| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
2100 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3100 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Inhibition |
'=' |
12 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
214 |
% |
| P59264 |
BXGT011265 |
Basic phospholipase A2 PLA-A |
reviewed |
- |
|
IC50 |
'=' |
2500 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Inhibition |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
5200 |
nM |
| P00690 |
BXGT005612 |
Pancreatic alpha-amylase |
reviewed |
- |
AMY2 |
IC50 |
'=' |
22600 |
nM |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
FC |
'=' |
0 |
- |
| Q76270 |
BXGT016848 |
GP41 |
unreviewed |
- |
HIV1 |
EC50 |
'>' |
100000 |
nM |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
IC50 |
'=' |
8500 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
- |
- |
- |
| P24666 |
BXGT008986 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
IC50 |
'=' |
7200 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
IC50 |
'=' |
9410 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
46 |
% |
| P02699 |
BXGT005925 |
Rhodopsin |
reviewed |
- |
RHO |
Activity |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
6000 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
16 |
% |
| P17706 |
BXGT008330 |
Tyrosine-protein phosphatase non-receptor type 2 |
reviewed |
- |
PTPN2 |
IC50 |
'=' |
3330 |
nM |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
Inhibition |
'=' |
55 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
86000 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
IC50 |
'=' |
130 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
4120 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
IC50 |
'>' |
1000000 |
nM |
| Q8WZA2 |
BXGT019025 |
Rap guanine nucleotide exchange factor 4 |
reviewed |
Enzyme modulator |
RAPGEF4 |
Potency |
- |
50118 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
19952 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
19952 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
14 |
ug.mL-1 |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3080 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
- |
- |
- |
| P05227 |
BXGT006343 |
Histidine-rich protein PFHRP-II |
reviewed |
- |
|
Ratio IC50 |
'>' |
3 |
- |
| Q8TDU6 |
BXGT018814 |
G-protein coupled bile acid receptor 1 |
reviewed |
G-protein coupled receptor |
GPBAR1 |
Efficacy |
'=' |
65 |
% |
| P30305 |
BXGT009419 |
M-phase inducer phosphatase 2 |
reviewed |
Enzyme |
CDC25B |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Activity |
- |
- |
- |
| P29350 |
BXGT009335 |
Tyrosine-protein phosphatase non-receptor type 6 |
reviewed |
- |
PTPN6 |
IC50 |
'=' |
25780 |
nM |
| P23469 |
BXGT008871 |
Receptor-type tyrosine-protein phosphatase epsilon |
reviewed |
Enzyme |
PTPRE |
IC50 |
'>' |
40000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3600 |
nM |
| Q9UGI9 |
BXGT021682 |
5'-AMP-activated protein kinase subunit gamma-3 |
reviewed |
Enzyme modulator |
PRKAG3 |
Activity |
- |
- |
- |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Activity |
- |
- |
- |
| Q9Y478 |
BXGT022271 |
5'-AMP-activated protein kinase subunit beta-1 |
reviewed |
Kinase |
PRKAB1 |
Activity |
- |
- |
- |
| Q9UGJ0 |
BXGT021683 |
5'-AMP-activated protein kinase subunit gamma-2 |
reviewed |
Enzyme modulator |
PRKAG2 |
Activity |
- |
- |
- |
| P54619 |
BXGT011060 |
5'-AMP-activated protein kinase subunit gamma-1 |
reviewed |
Kinase |
PRKAG1 |
Activity |
- |
- |
- |
| O43741 |
BXGT004620 |
5'-AMP-activated protein kinase subunit beta-2 |
reviewed |
Enzyme modulator |
PRKAB2 |
Activity |
- |
- |
- |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Activity |
- |
- |
- |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
EC50 |
'=' |
0 |
nM |
| P10520 |
BXGT007576 |
Streptokinase A |
reviewed |
- |
ska |
EC50 |
'=' |
1790 |
nM |
| P00489 |
BXGT005553 |
Glycogen phosphorylase, muscle form |
reviewed |
- |
PYGM |
IC50 |
'=' |
15300 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3500 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Activity |
- |
- |
- |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Inhibition |
- |
- |
- |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Inhibition |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3900 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3800 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
210000 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Activity |
- |
- |
- |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Inhibition |
- |
- |
- |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
195 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
23 |
% |
| P05227 |
BXGT006343 |
Histidine-rich protein PFHRP-II |
reviewed |
- |
|
IC50 |
'>' |
20000000 |
nM |
| P18433 |
BXGT008403 |
Receptor-type tyrosine-protein phosphatase alpha |
