| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Vmax |
'=' |
289 |
uM min-1 (mg of protein)-1 |
| Q9TVW2 |
BXGT021628 |
Adenosine kinase |
reviewed |
- |
AK |
Ki |
'=' |
8900 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Vmax |
'=' |
435 |
M min-1 mg-1 |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
9466 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ratio |
'=' |
80 |
- |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Ratio |
'=' |
80 |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ratio |
'=' |
80 |
- |
| O95398 |
BXGT005378 |
Rap guanine nucleotide exchange factor 3 |
reviewed |
Enzyme modulator |
RAPGEF3 |
Potency |
- |
125892 |
nM |
| P22629 |
BXGT008788 |
Streptavidin |
reviewed |
- |
|
Activity |
- |
- |
- |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Inhibition |
'=' |
15 |
% |
| Q9Y0I0 |
BXGT022205 |
Adenosine transporter 1 |
unreviewed |
- |
AT1 |
Km |
'=' |
700 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
EC50 |
'=' |
290 |
nM |
| P42356 |
BXGT010305 |
Phosphatidylinositol 4-kinase alpha |
reviewed |
Kinase |
PI4KA |
Ki |
'=' |
19200 |
nM |
| Q9UBF8 |
BXGT021653 |
Phosphatidylinositol 4-kinase beta |
reviewed |
Kinase |
PI4KB |
Ki |
'=' |
19200 |
nM |
| Q8TCG2 |
BXGT018798 |
Phosphatidylinositol 4-kinase type 2-beta |
reviewed |
Enzyme |
PI4K2B |
Ki |
'=' |
19200 |
nM |
| Q9BTU6 |
BXGT020127 |
Phosphatidylinositol 4-kinase type 2-alpha |
reviewed |
Kinase |
PI4K2A |
Ki |
'=' |
19200 |
nM |
| Q62674 |
BXGT016038 |
Sodium/nucleoside cotransporter 1 |
reviewed |
- |
Slc28a1 |
Activity |
- |
- |
- |
| Q9NFS5 |
BXGT021130 |
Spermidine synthase |
unreviewed |
- |
spds |
Activity |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
EC50 |
'=' |
730 |
nM |
| P42226 |
BXGT010288 |
Signal transducer and activator of transcription 6 |
reviewed |
Nucleic acid binding |
STAT6 |
Potency |
'=' |
1258 |
nM |
| P22629 |
BXGT008788 |
Streptavidin |
reviewed |
- |
|
Kd |
'=' |
168000 |
nM |
| O43868 |
BXGT004631 |
Sodium/nucleoside cotransporter 2 |
reviewed |
Transporter |
SLC28A2 |
Drug transport |
- |
- |
- |
| Q99808 |
BXGT019964 |
Equilibrative nucleoside transporter 1 |
reviewed |
Transporter |
SLC29A1 |
IC50 |
'=' |
17000 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
96 |
% |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
8436 |
nM |
| P00491 |
BXGT005555 |
Purine nucleoside phosphorylase |
reviewed |
Enzyme |
PNP |
Ki |
'=' |
2000000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
EC50 |
'=' |
310 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Relative Vmax |
'=' |
100 |
- |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Vmax |
'=' |
0 |
uM min-1 unit-1 |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
EC50 |
'=' |
51286 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
pKA |
'=' |
4 |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Affinity constant |
'=' |
0 |
uM |
| P00515 |
BXGT005566 |
cAMP-dependent protein kinase type II-alpha regulatory subunit |
reviewed |
- |
PRKAR2A |
Ki |
'=' |
15000 |
nM |
| P31322 |
BXGT009520 |
cAMP-dependent protein kinase type II-beta regulatory subunit |
reviewed |
- |
PRKAR2B |
Ki |
'=' |
15000 |
nM |
| P05131 |
BXGT006323 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
- |
PRKACB |
Ki |
'=' |
15000 |
nM |
| P00517 |
BXGT005568 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
