| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
Ki |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
8 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
8 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
8 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
8 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
8 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
8 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
8 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
8 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
8 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
8 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
8 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
8 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
8 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
8 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
8 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
8 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Ki |
'=' |
12 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
12 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
12 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
Ki |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
IC50 |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
IC50 |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
Ki |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
91 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
91 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
91 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
91 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
91 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
91 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
91 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
91 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
91 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
91 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
91 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
91 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
91 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
91 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
91 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
91 |
nM |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
Ratio |
'=' |
1 |
- |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
Ratio |
'=' |
1 |
- |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
Ratio |
'=' |
1 |
- |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
Ratio |
'=' |
1 |
- |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
Ratio |
'=' |
1 |
- |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
Ratio |
'=' |
1 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
6 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
6 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
6 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
6 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
6 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
6 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
6 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
6 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
6 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
6 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
6 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
6 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
6 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
6 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
6 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
6 |
nM |
| P16305 |
BXGT008215 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
85000 |
nM |
| P27681 |
BXGT009196 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
85000 |
nM |
| P63080 |
BXGT011492 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
85000 |
nM |
| Q9D6F4 |
BXGT020259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
85000 |
nM |
| P22933 |
BXGT008819 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
85000 |
nM |
| P26049 |
BXGT009086 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
85000 |
nM |
| Q9JLF1 |
BXGT020834 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
- |
Gabrq |
Ki |
'=' |
85000 |
nM |
| P62812 |
BXGT011459 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
85000 |
nM |
| A2AMW3 |
BXGT001075 |
Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon |
unreviewed |
- |
Gabre |
Ki |
'=' |
85000 |
nM |
| P22723 |
BXGT008798 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
85000 |
nM |
| Q9R0Y8 |
BXGT021410 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
85000 |
nM |
| P50571 |
BXGT010810 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
85000 |
nM |
| Q8QZW7 |
BXGT018675 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
85000 |
nM |
| P26048 |
BXGT009085 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
85000 |
nM |
| Q8BHJ7 |
BXGT017911 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
85000 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
17 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
17 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
17 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
TBPS shift |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
TBPS shift |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
TBPS shift |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
TBPS shift |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
TBPS shift |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
TBPS shift |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
TBPS shift |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
TBPS shift |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
TBPS shift |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
TBPS shift |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
TBPS shift |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
TBPS shift |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
TBPS shift |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
TBPS shift |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
TBPS shift |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
TBPS shift |
'=' |
1 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
ED50 |
'=' |
0 |
mg.kg-1 |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
ED50 |
'=' |
0 |
mg.kg-1 |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
ED50 |
'=' |
0 |
mg.kg-1 |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
ED50 |
'=' |
0 |
mg.kg-1 |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
ED50 |
'=' |
0 |
mg.kg-1 |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
ED50 |
'=' |
0 |
mg.kg-1 |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Control |
'=' |
7 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
[35S] TBPS shift |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
[35S] TBPS shift |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
[35S] TBPS shift |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
[35S] TBPS shift |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
[35S] TBPS shift |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
[35S] TBPS shift |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
[35S] TBPS shift |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
[35S] TBPS shift |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
[35S] TBPS shift |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
[35S] TBPS shift |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
[35S] TBPS shift |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
[35S] TBPS shift |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
[35S] TBPS shift |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
[35S] TBPS shift |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
[35S] TBPS shift |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
[35S] TBPS shift |
'=' |
1 |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Ki |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
Ki |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
4 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
4 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
4 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
4 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
4 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
4 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
4 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
4 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
4 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
4 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
4 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
4 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
4 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
4 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
4 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
4 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
2 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
2 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
2 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
IC50 |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
IC50 |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
- |
- |
- |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
74000 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
74000 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
74000 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
74000 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
74000 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
74000 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
74000 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
74000 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
74000 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
74000 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
74000 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
74000 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
74000 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
74000 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
74000 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
74000 |
nM |
| P21447 |
BXGT008651 |
ATP-dependent translocase ABCB1 |
reviewed |
- |
Abcb1a |
Activity |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
Ki |
- |
- |
- |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Inhibition |
'=' |
2 |
% |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
6 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
6 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
6 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
6 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
6 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
6 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
6 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
6 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
6 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
6 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
6 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
6 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
6 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
6 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
6 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
6 |
nM |
| P02770 |
BXGT005957 |
Serum albumin |
reviewed |
- |
Alb |
Kd |
'=' |
15100 |
nM |
| O60885 |
BXGT004906 |
Bromodomain-containing protein 4 |
reviewed |
Epigenetic regulator |
BRD4 |
Inhibition |
'=' |
43 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
5 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
5 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
5 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
5 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
5 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
5 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
5 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
5 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
5 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
5 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
5 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
5 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
5 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
5 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
5 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
5 |
nM |
| P02692 |
BXGT005921 |
Fatty acid-binding protein, liver |
