Showing entry for Serotonin



                             
General Compound Information
BXGC IdBXGC0005867
Compound NameSerotonin
Structure
FormulaC10H12N2O
InchiKeyQZAYGJVTTNCVMB-UHFFFAOYSA-N
SMILESNCCC1=CNC2=CC=C(O)C=C12
InchiInChI=1S/C10H12N2O/c11-4-3-7-6-12-10-2-1-8(13)5-9(7)10/h1-2,5-6,12-13H,3-4,11H2
IUPAC3-(2-aminoethyl)-1H-indol-5-ol
Molecular Weight176.22
Pubchem Id5202
Chembl IdCHEMBL39
Targets of Information Source
DrugBank DB08839
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
P31645 BXGT009558 Sodium-dependent serotonin transporter reviewed Transporter SLC6A4 investigational; nutraceutical -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A investigational; nutraceutical -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A investigational; nutraceutical -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B investigational; nutraceutical -
Q05940 BXGT012846 Synaptic vesicular amine transporter reviewed Transporter SLC18A2 investigational; nutraceutical -
PDB SRO
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Q9BIH3 BXGT020097 D7-related 4 protein unreviewed d7r4 - - - 2.4 -
Q8WSF8 BXGT018982 Soluble acetylcholine receptor unreviewed - - - 693000 -
P37231 BXGT009972 Peroxisome proliferator-activated receptor gamma reviewed PPARG Nuclear receptor - - 933000 -
Q09JR9 BXGT013045 Lipocalin unreviewed - - - <2 -
Q93NH4 BXGT019514 6-hydroxy-L-nicotine oxidase unreviewed 6-hlno - - - - -
Q5WPU9 BXGT015901 43.2 kDa salivary protein unreviewed LJM11_Clu9 - - - - -
P14779 BXGT008052 Bifunctional cytochrome P450/NADPH--P450 reductase reviewed cyp102A1 - - - 80000 -
P14779 BXGT008052 Bifunctional cytochrome P450/NADPH--P450 reductase reviewed cyp102A1 - - - 700 -
P14779 BXGT008052 Bifunctional cytochrome P450/NADPH--P450 reductase reviewed cyp102A1 - - - 3300 -
P01308 BXGT005749 Insulin reviewed INS - - - 3340000 -
P01308 BXGT005749 Insulin reviewed INS - - - 3120000 -
P01308 BXGT005749 Insulin reviewed INS - - - - -
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed Htr3a - - - - -
Q6ZJK7 BXGT024646 Tryptophan decarboxylase 1 reviewed TDC1 - - - - -
P00760 BXGT005644 Cationic trypsin reviewed - - - - -
Binding DB 10755
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 1049 - - 12
reviewed BXGT008187 Ribosyldihydronicotinamide dehydrogenase [quinone] reviewed NQO2 - 53900 - -
reviewed BXGT010360 Alpha-1A adrenergic receptor reviewed Adra1a 18000 - - -
reviewed BXGT010360 Alpha-1A adrenergic receptor reviewed Adra1a 23000 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 0.59 - - -
reviewed BXGT009486 5-hydroxytryptamine receptor 5A reviewed Htr5a 251.18 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 11 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 3.9 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 4.3 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 8.9 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 2.1 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 14 - - -
reviewed BXGT008708 D(1B) dopamine receptor reviewed G-protein coupled receptor DRD5 3000 - - -
reviewed BXGT008440 D(1A) dopamine receptor reviewed Drd1 5000 - - -
reviewed BXGT011367 D(2) dopamine receptor reviewed Drd2 >10000 - - -
reviewed BXGT008936 Sodium-dependent dopamine transporter reviewed Slc6a3 >10000 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 3.5 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 3 - - -
reviewed BXGT008728 Alpha-2C adrenergic receptor reviewed Adra2c >10000 - - -
reviewed BXGT026172 D(2) dopamine receptor reviewed DRD2 >10000 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 46.77 - - -
reviewed BXGT011367 D(2) dopamine receptor reviewed Drd2 1655 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 270 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 83 - - -
reviewed BXGT026170 5-hydroxytryptamine receptor 7 reviewed HTR7 1 - - -
reviewed BXGT010691 Melatonin receptor type 1B reviewed G-protein coupled receptor MTNR1B >10000 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 63.09 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 125.89 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 0.79 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b 10 - - -
reviewed BXGT026170 5-hydroxytryptamine receptor 7 reviewed HTR7 1.34 - - -
reviewed BXGT026170 5-hydroxytryptamine receptor 7 reviewed HTR7 0.25 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 151 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 56 - - -
reviewed BXGT009819 5-hydroxytryptamine receptor 5A reviewed Htr5a 1333 - - -
reviewed BXGT009820 5-hydroxytryptamine receptor 5B reviewed Htr5b 239 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 145 - - -
reviewed BXGT010608 Melatonin receptor type 1A reviewed MTNR1A >10000 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 0.26 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 1.25 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 12.58 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 0.79 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 3.98 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 102.32 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 15.84 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 4.26 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 1.09 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 3.98 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 0.57 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 15.84 - - -
reviewed BXGT009254 5-hydroxytryptamine receptor 1B reviewed Htr1b 39.81 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 5.24 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 3.01 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 0.57 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 8.91 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 2.08 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 3.89 - - -
reviewed BXGT009273 5-hydroxytryptamine receptor 1D reviewed Htr1d 2.51 - - -
reviewed BXGT007730 5-hydroxytryptamine receptor 1D reviewed HTR1D 5.01 - - -
reviewed BXGT007730 5-hydroxytryptamine receptor 1D reviewed HTR1D 15.84 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 10.96 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 7.24 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 6.16 - - -
reviewed BXGT012647 5-hydroxytryptamine receptor 1F reviewed Htr1f 125.89 - - -
reviewed BXGT009484 5-hydroxytryptamine receptor 1F reviewed Htr1f 67.6 - - -
reviewed BXGT009483 5-hydroxytryptamine receptor 1F reviewed G-protein coupled receptor HTR1F 10 - - -
reviewed BXGT009483 5-hydroxytryptamine receptor 1F reviewed G-protein coupled receptor HTR1F >10000 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 5.75 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 1.99 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 12.02 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 602.55 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 478.63 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 707.94 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 251.18 - - -
reviewed BXGT012637 5-hydroxytryptamine receptor 2B reviewed Htr2b 1258.92 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b 28.18 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b 10.23 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 0.7 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 22.9 - - -
reviewed BXGT008938 5-hydroxytryptamine receptor 3A reviewed Htr3a 269.15 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 79.43 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 50.11 - - -
reviewed BXGT009819 5-hydroxytryptamine receptor 5A reviewed Htr5a 239.88 - - -
reviewed BXGT009531 5-hydroxytryptamine receptor 5B reviewed Htr5b 251.18 - - -
reviewed BXGT009820 5-hydroxytryptamine receptor 5B reviewed Htr5b 1318.25 - - -
reviewed BXGT009820 5-hydroxytryptamine receptor 5B reviewed Htr5b 7.76 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 151.35 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 56.23 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 1.81 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 4.89 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 8.12 - - -
reviewed BXGT009620 5-hydroxytryptamine receptor 7 reviewed Htr7 5.01 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 1.51 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 25.11 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 0.6 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 9.8 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b 10.2 - - -
reviewed BXGT021415 5-hydroxytryptamine receptor 6 reviewed Htr6 39.81 - - -
reviewed BXGT009820 5-hydroxytryptamine receptor 5B reviewed Htr5b 7.8 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 200 - - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 56 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 8.1 - - -
reviewed BXGT005060 5-hydroxytryptamine receptor 3A reviewed HTR3A >10000 - - -
reviewed BXGT005060 5-hydroxytryptamine receptor 3A reviewed HTR3A 495 - - -
reviewed BXGT011367 D(2) dopamine receptor reviewed Drd2 7950 - - -
reviewed BXGT012624 Sodium-dependent dopamine transporter reviewed Transporter SLC6A3 >10000 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 1.83 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 1.52 - - -
