| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Inotropic effect |
'=' |
26 |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
6 |
nM |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Km |
'=' |
19400 |
nM |
| P23977 |
BXGT008936 |
Sodium-dependent dopamine transporter |
reviewed |
- |
Slc6a3 |
DA release |
'=' |
17 |
% |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
440 |
nM |
| P33535 |
BXGT009731 |
Mu-type opioid receptor |
reviewed |
- |
Oprm1 |
IC50 |
'=' |
3045 |
nM |
| P34975 |
BXGT009780 |
Kappa-type opioid receptor |
reviewed |
- |
Oprk1 |
IC50 |
'=' |
3045 |
nM |
| P33533 |
BXGT009729 |
Delta-type opioid receptor |
reviewed |
- |
Oprd1 |
IC50 |
'=' |
3045 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
251 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Kd |
'=' |
37000 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
EC50 |
'=' |
5000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
89125 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
3690 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Inhibition |
'=' |
83 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
2 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
2 |
nM |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
IC50 |
'=' |
2 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
2 |
nM |
| P25115 |
BXGT009024 |
D(1B) dopamine receptor |
reviewed |
- |
Drd5 |
IC50 |
'=' |
2 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
1 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
9 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
1100 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
57 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
36 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
51 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
15000 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Total binding inhibited |
'=' |
50 |
% |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Total binding inhibited |
'=' |
50 |
% |
| P21918 |
BXGT008708 |
D(1B) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD5 |
Total binding inhibited |
'=' |
50 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Total binding inhibited |
'=' |
50 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Total binding inhibited |
'=' |
50 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
1500 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5011 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
2350 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Log 1/Kd |
'=' |
-3 |
- |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
KL |
'=' |
4300 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ki |
'=' |
416 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
ED50 |
'=' |
3 |
uM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
High |
'=' |
31 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
35 |
nM |
| P21932 |
BXGT008709 |
Adenylate cyclase type 3 |
reviewed |
- |
Adcy3 |
EC50 |
'=' |
3500 |
nM |
| Q8CFM9 |
BXGT017933 |
Adenylyl cyclase 7 |
unreviewed |
- |
|
EC50 |
'=' |
3500 |
nM |
| P40146 |
BXGT010160 |
Adenylate cyclase type 8 |
reviewed |
- |
Adcy8 |
EC50 |
'=' |
3500 |
nM |
| Q03343 |
BXGT012709 |
Adenylate cyclase type 6 |
reviewed |
- |
Adcy6 |
EC50 |
'=' |
3500 |
nM |
| P26769 |
BXGT009133 |
Adenylate cyclase type 2 |
reviewed |
- |
Adcy2 |
EC50 |
'=' |
3500 |
nM |
| Q04400 |
BXGT012760 |
Adenylate cyclase type 5 |
reviewed |
- |
Adcy5 |
EC50 |
'=' |
3500 |
nM |
| P26770 |
BXGT009134 |
Adenylate cyclase type 4 |
reviewed |
- |
Adcy4 |
EC50 |
'=' |
3500 |
nM |
| D4A3N4 |
BXGT002921 |
Adenylate cyclase |
unreviewed |
- |
Adcy1 |
EC50 |
'=' |
3500 |
nM |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
'=' |
6 |
nM |
| P0DMM9 |
BXGT007504 |
Sulfotransferase 1A3 |
reviewed |
- |
SULT1A3 |
Activity |
- |
- |
- |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
22387 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
8 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
28183 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
724 |
nM |
| Q9HAW7 |
BXGT020508 |
UDP-glucuronosyltransferase 1-7 |
reviewed |
- |
UGT1A7 |
Activity |
'=' |
0 |
pm/min/mg |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
30131 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
470 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
4109 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ratio |
'=' |
31 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
8 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
Ki |
'=' |
101 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
3 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
2 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
89125 |
nM |
| Q3I4V7 |
BXGT014421 |
Carbonic anhydrase |
unreviewed |
- |
CAN2 |
KA |
'=' |
34 |
uM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
KA |
'=' |
9 |
uM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
2100 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
EC50 |
'=' |
1425 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
209 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
124 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
KA |
'=' |
13 |
uM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
KiL |
'=' |
3420 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
8 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
- |
- |
- |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
- |
- |
- |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
pD2 |
'=' |
7 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
100 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Intrinsic activity |
'=' |
100 |
nM |
| Q4Q090 |
BXGT014858 |
2,3-bisphosphoglycerate-independent phosphoglycerate mutase |
unreviewed |
- |
PGAM |
Potency |
- |
23934 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
Activity |
- |
- |
- |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
EC50 |
'=' |
1 |
nM |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
pD2 |
'=' |
5 |
- |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
pD2 |
'=' |
5 |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
pD2 |
'=' |
5 |
- |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
0 |
pm/min/mg |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
43 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
0 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
10000 |
nM |
| Q5AJ71 |
BXGT015288 |
Carbonic anhydrase |
reviewed |
- |
NCE103 |
KA |
'=' |
18 |
uM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
12000 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Emax |
'=' |
100 |
% |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
KA |
'=' |
30 |
uM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'>' |
10000 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'>' |