reviewed |
- |
Fabp1 |
Ki |
'=' |
115000 |
nM |
| O15245 |
BXGT004141 |
Solute carrier family 22 member 1 |
reviewed |
Transporter |
SLC22A1 |
Inhibition |
'=' |
5 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Kd |
'=' |
36 |
nM |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
Ki |
- |
- |
- |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
IC50 |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
IC50 |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
Ki |
- |
- |
- |
| P16305 |
BXGT008215 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Activity |
'=' |
1 |
- |
| P27681 |
BXGT009196 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Activity |
'=' |
1 |
- |
| P63080 |
BXGT011492 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Activity |
'=' |
1 |
- |
| Q9D6F4 |
BXGT020259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Activity |
'=' |
1 |
- |
| P22933 |
BXGT008819 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Activity |
'=' |
1 |
- |
| P26049 |
BXGT009086 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Activity |
'=' |
1 |
- |
| Q9JLF1 |
BXGT020834 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
- |
Gabrq |
Activity |
'=' |
1 |
- |
| P62812 |
BXGT011459 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Activity |
'=' |
1 |
- |
| A2AMW3 |
BXGT001075 |
Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon |
unreviewed |
- |
Gabre |
Activity |
'=' |
1 |
- |
| P22723 |
BXGT008798 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Activity |
'=' |
1 |
- |
| Q9R0Y8 |
BXGT021410 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Activity |
'=' |
1 |
- |
| P50571 |
BXGT010810 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Activity |
'=' |
1 |
- |
| Q8QZW7 |
BXGT018675 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Activity |
'=' |
1 |
- |
| P26048 |
BXGT009085 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Activity |
'=' |
1 |
- |
| Q8BHJ7 |
BXGT017911 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Activity |
'=' |
1 |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
20 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
20 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
20 |
nM |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
Ki |
'=' |
10 |
nM |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
Ki |
'=' |
10 |
nM |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
Ki |
'=' |
10 |
nM |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
Ki |
'=' |
10 |
nM |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
Ki |
'=' |
10 |
nM |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
Ki |
'=' |
10 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
7 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
7 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
7 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
7 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
7 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
7 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
7 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
7 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
7 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
7 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
7 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
7 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
7 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
7 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
7 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
7 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
5 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
1 |
- |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Activity |
'=' |
1 |
- |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Activity |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
20 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
20 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
20 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Efficacy |
'=' |
118 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
118 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
118 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA shift |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA shift |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA shift |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA shift |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA shift |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA shift |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA shift |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA shift |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA shift |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA shift |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA shift |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA shift |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA shift |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA shift |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA shift |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA shift |
'=' |
2 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
14 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
14 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
14 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
14 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
14 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
14 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
14 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
14 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
14 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
14 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
14 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
14 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
14 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
14 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
14 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
14 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
13 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
13 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
13 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
14 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
14 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
14 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
14 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
14 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
14 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'>' |
10000 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'>' |
10000 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'>' |
10000 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'>' |
10000 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
9 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
9 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
9 |
nM |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
IC50 |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
IC50 |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
IC50 |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
IC50 |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
IC50 |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ki |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
Ki |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
IC50 |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Ki |
'=' |
10 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Ki |
'=' |
10 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
10 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
Ki |
'=' |
10 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Ki |
'=' |
10 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
Ki |
'=' |
10 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
Ki |
'=' |
10 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
Ki |
'=' |
10 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
10 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
Ki |
'=' |
10 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
Ki |
'=' |
10 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
Ki |
'=' |
10 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
10 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
10 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
10 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
10 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
12 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Change in Cl- current |
'=' |
1 |
- |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Change in Cl- current |
'=' |
1 |
- |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Change in Cl- current |
'=' |
1 |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
IC50 |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ki |
- |
- |
- |
| O60885 |
BXGT004906 |
Bromodomain-containing protein 4 |
reviewed |
Epigenetic regulator |
BRD4 |
Delta Tm |
'=' |
1 |
degrees C |
| P02770 |
BXGT005957 |
Serum albumin |
reviewed |
- |
Alb |
PPB |
'=' |
92 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
EC50 |
'=' |
85 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
EC50 |
'=' |
85 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
EC50 |
'=' |
85 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Activity |
'=' |
207 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
207 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
207 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
9 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
9 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
9 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Ki |
'=' |
11 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
11 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
11 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
4 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
4 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
4 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
4 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
4 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
4 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
4 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
4 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
4 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
4 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
4 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
4 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
4 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
4 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
4 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
4 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Efficacy |
'=' |
211 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
211 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
211 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
20 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
20 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
20 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
20 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
20 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
20 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
20 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
20 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
20 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
20 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
20 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
20 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
20 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
20 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
20 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
20 |
nM |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
IC50 |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
5 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
5 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
5 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
5 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
5 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
5 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
5 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
5 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
5 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
5 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
