| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
IC50 |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
Ki |
- |
- |
- |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'=' |
10900 |
nM |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
Ki |
'=' |
4200 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
17782 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
Ki |
'=' |
606000 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
22387 |
nM |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
Ki |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Ki |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Ki |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
IC50 |
- |
- |
- |
| P07639 |
BXGT006652 |
3-dehydroquinate synthase |
reviewed |
- |
aroB |
Ki |
'=' |
630000 |
nM |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
IC50 |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
Ki |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
IC50 |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
IC50 |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Ki |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
IC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
- |
- |
- |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Inhibition |
- |
- |
- |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
39810 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Inhibition |
'=' |
10 |
% |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
10000 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'=' |
5 |
% |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'=' |
4003000 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
79432 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
10399 |
nM |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
IC50 |
- |
- |
- |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
5011 |
nM |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
IC50 |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
Ki |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
Ki |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
IC50 |
- |
- |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IC50 |
- |
- |
- |
| Q2PCB5 |
BXGT014154 |
Carbonic anhydrase |
unreviewed |
- |
ca |
Ki |
'=' |
14800 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1584 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
- |
- |
- |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
IC50 |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
- |
- |
- |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
30131 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
- |
- |
- |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
5623 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
- |
- |
- |
| Q99N23 |
BXGT019994 |
Carbonic anhydrase 15 |
reviewed |
- |
Ca15 |
Ki |
'=' |
10200 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
5358 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
5011 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
14125 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
Ki |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
IC50 |
- |
- |
- |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
Ki |
'=' |
48900 |
nM |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Ki |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
IC50 |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
- |
- |
- |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
730 |
nM |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
IC50 |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
- |
- |
- |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
2238 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
IC50 |
- |
- |
- |
| P07639 |
BXGT006652 |
3-dehydroquinate synthase |
reviewed |
- |
aroB |
Km |
'=' |
16000 |
nM |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
IC50 |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
IC50 |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
Ki |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Ki |
- |
- |
- |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
50118 |
nM |
| P07639 |
BXGT006652 |
3-dehydroquinate synthase |
reviewed |
- |
aroB |
Ki |
'=' |
880000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
'=' |
89 |
% |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
14125 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
39810 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
11917 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
115000 |
nM |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ki |
'=' |
13000 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
9900 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
12589 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
26679 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
35481 |
nM |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
IC50 |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
IC50 |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Ki |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
IC50 |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
'=' |
17431 |
nM |
| Q9Y468 |
BXGT022270 |
Lethal(3)malignant brain tumor-like protein 1 |
reviewed |
Epigenetic regulator |
L3MBTL1 |
Potency |
'=' |
17782 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
IC50 |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1258 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
19952 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Ki |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
Ki |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
IC50 |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
IC50 |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
Ki |
- |
- |
- |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
631 |
nM |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
Ki |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
Ki |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
Ki |
- |
- |
- |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Inhibition |
'=' |
47 |
% |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
- |
- |
- |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
Ki |
'=' |
55100 |
nM |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
Ki |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
Ki |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
Ki |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
Ki |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
Ki |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
Ki |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
IC50 |
- |
- |
- |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
714000 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
-41 |
% |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
8900 |
nM |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
115820 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
35481 |
nM |
| P22894 |
BXGT008815 |
Neutrophil collagenase |
reviewed |
Enzyme |
MMP8 |
Inhibition |
'=' |
31 |
% |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
15848 |
nM |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Inhibition |
'=' |
28 |
% |
| P54300 |
BXGT011042 |
Autoinducer 2-binding periplasmic protein LuxP |
reviewed |
- |
luxP |
IC50 |
'=' |
59000 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
9910 |
nM |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Inhibition |
'=' |
25 |
% |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
11220 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1584 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
23109 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
25118 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
IC50 |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Ki |
- |
- |
- |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
79432 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
- |
- |
- |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
Ki |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
IC50 |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Ki |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
Ki |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
