| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
25118 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
28183 |
nM |
| Q8TDS4 |
BXGT018812 |
Hydroxycarboxylic acid receptor 2 |
reviewed |
- |
HCAR2 |
Activity |
'=' |
4 |
% |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| O95149 |
BXGT005350 |
Snurportin-1 |
reviewed |
- |
SNUPN |
Potency |
- |
141253 |
nM |
| Q14974 |
BXGT013516 |
Importin subunit beta-1 |
reviewed |
Transporter |
KPNB1 |
Potency |
- |
141253 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
39810 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
1062 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
10 |
% |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
0 |
% |
| P03470 |
BXGT006081 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'>' |
100000 |
nM |
| P42330 |
BXGT010301 |
Aldo-keto reductase family 1 member C3 |
reviewed |
Enzyme |
AKR1C3 |
Inhibition |
'=' |
36 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
- |
- |
- |
| P0A6C1 |
BXGT007045 |
Endonuclease 4 |
reviewed |
- |
nfo |
Potency |
'=' |
25118 |
nM |
| Q76353 |
BXGT016849 |
Integrase |
unreviewed |
- |
|
IC50 |
'=' |
2800 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
IC50 |
'=' |
5551000 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
7079 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
32000 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
1000000 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
44668 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
141 |
nM |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
Ki |
'=' |
6490 |
nM |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'=' |
10100 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
562 |
nM |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
EC50 |
'=' |
97000 |
nM |
| Q76353 |
BXGT016849 |
Integrase |
unreviewed |
- |
|
IC50 |
'=' |
24000 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
35481 |
nM |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
Ki |
'=' |
8710 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Inhibition |
'=' |
16 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
16 |
% |
| Q12794 |
BXGT013265 |
Hyaluronidase-1 |
reviewed |
Enzyme |
HYAL1 |
IC50 |
'>' |
2000000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
1000 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
1000 |
nM |
| Q76353 |
BXGT016849 |
Integrase |
unreviewed |
- |
|
IC50 |
'>' |
100000 |
nM |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
Ki |
'=' |
7330 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
69 |
% |
| P24298 |
BXGT008960 |
Alanine aminotransferase 1 |
reviewed |
Enzyme |
GPT |
Activity |
'=' |
97 |
U/L |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
601 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
8912 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
20 |
% |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'=' |
18 |
% |
| P08238 |
BXGT006753 |
Heat shock protein HSP 90-beta |
reviewed |
Chaperone |
HSP90AB1 |
IC50 |
'>' |
50000 |
nM |
| P07900 |
BXGT006696 |
Heat shock protein HSP 90-alpha |
reviewed |
Chaperone |
HSP90AA1 |
IC50 |
'>' |
50000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
94 |
% |
| Q39830 |
BXGT014382 |
BiP isoform A |
unreviewed |
- |
|
IC50 |
'=' |
600000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
33587 |
nM |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
44668 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'>' |
350000 |
nM |
| Q57TT1 |
BXGT015153 |
Uncharacterized protein |
unreviewed |
- |
Tb927.8.6820 |
Potency |
- |
31622 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
Inhibition |
'=' |
0 |
% |
| P06280 |
BXGT006433 |
Alpha-galactosidase A |
reviewed |
- |
GLA |
Potency |
'=' |
50118 |
nM |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
IC50 |
'=' |
24 |
nM |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
'=' |
238 |
nM |
| O49150 |
BXGT004652 |
Lipoxygenase |
unreviewed |
- |
|
IC50 |
'=' |
4000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1200000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Activity |
- |
- |
- |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
56234 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'=' |
2380 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
3060 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
Activity |
'=' |
80 |
% |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
Activity |
'=' |
80 |
% |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Activity |
'=' |
80 |
% |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
Activity |
'=' |
80 |
% |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
Activity |
'=' |
80 |
% |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Activity |
'=' |
80 |
% |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Activity |
'=' |
80 |
% |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
Activity |
'=' |
80 |
% |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Activity |
'=' |
80 |
% |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Activity |
'=' |
80 |
% |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Activity |
'=' |
80 |
% |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
7870 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
43000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
22387 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
'=' |
22 |
% |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
10000 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
3000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1000000 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
IC50 |
'=' |
600000 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
7062 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
12589 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
15848 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Inhibition |
'=' |
600 |
% |
| P03070 |
BXGT006016 |
Large T antigen |
reviewed |
- |
|
IC50 |
- |
7300 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
IC50 |
'>' |
300000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
16700 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
'=' |
91 |
% |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
Ki |
'=' |
10900 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
8492 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
15848 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
25000 |
nM |
| P35236 |
BXGT009802 |
Tyrosine-protein phosphatase non-receptor type 7 |
reviewed |
Enzyme |