- |
PRKACA |
Ki |
'=' |
15000 |
nM |
| P00515 |
BXGT005566 |
cAMP-dependent protein kinase type II-alpha regulatory subunit |
reviewed |
- |
PRKAR2A |
IC50 |
'=' |
1100000 |
nM |
| P31322 |
BXGT009520 |
cAMP-dependent protein kinase type II-beta regulatory subunit |
reviewed |
- |
PRKAR2B |
IC50 |
'=' |
1100000 |
nM |
| P05131 |
BXGT006323 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
- |
PRKACB |
IC50 |
'=' |
1100000 |
nM |
| P00517 |
BXGT005568 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
- |
PRKACA |
IC50 |
'=' |
1100000 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
50000000 |
nM |
| Q61672 |
BXGT016021 |
Equilibrative nucleoside transporter 2 |
reviewed |
- |
Slc29a2 |
Activity |
- |
- |
- |
| Q9JIM1 |
BXGT020818 |
Equilibrative nucleoside transporter 1 |
reviewed |
- |
Slc29a1 |
Activity |
- |
- |
- |
| Q9X034 |
BXGT022047 |
5-methylthioadenosine/S-adenosylhomocysteine deaminase |
reviewed |
- |
mtaD |
Kcat/Km |
'=' |
9 |
10^3/M/s |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
33000 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
EC50 |
'=' |
40000 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
5 |
nM |
| P29276 |
BXGT009329 |
Adenosine receptor A2b |
reviewed |
- |
Adora2b |
Ki |
'=' |
5 |
nM |
| P03958 |
BXGT006121 |
Adenosine deaminase |
reviewed |
- |
Ada |
Km |
'=' |
7800 |
nM |
| O54699 |
BXGT004729 |
Equilibrative nucleoside transporter 2 |
reviewed |
- |
Slc29a2 |
Activity |
- |
- |
- |
| P47745 |
BXGT010581 |
Adenosine receptor A1 |
reviewed |
- |
ADORA1 |
EC50 |
'=' |
3388 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
k cat |
'=' |
76 |
s-1 |
| P00491 |
BXGT005555 |
Purine nucleoside phosphorylase |
reviewed |
Enzyme |
PNP |
Inhibition |
'=' |
30 |
% |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ratio |
'=' |
2 |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ratio |
'=' |
2 |
- |
| P29276 |
BXGT009329 |
Adenosine receptor A2b |
reviewed |
- |
Adora2b |
Ratio |
'=' |
2 |
- |
| O54698 |
BXGT004728 |
Equilibrative nucleoside transporter 1 |
reviewed |
- |
Slc29a1 |
Activity |
- |
- |
- |
| O00337 |
BXGT003911 |
Sodium/nucleoside cotransporter 1 |
reviewed |
Transporter |
SLC28A1 |
Drug transport |
- |
- |
- |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
42000 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
EC50 |
'=' |
51 |
nM |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
EC50 |
'=' |
51 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
29000 |
nM |
| P21802 |
BXGT008691 |
Fibroblast growth factor receptor 2 |
reviewed |
Kinase |
FGFR2 |
Concentration |
'=' |
50 |
uM |
| P22455 |
BXGT008772 |
Fibroblast growth factor receptor 4 |
reviewed |
Kinase |
FGFR4 |
Concentration |
'=' |
50 |
uM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Concentration |
'=' |
50 |
uM |
| P22607 |
BXGT008784 |
Fibroblast growth factor receptor 3 |
reviewed |
Kinase |
FGFR3 |
Concentration |
'=' |
50 |
uM |
| Q9GZV3 |
BXGT020427 |
High affinity choline transporter 1 |
reviewed |
Transporter |
SLC5A7 |
IC50 |
- |
570 |
nM |
| P23526 |
BXGT008878 |
Adenosylhomocysteinase |
reviewed |
Enzyme |
AHCY |
Km |
'=' |
820 |
nM |
| P23526 |
BXGT008878 |
Adenosylhomocysteinase |
reviewed |
Enzyme |
AHCY |
k cat |
'=' |
91 |
M-1 |
| P00515 |
BXGT005566 |
cAMP-dependent protein kinase type II-alpha regulatory subunit |
reviewed |
- |
PRKAR2A |