5 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
5 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
5 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
5 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
5 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
5 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
5 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
5 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
5 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
5 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
5 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
5 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
5 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
5 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
5 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
5 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
5 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
5 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
5 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
5 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
5 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
5 |
nM |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
IC50 |
- |
- |
- |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
IC50 |
- |
- |
- |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
Ki |
- |
- |
- |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Ki |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
IC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
6 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
6 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
6 |
nM |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
IC50 |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Ki |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Ki |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
IC50 |
- |
- |
- |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Activity |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
- |
- |
- |
| P04177 |
BXGT006162 |
Tyrosine 3-monooxygenase |
reviewed |
- |
Th |
Inhibition |
'=' |
23 |
% |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
GABA ratio |
'=' |
1 |
- |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
GABA ratio |
'=' |
1 |
- |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
GABA ratio |
'=' |
1 |
- |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
GABA ratio |
'=' |
1 |
- |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
GABA ratio |
'=' |
1 |
- |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
GABA ratio |
'=' |
1 |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
10 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
10 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
10 |
nM |
| P16305 |
BXGT008215 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
12 |
nM |
| P27681 |
BXGT009196 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
12 |
nM |
| P63080 |
BXGT011492 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
12 |
nM |
| Q9D6F4 |
BXGT020259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
12 |
nM |
| P22933 |
BXGT008819 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
12 |
nM |
| P26049 |
BXGT009086 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
12 |
nM |
| Q9JLF1 |
BXGT020834 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
- |
Gabrq |
IC50 |
'=' |
12 |
nM |
| P62812 |
BXGT011459 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
12 |
nM |
| A2AMW3 |
BXGT001075 |
Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon |
unreviewed |
- |
Gabre |
IC50 |
'=' |
12 |
nM |
| P22723 |
BXGT008798 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
12 |
nM |
| Q9R0Y8 |
BXGT021410 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
12 |
nM |
| P50571 |
BXGT010810 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
12 |
nM |
| Q8QZW7 |
BXGT018675 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
12 |
nM |
| P26048 |
BXGT009085 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
12 |
nM |
| Q8BHJ7 |
BXGT017911 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
12 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
144 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
144 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
144 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
144 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
144 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
144 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
144 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
144 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
144 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
144 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
144 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
144 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
144 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
144 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
144 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
144 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
1 |
- |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Log IC50 |
'=' |
-7 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Log IC50 |
'=' |
-7 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Log IC50 |
'=' |
-7 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
Log IC50 |
'=' |
-7 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Log IC50 |
'=' |
-7 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
Log IC50 |
'=' |
-7 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
Log IC50 |
'=' |
-7 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
Log IC50 |
'=' |
-7 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Log IC50 |
'=' |
-7 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
Log IC50 |
'=' |
-7 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
Log IC50 |
'=' |
-7 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
Log IC50 |
'=' |
-7 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Log IC50 |
'=' |
-7 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Log IC50 |
'=' |
-7 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Log IC50 |
'=' |
-7 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Log IC50 |
'=' |
-7 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Control |
'=' |
39 |
% |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Ki |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
IC50 |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
IC50 |
- |
- |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Efficacy |
'=' |
106 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
106 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
106 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
10 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
10 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
10 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
10 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
10 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
10 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
10 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
10 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
10 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
10 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
10 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
10 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
10 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
10 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
10 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
10 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
33 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
33 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
33 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
0 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
0 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Efficacy |
'=' |
0 |
% |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Ki |
'>' |
3000 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'>' |
3000 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'>' |
3000 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
33 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Efficacy |
'=' |
0 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
0 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
0 |
% |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Ki |
'>' |
7000 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'>' |
7000 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'>' |
7000 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Kd |
'=' |
23 |
nM |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
15 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
15 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
15 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Ki |
'=' |
11 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
11 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
11 |
nM |
| P02763 |
BXGT005951 |
Alpha-1-acid glycoprotein 1 |
reviewed |
- |
ORM1 |
Activity |
'=' |
10 |
uM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Efficacy |
'=' |
115 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
115 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
115 |
% |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
GR |
'=' |
1 |
- |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
GR |
'=' |
1 |
- |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
GR |
'=' |
1 |
- |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
GR |
'=' |
1 |
- |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
GR |
'=' |
1 |
- |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
GR |
'=' |
1 |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
Ki |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
IC50 |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
Ki |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
Ki |
- |
- |
- |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Ki |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
5 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
5 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
5 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
5 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
5 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
5 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
5 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
5 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
5 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
5 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
5 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
5 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
5 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
5 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
5 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
5 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
'=' |
8 |
uM |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
Ki |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Ki |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
- |
- |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
11 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
11 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
11 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Ka |
'=' |
1 |
10^5/M |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Binding |
'=' |
86 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
7 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
7 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
7 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
7 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
7 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
7 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
7 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
7 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
7 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
7 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
7 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
7 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
7 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
7 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
7 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
7 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
15 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