reviewed BXGT021415 5-hydroxytryptamine receptor 6 reviewed Htr6 5.01 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 134 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 5 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 102.3 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 656 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 2955 - - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 65 - - -
reviewed BXGT009486 5-hydroxytryptamine receptor 5A reviewed Htr5a 1100 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 4.2 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 3 - - -
reviewed BXGT009273 5-hydroxytryptamine receptor 1D reviewed Htr1d 18 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 7.77 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 9.46 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b 11.3 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 15.5 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 6.3 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 316.22 - - -
reviewed BXGT026171 5-hydroxytryptamine receptor 4 reviewed Htr4 79.43 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 2.6 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 2.3 - - -
reviewed BXGT026171 5-hydroxytryptamine receptor 4 reviewed Htr4 56.23 - - -
reviewed BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 >10000 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 2 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 7.94 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 0.63 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 7.94 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 0.4 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 218.77 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 120.22 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 1.17 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 56.23 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 87.09 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 7.94 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 125.89 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 199.52 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 12.58 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 234.42 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 0.38 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 7.94 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 3.98 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 38 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 9 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 3.4 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 158.48 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 39.81 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 56.23 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 38.9 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 0.12 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 1151 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 481.9 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 330 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 1.3 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 96 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 44 - - -
reviewed BXGT008938 5-hydroxytryptamine receptor 3A reviewed Htr3a 292 - - -
reviewed BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 >10000 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 6.31 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 4.07 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 3.38 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 11 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 159 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 0.13 - - -
reviewed BXGT026170 5-hydroxytryptamine receptor 7 reviewed HTR7 0.1 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 30.9 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 2.09 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 5.75 - - -
reviewed BXGT004042 5-hydroxytryptamine receptor 1B reviewed HTR1B 2.51 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 341 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 251.18 - - -
reviewed BXGT008936 Sodium-dependent dopamine transporter reviewed Slc6a3 2703 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 4 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 12.2 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 2.9 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 158.5 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 100 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 18.2 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 1 - - -
reviewed BXGT021415 5-hydroxytryptamine receptor 6 reviewed Htr6 95.5 - - -
reviewed BXGT009532 5-hydroxytryptamine receptor 6 reviewed Htr6 79.43 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 21 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 19 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 2.4 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 16.22 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 13.49 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 90 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 3 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 1.2 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 10 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 - - - 5
reviewed BXGT015984 5-hydroxytryptamine receptor 1D reviewed HTR1D - - - 8.5
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D - 3 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 10
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B - 5 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - 5.2 - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c - 81 - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 - - - 17
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a 87 - - -
reviewed BXGT016110 5-hydroxytryptamine receptor 1A reviewed Htr1a - 5 - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 10 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 3 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 2 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 5 - - -
reviewed BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E 4 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - 81 - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B - - - 30
reviewed BXGT015984 5-hydroxytryptamine receptor 1D reviewed HTR1D - - - 16
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - 5.2 - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b - 5 - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 1.5
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 1.7
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - 6 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 2.8 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - 2 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - 5.6 - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 5.4 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 1.7 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 930 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 7.8 - - -
reviewed BXGT009273 5-hydroxytryptamine receptor 1D reviewed Htr1d - - - 5.2
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - - - 10
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 230 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 6.8 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - 20 - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 20 - -
reviewed BXGT015984 5-hydroxytryptamine receptor 1D reviewed HTR1D - 3 - -
reviewed BXGT009273 5-hydroxytryptamine receptor 1D reviewed Htr1d - 3 - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 4 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 510 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c 23 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 5.5 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 1.7 - - -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a 320 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 1.7 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 5.06 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 2.48 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B - - - 4.82
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - 3 - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 1.4 - - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 33 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 0.8 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 2.5 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 5.1 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B - - - 4.7
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 2 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 1
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 0.94 - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 75 - - -
reviewed BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 - >50 - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 78 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 320 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 130 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 4 - - -