Ratio |
'=' |
6 |
- |
| P31322 |
BXGT009520 |
cAMP-dependent protein kinase type II-beta regulatory subunit |
reviewed |
- |
PRKAR2B |
Ratio |
'=' |
6 |
- |
| P05131 |
BXGT006323 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
- |
PRKACB |
Ratio |
'=' |
6 |
- |
| P00517 |
BXGT005568 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
- |
PRKACA |
Ratio |
'=' |
6 |
- |
| P00813 |
BXGT005667 |
Adenosine deaminase |
reviewed |
Enzyme |
ADA |
Ka |
'=' |
100000000 |
M-1 |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
50000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'~' |
1600000 |
nM |
| P42356 |
BXGT010305 |
Phosphatidylinositol 4-kinase alpha |
reviewed |
Kinase |
PI4KA |
Km |
'=' |
178900 |
nM |
| Q9UBF8 |
BXGT021653 |
Phosphatidylinositol 4-kinase beta |
reviewed |
Kinase |
PI4KB |
Km |
'=' |
178900 |
nM |
| Q8TCG2 |
BXGT018798 |
Phosphatidylinositol 4-kinase type 2-beta |
reviewed |
Enzyme |
PI4K2B |
Km |
'=' |
178900 |
nM |
| Q9BTU6 |
BXGT020127 |
Phosphatidylinositol 4-kinase type 2-alpha |
reviewed |
Kinase |
PI4K2A |
Km |
'=' |
178900 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
50450 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
EC50 |
'=' |
1040 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
100000000 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
37 |
nM |
| P29276 |
BXGT009329 |
Adenosine receptor A2b |
reviewed |
- |
Adora2b |
Ki |
'=' |
37 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
12 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
25000 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
- |
- |
- |
| Q62773 |
BXGT016044 |
Sodium/nucleoside cotransporter 2 |
reviewed |
- |
Slc28a2 |
Activity |
- |
- |
- |
| P23526 |
BXGT008878 |
Adenosylhomocysteinase |
reviewed |
Enzyme |
AHCY |
Inhibitory potency |
- |
- |
- |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
30000 |
nM |
| P00813 |
BXGT005667 |
Adenosine deaminase |
reviewed |
Enzyme |
ADA |
Ki |
'=' |
2180000 |
nM |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Emax |
'=' |
70 |
% |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
15848 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Relative Vmax |
'=' |
1 |
- |
| Q14542 |
BXGT013482 |
Equilibrative nucleoside transporter 2 |
reviewed |
Transporter |
SLC29A2 |
Ki |
'=' |
106000 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
EC50 |
'=' |
2511 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
'=' |
1 |
nM |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Activity |
'=' |
8 |
% |
| P02701 |
BXGT005926 |
Avidin |
reviewed |
- |
AVD |
Kq |
'=' |
1 |
10'11L/mol/s |
| P11142 |
BXGT007658 |
Heat shock cognate 71 kDa protein |
reviewed |
- |
HSPA8 |
Kd |
'=' |
110000 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Activity |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Activity |
- |
- |
- |
| P28647 |
BXGT009282 |
Adenosine receptor A3 |
reviewed |
- |
Adora3 |
Ki |
'=' |
100 |
nM |
| P02769 |
BXGT005956 |
Serum albumin |
reviewed |
- |
ALB |
Activity |
- |
- |
- |
| Q9X034 |
BXGT022047 |
5-methylthioadenosine/S-adenosylhomocysteine deaminase |
reviewed |
- |
mtaD |
Km |
'=' |
250000 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
EC50 |
'=' |
700 |
nM |
| O00337 |
BXGT003911 |
Sodium/nucleoside cotransporter 1 |
reviewed |
Transporter |
SLC28A1 |
Ki |
'=' |