PTPN7 |
IC50 |
'>' |
100000 |
nM |
| Q13093 |
BXGT013310 |
Platelet-activating factor acetylhydrolase |
reviewed |
Enzyme |
PLA2G7 |
Activity |
- |
- |
- |
| P51452 |
BXGT010849 |
Dual specificity protein phosphatase 3 |
reviewed |
- |
DUSP3 |
IC50 |
'>' |
100000 |
nM |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
Ki |
'=' |
9080 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
1610 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
50118 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
7943 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
32 |
% |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
2818 |
nM |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Potency |
- |
2511 |
nM |
| Q76353 |
BXGT016849 |
Integrase |
unreviewed |
- |
|
IC50 |
- |
- |
- |
| P17516 |
BXGT008313 |
Aldo-keto reductase family 1 member C4 |
reviewed |
Enzyme |
AKR1C4 |
Inhibition |
'=' |
0 |
% |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
25118 |
nM |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ki |
'=' |
10000 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
39810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
6309 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
31622 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
'=' |
400000 |
nM |
| O49150 |
BXGT004652 |
Lipoxygenase |
unreviewed |
- |
|
IC50 |
'=' |
3000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'>' |
10000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
24 |
% |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
3162 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
'=' |
12589 |
nM |
| P23739 |
BXGT008901 |
Sucrase-isomaltase, intestinal |
reviewed |
- |
Si |
IC50 |
'=' |
87450 |
nM |
| Q6P7A9 |
BXGT016460 |
Lysosomal alpha-glucosidase |
reviewed |
- |
Gaa |
IC50 |
'=' |
34690 |
nM |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
- |
- |
- |
| P52895 |
BXGT010961 |
Aldo-keto reductase family 1 member C2 |
reviewed |
Enzyme |
AKR1C2 |
Inhibition |
'=' |
19 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
90000 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
'=' |
21 |
nM |
| Q04828 |
BXGT012787 |
Aldo-keto reductase family 1 member C1 |
reviewed |
Enzyme |
AKR1C1 |
Inhibition |
'=' |
6 |
% |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
Inhibition |
'=' |
10 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
44668 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
14125 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
84921 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
2 |
% |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
'=' |
10 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23109 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
39810 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
44668 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
794 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
EC50 |
'=' |
216000 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
11220 |
nM |
| A0A0C7ACN7 |
BXGT000141 |
3-oxoacyl-ACP synthase |
unreviewed |
- |
pqsD |
Inhibition |
'=' |
26 |
% |
| P29372 |
BXGT009336 |
DNA-3-methyladenine glycosylase |
reviewed |
Enzyme |
MPG |
Inhibition |
'=' |
0 |
% |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1995 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
35397 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
9060 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
3162 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
10621 |
nM |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
6420 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
Ki |
'=' |
10840 |
nM |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
Ki |
'=' |
10840 |
nM |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
Ki |
'=' |
10840 |
nM |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
Ki |
'=' |
10840 |
nM |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
Ki |
'=' |
10840 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Ki |
'=' |
10840 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
Ki |
'=' |
10840 |
nM |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
Ki |
'=' |
10840 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
Ki |
'=' |
10840 |
nM |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
Ki |
'=' |
10840 |
nM |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
Ki |
'=' |
10840 |
nM |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
Activity |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
32800 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
25929 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'>' |
400000 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
17782 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
14125 |
nM |
| Q9GZT9 |
BXGT020425 |
Egl nine homolog 1 |
reviewed |
- |
EGLN1 |
Inhibition |
- |
- |
- |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
13 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
129700 |
nM |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
8500 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
IC50 |
'=' |
2540000 |
nM |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
IC50 |
'=' |
2540000 |
nM |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
IC50 |
'=' |
2540000 |
nM |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
IC50 |
'=' |
2540000 |
nM |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
IC50 |
'=' |
2540000 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
IC50 |
'=' |
2540000 |
nM |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
IC50 |
'=' |
2540000 |
nM |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
IC50 |
'=' |
2540000 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
IC50 |
'=' |
2540000 |
nM |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
IC50 |
'=' |
2540000 |
nM |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
IC50 |
'=' |
2540000 |
nM |
| Q06124 |
BXGT012856 |
Tyrosine-protein phosphatase non-receptor type 11 |
reviewed |
- |
PTPN11 |
Inhibition |
- |
- |
- |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Activity |
'=' |
104 |
% |
| Q8HY88 |
BXGT018198 |
Potassium channel subfamily K member 2 |
unreviewed |
- |
KCNK2 |
FC |
'=' |
1 |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'>' |
100000 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
1584893 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
15600 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
3370 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
1753000 |
nM |