reviewed BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A 126 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 160 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 150 - - -
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 120 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 3
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 11
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 14 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 12 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 6.9 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - - - 17
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - - 4 -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 2.1 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 0.92
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 0.21
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 1.9
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 0.5
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - - - 58
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 8.2 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 8.3 - - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c - - - 2.8
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B 13 - - -
reviewed BXGT009493 5-hydroxytryptamine receptor 2B reviewed Htr2b - - - 3.5
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 0.7
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 28
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 170
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 302
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 191
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 690 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 20 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 500 - - -
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 7.33 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 0.5 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 1.1 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 3 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - - - 323
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 0.09
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 0.5
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 5.8
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - - - 15
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 1.6 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 1258 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 100 - - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 - 3.7 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 43
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - 2.5 - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 - 1.2 - -
reviewed BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A - 1.8 - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b - 4.9 - -
reviewed BXGT010691 Melatonin receptor type 1B reviewed G-protein coupled receptor MTNR1B >100000 - - -
reviewed BXGT010607 Melatonin receptor type 1A reviewed G-protein coupled receptor MTNR1A >100000 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - 2.55 - -
reviewed BXGT007687 Tyrosinase reviewed Tyr - 550000 - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 6 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 - - - 5.8
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 25
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 11
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 47
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 15
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 - 27.5 - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 - - - 6.3
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 37 - - -
reviewed BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R - >50 - -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - >50 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - >50 - -
reviewed BXGT021317 Isocitrate lyase reviewed ICL1 - 301000 - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 6 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 560 - - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 2950 - - -
reviewed BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A - - - 141
reviewed BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A - - - 178
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 977 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 3.5 - - -
reviewed BXGT009818 5-hydroxytryptamine receptor 2A reviewed Htr2a 500 - - -
reviewed BXGT009818 5-hydroxytryptamine receptor 2A reviewed Htr2a - 680 - -
reviewed BXGT008938 5-hydroxytryptamine receptor 3A reviewed Htr3a 361 - - -
reviewed BXGT004563 Polyphenol oxidase 2 reviewed PPO2 - >350000 - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 950 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b - - - 26
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 4600 - -
reviewed BXGT015984 5-hydroxytryptamine receptor 1D reviewed HTR1D - - - 5.2
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 3600 - -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a 390 - - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - 3162 -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D - - 13 -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c - - 32 -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - 3.2 -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a - - - 12000
reviewed BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 - 0.0003 - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 35 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 25 - - -
reviewed BXGT008448 D(3) dopamine receptor reviewed Drd3 2338 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 4.3 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 2.5 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 2.1 - - -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a 66 - - -
reviewed BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D 4.8 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 7.1 - - -
reviewed BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 - - 9690 -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a - 2.6 - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 - 147 - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 2350 - -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a - 727 - -
reviewed BXGT006838 5-hydroxytryptamine receptor 2C reviewed Htr2c - 42 - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b - 4.6 - -
reviewed BXGT016041 5-hydroxytryptamine receptor 4 reviewed Htr4 187 - - -
reviewed BXGT009849 5-hydroxytryptamine receptor 3A reviewed Htr3a 120 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 7.3 - - -
reviewed BXGT009272 5-hydroxytryptamine receptor 1B reviewed Htr1b 1.1 - - -
reviewed BXGT009565 Sodium-dependent serotonin transporter reviewed Slc6a4 740 - - -
reviewed BXGT009483 5-hydroxytryptamine receptor 1F reviewed G-protein coupled receptor HTR1F - - - 7.9
reviewed BXGT009621 5-hydroxytryptamine receptor 7 reviewed Htr7 10 - - -
reviewed BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A 250 - - -
reviewed BXGT009486 5-hydroxytryptamine receptor 5A reviewed Htr5a 150 - - -
reviewed BXGT009835 D(3) dopamine receptor reviewed G-protein coupled receptor DRD3 - - - 523
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - - - 55.8
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - 1.2 - -
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - - - 351
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a - 0.9 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 3.7
reviewed BXGT008059 5-hydroxytryptamine receptor 2A reviewed Htr2a 0.3 - - -
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 4.8 - - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 100 - - -
reviewed BXGT007506 Adenosine receptor A3 reviewed G-protein coupled receptor ADORA3 - 79 - -
reviewed BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A - - - 457
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 24
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 5.8
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 70
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 - - - 100
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A 130 - - -
reviewed BXGT021317 Isocitrate lyase reviewed ICL1 - 301300 - -
reviewed BXGT008938 5-hydroxytryptamine receptor 3A reviewed Htr3a - - - 3400
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 150
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 147
reviewed BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B 14 - - -
reviewed BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A 170 - - -
reviewed BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 0.13 - - -
reviewed BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 84 - - -
reviewed BXGT008472 5-hydroxytryptamine receptor 1A reviewed Htr1a 2.6 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 214 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 1.63
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 445 - - -
reviewed BXGT008837 Prostaglandin G/H synthase 1 reviewed Enzyme PTGS1 - >400000 - -
reviewed BXGT009816 Prostaglandin G/H synthase 2 reviewed Enzyme PTGS2 - >400000 - -