1800 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Concentration |
'=' |
50 |
uM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
30 |
nM |
| P39069 |
BXGT010089 |
Adenylate kinase isoenzyme 1 |
reviewed |
- |
Ak1 |
Ki |
'=' |
19000000 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
24500 |
nM |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
ED50 |
'=' |
10 |
uM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
log(activity) |
'=' |
0 |
- |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Displacement |
'=' |
10 |
% |
| P20839 |
BXGT008608 |
Inosine-5'-monophosphate dehydrogenase 1 |
reviewed |
Enzyme |
IMPDH1 |
Ki |
'>' |
100000 |
nM |
| Q9QUK6 |
BXGT021375 |
Toll-like receptor 4 |
reviewed |
- |
Tlr4 |
Inhibition |
- |
- |
- |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
32000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
180 |
% |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Emax |
'=' |
65 |
% |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
35000000 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
1500 |
nM |
| Q9HAS3 |
BXGT020507 |
Solute carrier family 28 member 3 |
reviewed |
Transporter |
SLC28A3 |
IC50 |
'=' |
3300 |
nM |
| P00515 |
BXGT005566 |
cAMP-dependent protein kinase type II-alpha regulatory subunit |
reviewed |
- |
PRKAR2A |
IC50 |
'=' |
160000 |
nM |
| P31322 |
BXGT009520 |
cAMP-dependent protein kinase type II-beta regulatory subunit |
reviewed |
- |
PRKAR2B |
IC50 |
'=' |
160000 |
nM |
| P05131 |
BXGT006323 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
- |
PRKACB |
IC50 |
'=' |
160000 |
nM |
| P00517 |
BXGT005568 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
- |
PRKACA |
IC50 |
'=' |
160000 |
nM |
| P39069 |
BXGT010089 |
Adenylate kinase isoenzyme 1 |
reviewed |
- |
Ak1 |
Ki |
'=' |
82000000 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
EC50 |
'=' |
39 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
10 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Activity |
'=' |
10 |
% |
| O43318 |
BXGT004586 |
Mitogen-activated protein kinase kinase kinase 7 |
reviewed |
Kinase |
MAP3K7 |
Kd |
'=' |
34000 |
nM |
| P23526 |
BXGT008878 |
Adenosylhomocysteinase |
reviewed |
Enzyme |
AHCY |
Ki |
- |
- |
- |
| Q04400 |
BXGT012760 |
Adenylate cyclase type 5 |
reviewed |
- |
Adcy5 |
IC50 |
'>' |
300000 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Affinity constant |
'=' |
10 |
uM |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Affinity constant |
'=' |
10 |
uM |
| P28647 |
BXGT009282 |
Adenosine receptor A3 |
reviewed |
- |
Adora3 |
Ratio |
'=' |
100 |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ratio |
'=' |
100 |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
5 |
nM |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Ratio |
'=' |
1 |
- |
| P00491 |
BXGT005555 |
Purine nucleoside phosphorylase |
reviewed |
Enzyme |
PNP |
Activity |
'=' |
0 |
% |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Affinity constant |
'=' |
20 |
uM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Affinity constant |
'=' |
20 |
uM |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Affinity constant |
'=' |
20 |
uM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Affinity constant |
'=' |
20 |
uM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
'=' |
20 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
Ki |
'=' |
2500000 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
100000 |
nM |
| P28647 |
BXGT009282 |
Adenosine receptor A3 |
reviewed |
- |
Adora3 |
Displacement |
'=' |
10 |
% |
| P42356 |
BXGT010305 |
Phosphatidylinositol 4-kinase alpha |
reviewed |
Kinase |
PI4KA |
IC50 |
'=' |
30300 |
nM |
| Q9UBF8 |
BXGT021653 |
Phosphatidylinositol 4-kinase beta |
reviewed |
Kinase |
PI4KB |
IC50 |
'=' |
30300 |
nM |
| Q8TCG2 |
BXGT018798 |
Phosphatidylinositol 4-kinase type 2-beta |
reviewed |
Enzyme |
PI4K2B |
IC50 |
'=' |
30300 |
nM |
| Q9BTU6 |
BXGT020127 |
Phosphatidylinositol 4-kinase type 2-alpha |
reviewed |
Kinase |
PI4K2A |
IC50 |
'=' |
30300 |
nM |
| P12268 |
BXGT007783 |
Inosine-5'-monophosphate dehydrogenase 2 |
reviewed |
Enzyme |
IMPDH2 |
Ki |
'>' |
100000 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
29000 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Ratio |
'=' |
6 |
- |
| P07205 |
BXGT006568 |
Phosphoglycerate kinase 2 |
reviewed |
Kinase |
PGK2 |
IC50 |
'=' |
3000000 |
nM |
| P00558 |
BXGT005579 |
Phosphoglycerate kinase 1 |
reviewed |
Kinase |
PGK1 |
IC50 |
'=' |
3000000 |
nM |
| Q9TVW2 |
BXGT021628 |
Adenosine kinase |
reviewed |
- |
AK |
Km |
'=' |
2400 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
KD hydro |
- |
- |
- |
| P29410 |
BXGT009345 |
Adenylate kinase 2, mitochondrial |
reviewed |
- |
Ak2 |
Ki |
'=' |
92000000 |
nM |
| P00813 |
BXGT005667 |
Adenosine deaminase |
reviewed |
Enzyme |
ADA |
Km |
'=' |
5000 |
nM |
| P29410 |
BXGT009345 |
Adenylate kinase 2, mitochondrial |
reviewed |
- |
Ak2 |
Ki |
'=' |
87000000 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
43240 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
12589 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
IC50 |
'=' |
35000 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Kd |
- |
- |
- |
| P02701 |
BXGT005926 |
Avidin |
reviewed |
- |
AVD |
Activity |
- |
- |
- |
| O04417 |
BXGT003966 |
Calcium dependent protein kinase |
unreviewed |
- |
ZmCDPK1 |
IC50 |
'=' |
116000 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Displacement |
'=' |
25 |
% |
| P39069 |
BXGT010089 |
Adenylate kinase isoenzyme 1 |
reviewed |
- |
Ak1 |
Ki |
'=' |
580000 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
31000 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
31622 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
195000 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
EC50 |
'=' |
1410 |
nM |
| P22629 |
BXGT008788 |
Streptavidin |
reviewed |
- |
|
Kq |
'=' |
8 |
10'10L/mol/s |
| P02701 |
BXGT005926 |
Avidin |
reviewed |
- |
AVD |
Kd |
'=' |
117000 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
pKA |
'=' |
5 |
- |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Concentration |
'=' |
50 |
uM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
k cat/Km |
'=' |
3 |
uM-1 s-1 |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Activity |
- |
- |
- |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
Activity |
- |
- |
- |
| Q8TEK3 |
BXGT018822 |
Histone-lysine N-methyltransferase, H3 lysine-79 specific |
reviewed |
Epigenetic regulator |
DOT1L |
IC50 |
'=' |
100000 |
nM |
| P05771 |
BXGT006384 |
Protein kinase C beta type |
reviewed |
Kinase |
PRKCB |
IC50 |
'=' |
278000 |
nM |
| P56658 |
BXGT011188 |
Adenosine deaminase |
reviewed |
- |
ADA |
Km |
'=' |
45300 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
1122 |
nM |
| Q6DHV7 |
BXGT016246 |
Adenosine deaminase-like protein |
reviewed |
- |
ADAL |
Activity |
- |
- |
- |
| Q9GZV3 |
BXGT020427 |
High affinity choline transporter 1 |
reviewed |
Transporter |
SLC5A7 |
IC50 |
- |
199 |
nM |
| Q9X034 |
BXGT022047 |
5-methylthioadenosine/S-adenosylhomocysteine deaminase |
reviewed |
- |
mtaD |
Kcat |
'=' |
2 |
/s |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
EC50 |
'=' |
5754 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Emax |
'=' |
91 |
% |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
EC50 |
'=' |
24000 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Activity |
'=' |
-38 |
% |
| O88627 |
BXGT005278 |
Sodium/nucleoside cotransporter 2 |
reviewed |
- |
Slc28a2 |
Activity |
- |
- |
- |
| P11142 |
BXGT007658 |
Heat shock cognate 71 kDa protein |
reviewed |
- |
HSPA8 |
Kd |
'=' |
112201 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
25929 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
EC50 |
'>' |
112219 |
nM |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Drug metabolism |
'=' |
60 |
% |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Activity |
'=' |
20 |
% |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
EC50 |
'=' |
23500 |
nM |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Activity |
'=' |
100 |
% |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
log(activity) |
'=' |
0 |
- |
| Q9HAS3 |
BXGT020507 |
Solute carrier family 28 member 3 |
reviewed |
Transporter |
SLC28A3 |
Ki |
'=' |
2100 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
log(activity) |
'=' |
0 |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
'=' |
2 |
nM |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
1613 |
nM |
| O43318 |
BXGT004586 |
Mitogen-activated protein kinase kinase kinase 7 |
reviewed |
Kinase |
MAP3K7 |
Kd |
'=' |
4400 |
nM |
| Q99808 |
BXGT019964 |
Equilibrative nucleoside transporter 1 |
reviewed |
Transporter |
SLC29A1 |
Ki |
'=' |
12000 |
nM |
| Q13126 |
BXGT013313 |
S-methyl-5'-thioadenosine phosphorylase |
reviewed |
Enzyme |
MTAP |
Drug metabolism |
'=' |
596 |
nmol/mg/hr |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
4775 |
nM |
| O43868 |
BXGT004631 |
Sodium/nucleoside cotransporter 2 |
reviewed |
Transporter |
SLC28A2 |
Ki |
'=' |
5300 |
nM |
| Q14542 |
BXGT013482 |
Equilibrative nucleoside transporter 2 |
reviewed |
Transporter |
SLC29A2 |
IC50 |
'=' |
106000 |
nM |
| P50389 |
BXGT010795 |
Purine nucleoside phosphorylase |
reviewed |
- |
SSO2706 |
Drug metabolism |
'=' |
57000 |
nmol/mg/hr |
| O43868 |
BXGT004631 |
Sodium/nucleoside cotransporter 2 |
reviewed |
Transporter |
SLC28A2 |
IC50 |
'=' |
5500 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Activity |
'=' |
-66 |
% |
| O00337 |
BXGT003911 |
Sodium/nucleoside cotransporter 1 |
reviewed |
Transporter |
SLC28A1 |
IC50 |
'=' |
5500 |
nM |
| P0AF12 |
BXGT007340 |
5'-methylthioadenosine/S-adenosylhomocysteine nucleosidase |
reviewed |
- |
mtnN |
Drug metabolism |
'=' |
2100 |
nmol/mg/hr |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Kd |
'=' |
184000 |
nM |
| P29275 |
BXGT009328 |
Adenosine receptor A2b |
reviewed |
G-protein coupled receptor |
ADORA2B |
pKA |
'=' |
3 |
- |
| Q9HAS3 |
BXGT020507 |
Solute carrier family 28 member 3 |
reviewed |
Transporter |
SLC28A3 |
Drug transport |
- |
- |
- |