| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
56234 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
56234 |
nM |
| P62826 |
BXGT011463 |
GTP-binding nuclear protein Ran |
reviewed |
Enzyme modulator |
RAN |
Potency |
- |
56234 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
2511 |
nM |
| P22894 |
BXGT008815 |
Neutrophil collagenase |
reviewed |
Enzyme |
MMP8 |
Inhibition |
'=' |
9 |
% |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
Inhibition |
'=' |
-1 |
% |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Inhibition |
'=' |
20 |
% |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Inhibition |
'=' |
6 |
% |
| P52333 |
BXGT010928 |
Tyrosine-protein kinase JAK3 |
reviewed |
Kinase |
JAK3 |
Inhibition |
'=' |
78 |
% |
| Q13464 |
BXGT013357 |
Rho-associated protein kinase 1 |
reviewed |
Kinase |
ROCK1 |
Inhibition |
'=' |
28 |
% |
| P31751 |
BXGT009576 |
RAC-beta serine/threonine-protein kinase |
reviewed |
Kinase |
AKT2 |
Inhibition |
'=' |
7 |
% |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Inhibition |
'=' |
24 |
% |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Inhibition |
'=' |
17 |
% |
| P22612 |
BXGT008785 |
cAMP-dependent protein kinase catalytic subunit gamma |
reviewed |
Kinase |
PRKACG |
Inhibition |
'=' |
14 |
% |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Inhibition |
'=' |
14 |
% |
| P22694 |
BXGT008797 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
Kinase |
PRKACB |
Inhibition |
'=' |
14 |
% |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Inhibition |
'=' |
0 |
% |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Inhibition |
'=' |
-3 |
% |
| P08254 |
BXGT006758 |
Stromelysin-1 |
reviewed |
Enzyme |
MMP3 |
Inhibition |
'=' |
10 |
% |
| P04049 |
BXGT006133 |
RAF proto-oncogene serine/threonine-protein kinase |
reviewed |
Kinase |
RAF1 |
Inhibition |
'=' |
14 |
% |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
10890 |
nM |
| P11730 |
BXGT007741 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
- |
Camk2g |
Inhibition |
'=' |
0 |
% |
| P15791 |
BXGT008154 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
- |
Camk2d |
Inhibition |
'=' |
0 |
% |
| P08413 |
BXGT006769 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
- |
Camk2b |
Inhibition |
'=' |
0 |
% |
| P11275 |
BXGT007682 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
- |
Camk2a |
Inhibition |
'=' |
0 |
% |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
Inhibition |
'=' |
9 |
% |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Inhibition |
'=' |
7 |
% |
| P07332 |
BXGT006601 |
Tyrosine-protein kinase Fes/Fps |
reviewed |
Kinase |
FES |
Inhibition |
'=' |
20 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
11 |
% |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
Inhibition |
'=' |
45 |
% |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
Inhibition |
'=' |
66 |
% |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Inhibition |
'=' |
17 |
% |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Inhibition |
'=' |
6 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Inhibition |
'=' |
0 |
% |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Inhibition |
'=' |
3 |
% |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'=' |
61 |
% |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Inhibition |
'=' |
0 |
% |
| P49187 |
BXGT010683 |
Mitogen-activated protein kinase 10 |
reviewed |
- |
Mapk10 |
Inhibition |
'=' |
10 |
% |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Inhibition |
'=' |
19 |
% |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
200000 |
nM |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Inhibition |
'=' |
0 |
% |
| O14965 |
BXGT004117 |
Aurora kinase A |
reviewed |
Kinase |
AURKA |
Inhibition |
'=' |
90 |
% |
| P22629 |
BXGT008788 |
Streptavidin |
reviewed |
- |
|
Activity |
- |
- |
- |
| Q99816 |
BXGT019966 |
Tumor susceptibility gene 101 protein |
reviewed |
Enzyme |
TSG101 |
Potency |
- |
89125 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
'=' |
9 |
% |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Inhibition |
'=' |
88 |
% |
| Q96GD4 |
BXGT019667 |
Aurora kinase B |
reviewed |
Kinase |
AURKB |
Inhibition |
'=' |
99 |
% |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Inhibition |
'=' |
9 |
% |
| Q13177 |
BXGT013323 |
Serine/threonine-protein kinase PAK 2 |
reviewed |
Kinase |
PAK2 |
Inhibition |
'=' |
36 |
% |
| O00329 |
BXGT003909 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform |
reviewed |
Kinase |
PIK3CD |
Inhibition |
'=' |
68 |
% |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Inhibition |
'=' |
20 |
% |
| O00141 |
BXGT003882 |
Serine/threonine-protein kinase Sgk1 |
reviewed |
Kinase |
SGK1 |
Inhibition |
'=' |
76 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Inhibition |
'=' |
57 |
% |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
Inhibition |
'=' |
63 |
% |
| Q13148 |
BXGT013318 |
TAR DNA-binding protein 43 |
reviewed |
- |
TARDBP |
Potency |
- |
14125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
32642 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
29092 |
nM |
| P08069 |
BXGT006723 |
Insulin-like growth factor 1 receptor |
reviewed |
Kinase |
IGF1R |
Inhibition |
'=' |
44 |
% |
| Q13464 |
BXGT013357 |
Rho-associated protein kinase 1 |
reviewed |
Kinase |
ROCK1 |
Inhibition |
'=' |
80 |
% |
| Q08881 |
BXGT013012 |
Tyrosine-protein kinase ITK/TSK |
reviewed |
Kinase |
ITK |
Inhibition |
'=' |
87 |
% |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Inhibition |
'=' |
80 |
% |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Inhibition |
'=' |
16 |
% |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Inhibition |
'=' |
56 |
% |
| P08238 |
BXGT006753 |
Heat shock protein HSP 90-beta |
reviewed |
Chaperone |
HSP90AB1 |
IC50 |
'>' |
4000000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Inhibition |
'=' |
3 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
11 |
% |
| O14920 |
BXGT004110 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
reviewed |
Kinase |
IKBKB |
Inhibition |
'=' |
22 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
8 |
nM |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
Inhibition |
'=' |
5 |
% |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
Inhibition |
'=' |
11 |
% |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
90 |
% |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Inhibition |
'=' |
33 |
% |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
77 |
% |
| P49902 |
BXGT010758 |
Cytosolic purine 5'-nucleotidase |
reviewed |
Enzyme |
NT5C2 |
Inhibition |
'=' |
19 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
81 |
% |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'>' |
1000000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
'>' |
10000 |
nM |