15 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
15 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
15 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
15 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
15 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
15 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
15 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
15 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
15 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
15 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
15 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
15 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
15 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
15 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
15 |
nM |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
'>' |
100000 |
nM |
| P32239 |
BXGT009612 |
Gastrin/cholecystokinin type B receptor |
reviewed |
G-protein coupled receptor |
CCKBR |
IC50 |
'>' |
100000 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
1 |
- |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
123594743 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
123594743 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
123594743 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
123594743 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
123594743 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
123594743 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
123594743 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
123594743 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
123594743 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
123594743 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
123594743 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
123594743 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
123594743 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
123594743 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
123594743 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
123594743 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Activity |
'=' |
81 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
156 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
156 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Efficacy |
'=' |
156 |
% |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Efficacy |
'=' |
89 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
89 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
89 |
% |
| P30536 |
BXGT009435 |
Translocator protein |
reviewed |
- |
TSPO |
IC50 |
'=' |
123594743 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
8 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
8 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
8 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
8 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
8 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
8 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
8 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
8 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
8 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
8 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
8 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
8 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
8 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
8 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
8 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
8 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
1 |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Efficacy |
'=' |
138 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
138 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
138 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'>' |
1000 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'>' |
1000 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'>' |
1000 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'>' |
1000 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'>' |
1000 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'>' |
1000 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'>' |
1000 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'>' |
1000 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'>' |
1000 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'>' |
1000 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'>' |
1000 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'>' |
1000 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'>' |
1000 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'>' |
1000 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'>' |
1000 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'>' |
1000 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Shift |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Shift |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Shift |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Shift |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Shift |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Shift |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Shift |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Shift |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Shift |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Shift |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Shift |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Shift |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Shift |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Shift |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Shift |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Shift |
'=' |
1 |
- |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
12 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
12 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
12 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
12 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
12 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
12 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
12 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
12 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
12 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
12 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
12 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
12 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
12 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
12 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
12 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
12 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GS |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GS |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GS |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GS |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GS |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GS |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GS |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GS |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GS |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GS |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GS |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GS |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GS |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GS |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GS |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GS |
'=' |
2 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
0 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
0 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
0 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
0 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
0 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
0 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
0 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
0 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
0 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
0 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
0 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
0 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
0 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
0 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
0 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
0 |
- |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
13 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
- |
- |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Cl - current change |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Cl - current change |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Cl - current change |
'=' |
1 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
323 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
323 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
323 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
323 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
323 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
323 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
323 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
323 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
323 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
323 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
323 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
323 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
323 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
323 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
323 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
323 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
157 |
% |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Efficacy |
'=' |
157 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Efficacy |
'=' |
157 |
% |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Activity |
'=' |
508 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
508 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
508 |
% |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Activity |
'=' |
177 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
177 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
177 |
% |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Ratio |
'=' |
1 |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Ratio |
'=' |
1 |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ratio |
'=' |
1 |
- |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
Ratio |
'=' |
1 |
- |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Ratio |
'=' |
1 |
- |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
Ratio |
'=' |
1 |
- |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
Ratio |
'=' |
1 |
- |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
Ratio |
'=' |
1 |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ratio |
'=' |
1 |
- |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
Ratio |
'=' |
1 |
- |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
Ratio |
'=' |
1 |
- |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
Ratio |
'=' |
1 |
- |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ratio |
'=' |
1 |
- |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ratio |
'=' |
1 |
- |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ratio |
'=' |
1 |
- |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ratio |
'=' |
1 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
IC50 |
- |
- |
- |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
Ki |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
Ki |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
Ki |
- |
- |
- |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
IC50 |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
IC50 |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
IC50 |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Ki |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
- |
- |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
43 |
nM |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Ki |
'=' |
574 |
nM |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
- |
- |
- |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
Ki |
- |
- |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
Ki |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
IC50 |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
IC50 |
- |
