| P23977 |
BXGT008936 |
Sodium-dependent dopamine transporter |
reviewed |
- |
Slc6a3 |
FC |
'=' |
100 |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
38 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
38 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
38 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
37685 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
45 |
% |
| Q8K4Z4 |
BXGT018404 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
EC50 |
'=' |
213 |
nM |
| P26255 |
BXGT009093 |
Beta-3 adrenergic receptor |
reviewed |
- |
Adrb3 |
EC50 |
'=' |
1580 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
37 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
37 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
37 |
nM |
| Q8K4Z4 |
BXGT018404 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
pD2 |
'=' |
6 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
450 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
450 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
450 |
nM |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Selectivity |
- |
- |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Inhibition |
'=' |
18 |
% |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Inhibition |
'=' |
18 |
% |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Inhibition |
'=' |
18 |
% |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
Ki |
'=' |
400 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
pD2 |
'=' |
6 |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
pD2 |
'=' |
6 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
pD2 |
'=' |
6 |
- |
| Q8K4Z4 |
BXGT018404 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
IA |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
4000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
4000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
4000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3162 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
4456 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Intrinsic activity |
'=' |
1 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Intrinsic activity |
'=' |
1 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Intrinsic activity |
'=' |
1 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Kd |
'=' |
3981 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
3548 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
44668 |
nM |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
15848 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7079 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
25118 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
22 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
217000 |
nM |
| P14920 |
BXGT008067 |
D-amino-acid oxidase |
reviewed |
- |
DAO |
IC50 |
'>' |
10000000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
501 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
EC50 |
'=' |
6 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
EC50 |
'=' |
794 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
6309 |
nM |
| Q9GZT4 |
BXGT020424 |
Serine racemase |
reviewed |
Enzyme |
SRR |
IC50 |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
#NAME? |
'=' |
6 |
- |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
1500 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
30131 |
nM |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
6506 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
2 |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
17 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
17 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
17 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
IC50 |
'=' |
33 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
IC50 |
'=' |
33 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
IC50 |
'=' |
33 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
1995 |
nM |
| O70594 |
BXGT005072 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Activity |
- |
- |
- |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
26000 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
pD2 |
'=' |
6 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
pD2 |
'=' |
6 |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
pD2 |
'=' |
6 |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Log 1/Kd |
'=' |
-4 |
- |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
2119 |
nM |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
pD2 |
'=' |
6 |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
EC50 |
'=' |
5 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Emax |
'=' |
105 |
% |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Emax |
'=' |
215 |
% |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
112 |
% |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
1300 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
17782 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
2238 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
342000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
891 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IA |
'=' |
1 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IA |
'=' |
1 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IA |
'=' |
1 |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Relative affinity |
'=' |
106 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Relative affinity |
'=' |
106 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Relative affinity |
'=' |
106 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Relative affinity |
'=' |
106 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Relative affinity |
'=' |
106 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Relative affinity |
'=' |
106 |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
pD2 |
'=' |
4 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
pD2 |
'=' |
4 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
pD2 |
'=' |
4 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
pD2 |
'=' |
4 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
pD2 |
'=' |
4 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
pD2 |
'=' |
4 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
446 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
2238 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
290 |
nM |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
7943 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
61130 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
'=' |
63 |
nM |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
Intrinsic activity |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
pD2 |
'=' |
5 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
pD2 |
'=' |
5 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
pD2 |
'=' |
5 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
EC50 |
'=' |
1174 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
EC50 |
'=' |
10232 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
EC50 |
'=' |
12 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
39810 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
707 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
EC50 |
'=' |
2187 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
EC50 |
'=' |
371 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
'=' |
1620 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IC50 |
'=' |
1620 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
'=' |
1620 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
21192 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
4 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
4 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
4 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Emax |
'=' |
113 |
% |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
2590 |
nM |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
EC50 |
'=' |
10000 |
nM |
| Q8K4Z4 |
BXGT018404 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
EC50 |
'=' |