10000 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
9 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'>' |
1000 |
nM |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
'=' |
6400 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
843 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Inhibition |
'=' |
16 |
% |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
1258 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
3045 |
nM |
| P21918 |
BXGT008708 |
D(1B) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD5 |
Ki |
'=' |
2440 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
218 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio |
'=' |
400 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
'>' |
30000 |
nM |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
Ka |
'=' |
21 |
uM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
K Bind |
'=' |
0 |
uM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
K Bind |
'=' |
2 |
uM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Kd |
'=' |
17000 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
130 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
260 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
6309 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Inhibition |
'=' |
87 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Intrinsic activity |
'=' |
100 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
EC50 |
'=' |
3500 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
- |
- |
- |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
KL |
'=' |
580 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
1600 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
290 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
8912 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
79432 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ki |
'>' |
1000 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
11 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
1600 |
nM |
| P22909 |
BXGT008818 |
Alpha-2A adrenergic receptor |
reviewed |
- |
Adra2a |
Ki |
'=' |
58 |
nM |
| P19328 |
BXGT008473 |
Alpha-2B adrenergic receptor |
reviewed |
- |
Adra2b |
Ki |
'=' |
58 |
nM |
| P22086 |
BXGT008728 |
Alpha-2C adrenergic receptor |
reviewed |
- |
Adra2c |
Ki |
'=' |
58 |
nM |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Activity |
'>' |
10000 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
17 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
31622 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
51 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Inhibition |
'=' |
104 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
15 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
120 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
1062 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
ED20 |
'=' |
11 |
nM kg-1 |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
2 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
34 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Low |
'=' |
69 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Selectivity index |
'=' |
1 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Selectivity index |
'=' |
1 |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Km |
'=' |
280000 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
13 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
nH |
'=' |
0 |
- |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
3162 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
1600 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
39 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
3700 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ratio |
'=' |
1 |
- |
| P48039 |
BXGT010607 |
Melatonin receptor type 1A |
reviewed |
G-protein coupled receptor |
MTNR1A |
Ki |
'=' |
7100 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
1 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Kd |
'=' |
6200 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Inhibition |
'=' |
113 |
% |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Inhibition |
'=' |
110 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
1100 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
35481 |
nM |
| P53615 |
BXGT011003 |
Carbonic anhydrase |
reviewed |
- |
NCE103 |
Ka |
'=' |
13 |
uM |
| P23977 |
BXGT008936 |
Sodium-dependent dopamine transporter |
reviewed |
- |
Slc6a3 |
IC50 |
'=' |
200 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
- |
- |
- |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
KA |
'=' |
0 |
uM |
| O15245 |
BXGT004141 |
Solute carrier family 22 member 1 |
reviewed |
Transporter |
SLC22A1 |
Activity |
- |
- |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
12589 |
nM |
| P49286 |
BXGT010691 |
Melatonin receptor type 1B |
reviewed |
G-protein coupled receptor |
MTNR1B |
Ki |
'=' |
9100 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Inhibition |
- |
- |
- |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Km |
'=' |
330000 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
62 |
nM |
| Q16853 |
BXGT013683 |
Membrane primary amine oxidase |
reviewed |
- |
AOC3 |
Activity |
'=' |
0 |
% |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
0 |
pm/min/mg |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
3500 |
nM |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
EC50 |
'=' |
2 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
EC50 |
'=' |
8 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Efficacy |
'=' |
100 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
2200 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
7 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
EC50 |
'=' |
2 |
nM |
| Q6FTL6 |
BXGT016286 |
Carbonic anhydrase |
unreviewed |
- |
NCE103 |
Ka |
'=' |
27 |
uM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
1258 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
7940 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
501 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
843 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
3000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
8912 |
nM |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
KA |
'=' |
0 |
uM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
422 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Intrinsic activity |
'=' |
100 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
72 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'>' |
80000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
450 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
240 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
4 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Activity |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5173 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
124 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
