| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
39810 |
nM |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
Vmax |
'=' |
21 |
uM min-1mg-1 |
| Q13148 |
BXGT013318 |
TAR DNA-binding protein 43 |
reviewed |
- |
TARDBP |
Potency |
- |
2818 |
nM |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
Km |
'=' |
72000 |
nM |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
K cat/Km |
'=' |
5330 |
1/M.s |
| P30307 |
BXGT009421 |
M-phase inducer phosphatase 3 |
reviewed |
Enzyme |
CDC25C |
IC50 |
'=' |
19000 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
89125 |
nM |
| P30305 |
BXGT009419 |
M-phase inducer phosphatase 2 |
reviewed |
Enzyme |
CDC25B |
Inhibition |
'=' |
14 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
7943 |
nM |
| P16435 |
BXGT008226 |
NADPH--cytochrome P450 reductase |
reviewed |
- |
POR |
Activity |
- |
- |
- |
| Q9Z0U5 |
BXGT022402 |
Aldehyde oxidase 1 |
reviewed |
- |
Aox1 |
IC50 |
'=' |
190 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
8912 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
112 |
% |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
7079 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
17782 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
17782 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
3548 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
39810 |
nM |
| Q8WTS1 |
BXGT018985 |
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 |
reviewed |
- |
ABHD5 |
IC50 |
'=' |
9468 |
nM |
| Q00G26 |
BXGT012560 |
Perilipin-5 |
reviewed |
- |
PLIN5 |
IC50 |
'=' |
9468 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
8912 |
nM |
| P04406 |
BXGT006207 |
Glyceraldehyde-3-phosphate dehydrogenase |
reviewed |
Enzyme |
GAPDH |
Potency |
'=' |
10000 |
nM |
| P38435 |
BXGT010040 |
Vitamin K-dependent gamma-carboxylase |
reviewed |
- |
GGCX |
Activity |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
1584 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
6309 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
10000 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
2511 |
nM |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
Km |
'=' |
21000 |
nM |
| P04818 |
BXGT006269 |
Thymidylate synthase |
reviewed |
Enzyme |
TYMS |
k2 |
'=' |
0 |
M-1 s-1 |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Ratio |
'=' |
5 |
- |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Inhibition |
'=' |
43 |
% |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
25118 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
25118 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Km |
'=' |
1500 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
25929 |
nM |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
25118 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Km |
'=' |
1200 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
56234 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
12589 |
nM |
| P00883 |
BXGT005683 |
Fructose-bisphosphate aldolase A |
reviewed |
- |
ALDOA |
Potency |
'=' |
6309 |
nM |
| P00772 |
BXGT005648 |
Chymotrypsin-like elastase family member 1 |
reviewed |
- |
CELA1 |
Activity |
- |
- |
- |
| P08419 |
BXGT006770 |
Chymotrypsin-like elastase family member 2A |
reviewed |
- |
CELA2A |
Activity |
- |
- |
- |
| Q5FB27 |
BXGT015373 |
Aldehyde oxidase 1 |
reviewed |
- |
AOX1 |
IC50 |
'=' |
110 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
2909 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
10000 |
nM |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
Km |
'=' |
31200 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
k cat |
'=' |
700 |
s-1 |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7079 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
10000 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
11220 |
nM |
| Q13315 |
BXGT013339 |
Serine-protein kinase ATM |
reviewed |
Kinase |
ATM |
Potency |
'=' |
39810 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Vmax |
'=' |
0 |
uM s-1 |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
11220 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
12589 |
nM |
| P14902 |
BXGT008065 |
Indoleamine 2,3-dioxygenase 1 |
reviewed |
- |
IDO1 |
IC50 |
'=' |
1000 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
50118 |
nM |
| P30305 |
BXGT009419 |
M-phase inducer phosphatase 2 |
reviewed |
Enzyme |
CDC25B |
IC50 |
'=' |
3380 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Activity |
'=' |
50 |
% |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
6309 |
nM |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
x fold |
'=' |
375 |
uM |
| O15770 |
BXGT004187 |
Glutathione reductase |
reviewed |
- |
GR3 |
Km |
'=' |
82200 |
nM |
| P16435 |
BXGT008226 |
NADPH--cytochrome P450 reductase |
reviewed |
- |
POR |
Activity |
'=' |
2 |
umol/L/min |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
Ki |
'=' |
16100 |
nM |
| P00469 |
BXGT005550 |
Thymidylate synthase |
reviewed |
- |
thyA |
k |
'=' |
5 |
se-1 |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
561 |
nM |
| P68871 |
BXGT011615 |
Hemoglobin subunit beta |
reviewed |
- |
HBB |
Potency |
'=' |
12589 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
25118 |
nM |
| P28563 |
BXGT009271 |
Dual specificity protein phosphatase 1 |
reviewed |
- |
Dusp1 |
IC50 |
'=' |
24000 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
39810 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
35481 |
nM |
| P46426 |
BXGT010519 |
Glutathione S-transferase |
reviewed |
- |
|
Activity |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
20596 |
nM |
| P9WG47 |
BXGT012264 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'>' |
200000 |
nM |
| P9WG45 |
BXGT012263 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'>' |
200000 |
nM |
| P14902 |
BXGT008065 |
Indoleamine 2,3-dioxygenase 1 |
reviewed |
- |
IDO1 |
IC50 |
'=' |
370 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
- |
- |
- |
| P30307 |
BXGT009421 |
M-phase inducer phosphatase 3 |
reviewed |
Enzyme |
CDC25C |
IC50 |
'=' |
18800 |
nM |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
IC50 |
'=' |