30000 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Intrinsic activity |
'=' |
1 |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Intrinsic activity |
'=' |
1 |
- |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
IC50 |
'=' |
11000000 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
33807 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
134000 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
pD2 |
'=' |
8 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
pD2 |
'=' |
8 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
pD2 |
'=' |
8 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
pD2 |
'=' |
8 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
pD2 |
'=' |
8 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
pD2 |
'=' |
8 |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
EC50 |
'=' |
2600 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
EC50 |
'=' |
2600 |
nM |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
EC50 |
'=' |
2600 |
nM |
| Q28044 |
BXGT013944 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
Ki |
'=' |
6000 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
IC50 |
'=' |
16 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
IC50 |
'=' |
16 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
IC50 |
'=' |
16 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
'=' |
16 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IC50 |
'=' |
16 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
'=' |
16 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
340 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
340 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
340 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
490000 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Intrinsic activity |
'=' |
1 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Intrinsic activity |
'=' |
1 |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Intrinsic activity |
'=' |
1 |
- |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
Ki |
'=' |
20400 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
96700 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
3 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
3 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Activity |
- |
- |
- |
| Q8K4Z4 |
BXGT018404 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
Intrinsic activity |
'=' |
1 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
EC50 |
'=' |
118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
6500 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
6500 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
6500 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
191000 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
18 |
- |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
19952 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
1600 |
nM |
| P54833 |
BXGT011086 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
Ki |
'=' |
27000 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
'=' |
66 |
nM |
| P54833 |
BXGT011086 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
Ki |
'=' |
5000 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
EC50 |
- |
- |
- |
| P18130 |
BXGT008382 |
Alpha-1A adrenergic receptor |
reviewed |
- |
ADRA1A |
Ki |
'=' |
446 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
390 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
390 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
390 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Kd |
'=' |
50000 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Ki |
'=' |
1500 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
6 |
% |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
9 |
% |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
pD2 |
'=' |
6 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
pD2 |
'=' |
6 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
pD2 |
'=' |
6 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
pD2 |
'=' |
6 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
pD2 |
'=' |
6 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
pD2 |
'=' |
6 |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Intrinsic activity |
'=' |
1 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Intrinsic activity |
'=' |
1 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Intrinsic activity |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
3000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
3000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
3000 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Selectivity |
- |
- |
- |
| P26255 |
BXGT009093 |
Beta-3 adrenergic receptor |
reviewed |
- |
Adrb3 |
IC50 |
'=' |
1000 |
nM |
| P10608 |
BXGT007586 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
IC50 |
'=' |
1000 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
IC50 |
'=' |
1000 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
9 |
% |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
'=' |
30 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
'=' |
30 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
'=' |
30 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IA |
'=' |
1 |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IA |
'=' |
1 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IA |
'=' |
1 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Emax |
'=' |
100 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
2238 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
3981 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
'=' |
1500 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IC50 |
'=' |
1500 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
'=' |
1500 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
EC50 |
- |
- |
- |
| O75751 |
BXGT005150 |
Solute carrier family 22 member 3 |
reviewed |
Transporter |
SLC22A3 |
Km |
'=' |
510000 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
281 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
EC50 |
'=' |
15800 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
EC50 |
'=' |
15800 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
EC50 |
'=' |
15800 |
nM |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
Ki |
'=' |
2600 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
'=' |
2600 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Ki |
'=' |
2600 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
78 |
nM |
| Q9Y2I1 |
BXGT022235 |
Nischarin |
reviewed |
Enzyme modulator |
NISCH |
Ki |
'>' |
100000 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Selectivity |
'=' |
0 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Selectivity |
'=' |
0 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Emax |
'=' |
117 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
'=' |
0 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
6701 |
nM |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
9074 |
nM |
| Q62666 |
BXGT016037 |
Vesicular acetylcholine transporter |
reviewed |
- |
Slc18a3 |
Ki |
'>' |
10000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
8912 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
EC50 |
'=' |
1 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
EC50 |
'=' |
1 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
EC50 |
'=' |
1 |
nM |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Activity |
- |
- |
- |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
3548 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
EC50 |
'=' |
83200 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
EC50 |
'=' |
83200 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
EC50 |
'=' |
83200 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
5 |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
ISA |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
ISA |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
ISA |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
EC50 |
'=' |
110 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
EC50 |
