| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
4744 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
IC50 |
'>=' |
200000 |
nM |
| Q72874 |
BXGT016711 |
Pol polyprotein |
unreviewed |
- |
pol |
IC50 |
- |
- |
- |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
Activity |
- |
- |
- |
| P05186 |
BXGT006338 |
Alkaline phosphatase, tissue-nonspecific isozyme |
reviewed |
Enzyme |
ALPL |
IC50 |
'=' |
407 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
10000 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
- |
- |
- |
| Q05117 |
BXGT012807 |
Tartrate-resistant acid phosphatase type 5 |
reviewed |
- |
Acp5 |
Inhibition |
'=' |
159 |
% |
| P29474 |
BXGT009352 |
Nitric oxide synthase, endothelial |
reviewed |
- |
NOS3 |
Activity |
- |
- |
- |
| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
63095 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
63095 |
nM |
| Q9H0H5 |
BXGT020436 |
Rac GTPase-activating protein 1 |
reviewed |
Enzyme modulator |
RACGAP1 |
IC50 |
- |
205620 |
nM |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
7079 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
RU |
'=' |
431 |
- |
| P52209 |
BXGT010923 |
6-phosphogluconate dehydrogenase, decarboxylating |
reviewed |
Enzyme |
PGD |
IC50 |
'>' |
1000000 |
nM |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
35481 |
nM |
| Q05117 |
BXGT012807 |
Tartrate-resistant acid phosphatase type 5 |
reviewed |
- |
Acp5 |
Inhibition |
'=' |
83 |
% |
| P10415 |
BXGT007567 |
Apoptosis regulator Bcl-2 |
reviewed |
Signaling |
BCL2 |
Ki |
'>' |
100000 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
28 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Activity |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
3162 |
nM |
| P09923 |
BXGT006942 |
Intestinal-type alkaline phosphatase |
reviewed |
Enzyme |
ALPI |
EC50 |
'>' |
100000 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Kd |
'=' |
5190000 |
nM |
| P61823 |
BXGT011385 |
Ribonuclease pancreatic |
reviewed |
- |
RNASE1 |
Inhibition |
- |
- |
- |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
15848 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
IC50 |
'=' |
650000 |
nM |
| P9WMR3 |
BXGT012397 |
Replicative DNA helicase |
reviewed |
- |
dnaB |
AC50 |
'>' |
380000 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
100000 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Inhibition |
- |
- |
- |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Ka |
'=' |
1 |
10'2/M |
| P49327 |
BXGT010694 |
Fatty acid synthase |
reviewed |
Enzyme |
FASN |
IC50 |
'>' |
100000 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
12589 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
31622 |
nM |
| P10696 |
BXGT007603 |
Alkaline phosphatase, germ cell type |
reviewed |
Enzyme |
ALPG |
EC50 |
'=' |
51300 |
nM |
| Q29RK1 |
BXGT013982 |
Citrate synthase, mitochondrial |
reviewed |
- |
CS |
Activity |
'=' |
30 |
% |
| Q13093 |
BXGT013310 |
Platelet-activating factor acetylhydrolase |
reviewed |
Enzyme |
PLA2G7 |
Activity |
- |
- |
- |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'>' |
100000 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
Inhibition |
'=' |
61 |
% |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
IC50 |
'=' |
18500 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| Q72547 |
BXGT016709 |
Reverse transcriptase/RNaseH |
unreviewed |
- |
pol |
IC50 |
'>' |
100000 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1000 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Inhibition |
'=' |
41 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
10000 |
nM |
| P11412 |
BXGT007700 |
Glucose-6-phosphate 1-dehydrogenase |
reviewed |
- |
ZWF1 |
IC50 |
'>' |
1000000 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
11220 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1584 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
- |
- |
- |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
22387 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
89125 |
nM |
| P49327 |
BXGT010694 |
Fatty acid synthase |
reviewed |
Enzyme |
FASN |
Inhibition |
'=' |
10 |
% |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
Activity |
- |
- |
- |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
IC50 |
'=' |
1600 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
10 |
% |
| P07998 |
BXGT006711 |
Ribonuclease pancreatic |
reviewed |
- |
RNASE1 |
Ratio |
'=' |
0 |
- |
| Q05117 |
BXGT012807 |
Tartrate-resistant acid phosphatase type 5 |
reviewed |
- |
Acp5 |
Inhibition |
'=' |
170 |
% |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
0 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
-4 |
% |
| P00374 |
BXGT005520 |
Dihydrofolate reductase |
reviewed |
Enzyme |
DHFR |
Activity |
- |
- |
- |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
12200 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Activity |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
80 |
% |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'>' |
30000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
6513 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
- |
- |
- |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
- |
- |
- |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
77 |
% |
| P54803 |
BXGT011082 |
Galactocerebrosidase |
reviewed |
- |
GALC |
Potency |
- |
4466 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
IC50 |
'=' |
150000 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'=' |
2000 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Activity |
'=' |
5 |
% |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Kd |
'=' |
25900 |
nM |
| P07711 |
BXGT006661 |
Cathepsin L1 |
reviewed |
Enzyme |
CTSL |
IC50 |
'>' |
59642 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
89125 |
nM |
| Q8I2J3 |
BXGT018207 |
M18 aspartyl aminopeptidase |
unreviewed |
- |
PF3D7_0932300 |
IC50 |
'=' |
1376 |
nM |
| Q29RK1 |
BXGT013982 |
Citrate synthase, mitochondrial |
reviewed |
- |
CS |
Activity |
- |
- |
- |
| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
11582 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
11582 |
nM |
| P62826 |
BXGT011463 |
GTP-binding nuclear protein Ran |
reviewed |
Enzyme modulator |
RAN |
Potency |
- |
11582 |
nM |
| P9WHJ3 |
BXGT012297 |
Protein RecA |
reviewed |
- |
recA |
EC50 |
'>' |
380000 |
nM |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
Ki |
'=' |
200 |
nM |
| P29473 |
BXGT009351 |
Nitric oxide synthase, endothelial |
reviewed |
- |
NOS3 |
EC50 |
'=' |
2 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
2993 |
nM |
| P24822 |
BXGT008996 |
Intestinal-type alkaline phosphatase |
reviewed |
- |
Iap |
IC50 |
'=' |
1360 |
nM |
| Q05117 |
BXGT012807 |
Tartrate-resistant acid phosphatase type 5 |
reviewed |
- |
Acp5 |
Inhibition |
'=' |
78 |
% |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
12589 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
891 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat |
'=' |
41 |
/s |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Kcat/Km |
'=' |
68 |
/uM/s |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
Km |
'=' |
610 |
nM |