- |
- |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
Ratio |
'=' |
1 |
- |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
Ratio |
'=' |
1 |
- |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
Ratio |
'=' |
1 |
- |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
Ratio |
'=' |
1 |
- |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
Ratio |
'=' |
1 |
- |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
Ratio |
'=' |
1 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Inhibition |
'=' |
100 |
% |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Inhibition |
'=' |
100 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Inhibition |
'=' |
100 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Inhibition |
'=' |
100 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Inhibition |
'=' |
100 |
% |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Inhibition |
'=' |
100 |
% |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Inhibition |
'=' |
100 |
% |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Inhibition |
'=' |
100 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Inhibition |
'=' |
100 |
% |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Inhibition |
'=' |
100 |
% |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Inhibition |
'=' |
100 |
% |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Inhibition |
'=' |
100 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Inhibition |
'=' |
100 |
% |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Inhibition |
'=' |
100 |
% |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Inhibition |
'=' |
100 |
% |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Inhibition |
'=' |
100 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
20 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
IC50 |
- |
- |
- |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ki |
- |
- |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IC50 |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
IC50 |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
Ki |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
- |
- |
- |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'>' |
135000 |
nM |
| Q04828 |
BXGT012787 |
Aldo-keto reductase family 1 member C1 |
reviewed |
Enzyme |
AKR1C1 |
IC50 |
'=' |
5600 |
nM |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
IC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
ID50 |
'=' |
0 |
mg.kg-1 |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
ID50 |
'=' |
0 |
mg.kg-1 |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
ID50 |
'=' |
0 |
mg.kg-1 |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
ID50 |
'=' |
0 |
mg.kg-1 |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
ID50 |
'=' |
0 |
mg.kg-1 |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
ID50 |
'=' |
0 |
mg.kg-1 |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
16 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
16 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
16 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'>' |
7000 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'>' |
7000 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'>' |
7000 |
nM |
| Q9NY46 |
BXGT021248 |
Sodium channel protein type 3 subunit alpha |
reviewed |
Ion channel |
SCN3A |
Inhibition |
'=' |
15 |
% |
| Q99250 |
BXGT019913 |
Sodium channel protein type 2 subunit alpha |
reviewed |
Ion channel |
SCN2A |
Inhibition |
'=' |
15 |
% |
| P35498 |
BXGT009838 |
Sodium channel protein type 1 subunit alpha |
reviewed |
Ion channel |
SCN1A |
Inhibition |
'=' |
15 |
% |
| Q9NY46 |
BXGT021248 |
Sodium channel protein type 3 subunit alpha |
reviewed |
Ion channel |
SCN3A |
Inhibition |
'=' |
45 |
% |
| Q99250 |
BXGT019913 |
Sodium channel protein type 2 subunit alpha |
reviewed |
Ion channel |
SCN2A |
Inhibition |
'=' |
45 |
% |
| P35498 |
BXGT009838 |
Sodium channel protein type 1 subunit alpha |
reviewed |
Ion channel |
SCN1A |
Inhibition |
'=' |
45 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
98 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
98 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
98 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
103 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
103 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Efficacy |
'=' |
103 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
28 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
28 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
28 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
28 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
28 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
28 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
28 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
28 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
28 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
28 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
28 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
28 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
28 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
28 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
28 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
28 |
nM |
| P30551 |
BXGT009439 |
Cholecystokinin receptor type A |
reviewed |
- |
Cckar |
IC50 |
'>' |
100000 |
nM |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Kd |
'=' |
213 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA shift |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA shift |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA shift |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA shift |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA shift |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA shift |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA shift |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA shift |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA shift |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA shift |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA shift |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA shift |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA shift |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA shift |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA shift |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA shift |
'=' |
2 |
- |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Inhibition |
'=' |
0 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
77 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
77 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
77 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
77 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
77 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
77 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
77 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
77 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
77 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
77 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
77 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
77 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
77 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
77 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
77 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
77 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
IC50 |
- |
- |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
20 |
nM |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Activity |
'=' |
40 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
13 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
13 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
13 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Displacement |
'=' |
-13 |
% |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Displacement |
'=' |
-13 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Displacement |
'=' |
-13 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Displacement |
'=' |
-13 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Displacement |
'=' |
-13 |
% |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Displacement |
'=' |
-13 |
% |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Displacement |
'=' |
-13 |
% |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Displacement |
'=' |
-13 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Displacement |
'=' |
-13 |
% |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Displacement |
'=' |
-13 |
% |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Displacement |
'=' |
-13 |
% |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Displacement |
'=' |
-13 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Displacement |
'=' |
-13 |
% |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Displacement |
'=' |
-13 |
% |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Displacement |
'=' |
-13 |
% |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Displacement |
'=' |
-13 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
2 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
2 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
2 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
2 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
2 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
2 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
2 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
2 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
2 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
2 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
2 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
2 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
2 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
2 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
2 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
2 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Cl - current change |
'=' |
1 |
- |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
51 |
% |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
Ki |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
IC50 |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
Ki |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
IC50 |
- |
- |
- |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Km |
'=' |
72400 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'~' |
7 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'~' |
7 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'~' |
7 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'~' |
7 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'~' |
7 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'~' |
7 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'~' |
7 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'~' |
7 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'~' |
7 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'~' |
7 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'~' |
7 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'~' |
7 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'~' |
7 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'~' |
7 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'~' |
7 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'~' |
7 |
nM |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
IC50 |
'=' |
13 |
nM |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
IC50 |
'=' |
13 |
nM |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
IC50 |
'=' |
13 |
nM |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
IC50 |
'=' |
13 |
nM |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
IC50 |
'=' |
13 |
nM |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
IC50 |
'=' |
13 |
nM |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
Ki |
- |
- |
- |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
Ki |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
Ki |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ki |
- |
- |
- |
| P08104 |
BXGT006726 |
Sodium channel protein type 3 subunit alpha |
reviewed |
- |
Scn3a |
IC50 |
'=' |
152000 |
nM |
| P04774 |
BXGT006260 |
Sodium channel protein type 1 subunit alpha |
reviewed |
- |
Scn1a |
IC50 |
'=' |
152000 |
nM |
| P04775 |
BXGT006261 |
Sodium channel protein type 2 subunit alpha |
reviewed |
- |
Scn2a |
IC50 |
'=' |
152000 |
nM |
| P42330 |
BXGT010301 |