200 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
17782 |
nM |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
Reduction |
'=' |
8 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
- |
- |
- |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
157 |
% |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
158 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
50118 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
2511 |
nM |
| O15770 |
BXGT004187 |
Glutathione reductase |
reviewed |
- |
GR3 |
K cat |
'=' |
0 |
s-1 |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
6309 |
nM |
| P46426 |
BXGT010519 |
Glutathione S-transferase |
reviewed |
- |
|
Emax |
'=' |
22 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
17 |
% |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
- |
- |
- |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Ratio |
'=' |
0 |
- |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
K cat |
'=' |
0 |
s-1 |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
14125 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
2511 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
6309 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
2818 |
nM |
| O15770 |
BXGT004187 |
Glutathione reductase |
reviewed |
- |
GR3 |
K cat/Km |
'=' |
1991 |
1/M*s |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
14125 |
nM |
| P14902 |
BXGT008065 |
Indoleamine 2,3-dioxygenase 1 |
reviewed |
- |
IDO1 |
IC50 |
'=' |
1100 |
nM |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
22793 |
nM |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
IC50 |
'=' |
55000 |
nM |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
Ki |
'=' |
12100 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5011 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
-1 |
% |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
Ki |
'=' |
1500 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
7943 |
nM |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
k cat/Km |
'=' |
13 |
10e4 M-1 s-1 |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
Vmax |
'=' |
0 |
uM min-1mg-1 |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Vmax |
'=' |
0 |
uM s-1 |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
k cat |
'=' |
960 |
s-1 |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
22387 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
4610 |
nM |
| P30305 |
BXGT009419 |
M-phase inducer phosphatase 2 |
reviewed |
Enzyme |
CDC25B |
IC50 |
'=' |
2200 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
5623 |
nM |
| P15374 |
BXGT008113 |
Ubiquitin carboxyl-terminal hydrolase isozyme L3 |
reviewed |
Enzyme |
UCHL3 |
IC50 |
'=' |
71000 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
11220 |
nM |
| Q3B792 |
BXGT014403 |
NQO1 protein |
unreviewed |
- |
NQO1 |
Activity |
'=' |
1 |
umol/L/min |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
k cat/Km |
'=' |
1 |
10e4 M-1 s-1 |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
k cat/Km |
'=' |
10 |
10e4 M-1 s-1 |
| P14618 |
BXGT008027 |
Pyruvate kinase PKM |
reviewed |
Kinase |
PKM |
Potency |
'=' |
15848 |
nM |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
28183 |
nM |
| O60240 |
BXGT004860 |
Perilipin-1 |
reviewed |
- |
PLIN1 |
IC50 |
'=' |
7895 |
nM |
| Q8WTS1 |
BXGT018985 |
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 |
reviewed |
- |
ABHD5 |
IC50 |
'=' |
7895 |
nM |
| P09623 |
BXGT006912 |
Dihydrolipoyl dehydrogenase, mitochondrial |
reviewed |
- |
DLD |
Vmax |
'=' |
11 |
uM min-1mg-1 |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Activity |
'=' |
1225 |
umol/min/mg |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Vmax |
'=' |
7286 |
uM |
| P30305 |
BXGT009419 |
M-phase inducer phosphatase 2 |
reviewed |
Enzyme |
CDC25B |
Inhibition |
'=' |
27 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
19952 |
nM |
| O95398 |
BXGT005378 |
Rap guanine nucleotide exchange factor 3 |
reviewed |
Enzyme modulator |
RAPGEF3 |
Potency |
- |
25118 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
14125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
8199 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
3264 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
12589 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
7943 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
7943 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
8912 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
35481 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Activity |
'=' |
1315 |
micromol/min |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| Q9HC16 |
BXGT020525 |
DNA dC->dU-editing enzyme APOBEC-3G |
reviewed |
Enzyme |
APOBEC3G |
Potency |
- |
22387 |
nM |
| P15559 |
BXGT008139 |
NAD(P)H dehydrogenase [quinone] 1 |
reviewed |
- |
NQO1 |
Activity |
'=' |
1 |
umol/L/min |
| O54754 |
BXGT004731 |
Aldehyde oxidase 1 |
reviewed |
- |
Aox1 |
IC50 |
'=' |
150 |
nM |
| P80456 |
BXGT011910 |
Aldehyde oxidase 1 |
reviewed |
- |
AOX1 |
IC50 |
'=' |
2000 |
nM |
| P09936 |
BXGT006943 |
Ubiquitin carboxyl-terminal hydrolase isozyme L1 |
reviewed |
Enzyme |
UCHL1 |
IC50 |
'=' |
290000 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
33498 |
nM |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
Ratio Ki |
'=' |
10 |
- |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
Ratio Ki |
'=' |
3 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23109 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
7943 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Ki |
'=' |
400 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
6309 |
nM |
| P0DPI0 |
BXGT007528 |
Botulinum neurotoxin type A |
reviewed |
- |
botA |
Ratio |
'=' |
1 |
/M/s |
| Q64346 |
BXGT016113 |
Dual specificity protein phosphatase 6 |
reviewed |
- |
Dusp6 |
IC50 |
'=' |
20500 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
35481 |
nM |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
Ki |
'=' |
470 |
nM |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
14125 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
28183 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
'=' |
26000 |
nM |