reviewed BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B - - - 0.86
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 7.6
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 0.62 - - -
reviewed BXGT011863 5-hydroxytryptamine receptor 1D (Fragment) reviewed HTR1D - 10 - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 10000 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 29.51 - - -
reviewed BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 109.65 - - -
reviewed BXGT005068 5-hydroxytryptamine receptor 4 reviewed HTR4 - - - 10
reviewed BXGT016060 Solute carrier family 22 member 1 reviewed Slc22a1 390000 - - -
reviewed BXGT021408 Solute carrier family 22 member 2 reviewed Slc22a2 242000 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 0.87
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 2.6
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C 79 - - -
reviewed BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C - - - 44
reviewed BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A - - - 150
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A 0.9 - - -
reviewed BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A - - - 3.8
CHEMBL CHEMBL39
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 1258 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B EC50 '=' 30 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 8 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Intrinsic activity '=' 1 -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 120 nM
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 AC50 - - -
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Kd '=' 9690 nM
P30939 BXGT009483 5-hydroxytryptamine receptor 1F reviewed G-protein coupled receptor HTR1F EC50 '=' 7 nM
P35462 BXGT009835 D(3) dopamine receptor reviewed G-protein coupled receptor DRD3 EC50 '=' 523 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 8 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 4 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Efficacy '=' 98 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 11 nM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Inhibition - - -
Q9P8Q7 BXGT021317 Isocitrate lyase reviewed - ICL1 IC50 '=' 301000 nM
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 66 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 66 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A pD2 '=' 7 -
P28565 BXGT009273 5-hydroxytryptamine receptor 1D reviewed - Htr1d IC50 '=' 5 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 5 nM
P30940 BXGT009484 5-hydroxytryptamine receptor 1F reviewed - Htr1f IC50 '=' 5 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b IC50 '=' 5 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Activity '=' 100 %
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Emax '=' 100 %
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 Activity '=' 1 -
P19224 BXGT008468 UDP-glucuronosyltransferase 1-6 reviewed - UGT1A6 Activity - - -
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Activity '=' 99 %
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 2 nM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Ki - - -
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Emax - - -
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 EC50 - - -
P07451 BXGT006627 Carbonic anhydrase 3 reviewed - CA3 KA '=' 0 uM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 30600 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 Ki '=' 100 nM
P31652 BXGT009565 Sodium-dependent serotonin transporter reviewed - Slc6a4 Activity - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 2 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 Ki - - -
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D ED50 '=' 1 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 1 nM
Q9Z0E8 BXGT022397 Solute carrier family 22 member 5 reviewed - Slc22a5 Activity '=' 51 %
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 AC50 - - -
P22303 BXGT008751 Acetylcholinesterase reviewed Enzyme ACHE IC50 - - -
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 Potency '=' 15848 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 1 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 5 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IA '=' 1 -
P23280 BXGT008844 Carbonic anhydrase 6 reviewed - CA6 KA '=' 19 uM
P00918 BXGT005690 Carbonic anhydrase 2 reviewed - CA2 KA '=' 50 uM
Q63089 BXGT016060 Solute carrier family 22 member 1 reviewed - Slc22a1 Km '=' 37600 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 0 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Emax '=' 91 %
O97447 BXGT005436 Putative fructose-1,6-bisphosphate aldolase unreviewed - ald Potency '=' 15811 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Emax '=' 100 %
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 Ki '=' 1049 nM
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 EC50 '=' 12 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IC50 '=' 29 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 120 nM
P28565 BXGT009273 5-hydroxytryptamine receptor 1D reviewed - Htr1d EC50 '=' 5 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Emax '=' 100 %
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 93 nM
P00915 BXGT005689 Carbonic anhydrase 1 reviewed - CA1 KA '=' 45 uM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Activity - - -
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 23 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C IC50 '=' 81 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 43 nM
O43570 BXGT004601 Carbonic anhydrase 12 reviewed - CA12 KA '=' 0 uM
Q9S446 BXGT021560 Class A sortase SrtA unreviewed - srtA IC50 '>' 100 ug.mL-1
Q9R0W2 BXGT021408 Solute carrier family 22 member 2 reviewed - Slc22a2 Ki '=' 242000 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Max '=' 100 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 1 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 6 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 1 nM
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 Ki '=' 109 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 2 nM
P14679 BXGT008039 Tyrosinase reviewed Enzyme TYR Activity '=' 15 %
P16662 BXGT008253 UDP-glucuronosyltransferase 2B7 reviewed - UGT2B7 Activity '=' 0 pm/min/mg
P06133 BXGT006414 UDP-glucuronosyltransferase 2B4 reviewed - UGT2B4 Activity '=' 0 pm/min/mg
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 13000 nM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Imax - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 320 nM
Q3I4V7 BXGT014421 Carbonic anhydrase unreviewed - CAN2 KA '=' 46 uM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IC50 '=' 16 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 5 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 - - -
Q5AJ71 BXGT015288 Carbonic anhydrase reviewed - NCE103 KA '=' 28 uM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 - - -
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 20900 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 5100 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 1 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 1 nM
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 Activity '=' 99 %
P22748 BXGT008802 Carbonic anhydrase 4 reviewed - CA4 Ka '=' 3 uM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 18 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 180 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 170000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 90000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 63000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 15000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 140000 nM
Q99N23 BXGT019994 Carbonic anhydrase 15 reviewed - Ca15 KA '=' 7 uM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Activity - - -
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 11 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 2350 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 7 nM
Q16445 BXGT013629 Gamma-aminobutyric acid receptor subunit alpha-6 reviewed Ion channel GABRA6 IC50 - - -
P31644 BXGT009557 Gamma-aminobutyric acid receptor subunit alpha-5 reviewed Ion channel GABRA5 IC50 - - -
P47869 BXGT010590 Gamma-aminobutyric acid receptor subunit alpha-2 reviewed Ion channel GABRA2 IC50 - - -
P78334 BXGT011834 Gamma-aminobutyric acid receptor subunit epsilon reviewed Ion channel GABRE IC50 - - -
P18505 BXGT008409 Gamma-aminobutyric acid receptor subunit beta-1 reviewed Ion channel GABRB1 IC50 - - -
Q8N1C3 BXGT018498 Gamma-aminobutyric acid receptor subunit gamma-1 reviewed Ion channel GABRG1 IC50 - - -
O14764 BXGT004094 Gamma-aminobutyric acid receptor subunit delta reviewed Ion channel GABRD IC50 - - -
O00591 BXGT003939 Gamma-aminobutyric acid receptor subunit pi reviewed Ion channel GABRP IC50 - - -
P34903 BXGT009769 Gamma-aminobutyric acid receptor subunit alpha-3 reviewed Ion channel GABRA3 IC50 - - -
Q9UN88 BXGT021783 Gamma-aminobutyric acid receptor subunit theta reviewed Ion channel GABRQ IC50 - - -
Q99928 BXGT019975 Gamma-aminobutyric acid receptor subunit gamma-3 reviewed Ion channel GABRG3 IC50 - - -
P48169 BXGT010622 Gamma-aminobutyric acid receptor subunit alpha-4 reviewed Ion channel GABRA4 IC50 - - -