'=' |
61 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
1776000 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
2700 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
1000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
1000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
1000 |
nM |
| Q28044 |
BXGT013944 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
#NAME? |
- |
- |
- |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
EC50 |
'=' |
30 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
378000 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
1 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ratio Ki |
'=' |
1 |
- |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
707 |
nM |
| P54833 |
BXGT011086 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
Ki |
'=' |
11000 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ratio |
'=' |
1 |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ratio |
'=' |
1 |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ratio |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ratio |
'=' |
1 |
- |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ratio |
'=' |
1 |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ratio |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
500 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
500 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
500 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
794 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Intrinsic activity |
'=' |
1 |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Activity |
'>' |
10000 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
410 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Intrinsic activity |
'=' |
1 |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Intrinsic activity |
'=' |
1 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Intrinsic activity |
'=' |
1 |
- |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
4400000 |
nM |
| P18841 |
BXGT008428 |
Alpha-1B adrenergic receptor |
reviewed |
- |
ADRA1B |
Ki |
'=' |
263 |
nM |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
Selectivity |
'=' |
0 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Selectivity |
'=' |
0 |
- |
| P26255 |
BXGT009093 |
Beta-3 adrenergic receptor |
reviewed |
- |
Adrb3 |
EC50 |
'=' |
52 |
nM |
| P10608 |
BXGT007586 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
EC50 |
'=' |
52 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
EC50 |
'=' |
52 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
pD2 |
'=' |
6 |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
pD2 |
'=' |
6 |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
pD2 |
'=' |
6 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
14 |
% |
| P0DMM9 |
BXGT007504 |
Sulfotransferase 1A3 |
reviewed |
- |
SULT1A3 |
Activity |
- |
- |
- |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
IC50 |
'=' |
750 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
IC50 |
'=' |
750 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
IC50 |
'=' |
750 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
KL |
'=' |
4141 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
KL |
'=' |
126000 |
nM |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
EC50 |
'=' |
350 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
1258 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3548 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
11 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Control response |
'=' |
6 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3981 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
EC50 |
'=' |
200 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
EC50 |
'=' |
200 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
EC50 |
'=' |
200 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
30 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
30 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
30 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
126 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
EC50 |
'=' |
166 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
EC50 |
'=' |
166 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
EC50 |
'=' |
166 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Intrinsic activity |
'=' |
96 |
% |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Activity |
- |
- |
- |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
11000000 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
IC50 |
'=' |
5000 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
IC50 |
'=' |
5000 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
IC50 |
'=' |
5000 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
'=' |
5000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IC50 |
'=' |
5000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
'=' |
5000 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
15848 |
nM |
| Q01338 |
BXGT012584 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
5800 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
9466 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
102 |
% |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Km |
'=' |
1900000 |
nM |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Activity |
- |
- |
- |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
707 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5623 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
25118 |
nM |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
37933 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
56234 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
891 |
nM |
| B0FL73 |
BXGT001833 |
Beta-1 adrenergic receptor |
unreviewed |
- |
ADRB1 |
IA |
'=' |
1 |
- |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
1901 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
50118 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Kd |
'=' |
3980 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
IC50 |
'=' |
434000 |
nM |
| Q9Z0E8 |
BXGT022397 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Activity |
'=' |
70 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
1300 |
nM |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
EC50 |
- |
- |
- |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
3981 |
nM |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
EC50 |
'=' |
128 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
756 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Activity |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
28183 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
28183 |
nM |
| Q01337 |
BXGT012583 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
650 |
nM |
| Q99489 |
BXGT019924 |
D-aspartate oxidase |
reviewed |
- |
DDO |
IC50 |
- |
- |
- |
| P10608 |
BXGT007586 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
Ki |
'=' |
4200 |
nM |
| P26255 |
BXGT009093 |
Beta-3 adrenergic receptor |
reviewed |
- |
Adrb3 |
EC50 |
'=' |
100000 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
20 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
20 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
20 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
#NAME? |
'=' |
8 |
- |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
PD2 |
'=' |
7 |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
PD2 |
'=' |
7 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
PD2 |
'=' |
7 |
- |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
E |
'=' |
100 |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
E |
'=' |
100 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
E |
'=' |
100 |
- |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'>' |
1000000 |
nM |
| P10608 |
BXGT007586 |
Beta-2 adrenergic receptor |
reviewed |
- |
Adrb2 |
Activity |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
10000 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
EC50 |
'=' |
9 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
3300 |
nM |