'=' |
868 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
44668 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
37685 |
nM |
| Q9HC16 |
BXGT020525 |
DNA dC->dU-editing enzyme APOBEC-3G |
reviewed |
Enzyme |
APOBEC3G |
Potency |
- |
31622 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
5972 |
nM |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
IC50 |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
IC50 |
- |
- |
- |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
Ki |
- |
- |
- |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
25118 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
11220 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
35481 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
Ki |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
Ki |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
IC50 |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
Ki |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
IC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Ki |
- |
- |
- |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
31622 |
nM |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
IC50 |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
1412 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
23280 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
17782 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
25118 |
nM |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
IC50 |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
Ki |
- |
- |
- |
| Q3SZX4 |
BXGT014517 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ki |
'=' |
3480 |
nM |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
Ki |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
Ki |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ki |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Ki |
- |
- |
- |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
17782 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
18887 |
nM |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
Ki |
'=' |
12200 |
nM |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
IC50 |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
- |
- |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
- |
- |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
- |
- |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IC50 |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IC50 |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
- |
- |
- |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
15848 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Potency |
- |
5955 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
'=' |
11220 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
Ki |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
Ki |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
- |
- |
- |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
44668 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
12589 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
- |
- |
- |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
Inhibition |
'=' |
10 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
28183 |
nM |
| P07639 |
BXGT006652 |
3-dehydroquinate synthase |
reviewed |
- |
aroB |
Km |
'=' |
18000 |
nM |
| P08254 |
BXGT006758 |
Stromelysin-1 |
reviewed |
Enzyme |
MMP3 |
Inhibition |
'=' |
1 |
% |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
- |
- |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
2511 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
70794 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29092 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
Inhibition |
'=' |
87 |
% |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
IC50 |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
26043 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ki |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
IC50 |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
IC50 |
- |
- |
- |
| Q9GZT9 |
BXGT020425 |
Egl nine homolog 1 |
reviewed |
- |
EGLN1 |
Inhibition |
- |
- |
- |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
IC50 |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
IC50 |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
IC50 |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
IC50 |
- |
- |
- |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
IC50 |
- |
- |
- |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
Ki |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
Ki |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
IC50 |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
Ki |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
Ki |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
IC50 |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1778 |
nM |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
IC50 |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ki |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
- |
- |
- |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
Ki |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Ki |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
- |
- |
- |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
35481 |
nM |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
Ki |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
IC50 |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
IC50 |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
Ki |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Ki |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
'=' |
23367 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
50118 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
75686 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
39810 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
- |
- |
- |
| P0A6C1 |
BXGT007045 |
Endonuclease 4 |
reviewed |
- |
nfo |
Potency |
'=' |
19952 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
926 |
nM |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
13091 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
15848 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
IC50 |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
Ki |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
Ki |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
Ki |
- |
- |
- |
| P51151 |
BXGT010837 |
Ras-related protein Rab-9A |
reviewed |
- |
RAB9A |
Potency |
'=' |
73078 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
26679 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
12589 |
nM |
| P10145 |
BXGT007542 |
Interleukin-8 |
reviewed |
Signaling |
CXCL8 |
Potency |
- |
74978 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
10322 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Ki |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
Ki |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ki |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
IC50 |
- |
- |
- |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
79432 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
18833 |
nM |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
IC50 |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
Ki |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
Ki |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ki |
- |
- |
- |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Ki |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
IC50 |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
IC50 |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Ki |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
IC50 |
- |
- |
- |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
IC50 |
'=' |
33000 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
29849 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
35481 |
nM |
| P14902 |
BXGT008065 |
Indoleamine 2,3-dioxygenase 1 |
reviewed |
- |
IDO1 |
Inhibition |
'=' |
-8 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
35481 |
nM |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
44668 |
nM |
| Q00987 |
BXGT012559 |
E3 ubiquitin-protein ligase Mdm2 |
reviewed |
Nucleic acid binding |
MDM2 |
IC50 |
'>' |
100000 |
nM |