| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
10000 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
1 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
IC50 |
'=' |
22000 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
15848 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
45 |
% |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
12589 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
19952 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Inhibition |
- |
- |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
Inhibition |
- |
- |
- |
| P21447 |
BXGT008651 |
ATP-dependent translocase ABCB1 |
reviewed |
- |
Abcb1a |
Kd |
'=' |
6700 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
7943 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'>' |
10000 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
'=' |
6000 |
nM |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
56234 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
103 |
% |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| Q86831 |
BXGT017584 |
Polyprotein II |
unreviewed |
- |
|
Inhibition |
'=' |
72 |
% |
| P03469 |
BXGT006080 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
85200 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
112 |
% |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'>' |
10000 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
37 |
% |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
23 |
nmol/min |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
38 |
% |
| O95067 |
BXGT005347 |
G2/mitotic-specific cyclin-B2 |
reviewed |
Enzyme modulator |
CCNB2 |
IC50 |
'=' |
41000 |
nM |
| Q8WWL7 |
BXGT019000 |
G2/mitotic-specific cyclin-B3 |
reviewed |
Enzyme modulator |
CCNB3 |
IC50 |
'=' |
41000 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
41000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
41000 |
nM |
| P00441 |
BXGT005540 |
Superoxide dismutase [Cu-Zn] |
reviewed |
Enzyme |
SOD1 |
Activity |
- |
- |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
1 |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
5 |
% |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
Ki |
'=' |
21100 |
nM |
| Q13332 |
BXGT013342 |
Receptor-type tyrosine-protein phosphatase S |
reviewed |
Enzyme |
PTPRS |
IC50 |
- |
- |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
3981 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'>' |
50 |
% |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
'=' |
2200 |
nM |
| Q9NZ45 |
BXGT021269 |
CDGSH iron-sulfur domain-containing protein 1 |
reviewed |
- |
CISD1 |
Ki |
'=' |
132 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
IC50 |
'<' |
150 |
ug.mL-1 |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
84 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
7943 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
IC50 |
'=' |
55000 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
13 |
% |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
11220 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
15848 |
nM |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
13 |
nmol/min |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
716 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
2400 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
6309 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
15848 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
'=' |
55 |
uM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
3 |
- |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
97800 |
nM |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
28 |
nmol/min |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
Inhibition |
'=' |
60 |
% |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
IC50 |
'=' |
28 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Ka |
'=' |
1 |
10'5/M |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
28183 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
14700 |
nM |
| P24135 |
BXGT008949 |
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-2 |
reviewed |
- |
Plcg2 |
Activity |
- |
- |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
8 |
% |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
20000 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
58600 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
12589 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3 |
ug.mL-1 |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
Activity |
'=' |
4 |
% |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
15848 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
4700 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
1584 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
35481 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
15848 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
ID50 |
'=' |
67 |
ug ml-1 |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
21689 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
10000 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
Activity |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Potency |
- |
2 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
5011 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
8000 |
nM |
| Q12791 |
BXGT013264 |
Calcium-activated potassium channel subunit alpha-1 |
reviewed |
Ion channel |
KCNMA1 |
Control |
'=' |
167 |
% |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
7 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
20596 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
12 |
% |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
1330 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
IC50 |
'=' |
1200 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
7943 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
132000 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
64700 |
nM |
| Q03114 |
BXGT012692 |
Cyclin-dependent-like kinase 5 |
reviewed |
- |
Cdk5 |
EC50 |
'=' |
66100 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
24 |
% |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
1060 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
31622 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
7 |
% |
| P48147 |
BXGT010620 |
Prolyl endopeptidase |
reviewed |
Enzyme |
PREP |
IC50 |
'>' |
200000 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
15355 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
632 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
47 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
38100 |
nM |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
118 |
% |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
43100 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
79432 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
3548 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
11220 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
35481 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
- |
- |
- |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
16 |
ug.mL-1 |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'>' |
100000 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Kd |
'=' |
6760 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
12589 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
7 |
- |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
44668 |
nM |
| P00760 |
BXGT005644 |
Cationic trypsin |
reviewed |
- |
|
IC50 |
'=' |
105900 |
nM |
| Q63470 |
BXGT016073 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
reviewed |
- |
Dyrk1a |
AC50 |
'=' |
1259 |
nM |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
15 |
nmol/min |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
8912 |
nM |
| P11166 |
BXGT007661 |
Solute carrier family 2, facilitated glucose transporter member 1 |
reviewed |
Transporter |
SLC2A1 |
IC50 |
'=' |
4000 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
44668 |
nM |
| P11474 |
BXGT007710 |
Steroid hormone receptor ERR1 |
reviewed |
Nuclear receptor |
ESRRA |
IC50 |
'=' |
9640 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
IC50 |
'=' |