P28472 BXGT009260 Gamma-aminobutyric acid receptor subunit beta-3 reviewed Ion channel GABRB3 IC50 - - -
P18507 BXGT008411 Gamma-aminobutyric acid receptor subunit gamma-2 reviewed Ion channel GABRG2 IC50 - - -
P47870 BXGT010591 Gamma-aminobutyric acid receptor subunit beta-2 reviewed Ion channel GABRB2 IC50 - - -
P14867 BXGT008061 Gamma-aminobutyric acid receptor subunit alpha-1 reviewed Ion channel GABRA1 IC50 - - -
P11344 BXGT007687 Tyrosinase reviewed - Tyr IC50 '=' 550000 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 21192 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Ki '=' 13 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Activity '=' 100 %
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 1 nM
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Intrinsic activity - - -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Intrinsic activity - - -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Intrinsic activity - - -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Intrinsic activity - - -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Intrinsic activity - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 2 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 '=' 5 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 3600 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 3600 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b IC50 '=' 3600 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 2 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 1 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 37000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 4400 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 49000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 6200 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 1300 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B EC50 '=' 4 nM
P31652 BXGT009565 Sodium-dependent serotonin transporter reviewed - Slc6a4 Ki '=' 740 nM
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 120 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 120 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D IC50 '=' 3 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 '=' 2 nM
Q9Y2D0 BXGT022229 Carbonic anhydrase 5B, mitochondrial reviewed - CA5B KA '=' 0 uM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 EC50 '=' 5 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 930 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 930 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 930 nM
Q16790 BXGT013670 Carbonic anhydrase 9 reviewed - CA9 KA '=' 33 uM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 78 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 pD2 '=' 7 -
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 8 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Ki '=' 12 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Emax '=' 100 %
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 0 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 126 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C pKD '=' 5 -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A pKD '=' 5 -
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B pKD '=' 5 -
Q7Z2W7 BXGT017248 Transient receptor potential cation channel subfamily M member 8 reviewed Ion channel TRPM8 Inhibition - - -
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 Ki '=' 29 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 IC50 '=' 147 nM
Q9P8Q7 BXGT021317 Isocitrate lyase reviewed - ICL1 IC50 '=' 53 ug.mL-1
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 560 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 560 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 560 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 3 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 10 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 10 nM
Q50565 BXGT014936 Carbonic anhydrase unreviewed - MTH_1582 Ka '=' 62 uM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 0 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 0 nM
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 398 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 398 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 2 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 31 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 4 nM
P22310 BXGT008754 UDP-glucuronosyltransferase 1-4 reviewed - UGT1A4 Activity '=' 0 pm/min/mg
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 81 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 5 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 10 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 4 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 3 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 1 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 IC50 - - -
O15244 BXGT004140 Solute carrier family 22 member 2 reviewed Transporter SLC22A2 Km '=' 80000 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 214 nM
P79400 BXGT011863 5-hydroxytryptamine receptor 1D reviewed - HTR1D IC50 '=' 10 nM
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 AC50 - - -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A EC50 '=' 457 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 1 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A EC50 '=' 500 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a EC50 '=' 10 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c pKD '=' 7 -
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 390 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 390 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 2 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 7 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D IA '=' 1 -
O15244 BXGT004140 Solute carrier family 22 member 2 reviewed Transporter SLC22A2 Activity - - -
P79400 BXGT011863 5-hydroxytryptamine receptor 1D reviewed - HTR1D Relative maximum '=' 1 -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 70 nM
P28565 BXGT009273 5-hydroxytryptamine receptor 1D reviewed - Htr1d IC50 '=' 3 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 3 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 42 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 Activity - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 690 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 17 nM
O70212 BXGT005060 5-hydroxytryptamine receptor 3A reviewed - HTR3A Intrinsic activity '=' 1 -
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 17200 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 15 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 0 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Emax '=' 98 %
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Emax '=' 97 %
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Efficacy '=' 101 %
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 1 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Intrinsic activity '=' 1 %
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 229 nM
P36544 BXGT009926 Neuronal acetylcholine receptor subunit alpha-7 reviewed - CHRNA7 EC50 - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 14 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 '=' 1 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Emax '=' 100 %
P15289 BXGT008102 Arylsulfatase A reviewed Enzyme ARSA Potency - 4256 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A EC50 '=' 178 nM
Q9R0W2 BXGT021408 Solute carrier family 22 member 2 reviewed - Slc22a2 Km '=' 3600000 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A EC50 '=' 141 nM
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Agonist activity '=' 0 -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Agonist activity '=' 0 -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Agonist activity '=' 0 -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Agonist activity '=' 0 -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Agonist activity '=' 0 -
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 3 nM
P16473 BXGT008234 Thyrotropin receptor reviewed G-protein coupled receptor TSHR Potency '=' 31622 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 130 nM
P97697 BXGT012214 Inositol monophosphatase 1 reviewed - Impa1 Potency '=' 19952 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 6 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 160 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 2 nM
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 EC50 '=' 100 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 180 nM
O70212 BXGT005060 5-hydroxytryptamine receptor 3A reviewed - HTR3A pD2 '=' 6 -
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 361 nM
Q9JHJ5 BXGT020810 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 361 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 3 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Ki '=' 13 nM
P31645 BXGT009558 Sodium-dependent serotonin transporter reviewed Transporter SLC6A4 Activity '>' 10000 %