Aldo-keto reductase family 1 member C3 |
reviewed |
Enzyme |
AKR1C3 |
IC50 |
'=' |
84000 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
'=' |
54 |
% |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
IC50 |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
- |
- |
- |
| P30553 |
BXGT009440 |
Gastrin/cholecystokinin type B receptor |
reviewed |
- |
Cckbr |
IC50 |
'>' |
100000 |
nM |
| P30551 |
BXGT009439 |
Cholecystokinin receptor type A |
reviewed |
- |
Cckar |
IC50 |
'>' |
100000 |
nM |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
IC50 |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
IC50 |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
Ki |
- |
- |
- |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
345 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
345 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Activity |
'=' |
345 |
% |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
Ki |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
Ki |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
IC50 |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Change in Cl- current |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
12 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
12 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
12 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Displacement |
'=' |
25 |
% |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Displacement |
'=' |
25 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Displacement |
'=' |
25 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Displacement |
'=' |
25 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Displacement |
'=' |
25 |
% |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Displacement |
'=' |
25 |
% |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Displacement |
'=' |
25 |
% |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Displacement |
'=' |
25 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Displacement |
'=' |
25 |
% |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Displacement |
'=' |
25 |
% |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Displacement |
'=' |
25 |
% |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Displacement |
'=' |
25 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Displacement |
'=' |
25 |
% |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Displacement |
'=' |
25 |
% |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Displacement |
'=' |
25 |
% |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Displacement |
'=' |
25 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA current |
'=' |
300 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA current |
'=' |
300 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA current |
'=' |
300 |
% |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ki |
- |
- |
- |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
Ki |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
Ki |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
Ki |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
Ki |
- |
- |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Activity |
'=' |
420 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
420 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
420 |
% |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
IC50 |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
IC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
IC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA ratio |
- |
- |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA ratio |
- |
- |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA ratio |
- |
- |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA ratio |
- |
- |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA ratio |
- |
- |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA ratio |
- |
- |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA ratio |
- |
- |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA ratio |
- |
- |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA ratio |
- |
- |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA ratio |
- |
- |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA ratio |
- |
- |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA ratio |
- |
- |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA ratio |
- |
- |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA ratio |
- |
- |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA ratio |
- |
- |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA ratio |
- |
- |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Activity |
'=' |
72 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Activity |
'=' |
72 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Activity |
'=' |
72 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
12 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
12 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
12 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
12 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
12 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
12 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
12 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
12 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
12 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
12 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
12 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
12 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
12 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
12 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
12 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
12 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ratio |
'=' |
1 |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
14 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
14 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
PPB |
'=' |
93 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
15 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Activity |
'=' |
71 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Activity |
'=' |
71 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Activity |
'=' |
71 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
6 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
6 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
6 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
6 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
6 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
6 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
6 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
6 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
6 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
6 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
6 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
6 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
6 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
6 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
6 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
6 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
5 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
5 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
5 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
5 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
5 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
5 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
5 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
5 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
5 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
5 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
5 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
5 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
5 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
5 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
5 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
5 |
nM |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
IC50 |
'=' |
25 |
nM |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
IC50 |
'=' |
25 |
nM |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
IC50 |
'=' |
25 |
nM |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
IC50 |
'=' |
25 |
nM |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
IC50 |
'=' |
25 |
nM |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
IC50 |
'=' |
25 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Displacement |
'=' |
33 |
% |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Displacement |
'=' |
33 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Displacement |
'=' |
33 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Displacement |
'=' |
33 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Displacement |
'=' |
33 |
% |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Displacement |
'=' |
33 |
% |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Displacement |
'=' |
33 |
% |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Displacement |
'=' |
33 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Displacement |
'=' |
33 |
% |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Displacement |
'=' |
33 |
% |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Displacement |
'=' |
33 |
% |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Displacement |
'=' |
33 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Displacement |
'=' |
33 |
% |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Displacement |
'=' |
33 |
% |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Displacement |
'=' |
33 |
% |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Displacement |
'=' |
33 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
20 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
20 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
20 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
20 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
20 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
20 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
20 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
20 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
20 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
20 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
20 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
20 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
20 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
20 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
20 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
20 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Kd |
'=' |
24547 |
nM |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
IC50 |
- |
- |
- |
| P22300 |
BXGT008750 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
GABRG2 |
IC50 |
'=' |
41 |
nM |
| P10064 |
BXGT007533 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
GABRA3 |
IC50 |
'=' |
41 |
nM |
| P08219 |
BXGT006749 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
GABRA1 |
IC50 |
'=' |
41 |
nM |
| P20237 |
BXGT008552 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
GABRA4 |
IC50 |
'=' |
41 |
nM |
| P08220 |
BXGT006750 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
GABRB1 |
IC50 |
'=' |
41 |
nM |
| P10063 |
BXGT007532 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
GABRA2 |
IC50 |
'=' |
41 |
nM |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
8 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
8 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
8 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
8 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
8 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
8 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
8 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
8 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
8 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
8 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
8 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
8 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
8 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
8 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
8 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
8 |
nM |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Inhibition |
'=' |
51 |
% |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
14 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