467 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Kd |
'=' |
64560 |
nM |
| Q50565 |
BXGT014936 |
Carbonic anhydrase |
unreviewed |
- |
MTH_1582 |
Ka |
'=' |
51 |
uM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
1 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
4700 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
5 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
5340 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
5340 |
nM |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
IC50 |
'=' |
5340 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
5340 |
nM |
| P25115 |
BXGT009024 |
D(1B) dopamine receptor |
reviewed |
- |
Drd5 |
IC50 |
'=' |
5340 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Efficacy |
'=' |
100 |
% |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
Efficacy |
'=' |
100 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
7 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
Ki |
'=' |
49 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'>' |
10000 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
50 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Activity |
'=' |
19 |
% |
| P50130 |
BXGT010775 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
52 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ki |
'=' |
4400 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
650 |
nM |
| P21932 |
BXGT008709 |
Adenylate cyclase type 3 |
reviewed |
- |
Adcy3 |
Activity |
'=' |
150 |
% |
| Q8CFM9 |
BXGT017933 |
Adenylyl cyclase 7 |
unreviewed |
- |
|
Activity |
'=' |
150 |
% |
| P40146 |
BXGT010160 |
Adenylate cyclase type 8 |
reviewed |
- |
Adcy8 |
Activity |
'=' |
150 |
% |
| Q03343 |
BXGT012709 |
Adenylate cyclase type 6 |
reviewed |
- |
Adcy6 |
Activity |
'=' |
150 |
% |
| P26769 |
BXGT009133 |
Adenylate cyclase type 2 |
reviewed |
- |
Adcy2 |
Activity |
'=' |
150 |
% |
| Q04400 |
BXGT012760 |
Adenylate cyclase type 5 |
reviewed |
- |
Adcy5 |
Activity |
'=' |
150 |
% |
| P26770 |
BXGT009134 |
Adenylate cyclase type 4 |
reviewed |
- |
Adcy4 |
Activity |
'=' |
150 |
% |
| D4A3N4 |
BXGT002921 |
Adenylate cyclase |
unreviewed |
- |
Adcy1 |
Activity |
'=' |
150 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Intrinsic activity |
'=' |
100 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'=' |
103 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
'=' |
15 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
'=' |
15 |
nM |
| P21918 |
BXGT008708 |
D(1B) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD5 |
IC50 |
'=' |
15 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
'=' |
15 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
'=' |
15 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Activity |
'=' |
439 |
/s |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Intrinsic activity |
'=' |
100 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
5340 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
240 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
28183 |
nM |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
2100000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
102 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
14125 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
6294 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
1584 |
nM |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
'=' |
460 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ratio |
'=' |
9 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio |
'=' |
9 |
- |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
4300 |
nM |
| P23977 |
BXGT008936 |
Sodium-dependent dopamine transporter |
reviewed |
- |
Slc6a3 |
Ki |
'>' |
5000 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
K bind |
'=' |
150 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Displacement |
- |
- |
- |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
200 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
0 |
pm/min/mg |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
1860 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
3260 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Activity |
'>' |
75 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
192 |
nM |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Ki |
'=' |
603000 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
15848 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
31622 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
1700 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
18200 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
97 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
64 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
64 |
nM |
| O95622 |
BXGT005386 |
Adenylate cyclase type 5 |
reviewed |
- |
ADCY5 |
Response |
'=' |
100 |
% |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
39810 |
nM |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
KA |
'=' |
27 |
uM |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
KA |
'=' |
7 |
uM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ki |
'=' |
150 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
18 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
EC50 |
'=' |
3 |
- |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
26121 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
15848 |
nM |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
EC50 |
'=' |
2 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Efficacy |
'=' |
100 |
% |
| P21932 |
BXGT008709 |
Adenylate cyclase type 3 |
reviewed |
- |
Adcy3 |
Cyclase stimulation |
'=' |
58 |
% |
| Q8CFM9 |
BXGT017933 |
Adenylyl cyclase 7 |
unreviewed |
- |
|
Cyclase stimulation |
'=' |
58 |
% |
| P40146 |
BXGT010160 |
Adenylate cyclase type 8 |
reviewed |
- |
Adcy8 |
Cyclase stimulation |
'=' |
58 |
% |
| Q03343 |
BXGT012709 |
Adenylate cyclase type 6 |
reviewed |
- |
Adcy6 |
Cyclase stimulation |
'=' |
58 |
% |
| P26769 |
BXGT009133 |
Adenylate cyclase type 2 |
reviewed |
- |
Adcy2 |
Cyclase stimulation |
'=' |
58 |
% |
| Q04400 |
BXGT012760 |
Adenylate cyclase type 5 |
reviewed |
- |
Adcy5 |
Cyclase stimulation |
'=' |
58 |
% |
| P26770 |
BXGT009134 |
Adenylate cyclase type 4 |
reviewed |
- |
Adcy4 |
Cyclase stimulation |
'=' |
58 |
% |
| D4A3N4 |
BXGT002921 |
Adenylate cyclase |
unreviewed |
- |
Adcy1 |
Cyclase stimulation |
'=' |
58 |
% |
| Q99N23 |
BXGT019994 |
Carbonic anhydrase 15 |
reviewed |
- |
Ca15 |
KA |
'=' |
7 |
uM |
| P29276 |
BXGT009329 |
Adenosine receptor A2b |
reviewed |
- |
Adora2b |
Ki |
'=' |
977 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
1900 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Inhibition |
'=' |
92 |
% |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Inhibition |
'=' |
151 |
% |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
12000000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