P32305 BXGT009621 5-hydroxytryptamine receptor 7 reviewed - Htr7 Ki '=' 10 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 65 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 125 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 25 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 50 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Emax '=' 94 %
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 250 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 42000 nM
O70212 BXGT005060 5-hydroxytryptamine receptor 3A reviewed - HTR3A pD2 '=' 5 -
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A pKD '=' 8 -
P43166 BXGT010364 Carbonic anhydrase 7 reviewed - CA7 KA '=' 0 uM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 20 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 7100 nM
P05177 BXGT006336 Cytochrome P450 1A2 reviewed Enzyme CYP1A2 AC50 '=' 7943 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 51000 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 130 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 10000 nM
O70212 BXGT005060 5-hydroxytryptamine receptor 3A reviewed - HTR3A pD2 '=' 4 -
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 24000 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 2900 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Inhibition '=' 71 %
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 100 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a EC50 '=' 55 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 Ki '=' 187 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 5 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B EC50 '=' 4 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Activity '=' 100 %
P11344 BXGT007687 Tyrosinase reviewed - Tyr Activity '=' 22 %
P49286 BXGT010691 Melatonin receptor type 1B reviewed G-protein coupled receptor MTNR1B Ki '>' 100000 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 600 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 2 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Relative efficacy '=' 99 %
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 0 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a EC50 '=' 351 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 2950 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 2950 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 2950 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 977 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 977 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 977 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 600 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 600 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 IC50 '=' 3 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 Ki '=' 230 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 4 nM
O70212 BXGT005060 5-hydroxytryptamine receptor 3A reviewed - HTR3A pD2 '=' 5 -
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 4 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 6 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 6 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c EC50 '=' 2 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Potency '=' 39810 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 100 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 0 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 4600 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 4600 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b IC50 '=' 4600 nM
P18090 BXGT008380 Beta-1 adrenergic receptor reviewed - Adrb1 Ki - - -
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 2 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 4 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 ED50 '=' 16 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 Intrinsic activity '=' 1 -
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 14 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 70 nM
P22303 BXGT008751 Acetylcholinesterase reviewed Enzyme ACHE Inhibition '=' 28 %
P49798 BXGT010745 Regulator of G-protein signaling 4 reviewed Enzyme modulator RGS4 Potency - 4739 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki - - -
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Potency '=' 25118 nM
P28565 BXGT009273 5-hydroxytryptamine receptor 1D reviewed - Htr1d Ki '=' 2 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 2 nM
P30940 BXGT009484 5-hydroxytryptamine receptor 1F reviewed - Htr1f Ki '=' 2 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 2 nM
P07265 BXGT006583 Alpha-glucosidase MAL62 reviewed - MAL62 IC50 '>' 300000 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a nH '=' 0 -
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c nH '=' 0 -
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 pIC50 - - -
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 - - -
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 3 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b IC50 '=' 5 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 3 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Emax '=' 224 -
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Agonist activity '=' 76 -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Agonist activity '=' 76 -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Agonist activity '=' 76 -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Agonist activity '=' 76 -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Agonist activity '=' 76 -
P23415 BXGT008864 Glycine receptor subunit alpha-1 reviewed Ion channel GLRA1 EC50 - - -
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 3 nM
P32305 BXGT009621 5-hydroxytryptamine receptor 7 reviewed - Htr7 Ki '=' 7 nM
P61169 BXGT011367 D(2) dopamine receptor reviewed - Drd2 KL '=' 183000 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 0 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 pEC50 - - -
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b EC50 '=' 3 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 150 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C log(ratio) '=' 7 -
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 pD2 '=' 7 -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 5 nM
P28566 BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E Ki '=' 11 nM
P21398 BXGT008645 Amine oxidase [flavin-containing] A reviewed - MAOA Activity - - -
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Stimulation '=' 126 %
Q64264 BXGT016110 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki - - -
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 262 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 EC50 '=' 17 nM
P35218 BXGT009796 Carbonic anhydrase 5A, mitochondrial reviewed - CA5A KA '=' 6 uM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 1 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Simulation '=' 219 %
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 210000 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B Ki '=' 5 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 7 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 7 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 7 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IA '=' 1 -
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 10 nM
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 EC50 '=' 6 nM
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 320 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 320 nM
Q9P8Q7 BXGT021317 Isocitrate lyase reviewed - ICL1 IC50 '=' 301300 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 2 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 9600 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B Relative efficacy '=' 101 %
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 200 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 27000 nM
Q6FTL6 BXGT016286 Carbonic anhydrase unreviewed - NCE103 Ka '=' 16 uM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '<' 50 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 8 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 25 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IC50 '=' 5 nM
Q60484 BXGT015984 5-hydroxytryptamine receptor 1D reviewed - HTR1D EC50 '=' 5 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 pD2 '=' 8 -
Q64264 BXGT016110 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 5 nM
P35363 BXGT009818 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 500 nM
P34968 BXGT009776 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 500 nM
Q02152 BXGT012637 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 500 nM
P35363 BXGT009818 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 680 nM
P34968 BXGT009776 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 680 nM
Q02152 BXGT012637 5-hydroxytryptamine receptor 2B reviewed - Htr2b IC50 '=' 680 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 170 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 0 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 5 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 50 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 3 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 950 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 950 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 950 nM
P43140 BXGT010360 Alpha-1A adrenergic receptor reviewed - Adra1a Inhibition '<' 50 %