14 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
14 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
14 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
14 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
14 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
14 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
14 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
14 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
14 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
14 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
14 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
14 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
14 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
14 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
14 |
nM |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Activity |
'=' |
3 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Activity |
'=' |
776 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
9 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
9 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA ratio |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA ratio |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA ratio |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA ratio |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA ratio |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA ratio |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA ratio |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA ratio |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA ratio |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA ratio |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA ratio |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA ratio |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA ratio |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA ratio |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA ratio |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA ratio |
'=' |
2 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
4 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
4 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
4 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
4 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
4 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
4 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
4 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
4 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
4 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
4 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
4 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
4 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
4 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
4 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
4 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
4 |
nM |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
IC50 |
'=' |
194 |
nM |
| Q63931 |
BXGT016083 |
Cholecystokinin receptor type A |
reviewed |
- |
CCKAR |
IC50 |
'>' |
100000 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
14 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
14 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
14 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Efficacy |
'=' |
73 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
73 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Efficacy |
'=' |
73 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
9 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
9 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
9 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
9 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
9 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
9 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
9 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
9 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
9 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
9 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
9 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
9 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
9 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
9 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
9 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
9 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
13 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
13 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
13 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
13 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
13 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
13 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
13 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
13 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
13 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
13 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
13 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
13 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
13 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
13 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
13 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
13 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Efficacy |
'=' |
157 |
% |
| P16305 |
BXGT008215 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
- |
- |
| P27681 |
BXGT009196 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
- |
- |
| P63080 |
BXGT011492 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
- |
- |
| Q9D6F4 |
BXGT020259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
- |
- |
| P22933 |
BXGT008819 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
- |
- |
| P26049 |
BXGT009086 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
- |
- |
| Q9JLF1 |
BXGT020834 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
- |
Gabrq |
IC50 |
'=' |
- |
- |
| P62812 |
BXGT011459 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
- |
- |
| A2AMW3 |
BXGT001075 |
Gamma-aminobutyric acid (GABA) A receptor, subunit epsilon |
unreviewed |
- |
Gabre |
IC50 |
'=' |
- |
- |
| P22723 |
BXGT008798 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
- |
- |
| Q9R0Y8 |
BXGT021410 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
- |
- |
| P50571 |
BXGT010810 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
- |
- |
| Q8QZW7 |
BXGT018675 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
- |
- |
| P26048 |
BXGT009085 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
- |
- |
| Q8BHJ7 |
BXGT017911 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA shift |
'=' |
3 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA shift |
'=' |
3 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA shift |
'=' |
3 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA shift |
'=' |
3 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA shift |
'=' |
3 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA shift |
'=' |
3 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA shift |
'=' |
3 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA shift |
'=' |
3 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA shift |
'=' |
3 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA shift |
'=' |
3 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA shift |
'=' |
3 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA shift |
'=' |
3 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA shift |
'=' |
3 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA shift |
'=' |
3 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA shift |
'=' |
3 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA shift |
'=' |
3 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
ID50 |
'=' |
5 |
mg.kg-1 |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
ID50 |
'=' |
5 |
mg.kg-1 |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
ID50 |
'=' |
5 |
mg.kg-1 |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
ID50 |
'=' |
5 |
mg.kg-1 |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
ID50 |
'=' |
5 |
mg.kg-1 |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
ID50 |
'=' |
5 |
mg.kg-1 |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
IC50 |
- |
- |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
14 |
nM |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
'=' |
14 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
14 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
'=' |
14 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
'=' |
14 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
'=' |
14 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
'=' |
14 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
'=' |
14 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
'=' |
14 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
'=' |
14 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
'=' |
14 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
'=' |
14 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
'=' |
14 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
14 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
14 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
'=' |
14 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
'=' |
14 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
6 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
6 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
6 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
6 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
6 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
6 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
6 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
6 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
6 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
6 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
6 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
6 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
6 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
6 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
6 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
6 |
nM |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
IC50 |
- |
- |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
Ki |
- |
- |
- |
| P02692 |
BXGT005921 |
Fatty acid-binding protein, liver |
reviewed |
- |
Fabp1 |
Ki |
'=' |
531 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
4 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
4 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
4 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
4 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
4 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
4 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
4 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
4 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
4 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
4 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
4 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
4 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
4 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
4 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
4 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
4 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Binding affinity |
'=' |
29 |
spec bound mg-1 |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Inhibition |
'<' |
50 |
% |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Inhibition |
'<' |
50 |
% |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Inhibition |
'<' |
50 |
% |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Inhibition |
'<' |
50 |
% |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Inhibition |
'<' |
50 |
% |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Inhibition |
'<' |
50 |
% |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Inhibition |
'<' |
50 |
% |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Inhibition |
'<' |
50 |
% |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Inhibition |
'<' |
50 |
% |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Inhibition |
'<' |
50 |
% |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Inhibition |
'<' |
50 |
% |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Inhibition |
'<' |
50 |
% |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Inhibition |
'<' |
50 |
% |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Inhibition |
