| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
Inhibition |
'=' |
96 |
% |
| P08151 |
BXGT006731 |
Zinc finger protein GLI1 |
reviewed |
- |
GLI1 |
Activity |
- |
- |
- |
| Q9UGI9 |
BXGT021682 |
5'-AMP-activated protein kinase subunit gamma-3 |
reviewed |
Enzyme modulator |
PRKAG3 |
Activity |
- |
- |
- |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Activity |
- |
- |
- |
| Q9Y478 |
BXGT022271 |
5'-AMP-activated protein kinase subunit beta-1 |
reviewed |
Kinase |
PRKAB1 |
Activity |
- |
- |
- |
| Q9UGJ0 |
BXGT021683 |
5'-AMP-activated protein kinase subunit gamma-2 |
reviewed |
Enzyme modulator |
PRKAG2 |
Activity |
- |
- |
- |
| P54619 |
BXGT011060 |
5'-AMP-activated protein kinase subunit gamma-1 |
reviewed |
Kinase |
PRKAG1 |
Activity |
- |
- |
- |
| O43741 |
BXGT004620 |
5'-AMP-activated protein kinase subunit beta-2 |
reviewed |
Enzyme modulator |
PRKAB2 |
Activity |
- |
- |
- |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Activity |
- |
- |
- |
| Q13133 |
BXGT013315 |
Oxysterols receptor LXR-alpha |
reviewed |
Nuclear receptor |
NR1H3 |
FC |
- |
- |
- |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Inhibition |
- |
- |
- |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
Ratio |
'=' |
0 |
- |
| P55055 |
BXGT011101 |
Oxysterols receptor LXR-beta |
reviewed |
Nuclear receptor |
NR1H2 |
FC |
- |
- |
- |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
3162 |
nM |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
FC |
'=' |
2 |
- |
| Q13133 |
BXGT013315 |
Oxysterols receptor LXR-alpha |
reviewed |
Nuclear receptor |
NR1H3 |
LC50 |
'=' |
25000 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
IC50 |
'=' |
33700 |
nM |
| P55055 |
BXGT011101 |
Oxysterols receptor LXR-beta |
reviewed |
Nuclear receptor |
NR1H2 |
EC50 |
'>' |
50000 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
6513 |
nM |
| P00489 |
BXGT005553 |
Glycogen phosphorylase, muscle form |
reviewed |
- |
PYGM |
IC50 |
'=' |
43000 |
nM |
| P0DPI0 |
BXGT007528 |
Botulinum neurotoxin type A |
reviewed |
- |
botA |
Ki |
'=' |
14300 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Activity |
- |
- |
- |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
3162 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Activity |
- |
- |
- |
| Q9UBT2 |
BXGT021663 |
SUMO-activating enzyme subunit 2 |
reviewed |
Enzyme |
UBA2 |
IC50 |
'=' |
9240 |
nM |
| Q9UBE0 |
BXGT021651 |
SUMO-activating enzyme subunit 1 |
reviewed |
Enzyme |
SAE1 |
IC50 |
'=' |
9240 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
IC50 |
'=' |
46250 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
IC50 |
'=' |
43600 |
nM |
| Q9UBT2 |
BXGT021663 |
SUMO-activating enzyme subunit 2 |
reviewed |
Enzyme |
UBA2 |
IC50 |
'=' |
13160 |
nM |
| Q9UBE0 |
BXGT021651 |
SUMO-activating enzyme subunit 1 |
reviewed |
Enzyme |
SAE1 |
IC50 |
'=' |
13160 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
CD |
'>' |
20 |
ug ml-1 |
| Q72874 |
BXGT016711 |
Pol polyprotein |
unreviewed |
- |
pol |
IC50 |
'>' |
219000 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
EC50 |
'=' |
0 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5804 |
nM |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
7079 |
nM |
| Q8TDU6 |
BXGT018814 |
G-protein coupled bile acid receptor 1 |
reviewed |
G-protein coupled receptor |
GPBAR1 |
Efficacy |
'=' |
83 |
% |
| Q8WZA2 |
BXGT019025 |
Rap guanine nucleotide exchange factor 4 |
reviewed |
Enzyme modulator |
RAPGEF4 |
Potency |
- |
100000 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
3981 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
101 |
% |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
IC50 |
'=' |
14000 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
3162 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
Inhibition |
- |
- |