572 |
nM |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
'>' |
1100000 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
'>' |
100000 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
8 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Kd |
'=' |
267000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
nH |
'=' |
0 |
- |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Activity |
- |
- |
- |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
KA |
'=' |
0 |
uM |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Activity |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
6 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Kd |
'=' |
49000 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IA |
'=' |
100 |
% |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
2300000 |
nM |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
8087 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio |
'=' |
8 |
- |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
800 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
26854 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
1520 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
150000 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
150000 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
1700 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
1700 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
nH |
'=' |
0 |
- |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
15 |
nM |
| O70127 |
BXGT005057 |
Bile salt export pump |
reviewed |
- |
Abcb11 |
IC50 |
'>' |
1000000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'=' |
18 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
34 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
20 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
20 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
42 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
483 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
483 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
759 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
1200 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
'=' |
90000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
IC50 |
'=' |
90000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
'=' |
90000 |
nM |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
pD2 |
'=' |
4 |
- |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
pD2 |
'=' |
4 |
- |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
pD2 |
'=' |
4 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
190 |
nM |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1778 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IA |
'=' |
100 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
2 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
IC50 |
'=' |
2 |
nM |
| P30729 |
BXGT009461 |
D(4) dopamine receptor |
reviewed |
- |
Drd4 |
IC50 |
'=' |
2 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
2 |
nM |
| P25115 |
BXGT009024 |
D(1B) dopamine receptor |
reviewed |
- |
Drd5 |
IC50 |
'=' |
2 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
8000 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
3380 |
nM |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
KA |
'=' |
14 |
uM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
296 |
nM |
| O15245 |
BXGT004141 |
Solute carrier family 22 member 1 |
reviewed |
Transporter |
SLC22A1 |
Activity |
'=' |
487 |
uM |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Km |
'=' |
520000 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
EC50 |
'=' |
10 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Ki |
'=' |
347000 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
22387 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
891 |
nM |
| Q8BW75 |
BXGT017924 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
Maob |
Activity |
- |
- |
- |
| O15245 |
BXGT004141 |
Solute carrier family 22 member 1 |
reviewed |
Transporter |
SLC22A1 |
Inhibition |
'=' |
11 |
% |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
Ki |
'=' |
7 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Kb |
'=' |
2350 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
'=' |
0 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Kd |
'=' |
2500 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
10 |
% |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
293 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio Ki |
'=' |
724 |
- |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
104 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
'=' |
61000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
8 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
170 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
446 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
110 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Inhibition |
'=' |
95 |
% |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
'=' |
14000 |
nM |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Ki |
'=' |
14000 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
'=' |
14000 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
'=' |
10000 |
nM |
| P54833 |
BXGT011086 |
Beta-2 adrenergic receptor |
reviewed |
- |
ADRB2 |
Ki |
'=' |
50000 |
nM |
| Q712U5 |
BXGT016689 |
cAMP-regulated phosphoprotein 19 |
reviewed |
- |
Arpp19 |
EC50 |
'=' |
3500 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
5 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
K0.5 |
'=' |
267 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
K0.5 |
'=' |
36 |
nM |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ka |
'=' |
33 |
uM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
EC50 |
'=' |
5 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
156 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Ki |
'=' |
309 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
100 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
510 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
510 |
nM |
| P35368 |
BXGT009822 |
Alpha-1B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1B |
Ki |
'=' |
2511 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
'=' |
2511 |
nM |
| P35348 |
BXGT009814 |
Alpha-1A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1A |
Ki |
'=' |
2511 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
617 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
990 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
89125 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
4 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
4 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
IC50 |
'=' |
3 |
nM |
| Q95136 |
BXGT019575 |
D(1A) dopamine receptor |
reviewed |
- |
DRD1 |
IC50 |
'=' |
3 |
nM |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Km |
