| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
CC50 |
'=' |
76 |
ug.mL-1 |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
117 |
% |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
25118 |
nM |
| Q92793 |
BXGT019374 |
CREB-binding protein |
reviewed |
- |
CREBBP |
Potency |
'=' |
25118 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
398 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
31622 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
12589 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'=' |
12 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
1995 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
Ki |
'=' |
170 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Ki |
'=' |
170 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
Ki |
'=' |
170 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
90000 |
nM |
| O95067 |
BXGT005347 |
G2/mitotic-specific cyclin-B2 |
reviewed |
Enzyme modulator |
CCNB2 |
IC50 |
'=' |
790 |
nM |
| Q8WWL7 |
BXGT019000 |
G2/mitotic-specific cyclin-B3 |
reviewed |
Enzyme modulator |
CCNB3 |
IC50 |
'=' |
790 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
790 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
790 |
nM |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
0 |
pm/min/mg |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
'=' |
100200 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'<' |
1000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'<' |
1000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'<' |
1000 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
22387 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
2511 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
- |
- |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
31622 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'<' |
50 |
% |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
11220 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
15848 |
nM |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
64 |
pm/min/mg |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
15000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7943 |
nM |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
Potency |
'=' |
15848 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
0 |
% |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
15848 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Activity |
- |
- |
- |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
IC50 |
'>' |
100000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
39810 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
EC50 |
'=' |
19000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
12589 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
891 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
11220 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1258 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'=' |
30000 |
nM |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
Potency |
'=' |
19952 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
IC50 |
'=' |
4100 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
8500 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
28183 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
28183 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
28400 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5011 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'>' |
60000 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
'=' |
19600 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
8912 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
8912 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
37 |
% |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
65 |
pm/min/mg |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
891 |
nM |
| P07824 |
BXGT006682 |
Arginase-1 |
reviewed |
- |
Arg1 |
IC50 |
'=' |
1400 |
nM |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P19224 |
BXGT008468 |
UDP-glucuronosyltransferase 1-6 |
reviewed |
- |
UGT1A6 |
Activity |
'=' |
0 |
pm/min/mg |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
27 |
% |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
25059 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
8 |
ug.mL-1 |
| Q9Z1B7 |
BXGT022403 |
Mitogen-activated protein kinase 13 |
reviewed |
- |
Mapk13 |
Activity |
- |
- |
- |
| Q9WUI1 |
BXGT021940 |
Mitogen-activated protein kinase 11 |
reviewed |
- |
Mapk11 |
Activity |
- |
- |
- |
| O08911 |
BXGT004043 |
Mitogen-activated protein kinase 12 |
reviewed |
- |
Mapk12 |
Activity |
- |
- |
- |
| P47811 |
BXGT010587 |
Mitogen-activated protein kinase 14 |
reviewed |
- |
Mapk14 |
Activity |
- |
- |
- |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
85 |
% |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Activity |
- |
- |
- |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
IC50 |
'=' |
950 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
Ki |
'=' |
7 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
1995 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
14125 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
7943 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
4330 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
1000 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
IC50 |
'=' |
5000 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
'=' |
4 |
ug.mL-1 |
| P0AES4 |
BXGT007329 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'=' |
83 |
ug.mL-1 |
| P0AES6 |
BXGT007331 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'=' |
83 |
ug.mL-1 |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
IC50 |
'=' |
850 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
5011 |
nM |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
15848 |
nM |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
570 |
pm/min/mg |
| O60656 |
BXGT004889 |
UDP-glucuronosyltransferase 1-9 |
reviewed |
- |
UGT1A9 |
Activity |
'=' |
1700 |
pm/min/mg |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
2000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
56 |
% |
| Q92793 |
BXGT019374 |
CREB-binding protein |
reviewed |
- |
CREBBP |
Potency |
'=' |
10000 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
IC50 |
'=' |
1400 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
28183 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
25118 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
25118 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
8912 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
- |
- |
- |
| Q92793 |
BXGT019374 |
CREB-binding protein |
reviewed |
- |
CREBBP |
Potency |
'=' |
7943 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5956 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
19952 |
nM |
| Q15078 |
BXGT013534 |
Cyclin-dependent kinase 5 activator 1 |
reviewed |
Enzyme modulator |
CDK5R1 |
IC50 |
'=' |
570 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
IC50 |
'=' |
570 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
25118 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
562 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
19952 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
1 |
- |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
350 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
350 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
350 |
nM |
| P35503 |
BXGT009840 |
UDP-glucuronosyltransferase 1-3 |
reviewed |
- |
UGT1A3 |
Activity |
'=' |
276 |
pm/min/mg |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
598 |
pm/min/mg |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
3162 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
420 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
IC50 |
'=' |
420 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
2 |
% |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
6683 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
25118 |
nM |
| P68871 |
BXGT011615 |
Hemoglobin subunit beta |
reviewed |
- |
HBB |
Potency |
'=' |
31622 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
108 |
% |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
Inhibition |
- |
- |
- |