB2A IC50 '=' 1020 nM
Q6PEY2 BXGT016465 Tubulin alpha-3E chain reviewed Cellular structure TUBA3E IC50 '=' 1020 nM
Q9BQE3 BXGT020109 Tubulin alpha-1C chain reviewed Cellular structure TUBA1C IC50 '=' 1020 nM
P68363 BXGT011594 Tubulin alpha-1B chain reviewed Cellular structure TUBA1B IC50 '=' 1020 nM
P07437 BXGT006624 Tubulin beta chain reviewed Cellular structure TUBB IC50 '=' 1020 nM
Q3ZCM7 BXGT014551 Tubulin beta-8 chain reviewed - TUBB8 IC50 '=' 1020 nM
P04350 BXGT006193 Tubulin beta-4A chain reviewed Cellular structure TUBB4A IC50 '=' 1020 nM
Q71U36 BXGT016705 Tubulin alpha-1A chain reviewed Cellular structure TUBA1A IC50 '=' 1020 nM
Q13509 BXGT013366 Tubulin beta-3 chain reviewed Cellular structure TUBB3 IC50 '=' 1020 nM
P68366 BXGT011595 Tubulin alpha-4A chain reviewed Cellular structure TUBA4A IC50 '=' 1020 nM
P0DPH7 BXGT007527 Tubulin alpha-3C chain reviewed - TUBA3C IC50 '=' 1020 nM
Q9H4B7 BXGT020475 Tubulin beta-1 chain reviewed Cellular structure TUBB1 IC50 '=' 1020 nM
P68371 BXGT011597 Tubulin beta-4B chain reviewed Cellular structure TUBB4B IC50 '=' 1020 nM
P02550 BXGT005891 Tubulin alpha-1A chain reviewed - TUBA1A Inhibition '=' 87 %
P02554 BXGT005892 Tubulin beta chain reviewed - Inhibition '=' 87 %
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - IC50 '=' 1200 nM
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B IC50 '=' 1200 nM
Q862F3 BXGT017581 Similar to alpha-tubulin isoform 1 unreviewed - Inhibition '=' 99 %
Q6B856 BXGT016212 Tubulin beta-2B chain reviewed - TUBB2B Inhibition '=' 99 %
Q8TCC7 BXGT018794 Solute carrier family 22 member 8 reviewed Transporter SLC22A8 Drug uptake - - -
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 Drug uptake - - -
O94956 BXGT005343 Solute carrier organic anion transporter family member 2B1 reviewed Transporter SLCO2B1 Drug uptake - - -
Q4U2R8 BXGT014891 Solute carrier family 22 member 6 reviewed Transporter SLC22A6 Inhibition - - -
O94956 BXGT005343 Solute carrier organic anion transporter family member 2B1 reviewed Transporter SLCO2B1 IC50 '=' 12270 nM
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF04750 Scutellaria baicalensis Scutellaria baicalensis Medicinal Plant
BXGF05037 combretum caffrum combretum caffrum Others
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease