| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
35000 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
10322 |
nM |
| P33437 |
BXGT009725 |
Collagenase |
reviewed |
- |
prtC |
Activity |
'=' |
82 |
% |
| P33437 |
BXGT009725 |
Collagenase |
reviewed |
- |
prtC |
Activity |
'=' |
48 |
% |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
39810 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
8196 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'>' |
100000 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
50118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
11220 |
nM |
| P36544 |
BXGT009926 |
Neuronal acetylcholine receptor subunit alpha-7 |
reviewed |
- |
CHRNA7 |
Ratio |
'=' |
6 |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Potency |
- |
3981 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
3 |
ug.mL-1 |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
10691 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
IC50 |
'=' |
32000 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
IC50 |
'=' |
32000 |
nM |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
IC50 |
'=' |
32000 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
7943 |
nM |
| P37840 |
BXGT010015 |
Alpha-synuclein |
reviewed |
Transporter |
SNCA |
Potency |
- |
32642 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'=' |
3 |
uM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Potency |
- |
16360 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'>' |
50000 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'=' |
11 |
uM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
15848 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
15848 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
26121 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
1778 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
Activity |
'=' |
1 |
uM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
130000 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
130000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
210 |
% |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
'=' |
11220 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Inhibition |
'=' |
10 |
% |
| Q6W5P4 |
BXGT016588 |
Neuropeptide S receptor |
reviewed |
- |
NPSR1 |
Potency |
'=' |
31622 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
- |
50118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7943 |
nM |
| P33437 |
BXGT009725 |
Collagenase |
reviewed |
- |
prtC |
Activity |
'=' |
78 |
% |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Inhibition |
'=' |
14 |
% |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
3 |
ug.mL-1 |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
0 |
% |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Inhibition |
- |
- |
- |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
2930 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
44668 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
119 |
% |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
79432 |
nM |
| P21802 |
BXGT008691 |
Fibroblast growth factor receptor 2 |
reviewed |
Kinase |
FGFR2 |
Inhibition |
'=' |
0 |
% |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
35481 |
nM |
| P0A6C1 |
BXGT007045 |
Endonuclease 4 |
reviewed |
- |
nfo |
Potency |
'=' |
631 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
6309 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
'=' |
3981 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'=' |
3 |
uM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
1 |
- |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Inhibition |
'=' |
0 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'>' |
60000 |
nM |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
19952 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
1995 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
Activity |
'=' |
2 |
uM |
| Q04759 |
BXGT012781 |
Protein kinase C theta type |
reviewed |
Kinase |
PRKCQ |
Inhibition |
- |
- |
- |
| Q15139 |
BXGT013546 |
Serine/threonine-protein kinase D1 |
reviewed |
Kinase |
PRKD1 |
Inhibition |
- |
- |
- |
| P24723 |
BXGT008989 |
Protein kinase C eta type |
reviewed |
Kinase |
PRKCH |
Inhibition |
- |
- |
- |
| Q02156 |
BXGT012639 |
Protein kinase C epsilon type |
reviewed |
Kinase |
PRKCE |
Inhibition |
- |
- |
- |
| Q05513 |
BXGT012820 |
Protein kinase C zeta type |
reviewed |
Kinase |
PRKCZ |
Inhibition |
- |
- |
- |
| P05771 |
BXGT006384 |
Protein kinase C beta type |
reviewed |
Kinase |
PRKCB |
Inhibition |
- |
- |
- |
| Q05655 |
BXGT012832 |
Protein kinase C delta type |
reviewed |
Kinase |
PRKCD |
Inhibition |
- |
- |
- |
| P05129 |
BXGT006322 |
Protein kinase C gamma type |
reviewed |
Kinase |
PRKCG |
Inhibition |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Inhibition |
- |
- |
- |
| P41743 |
BXGT010270 |
Protein kinase C iota type |
reviewed |
Kinase |
PRKCI |
Inhibition |
- |
- |
- |
| O94806 |
BXGT005335 |
Serine/threonine-protein kinase D3 |
reviewed |
Kinase |
PRKD3 |
Inhibition |
- |
- |
- |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
28183 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
10000 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
10 |
ug.mL-1 |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
1778 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
7943 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
'=' |
15848 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
100000 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
28183 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
22387 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
1 |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
3981 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
39810 |
nM |
| Q194T2 |
BXGT013743 |
Non-structural protein 1 |
unreviewed |
- |
NS1 |
Potency |
'=' |
15848 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
15101 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
6309 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
8 |
ug.mL-1 |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
320 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Activity |
'=' |
67 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
15848 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
3981 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
11220 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
10322 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
29934 |
nM |
| P51531 |
BXGT010851 |
Probable global transcription activator SNF2L2 |
reviewed |
Epigenetic regulator |
SMARCA2 |
EC50 |
'>' |
91140 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
89125 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
8436 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
31622 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
50118 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
79432 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
1122 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
12589 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
23109 |
nM |
| P36544 |
BXGT009926 |
Neuronal acetylcholine receptor subunit alpha-7 |
reviewed |
- |
CHRNA7 |
Activity |
- |
- |
- |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
112201 |
nM |
| Q4Q090 |
BXGT014858 |
2,3-bisphosphoglycerate-independent phosphoglycerate mutase |
unreviewed |
- |
PGAM |
Potency |
- |
37933 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
39810 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
'=' |
4466 |
nM |
| P19643 |
BXGT008505 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
Maob |
IC50 |
'=' |
47200 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
12995 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
Activity |
'=' |
9 |
uM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
94 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3548 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
3768 |
nM |
| P33437 |
BXGT009725 |
Collagenase |
reviewed |
- |
prtC |
Inhibition |
'=' |
52 |
% |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
2310 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Inhibition |
'=' |
13 |
% |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
400 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'=' |
360 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
4 |
- |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
25118 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
20596 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
'=' |
2830 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
1000 |
nM |
| P05412 |
BXGT006354 |
Transcription factor AP-1 |
reviewed |
Transcription factor |
JUN |
Inhibition |
- |
- |
- |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
'=' |
19952 |
nM |
| P21396 |
BXGT008643 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
Maoa |
IC50 |
'=' |
13900 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23109 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
21331 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
14581 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
25929 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
- |
- |
- |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
10000 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
79432 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
89125 |
nM |
| Q63921 |
BXGT016082 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
Ptgs1 |
IC50 |
'=' |
35000 |
nM |
| P35355 |
BXGT009817 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
Ptgs2 |
IC50 |
'=' |
35000 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
11 |
ug.mL-1 |
| P21396 |
BXGT008643 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
Maoa |
IC50 |
'=' |
17300 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
5 |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Activity |
'=' |
91 |
% |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
98 |
% |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
44668 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
70794 |
nM |
| P36544 |
BXGT009926 |
Neuronal acetylcholine receptor subunit alpha-7 |
reviewed |
- |
CHRNA7 |
EC50 |
'=' |
11600 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
10000 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
12589 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
19700 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
33000 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Activity |
'=' |
97 |
% |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
35481 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
89125 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
51500 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
8912 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
14 |
% |
| Q9Z1B7 |
BXGT022403 |
Mitogen-activated protein kinase 13 |
reviewed |
- |
Mapk13 |
FC |
'=' |
1 |
- |
| Q9WUI1 |
BXGT021940 |
Mitogen-activated protein kinase 11 |
reviewed |
- |
Mapk11 |
FC |
'=' |
1 |
- |
| O08911 |
BXGT004043 |
Mitogen-activated protein kinase 12 |
reviewed |
- |
Mapk12 |
FC |
'=' |
1 |
- |
| P47811 |
BXGT010587 |
Mitogen-activated protein kinase 14 |
reviewed |
- |
Mapk14 |
FC |
'=' |
1 |
- |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Inhibition |
'=' |
48 |
% |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
9 |
ug.mL-1 |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
28183 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Inhibition |
'=' |
50 |
% |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
6012 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Inhibition |
'=' |
3 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
269 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
48 |
% |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
1 |
- |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
15 |
% |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
47300 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Inhibition |
'=' |
22 |
% |
| Q96P20 |
BXGT019704 |
NACHT, LRR and PYD domains-containing protein 3 |
reviewed |
- |
NLRP3 |
IC50 |
'=' |
1540 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
1870 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
3800 |
nM |