P23944 BXGT008930 Alpha-1D adrenergic receptor reviewed - Adra1d Inhibition '<' 50 %
P15823 BXGT008160 Alpha-1B adrenergic receptor reviewed - Adra1b Inhibition '<' 50 %
Q62758 BXGT016041 5-hydroxytryptamine receptor 4 reviewed - Htr4 Ki '=' 37 nM
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b IC50 '=' 727 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a IC50 '=' 727 nM
P53615 BXGT011003 Carbonic anhydrase reviewed - NCE103 Ka '=' 15 uM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 3 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 0 nM
O88446 BXGT005272 Solute carrier family 22 member 3 reviewed - Slc22a3 IC50 '=' 97000 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Imax - - -
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 25 nM
P19020 BXGT008448 D(3) dopamine receptor reviewed - Drd3 Ki '=' 2338 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 '=' 6 nM
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 Activity '=' 100 %
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Agonist activity '=' 41 -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Agonist activity '=' 41 -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Agonist activity '=' 41 -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Agonist activity '=' 41 -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Agonist activity '=' 41 -
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Agonist activity '=' 90 -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Agonist activity '=' 90 -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Agonist activity '=' 90 -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Agonist activity '=' 90 -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Agonist activity '=' 90 -
P48039 BXGT010607 Melatonin receptor type 1A reviewed G-protein coupled receptor MTNR1A Ki '>' 100000 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 160 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 9 nM
Q60484 BXGT015984 5-hydroxytryptamine receptor 1D reviewed - HTR1D EC50 '=' 16 nM
P22309 BXGT008753 UDP-glucuronosyltransferase 1-1 reviewed - UGT1A1 Activity '=' 0 pm/min/mg
O75795 BXGT005152 UDP-glucuronosyltransferase 2B17 reviewed - UGT2B17 Activity '=' 0 pm/min/mg
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 12000 nM
P46063 BXGT010501 ATP-dependent DNA helicase Q1 reviewed Enzyme RECQL Potency '=' 39810 nM
P08482 BXGT006775 Muscarinic acetylcholine receptor M1 reviewed - Chrm1 Potency '=' 22387 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 147 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 5 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 33 nM
Q9ULX7 BXGT021769 Carbonic anhydrase 14 reviewed - CA14 KA '=' 6 uM
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Ki '=' 120 nM
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Ki '=' 120 nM
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Ki '=' 120 nM
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Ki '=' 120 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Ki '=' 120 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 1258 nM
P30966 BXGT009486 5-hydroxytryptamine receptor 5A reviewed - Htr5a Ki '=' 150 nM
P23219 BXGT008837 Prostaglandin G/H synthase 1 reviewed Enzyme PTGS1 IC50 '>' 400000 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b IC50 '=' 4 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 75 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 84 nM
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 AC50 '=' 10000 nM
P28566 BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E Ki '=' 4 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Selectivity '=' 0 -
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 0 nM
P07265 BXGT006583 Alpha-glucosidase MAL62 reviewed - MAL62 Inhibition '=' 25 %
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 445 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 510 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 35 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 6 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c Ki '=' 6 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Ki '=' 6 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a EC50 '=' 57 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Efficacy '=' 99 %
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b Ki '=' 25 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A IC50 '=' 5 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 1 nM
P18901 BXGT008440 D(1A) dopamine receptor reviewed - Drd1 KL '=' 6543 nM
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 AC50 - - -
Q92830 BXGT019379 Histone acetyltransferase KAT2A reviewed - KAT2A Potency - 11220 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Emax '=' 99 %
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Ki '=' 87 nM
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Ki '=' 87 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 11000 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D Ki '=' 2 nM
O42713 BXGT004563 Polyphenol oxidase 2 reviewed - PPO2 IC50 '>' 350000 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 184 nM
P30939 BXGT009483 5-hydroxytryptamine receptor 1F reviewed G-protein coupled receptor HTR1F Emax '=' 100 %
Q13639 BXGT013389 5-hydroxytryptamine receptor 4 reviewed G-protein coupled receptor HTR4 Ki '=' 500 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 Imax - - -
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 1 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 1 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 51 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b EC50 '=' 4 nM
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 Potency '=' 10000 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a IC50 '=' 20 nM
P08909 BXGT006838 5-hydroxytryptamine receptor 2C reviewed - Htr2c IC50 '=' 20 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b IC50 '=' 20 nM
P35462 BXGT009835 D(3) dopamine receptor reviewed G-protein coupled receptor DRD3 Activity '=' 30 uM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 2 nM
Q60484 BXGT015984 5-hydroxytryptamine receptor 1D reviewed - HTR1D EC50 '=' 8 nM
P32305 BXGT009621 5-hydroxytryptamine receptor 7 reviewed - Htr7 Ki '=' 0 nM
P32305 BXGT009621 5-hydroxytryptamine receptor 7 reviewed - Htr7 Increase - - -
P18417 BXGT008401 Strictosidine synthase reviewed - STR1 Km '=' 1200000 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b EC50 '=' 26 nM
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 AC50 '=' 15848 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Emax '=' 100 %
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Activity - - -
P05177 BXGT006336 Cytochrome P450 1A2 reviewed Enzyme CYP1A2 AC50 '=' 1995 nM
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 Log 1/Kd '=' -3 -
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 1 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Kd '=' 3 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Inhibition '=' 97 %
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 0 nM
P31652 BXGT009565 Sodium-dependent serotonin transporter reviewed - Slc6a4 Ki - - -
O75751 BXGT005150 Solute carrier family 22 member 3 reviewed Transporter SLC22A3 Activity - - -
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 24 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 15 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 44 nM
Q60484 BXGT015984 5-hydroxytryptamine receptor 1D reviewed - HTR1D IC50 '=' 3 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 IC50 '=' 0 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 9 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b IC50 '=' 4 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 2 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Activity '=' 100 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 16 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P54855 BXGT011088 UDP-glucuronosyltransferase 2B15 reviewed - UGT2B15 Activity '=' 0 pm/min/mg
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 43 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 Inhibition - - -
Q9JJ16 BXGT020824 5-hydroxytryptamine receptor 3B reviewed - Htr3b Intrinsic efficacy - - -
P35563 BXGT009849 5-hydroxytryptamine receptor 3A reviewed - Htr3a Intrinsic efficacy - - -
Q63089 BXGT016060 Solute carrier family 22 member 1 reviewed - Slc22a1 Ki '=' 390000 nM
O88446 BXGT005272 Solute carrier family 22 member 3 reviewed - Slc22a3 Activity '=' 30 %
Q05940 BXGT012846 Synaptic vesicular amine transporter reviewed Transporter SLC18A2 Ki '=' 640000 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Inhibition '=' 100 %
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 IC50 - - -
P21728 BXGT008686 D(1A) dopamine receptor reviewed G-protein coupled receptor DRD1 IC50 - - -
O70528 BXGT005068 5-hydroxytryptamine receptor 4 reviewed - HTR4 EC50 '=' 10 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 15848 nM
P08482 BXGT006775 Muscarinic acetylcholine receptor M1 reviewed - Chrm1 Potency '=' 100 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 3400 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 3300 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 980 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Emax '=' 0 %