'=' |
51000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
227 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
IC50 |
'=' |
62000 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
pEC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
6 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
23280 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Activity |
'>' |
75 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
%max |
'=' |
106 |
% |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
582 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
582 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Activity |
'=' |
100 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
35481 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
65 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
21 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
20 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
5 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio |
'=' |
8 |
- |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
14125 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
226 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
KA |
'=' |
0 |
uM |
| P16662 |
BXGT008253 |
UDP-glucuronosyltransferase 2B7 |
reviewed |
- |
UGT2B7 |
Activity |
'=' |
0 |
pm/min/mg |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Km |
'=' |
390000 |
nM |
| Q9Z0E8 |
BXGT022397 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Activity |
'=' |
70 |
% |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
8 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
log(activity) |
'=' |
0 |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
'>' |
28000 |
nM |
| P20288 |
BXGT008560 |
D(2) dopamine receptor |
reviewed |
- |
DRD2 |
Ki |
'=' |
14 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
Ki |
'=' |
11 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
360 |
nM |
| Q64133 |
BXGT016109 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
Maoa |
Activity |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
82 |
nM |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'>' |
1000000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
96 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio EC50 |
'=' |
2 |
- |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
650000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
0 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'=' |
101 |
% |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
IC50 |
'=' |
111 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
4470 |
nM |
| P40881 |
BXGT010205 |
Carbonic anhydrase |
reviewed |
- |
|
KA |
'=' |
54 |
uM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Activity |
- |
- |
- |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
IC50 |
'=' |
3140 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
IC50 |
'=' |
3000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
31622 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
1 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
100 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
Ki |
'=' |
197 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'=' |
101 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
KiH |
'=' |
58 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
pKA |
'=' |
7 |
- |
| P50225 |
BXGT010781 |
Sulfotransferase 1A1 |
reviewed |
- |
SULT1A1 |
Activity |
- |
- |
- |
| O43704 |
BXGT004615 |
Sulfotransferase family cytosolic 1B member 1 |
reviewed |
- |
SULT1B1 |
Activity |
- |
- |
- |
| O70594 |
BXGT005072 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Inhibition |
- |
- |
- |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
31622 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
183 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
1584 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
36 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
IC50 |
'=' |
384000 |
nM |
| O70423 |
BXGT005066 |
Membrane primary amine oxidase |
reviewed |
- |
Aoc3 |
Activity |
'=' |
0 |
% |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Activity |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
48 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
%max |
'=' |
100 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Emax |
'=' |
97 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
113 |
% |
| P54803 |
BXGT011082 |
Galactocerebrosidase |
reviewed |
- |
GALC |
Potency |
- |
4466 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
0 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
92 |
% |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
pEC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
97 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
'=' |
16 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ratio |
'=' |
8 |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
93 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
390 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
10 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18837 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
87 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
%max |
'=' |
100 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
2 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
7 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
31622 |
nM |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
IC50 |
'=' |
2300000 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
200 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
3 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
163 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'>' |
75 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
4 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
Activity |
'=' |
60 |
% |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
2 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
90 |
% |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
EC50 |
'=' |
12 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
115 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
'=' |
232 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
'=' |
2 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
160 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
0 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Activity |
'=' |
100 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
EC50 |
'=' |
19 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Emax |
'=' |
95 |
% |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
'=' |
243 |
nM |
| Q4CVY4 |
BXGT026093 |
Carbonic anhydrase-like protein, putative |
unreviewed |
- |
Tc00.1047053509597.20 |
KA |
'>' |
100 |
uM |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
EC50 |
'=' |
91 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Activity |
'=' |
86 |
% |