'<' |
50 |
% |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Inhibition |
'<' |
50 |
% |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Inhibition |
'<' |
50 |
% |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
26 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
26 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
26 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
15 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
15 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
15 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
11 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
11 |
nM |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
Ki |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Ki |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
Ki |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IC50 |
- |
- |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
EC50 |
'=' |
131 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
EC50 |
'=' |
131 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
EC50 |
'=' |
131 |
nM |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
IC50 |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
- |
- |
- |
| Q60484 |
BXGT015984 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
EC50 |
- |
- |
- |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Inhibition |
'=' |
97 |
% |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
IC50 |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
IC50 |
- |
- |
- |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
IC50 |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
Ki |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
IC50 |
- |
- |
- |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
PPB |
'=' |
94 |
% |
| O60885 |
BXGT004906 |
Bromodomain-containing protein 4 |
reviewed |
Epigenetic regulator |
BRD4 |
Delta Tm |
'=' |
1 |
degrees C |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
IC50 |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
IC50 |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
Ki |
- |
- |
- |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
'=' |
61 |
% |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
IC50 |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
- |
- |
- |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
22387 |
nM |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
IC50 |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Inhibition |
- |
- |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Inhibition |
- |
- |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Inhibition |
- |
- |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Inhibition |
- |
- |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Inhibition |
- |
- |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Inhibition |
- |
- |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Inhibition |
- |
- |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Inhibition |
- |
- |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Inhibition |
- |
- |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Inhibition |
- |
- |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Inhibition |
- |
- |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Inhibition |
- |
- |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Inhibition |
- |
- |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Inhibition |
- |
- |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Inhibition |
- |
- |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Inhibition |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA shift |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA shift |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA shift |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA shift |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA shift |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA shift |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA shift |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA shift |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA shift |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA shift |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA shift |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA shift |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA shift |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA shift |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA shift |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA shift |
'=' |
2 |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
5011 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Ki |
'=' |
251188 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
9 |
% |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
- |
- |
- |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
IC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
Ki |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
Ki |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Ki |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
Ki |
- |
- |
- |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
- |
- |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IC50 |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Ki |
- |
- |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
Ki |
- |
- |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
- |
- |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
EC50 |
'=' |
35 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
EC50 |
'=' |
35 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
EC50 |
'=' |
35 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
192 |
% |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Activity |
'=' |
192 |
% |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Activity |
'=' |
192 |
% |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Activity |
'=' |
153 |
% |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
'=' |
153 |
% |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
'=' |
153 |
% |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
'=' |
6 |
% |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Ki |
'=' |
13000 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
'=' |
17 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
'=' |
17 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
'=' |
17 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA ratio |
'=' |
2 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA ratio |
'=' |
2 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA ratio |
'=' |
2 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA ratio |
'=' |
2 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA ratio |
'=' |
2 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA ratio |
'=' |
2 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA ratio |
'=' |
2 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA ratio |
'=' |
2 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA ratio |
'=' |
2 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA ratio |
'=' |
2 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA ratio |
'=' |
2 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA ratio |
'=' |
2 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA ratio |
'=' |
2 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA ratio |
'=' |
2 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA ratio |
'=' |
2 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA ratio |
'=' |
2 |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
IC50 |
'=' |
30 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
IC50 |
'=' |
30 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
IC50 |
'=' |
30 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
IC50 |
'=' |
30 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
IC50 |
'=' |
30 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
IC50 |
'=' |
30 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
IC50 |
'=' |
30 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
IC50 |
'=' |
30 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
IC50 |
'=' |
30 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
IC50 |
'=' |
30 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
IC50 |
'=' |
30 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
IC50 |
'=' |
30 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
IC50 |
'=' |
30 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
IC50 |
'=' |
30 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
IC50 |
'=' |
30 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
IC50 |
'=' |
30 |
nM |
| O60885 |
BXGT004906 |
Bromodomain-containing protein 4 |
reviewed |
Epigenetic regulator |
BRD4 |
IC50 |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
Ki |
- |
- |
- |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Inhibition |
'=' |
34 |
% |
| O15439 |
BXGT004169 |
Multidrug resistance-associated protein 4 |
reviewed |
Transporter |
ABCC4 |
IC50 |
'=' |
133000 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
- |
- |
- |
| O60840 |
BXGT004901 |
Voltage-dependent L-type calcium channel subunit alpha-1F |
reviewed |
Ion channel |
CACNA1F |
IC50 |
'=' |
30500 |
nM |
| Q01668 |
BXGT012605 |
Voltage-dependent L-type calcium channel subunit alpha-1D |
reviewed |
Ion channel |
CACNA1D |
IC50 |
'=' |
30500 |
nM |
| Q13698 |
BXGT013392 |
Voltage-dependent L-type calcium channel subunit alpha-1S |
reviewed |
Ion channel |
CACNA1S |
IC50 |
'=' |
30500 |
nM |
| Q13936 |
BXGT013404 |
Voltage-dependent L-type calcium channel subunit alpha-1C |
reviewed |
Ion channel |
CACNA1C |
IC50 |
'=' |
30500 |
nM |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Ki |
- |
- |
- |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA ratio |
'=' |
1 |
- |
| P52895 |
BXGT010961 |
Aldo-keto reductase family 1 member C2 |
reviewed |
Enzyme |
AKR1C2 |
IC50 |
'=' |
2400 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
33498 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
Ki |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Ki |
- |
- |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
EC50 |
'=' |
45 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
EC50 |
'=' |
45 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
EC50 |
'=' |
45 |
nM |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
Ki |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
23 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
23 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
23 |
nM |
| P02768 |
BXGT005955 |
Serum albumin |
reviewed |
Transporter |
ALB |
Activity |
'=' |
6 |
% |
| P16257 |
BXGT008211 |
Translocator protein |
reviewed |
- |
Tspo |
Inhibition |
'=' |
85 |
% |
| O60885 |
BXGT004906 |
Bromodomain-containing protein 4 |
reviewed |
Epigenetic regulator |
BRD4 |
Delta Tm |
'=' |
1 |
degrees C |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
11 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
- |
- |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
14 |
nM |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'=' |
133000 |
nM |
| O15438 |
BXGT004168 |
Canalicular multispecific organic anion transporter 2 |
reviewed |
Transporter |
ABCC3 |
IC50 |
'=' |
133000 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
15 |
nM |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Activity |
- |
- |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Activity |
- |
- |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Activity |
- |
- |
- |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
Activity |
- |
- |
- |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Activity |
- |
- |
- |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
Activity |
- |
- |
- |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
Activity |
- |
- |
- |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
Activity |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Activity |
- |
- |
- |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
Activity |
- |
- |
- |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
Activity |
- |
- |
- |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
Activity |
- |
- |
- |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Activity |
- |
- |
- |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Activity |
- |
- |
- |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Activity |
- |
- |
- |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Activity |
- |
- |
- |