| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Inhibition |
- |
- |
- |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
15848 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
3162 |
nM |
| Q9XUB2 |
BXGT022194 |
Zinc finger protein mex-5 |
reviewed |
- |
mex-5 |
EC50 |
'=' |
21569 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
50118 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
12589 |
nM |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Inhibition |
- |
- |
- |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
35481 |
nM |
| Q15149 |
BXGT013547 |
Plectin |
reviewed |
Cellular structure |
PLEC |
IC50 |
'=' |
155815 |
nM |
| Q99816 |
BXGT019966 |
Tumor susceptibility gene 101 protein |
reviewed |
Enzyme |
TSG101 |
Potency |
- |
36587 |
nM |
| P35236 |
BXGT009802 |
Tyrosine-protein phosphatase non-receptor type 7 |
reviewed |
Enzyme |
PTPN7 |
IC50 |
'=' |
19620 |
nM |
| P30204 |
BXGT009411 |
Macrophage scavenger receptor types I and II |
reviewed |
- |
Msr1 |
Inhibition |
- |
- |
- |
| Q14191 |
BXGT013452 |
Werner syndrome ATP-dependent helicase |
reviewed |
Enzyme |
WRN |
Potency |
- |
26679 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P08238 |
BXGT006753 |
Heat shock protein HSP 90-beta |
reviewed |
Chaperone |
HSP90AB1 |
IC50 |
'=' |
3339 |
nM |
| P07900 |
BXGT006696 |
Heat shock protein HSP 90-alpha |
reviewed |
Chaperone |
HSP90AA1 |
IC50 |
'=' |
3339 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
15848 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
35481 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
25929 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
100000 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
22334 |
nM |
| P00766 |
BXGT005647 |
Chymotrypsinogen A |
reviewed |
- |
|
Inhibition |
'=' |
- |
- |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
Potency |
'=' |
25118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
35481 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
501 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
25118 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
11220 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
39810 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
'=' |
49 |
% |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'>' |
10000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
794 |
nM |
| Q9Z0J5 |
BXGT022399 |
Thioredoxin reductase 2, mitochondrial |
reviewed |
- |
Txnrd2 |
IC50 |
'=' |
123000 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
39810 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
125892 |
nM |
| G5EF15 |
BXGT003524 |
Cytoplasmic zinc-finger protein |
unreviewed |
- |
pos-1 |
EC50 |
'=' |
29176 |
nM |
| P08419 |
BXGT006770 |
Chymotrypsin-like elastase family member 2A |
reviewed |
- |
CELA2A |
Inhibition |
- |
- |
- |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Potency |
- |
37578 |
nM |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
15848 |
nM |
| P10145 |
BXGT007542 |
Interleukin-8 |
reviewed |
Signaling |
CXCL8 |
Potency |
- |
74978 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
28183 |
nM |
| Q15149 |
BXGT013547 |
Plectin |
reviewed |
Cellular structure |
PLEC |
IC50 |
'>' |
200000 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
15848 |
nM |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
130000 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
35481 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
4256 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
28183 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
50118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Inhibition |
'=' |
40 |
% |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
IC50 |
'=' |
84000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
28183 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
'=' |
28183 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
28183 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
- |
- |
- |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
25118 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
31622 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Control |
'=' |
96 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Control |
'=' |
96 |
% |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
56234 |
nM |
| Q99816 |
BXGT019966 |
Tumor susceptibility gene 101 protein |
reviewed |
Enzyme |
TSG101 |
Potency |
- |
50118 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
2511 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Control |
'=' |
99 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Control |
'=' |
99 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
17782 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
11220 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
79432 |
nM |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
15848 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
33491 |
nM |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Inhibition |
'=' |
22 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| Q15149 |
BXGT013547 |
Plectin |
reviewed |
Cellular structure |
PLEC |
IC50 |
'=' |
32104 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Inhibition |
'=' |
3 |
% |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
39810 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
50118 |
nM |
| P16234 |
BXGT008209 |
Platelet-derived growth factor receptor alpha |
reviewed |
Kinase |
PDGFRA |
Activity |
- |
- |
- |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Control |
'=' |
97 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Control |
'=' |
97 |
% |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
12589 |
nM |
| P11308 |
BXGT007684 |
Transcriptional regulator ERG |
reviewed |
Transcription factor |
ERG |
Potency |
- |
14125 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
28183 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
67015 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
2818 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
3162 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
50118 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
50118 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18356 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
'=' |
17000 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
25118 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
10000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
47443 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
22387 |
nM |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
2511 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
12589 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
10000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Potency |
- |
21192 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
25118 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
29092 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
75686 |
nM |
| P37136 |
BXGT009967 |
Acetylcholinesterase |
reviewed |
- |
Ache |
Inhibition |
'<' |
10 |
% |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
12589 |
nM |
| Q9NXA8 |
BXGT021245 |
NAD-dependent protein deacylase sirtuin-5, mitochondrial |
reviewed |
Epigenetic regulator |
SIRT5 |
AC50 |
'>' |
30000 |
nM |
| P54149 |
BXGT011034 |
Mitochondrial peptide methionine sulfoxide reductase |
reviewed |
- |
MSRA |
IC50 |
- |
155058 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
39810 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
35481 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
316 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
IC50 |
'=' |
637 |
nM |