- |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
Emax |
- |
- |
- |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
8912 |
nM |
| P05771 |
BXGT006384 |
Protein kinase C beta type |
reviewed |
Kinase |
PRKCB |
IC50 |
'>' |
150000 |
nM |
| Q8TDU6 |
BXGT018814 |
G-protein coupled bile acid receptor 1 |
reviewed |
G-protein coupled receptor |
GPBAR1 |
EC50 |
'=' |
1040 |
nM |
| P08151 |
BXGT006731 |
Zinc finger protein GLI1 |
reviewed |
- |
GLI1 |
IC50 |
'=' |
32000 |
nM |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
Inhibition |
'=' |
63 |
% |
| P00489 |
BXGT005553 |
Glycogen phosphorylase, muscle form |
reviewed |
- |
PYGM |
IC50 |
'=' |
42657 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
55820 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Kd |
'=' |
593 |
nM |
| Q02156 |
BXGT012639 |
Protein kinase C epsilon type |
reviewed |
Kinase |
PRKCE |
IC50 |
'>' |
150000 |
nM |
| Q8IUX4 |
BXGT018337 |
DNA dC->dU-editing enzyme APOBEC-3F |
reviewed |
Enzyme |
APOBEC3F |
Potency |
- |
6309 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
20596 |
nM |
| P55055 |
BXGT011101 |
Oxysterols receptor LXR-beta |
reviewed |
Nuclear receptor |
NR1H2 |
LC50 |
'>' |
25000 |
nM |
| P0DPI0 |
BXGT007528 |
Botulinum neurotoxin type A |
reviewed |
- |
botA |
IC50 |
'=' |
20000 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
11000 |
nM |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
IC50 |
'=' |
6500 |
nM |
| Q76270 |
BXGT016848 |
GP41 |
unreviewed |
- |
HIV1 |
EC50 |
'>' |
100000 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
Inhibition |
'<' |
10 |
% |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Ka |
'=' |
1 |
10'6/M |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Inhibition |
- |
- |
- |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'>' |
10 |
ug ml-1 |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
38 |
% |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
EC50 |
'>' |
100000 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
2 |
% |
| P00690 |
BXGT005612 |
Pancreatic alpha-amylase |
reviewed |
- |
AMY2 |
IC50 |
'>' |
200000 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
Ratio |
'=' |
0 |
- |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Kd |
'=' |
4500 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
18356 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
920 |
nM |
| Q9HC16 |
BXGT020525 |
DNA dC->dU-editing enzyme APOBEC-3G |
reviewed |
Enzyme |
APOBEC3G |
Potency |
- |
8912 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
6513 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
112 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
3662 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Kd |
'=' |
1300 |
nM |
| P13726 |
BXGT007950 |
Tissue factor |
reviewed |
Receptor |
F3 |
IC50 |
- |
- |
- |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
-5 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
7307 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Activity |
- |
- |
- |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
37685 |
nM |
| Q13133 |
BXGT013315 |
Oxysterols receptor LXR-alpha |
reviewed |
Nuclear receptor |
NR1H3 |
EC50 |
'>' |
50000 |
nM |
| P11597 |
BXGT007727 |
Cholesteryl ester transfer protein |
reviewed |
- |
CETP |
IC50 |
- |
- |
- |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
25 |
% |
| Q923J1 |
BXGT019344 |
Transient receptor potential cation channel subfamily M member 7 |
reviewed |
- |
Trpm7 |
Inhibition |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
2000 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
IC50 |
'>' |
10000 |
nM |
| P11597 |
BXGT007727 |
Cholesteryl ester transfer protein |
reviewed |
- |
CETP |
Inhibition |
'=' |
31 |
% |
| Q9QUK6 |
BXGT021375 |
Toll-like receptor 4 |
reviewed |
- |
Tlr4 |
Inhibition |
- |
- |
- |