reviewed |
Enzyme |
PTPRA |
Inhibition |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
15500 |
nM |
| P00489 |
BXGT005553 |
Glycogen phosphorylase, muscle form |
reviewed |
- |
PYGM |
IC50 |
'=' |
9000 |
nM |
| P00599 |
BXGT005596 |
Basic phospholipase A2 1 |
reviewed |
- |
|
IC50 |
'=' |
2900 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Ki |
'=' |
3400 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Km |
- |
- |
- |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
113 |
% |
| P10586 |
BXGT007581 |
Receptor-type tyrosine-protein phosphatase F |
reviewed |
Enzyme |
PTPRF |
Inhibition |
- |
- |
- |
| P17706 |
BXGT008330 |
Tyrosine-protein phosphatase non-receptor type 2 |
reviewed |
- |
PTPN2 |
IC50 |
'=' |
6700 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
Inhibition |
- |
- |
- |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
Inhibition |
- |
- |
- |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Inhibition |
- |
- |
- |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
Inhibition |
- |
- |
- |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
Inhibition |
- |
- |
- |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Inhibition |
- |
- |
- |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Inhibition |
- |
- |
- |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
Inhibition |
- |
- |
- |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Inhibition |
- |
- |
- |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Inhibition |
- |
- |
- |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Inhibition |
- |
- |
- |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Inhibition |
- |
- |
- |
| P11597 |
BXGT007727 |
Cholesteryl ester transfer protein |
reviewed |
- |
CETP |
IC50 |
'=' |
46600 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
158 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
IC50 |
'=' |
18600 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| P05227 |
BXGT006343 |
Histidine-rich protein PFHRP-II |
reviewed |
- |
|
Inhibition |
'=' |
17 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
185 |
% |
| Q9YQ12 |
BXGT022394 |
Protease |
unreviewed |
- |
protease |
IC50 |
'=' |
8000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3400 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
3700 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
15 |
% |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
499 |
nM |
| Q7T3S7 |
BXGT017140 |
Acidic phospholipase A2 EC-I |
reviewed |
- |
|
IC50 |
'=' |
2300 |
nM |
| P00489 |
BXGT005553 |
Glycogen phosphorylase, muscle form |
reviewed |
- |
PYGM |
IC50 |
'=' |
8912 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
70 |
% |
| Q9YQ12 |
BXGT022394 |
Protease |
unreviewed |
- |
protease |
Inhibition |
'=' |
85 |
% |
| Q8TDU6 |
BXGT018814 |
G-protein coupled bile acid receptor 1 |
reviewed |
G-protein coupled receptor |
GPBAR1 |
EC50 |
'=' |
1430 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Activity |
- |
- |
- |
| P10586 |
BXGT007581 |
Receptor-type tyrosine-protein phosphatase F |
reviewed |
Enzyme |
PTPRF |
IC50 |
'=' |
3800 |
nM |
| P22513 |
BXGT008777 |
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal |
reviewed |
- |
|
Inhibition |
'=' |
25 |
% |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
Inhibition |
'=' |
90 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
4000 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
28070 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
11220 |
nM |
| P24666 |
BXGT008986 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
IC50 |
'=' |
11100 |
nM |
| P28845 |
BXGT009297 |
Corticosteroid 11-beta-dehydrogenase isozyme 1 |
reviewed |
- |
HSD11B1 |
Inhibition |
- |
- |
- |
| P80365 |
BXGT011895 |
Corticosteroid 11-beta-dehydrogenase isozyme 2 |
reviewed |
Enzyme |
HSD11B2 |
Activity |
- |
- |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
32000 |
nM |
| P29350 |
BXGT009335 |
Tyrosine-protein phosphatase non-receptor type 6 |
reviewed |
- |
PTPN6 |
IC50 |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
4000 |
nM |
| P10586 |
BXGT007581 |
Receptor-type tyrosine-protein phosphatase F |
reviewed |
Enzyme |
PTPRF |
IC50 |
'>' |
40000 |
nM |
| P18433 |
BXGT008403 |
Receptor-type tyrosine-protein phosphatase alpha |
reviewed |
Enzyme |
PTPRA |
IC50 |
'>' |
40000 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
707 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
18356 |
nM |
| P28845 |
BXGT009297 |
Corticosteroid 11-beta-dehydrogenase isozyme 1 |
reviewed |
- |
HSD11B1 |
IC50 |
'=' |
1900 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
1021 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
130000 |
nM |
| Q2M2H8 |
BXGT026100 |
Probable maltase-glucoamylase 2 |
reviewed |
Enzyme |
MGAM2 |
IC50 |
- |
- |
- |
| P14410 |
BXGT008009 |
Sucrase-isomaltase, intestinal |
