| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Potency |
'=' |
3162 |
nM |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
IC50 |
'=' |
4000 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
39810 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
85 |
% |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
EC50 |
'>' |
300000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
28183 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
40 |
ug.mL-1 |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
3162 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
10000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
10000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
10000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
24 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
2377 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
2927 |
nM |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
Potency |
'=' |
15848 |
nM |
| Q96S37 |
BXGT019737 |
Solute carrier family 22 member 12 |
reviewed |
Transporter |
SLC22A12 |
Ki |
'=' |
5740 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
19952 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
50118 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
1 |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
28183 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
28183 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
35481 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
39810 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
31622 |
nM |
| Q07820 |
BXGT012942 |
Induced myeloid leukemia cell differentiation protein Mcl-1 |
reviewed |
Signaling |
MCL1 |
IC50 |
'=' |
2988 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
28183 |
nM |
| Q9S446 |
BXGT021560 |
Class A sortase SrtA |
unreviewed |
- |
srtA |
IC50 |
'=' |
37390 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
4466 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
76500 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
10000 |
nM |
| Q96S37 |
BXGT019737 |
Solute carrier family 22 member 12 |
reviewed |
Transporter |
SLC22A12 |
IC50 |
'=' |
2000 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
5000 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
12589 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
21192 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
31700 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
79432 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
IC50 |
'=' |
1600 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
-3 |
% |
| P0A6C1 |
BXGT007045 |
Endonuclease 4 |
reviewed |
- |
nfo |
Potency |
'=' |
3548 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
21000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
25118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
11220 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
10100 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
28183 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
28183 |
nM |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
8000 |
nM |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
18492 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
10000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
31622 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
'=' |
34000 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
30300 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
15848 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
15848 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
4 |
% |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
3162 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
13800 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
25118 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
25118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
12589 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
21700 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
11220 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
11220 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
22387 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
23934 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
4228 |
nM |
| P13267 |
BXGT007895 |
DNA polymerase III PolC-type |
reviewed |
- |
polC |
Potency |
- |
18887 |
nM |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Potency |
'=' |
39810 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
78 |
% |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
10000 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
15848 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
50118 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
IC50 |
'=' |
2300 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| P08482 |
BXGT006775 |
Muscarinic acetylcholine receptor M1 |
reviewed |
- |
Chrm1 |
Potency |
'=' |
20 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
112 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'<' |
50 |
% |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
28183 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
50 |
% |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Efficacy |
'=' |
284 |
picometer |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
22387 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
12300 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
15848 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
Ki |
'=' |
3 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
7079 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
28000 |
nM |
| P00760 |
BXGT005644 |
Cationic trypsin |
reviewed |
- |
|
IC50 |
'=' |
110800 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
7943 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
3793 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
18 |
% |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
11000 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
5011 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
35481 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
39810 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
19952 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
19952 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
IC50 |
'=' |
12600 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Activity |
- |
- |
- |
| Q14790 |
BXGT013505 |
Caspase-8 |
reviewed |
Enzyme |
CASP8 |
Inhibition |
- |
- |
- |
| Q3ZAV1 |
BXGT014546 |
Solute carrier family 22 member 12 |
reviewed |
- |
Slc22a12 |
IC50 |
'=' |
18000 |
nM |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
15848 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
