| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
25118 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
22387 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
3162 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
28183 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
125 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
7943 |
nM |
| Q9HC16 |
BXGT020525 |
DNA dC->dU-editing enzyme APOBEC-3G |
reviewed |
Enzyme |
APOBEC3G |
Potency |
- |
26608 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
42163 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
39810 |
nM |
| P00761 |
BXGT005645 |
Trypsin |
reviewed |
- |
|
IC50 |
'>' |
200000 |
nM |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'=' |
12000 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
44668 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
15848 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
8912 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
15848 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
12589 |
nM |
| Q9Y468 |
BXGT022270 |
Lethal(3)malignant brain tumor-like protein 1 |
reviewed |
Epigenetic regulator |
L3MBTL1 |
Potency |
'=' |
31622 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
10000 |
nM |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
93000 |
nM |
| Q9UGP5 |
BXGT021689 |
DNA polymerase lambda |
reviewed |
Enzyme |
POLL |
Inhibition |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
5011 |
nM |
| P13726 |
BXGT007950 |
Tissue factor |
reviewed |
Receptor |
F3 |
IC50 |
'=' |
30000 |
nM |
| P08709 |
BXGT006818 |
Coagulation factor VII |
reviewed |
Enzyme |
F7 |
IC50 |
'=' |
30000 |
nM |
| P04054 |
BXGT006136 |
Phospholipase A2 |
reviewed |
Enzyme |
PLA2G1B |
IC50 |
'=' |
22300 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
28183 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
22387 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
10000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
28183 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
17782 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
12589 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
79432 |
nM |
| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
125892 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
125892 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
794 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
96 |
% |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
Activity |
- |
- |
- |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
EC50 |
'=' |
2600 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Inhibition |
'=' |
100 |
% |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
35481 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
39810 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
Activity |
'=' |
100 |
% |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
'=' |
4000 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
0 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
25118 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
IC50 |
'=' |
1200 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
5200 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
56234 |
nM |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
EC50 |
'=' |
3235 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1778 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
10 |
- |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
14125 |
nM |
| Q14191 |
BXGT013452 |
Werner syndrome ATP-dependent helicase |
reviewed |
Enzyme |
WRN |
Potency |
- |
17782 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
92 |
% |
| Q8IUX4 |
BXGT018337 |
DNA dC->dU-editing enzyme APOBEC-3F |
reviewed |
Enzyme |
APOBEC3F |
Potency |
- |
22387 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
3548 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
44200 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Kd |
'=' |
7 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
22387 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
39810 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
5011 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
79432 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Inhibition |
- |
- |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
49 |
% |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
IC50 |
'=' |
6000 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
17782 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
IC50 |
'=' |
16000 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Kd |
'=' |
2000 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
35481 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
35481 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
31622 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
28183 |
nM |
| Q9Y4P1 |
BXGT022283 |
Cysteine protease ATG4B |
reviewed |
Enzyme |
ATG4B |
IC50 |
'=' |
15300 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
8912 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
31622 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
22387 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
4109 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
9466 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
50118 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
17782 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
10000 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
23934 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
29934 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
2884 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
39810 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
19952 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
22387 |
nM |
| O75469 |
BXGT005128 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
Nuclear receptor |
NR1I2 |
Efficacy |
'=' |
110 |
% |
| Q9R1A7 |
BXGT021413 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
- |
Nr1i2 |
Activity |
- |
- |
- |
| O75469 |
BXGT005128 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
Nuclear receptor |
NR1I2 |
Activity |
- |
- |
- |
| O75469 |
BXGT005128 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
Nuclear receptor |
NR1I2 |
EC50 |
'=' |
2500 |
nM |
| O14746 |
BXGT004091 |
Telomerase reverse transcriptase |
reviewed |
Enzyme |
TERT |
Activity |
'=' |
20 |
% |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
3162 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
56234 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
150 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
Activity |
'=' |
100 |
% |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
66824 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
12589 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
19952 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
3000 |
nM |
| Q5NUL3 |
BXGT015621 |
Free fatty acid receptor 4 |
reviewed |
- |
FFAR4 |
Efficacy |
'=' |
99 |
% |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
Efficacy |
'=' |
88 |
% |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Potency |
- |
16833 |
nM |
| O75469 |
BXGT005128 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
Nuclear receptor |
NR1I2 |
Efficacy |
'=' |
16 |
% |
| O75469 |
BXGT005128 |
Nuclear receptor subfamily 1 group I member 2 |
reviewed |
Nuclear receptor |
NR1I2 |
EC50 |
'=' |
2 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
EC50 |
'=' |
11090 |
nM |
| O14842 |
BXGT004106 |
Free fatty acid receptor 1 |
reviewed |
G-protein coupled receptor |
FFAR1 |
Emax |
'=' |
100 |
% |