reviewed |
Enzyme |
SI |
IC50 |
- |
- |
- |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
IC50 |
- |
- |
- |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
IC50 |
- |
- |
- |
| Q77YF9 |
BXGT016886 |
Protein Vpr |
unreviewed |
- |
vpr |
Potency |
- |
5623 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Imax |
'=' |
63 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
IC50 |
'=' |
11481 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
2800 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Ki |
'=' |
6400 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
102 |
% |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
89125 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
41000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
120 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
134 |
% |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
5 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
45 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
22200 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
96 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
2750 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
EC50 |
'=' |
41310 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
2000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
2300 |
nM |
| P12276 |
BXGT007788 |
Fatty acid synthase |
reviewed |
- |
FASN |
IC50 |
'=' |
59300 |
nM |
| P12276 |
BXGT007788 |
Fatty acid synthase |
reviewed |
- |
FASN |
IC50 |
'=' |
13100 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
1000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
2500 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
259 |
% |
| P08047 |
BXGT006720 |
Transcription factor Sp1 |
reviewed |
Nucleic acid binding |
SP1 |
Activity |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Vmax |
- |
- |
- |
| Q96K76 |
BXGT026122 |
Ubiquitin carboxyl-terminal hydrolase 47 |
reviewed |
Enzyme |
USP47 |
IC50 |
'=' |
26000 |
nM |
| Q93009 |
BXGT019455 |
Ubiquitin carboxyl-terminal hydrolase 7 |
reviewed |
Enzyme |
USP7 |
IC50 |
'=' |
7000 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Imax |
'=' |
76 |
% |
| P09810 |
BXGT006924 |
Tryptophan 5-hydroxylase 1 |
reviewed |
- |
Tph1 |
Inhibition |
'=' |
6 |
% |
| Q9QUK6 |
BXGT021375 |
Toll-like receptor 4 |
reviewed |
- |
Tlr4 |
Inhibition |
- |
- |
- |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
IC50 |
'=' |
4 |
ug.mL-1 |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
IC50 |
'=' |
15848 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
17782 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
Inhibition |
'=' |
31 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
28 |
% |
| Q2M2H8 |
BXGT026100 |
Probable maltase-glucoamylase 2 |
reviewed |
Enzyme |
MGAM2 |
Inhibition |
- |
- |
- |
| P14410 |
BXGT008009 |
Sucrase-isomaltase, intestinal |
reviewed |
Enzyme |
SI |
Inhibition |
- |
- |
- |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Inhibition |
- |
- |
- |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
Inhibition |
- |
- |
- |
| Q6P7A9 |
BXGT016460 |
Lysosomal alpha-glucosidase |
reviewed |
- |
Gaa |
Inhibition |
'<' |
50 |
% |
| P07339 |
BXGT006604 |
Cathepsin D |
reviewed |
Enzyme |
CTSD |
IC50 |
'=' |
18200 |
nM |
| P06766 |
BXGT006502 |
DNA polymerase beta |
reviewed |
- |
Polb |
IC50 |
'=' |
4800 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Inhibition |
- |
- |
- |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
IC50 |
'=' |
1060 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Inhibition |
'=' |
97 |
% |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
5400 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Ki |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
8900 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
44668 |
nM |
| P11597 |
BXGT007727 |
Cholesteryl ester transfer protein |
reviewed |
- |
CETP |
Inhibition |
'=' |
31 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
24 |
% |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
Activity |
'=' |
156 |
% |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
IC50 |
'=' |
680 |
nM |
| P17706 |
BXGT008330 |
Tyrosine-protein phosphatase non-receptor type 2 |
reviewed |
- |
PTPN2 |
IC50 |
'=' |
2400 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
IC50 |
'=' |
31 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
5460 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Activity |
- |
- |
- |
| Q2M2H8 |
BXGT026100 |
Probable maltase-glucoamylase 2 |
reviewed |
Enzyme |
MGAM2 |
Ki |
- |
- |
- |
| P14410 |
BXGT008009 |
Sucrase-isomaltase, intestinal |
reviewed |
Enzyme |
SI |
Ki |
- |
- |
- |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Ki |
- |
- |
- |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
Ki |
- |
- |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
82 |
% |