17300 |
nM |
| P29276 |
BXGT009329 |
Adenosine receptor A2b |
reviewed |
- |
Adora2b |
Ki |
'=' |
17300 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
29934 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
50118 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
14125 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
29934 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
39810 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
39810 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
553 |
% |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
19952 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
100000 |
nM |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Potency |
- |
3162 |
nM |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
23934 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
14125 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
14125 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
49000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
199 |
nM |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Inhibition |
'=' |
71 |
% |
| Q27686 |
BXGT013930 |
Pyruvate kinase |
reviewed |
- |
PYK |
Potency |
'=' |
19952 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
4466 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
28183 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| P11064 |
BXGT007646 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
Inhibition |
'=' |
35 |
% |
| P28647 |
BXGT009282 |
Adenosine receptor A3 |
reviewed |
- |
Adora3 |
Ratio |
'=' |
0 |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ratio |
'=' |
0 |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
562 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
1600 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
103 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
6012 |
nM |
| Q13332 |
BXGT013342 |
Receptor-type tyrosine-protein phosphatase S |
reviewed |
Enzyme |
PTPRS |
IC50 |
'=' |
4300 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
26 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
5011 |
nM |
| Q9BUF5 |
BXGT020135 |
Tubulin beta-6 chain |
reviewed |
Cellular structure |
TUBB6 |
Kd |
'>' |
100000 |
nM |
| Q9BVA1 |
BXGT020142 |
Tubulin beta-2B chain |
reviewed |
- |
TUBB2B |
Kd |
'>' |
100000 |
nM |
| Q13885 |
BXGT013400 |
Tubulin beta-2A chain |
reviewed |
Cellular structure |
TUBB2A |
Kd |
'>' |
100000 |
nM |
| Q6PEY2 |
BXGT016465 |
Tubulin alpha-3E chain |
reviewed |
Cellular structure |
TUBA3E |
Kd |
'>' |
100000 |
nM |
| Q9BQE3 |
BXGT020109 |
Tubulin alpha-1C chain |
reviewed |
Cellular structure |
TUBA1C |
Kd |
'>' |
100000 |
nM |
| P68363 |
BXGT011594 |
Tubulin alpha-1B chain |
reviewed |
Cellular structure |
TUBA1B |
Kd |
'>' |
100000 |
nM |
| P07437 |
BXGT006624 |
Tubulin beta chain |
reviewed |
Cellular structure |
TUBB |
Kd |
'>' |
100000 |
nM |
| Q3ZCM7 |
BXGT014551 |
Tubulin beta-8 chain |
reviewed |
- |
TUBB8 |
Kd |
'>' |
100000 |
nM |
| P04350 |
BXGT006193 |
Tubulin beta-4A chain |
reviewed |
Cellular structure |
TUBB4A |
Kd |
'>' |
100000 |
nM |
| Q71U36 |
BXGT016705 |
Tubulin alpha-1A chain |
reviewed |
Cellular structure |
TUBA1A |
Kd |
'>' |
100000 |
nM |
| Q13509 |
BXGT013366 |
Tubulin beta-3 chain |
reviewed |
Cellular structure |
TUBB3 |
Kd |
'>' |
100000 |
nM |
| P68366 |
BXGT011595 |
Tubulin alpha-4A chain |
reviewed |
Cellular structure |
TUBA4A |
Kd |
'>' |
100000 |
nM |
| P0DPH7 |
BXGT007527 |
Tubulin alpha-3C chain |
reviewed |
- |
TUBA3C |
Kd |
'>' |
100000 |
nM |
| Q9H4B7 |
BXGT020475 |
Tubulin beta-1 chain |
reviewed |
Cellular structure |
TUBB1 |
Kd |
'>' |
100000 |
nM |
| P68371 |
BXGT011597 |
Tubulin beta-4B chain |
reviewed |
Cellular structure |
TUBB4B |
Kd |
'>' |
100000 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
3981 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
3981 |
nM |
| Q9BUF5 |
BXGT020135 |
Tubulin beta-6 chain |
reviewed |
Cellular structure |
TUBB6 |
Kd |
'=' |
199526 |
nM |
| Q9BVA1 |
BXGT020142 |
Tubulin beta-2B chain |
reviewed |
- |
TUBB2B |
Kd |
'=' |
199526 |
nM |
| Q13885 |
BXGT013400 |
Tubulin beta-2A chain |
reviewed |
Cellular structure |
TUBB2A |
Kd |
'=' |
199526 |
nM |
| Q6PEY2 |
BXGT016465 |
Tubulin alpha-3E chain |
reviewed |
Cellular structure |
TUBA3E |
Kd |
'=' |
199526 |
nM |
| Q9BQE3 |
BXGT020109 |
Tubulin alpha-1C chain |
reviewed |
Cellular structure |
TUBA1C |
Kd |
'=' |
199526 |
nM |
| P68363 |
BXGT011594 |
Tubulin alpha-1B chain |
reviewed |
Cellular structure |
TUBA1B |
Kd |
'=' |
199526 |
nM |
| P07437 |
BXGT006624 |
Tubulin beta chain |
reviewed |
Cellular structure |
TUBB |
Kd |
'=' |
199526 |
nM |
| Q3ZCM7 |
BXGT014551 |
Tubulin beta-8 chain |
reviewed |
- |
TUBB8 |
Kd |
'=' |
199526 |
nM |
| P04350 |
BXGT006193 |
Tubulin beta-4A chain |
reviewed |
Cellular structure |
TUBB4A |
Kd |
'=' |
199526 |
nM |
| Q71U36 |
BXGT016705 |
Tubulin alpha-1A chain |
reviewed |
Cellular structure |
TUBA1A |
Kd |
'=' |
199526 |
nM |
| Q13509 |
BXGT013366 |
Tubulin beta-3 chain |
reviewed |
Cellular structure |
TUBB3 |
Kd |
'=' |
199526 |
nM |
| P68366 |
BXGT011595 |
Tubulin alpha-4A chain |
reviewed |
Cellular structure |
TUBA4A |
Kd |
'=' |
199526 |
nM |
| P0DPH7 |
BXGT007527 |
Tubulin alpha-3C chain |
reviewed |
- |
TUBA3C |
Kd |
'=' |
199526 |
nM |
| Q9H4B7 |
BXGT020475 |
Tubulin beta-1 chain |
reviewed |
Cellular structure |
TUBB1 |
Kd |
'=' |
199526 |
nM |
| P68371 |
BXGT011597 |
Tubulin beta-4B chain |
reviewed |
Cellular structure |
TUBB4B |
Kd |
'=' |
199526 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
546 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
3981 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
14125 |
nM |
| O00167 |
BXGT003887 |
Eyes absent homolog 2 |
reviewed |
- |
EYA2 |
Potency |
- |
8493 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
7079 |
nM |
| Q13332 |
BXGT013342 |
Receptor-type tyrosine-protein phosphatase S |
reviewed |
Enzyme |
PTPRS |
Inhibition |
'=' |
84 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
TIME |
'=' |
10 |
hr |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
4466 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
1330 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
11200 |
nM |
| P11064 |
BXGT007646 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
IC50 |
'=' |
10000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
22387 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Activity |
- |
- |
- |
| Q86831 |
BXGT017584 |
Polyprotein II |
unreviewed |
- |
|
Inhibition |
'=' |
40 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
45 |
% |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Ratio |
'=' |
9 |
- |