2320 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'>' |
100000 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
20 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
75100 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
10000 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
14 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
38 |
% |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
logIC50 |
'=' |
1 |
- |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
39810 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
1 |
- |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
2 |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
10000 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
- |
- |
- |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
25118 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
2700 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
3500 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
IC50 |
'=' |
3500 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
60 |
% |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
18 |
% |
| P10686 |
BXGT007601 |
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-1 |
reviewed |
- |
Plcg1 |
Activity |
- |
- |
- |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
Activity |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'=' |
360 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'>' |
100000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
79432 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
28183 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
43 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
10000 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
10000 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
46400 |
nM |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
IC50 |
'>' |
20000 |
nM |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
105 |
% |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
8412 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
TIME |
'=' |
3 |
hr |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
Activity |
- |
- |
- |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
11200 |
nM |
| Q9GZU7 |
BXGT020426 |
Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1 |
reviewed |
- |
CTDSP1 |
IC50 |
'=' |
9933 |
nM |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
230000 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
7943 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
22387 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
1 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
'=' |
55 |
uM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23715 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
'=' |
2240 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
81 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
- |
- |
- |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Activity |
- |
- |
- |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
Inhibition |
- |
- |
- |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
- |
- |
- |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
FC |
'=' |
1 |
- |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'>' |
95 |
% |
| Q9BJJ9 |
BXGT020099 |
Enoyl-ACP reductase |
unreviewed |
- |
FabI |
Inhibition |
'=' |
6 |
% |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
5 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
171400 |
nM |
| P21447 |
BXGT008651 |
ATP-dependent translocase ABCB1 |
reviewed |
- |
Abcb1a |
Delta Fmax |
'=' |
97 |
% |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
28183 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
7943 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
29849 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
1 |
- |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
KSV |
'=' |
1 |
10'5/M |
| Q6P7A9 |
BXGT016460 |
Lysosomal alpha-glucosidase |
reviewed |
- |
Gaa |
Inhibition |
'=' |
99 |
% |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
39810 |
nM |
| P98170 |
BXGT012231 |
E3 ubiquitin-protein ligase XIAP |
reviewed |
Enzyme modulator |
XIAP |
IC50 |
'>' |
100000 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
35481 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
196 |
% |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
IC50 |
'=' |
1000 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Ki |
'=' |
750 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
34 |
% |
| Q9NZ45 |
BXGT021269 |
CDGSH iron-sulfur domain-containing protein 1 |
reviewed |
- |
CISD1 |
IC50 |
'=' |
3100 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
280 |
% |
| Q9H0H5 |
BXGT020436 |
Rac GTPase-activating protein 1 |
reviewed |
Enzyme modulator |
RACGAP1 |
IC50 |
- |
44490 |
nM |
| Q6P7A9 |
BXGT016460 |
Lysosomal alpha-glucosidase |
reviewed |
- |
Gaa |
IC50 |
'=' |
59540 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
145 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
IC50 |
'=' |
20600 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
1995 |
nM |
| Q9BJJ9 |
BXGT020099 |
Enoyl-ACP reductase |
unreviewed |
- |
FabI |
IC50 |
- |
- |
- |
| Q15078 |
BXGT013534 |
Cyclin-dependent kinase 5 activator 1 |
reviewed |
Enzyme modulator |
CDK5R1 |
IC50 |
'=' |
51000 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
IC50 |
'=' |
51000 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
IC50 |
'=' |
9700 |
nM |
| Q8BRK8 |
BXGT017920 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
- |
Prkaa2 |
Activity |
- |
- |
- |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
21136 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
15848 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
9525 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
0 |
% |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
6309 |
nM |
| P29372 |
BXGT009336 |
DNA-3-methyladenine glycosylase |
reviewed |
Enzyme |
MPG |
Inhibition |
'=' |
25 |
% |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
99 |
nmol/min |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
25118 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
6200 |
nM |
| Q64725 |
BXGT016130 |
Tyrosine-protein kinase SYK |
reviewed |
- |
Syk |
Activity |
- |
- |
- |
| Q13332 |
BXGT013342 |
Receptor-type tyrosine-protein phosphatase S |
reviewed |
Enzyme |
PTPRS |
Inhibition |
'=' |
22 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
28183 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
'=' |
1050 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
'=' |
92800 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
4 |
- |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
50118 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Potency |
- |
74978 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
388900 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
IC50 |
'=' |
4000 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
5011 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
50 |
% |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
39810 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'<' |
1000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'<' |
1000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'<' |
1000 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Kq |
'=' |
1 |
10'12/M/s |
| P04040 |
BXGT006132 |
Catalase |
reviewed |
Enzyme |
CAT |
Activity |
'<=' |
95 |
% |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
79 |
nM |
| P03469 |
BXGT006080 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
42200 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
70000 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
100000 |
nM |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
25 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
78 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
17782 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
398107 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
IC50 |
- |
- |
- |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
10000 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
490 |
nM |