Q63089 BXGT016060 Solute carrier family 22 member 1 reviewed - Slc22a1 Activity - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Relative efficacy '=' 98 %
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 0 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 150 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki - - -
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 0 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 0 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 323 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 147 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 79 nM
Q9D6N1 BXGT020260 Carbonic anhydrase 13 reviewed - Ca13 KA '=' 0 uM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 0 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 1 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 1 nM
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C #NAME? '=' 7 -
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D #NAME? '=' 7 -
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B #NAME? '=' 7 -
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E #NAME? '=' 7 -
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A #NAME? '=' 7 -
Q8WXA8 BXGT019008 5-hydroxytryptamine receptor 3C reviewed Ion channel HTR3C Ki '=' 144 nM
Q70Z44 BXGT016686 5-hydroxytryptamine receptor 3D reviewed Ion channel HTR3D Ki '=' 144 nM
O95264 BXGT005367 5-hydroxytryptamine receptor 3B reviewed Ion channel HTR3B Ki '=' 144 nM
A5X5Y0 BXGT001376 5-hydroxytryptamine receptor 3E reviewed Ion channel HTR3E Ki '=' 144 nM
P46098 BXGT010507 5-hydroxytryptamine receptor 3A reviewed Ion channel HTR3A Ki '=' 144 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 150 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IC50 '=' 6 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a EC50 '=' 323 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 79 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 61 nM
P30994 BXGT009493 5-hydroxytryptamine receptor 2B reviewed - Htr2b Emax '=' 74 %
Q05940 BXGT012846 Synaptic vesicular amine transporter reviewed Transporter SLC18A2 IC50 '=' 1430 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 1 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 27 nM
P28221 BXGT009237 5-hydroxytryptamine receptor 1D reviewed G-protein coupled receptor HTR1D pKD '=' 7 -
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Activity '=' 99 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 1 nM
Q8BRU6 BXGT026111 Synaptic vesicular amine transporter reviewed - Slc18a2 IC50 '=' 98 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 15 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Activity '=' 102 %
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Ki '=' 79 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 39 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Inhibition - - -
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 110 nM
P14416 BXGT008011 D(2) dopamine receptor reviewed G-protein coupled receptor DRD2 Activity '>' 75 %
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 0 nM
Q4CVY4 BXGT026093 Carbonic anhydrase-like protein, putative unreviewed - Tc00.1047053509597.20 KA '=' 1 uM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Imax - - -
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 1 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C Activity '>' 75 %
P40881 BXGT010205 Carbonic anhydrase reviewed - KA '=' 38 uM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 280 nM
P28222 BXGT009238 5-hydroxytryptamine receptor 1B reviewed G-protein coupled receptor HTR1B IC50 '=' 12 nM
O70594 BXGT005072 Solute carrier family 22 member 5 reviewed - Slc22a5 Activity - - -
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 0 nM
P23979 BXGT008938 5-hydroxytryptamine receptor 3A reviewed - Htr3a EC50 '=' 1320 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a Ki '=' 2 nM
P12392 BXGT007812 Neuronal acetylcholine receptor subunit beta-4 reviewed - Chrnb4 EC50 - - -
P04757 BXGT006258 Neuronal acetylcholine receptor subunit alpha-3 reviewed - Chrna3 EC50 - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 7 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 398 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Ki '=' 125 nM
P28565 BXGT009273 5-hydroxytryptamine receptor 1D reviewed - Htr1d IC50 '=' 20 nM
P19327 BXGT008472 5-hydroxytryptamine receptor 1A reviewed - Htr1a IC50 '=' 20 nM
P30940 BXGT009484 5-hydroxytryptamine receptor 1F reviewed - Htr1f IC50 '=' 20 nM
P28564 BXGT009272 5-hydroxytryptamine receptor 1B reviewed - Htr1b IC50 '=' 20 nM
O42275 BXGT004559 Acetylcholinesterase reviewed - ache Inhibition '=' 62 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 18 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 169 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A FC '=' 6 -
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Activity '=' 52 %
P28566 BXGT009274 5-hydroxytryptamine receptor 1E reviewed G-protein coupled receptor HTR1E Ki '=' 10 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 1 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 IC50 '=' 0 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 190 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A IC50 '=' 260 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 15 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 10 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ki '=' 600 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 2 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 AC50 '=' 25118 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C EC50 '=' 0 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Activity '>' 75 %
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 5 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 0 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 302 nM
P05164 BXGT006333 Myeloperoxidase reviewed Enzyme MPO IC50 - - -
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 47 nM
Q05940 BXGT012846 Synaptic vesicular amine transporter reviewed Transporter SLC18A2 Ki '=' 2290 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 7 nM
P14842 BXGT008059 5-hydroxytryptamine receptor 2A reviewed - Htr2a Ratio Ki '=' 50 -
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 5 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 6 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Activity - - -
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 82 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 1 nM
P28335 BXGT009255 5-hydroxytryptamine receptor 2C reviewed G-protein coupled receptor HTR2C log(ratio) '=' 9 -
P35354 BXGT009816 Prostaglandin G/H synthase 2 reviewed Enzyme PTGS2 IC50 '>' 400000 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 IC50 '=' 130 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 1 nM
P47898 BXGT010594 5-hydroxytryptamine receptor 5A reviewed G-protein coupled receptor HTR5A Ki '=' 130 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 Ki '=' 0 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 69 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Activity '=' 94 %
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 EC50 '=' 43 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 47 nM
Q05940 BXGT012846 Synaptic vesicular amine transporter reviewed Transporter SLC18A2 Ki '=' 7690 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 5 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 97 nM
P41595 BXGT010267 5-hydroxytryptamine receptor 2B reviewed G-protein coupled receptor HTR2B EC50 '=' 4 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 27 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Ki '=' 1 nM
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A Ki '=' 11 nM
P50406 BXGT010796 5-hydroxytryptamine receptor 6 reviewed G-protein coupled receptor HTR6 Activity '=' 98 %
P28223 BXGT009239 5-hydroxytryptamine receptor 2A reviewed G-protein coupled receptor HTR2A EC50 '=' 1 nM
P34969 BXGT009777 5-hydroxytryptamine receptor 7 reviewed G-protein coupled receptor HTR7 EC50 '=' 48 nM
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A Emax '=' 2 %
P08908 BXGT006837 5-hydroxytryptamine receptor 1A reviewed G-protein coupled receptor HTR1A EC50 '=' 19 nM
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF00012 Pineapple Ananas comosus Fruits
BXGF00013 Dill Anethum graveolens Herbs and Spices
BXGF00022 Oat Avena sativa Cereals and cereal products
BXGF00041 Papaya Carica papaya Fruits
BXGF00087 Sea-buckthornberry Hippophae rhamnoides Fruits
BXGF00088 Barley Hordeum vulgare Cereals and cereal products
BXGF00093 Black walnut Juglans nigra Nuts
BXGF00094 Common walnut Juglans regia Nuts
BXGF00115 Bitter gourd Momordica charantia Gourds
BXGF00130 Avocado Persea americana Vegetables
BXGF00132 Scarlet bean Phaseolus coccineus Pulses
BXGF00135 Date Phoenix dactylifera Fruits
BXGF00141 Common pea Pisum sativum Pulses
BXGF00147 European plum Prunus domestica Fruits
BXGF00151 Pomegranate Punica granatum Fruits
BXGF00169 Rye Secale cereale Cereals and cereal products
BXGF00173 Garden tomato (var.) Solanum lycopersicum var. lycopersicum Vegetables
BXGF00174 Eggplant Solanum melongena Vegetables
BXGF00175 Potato Solanum tuberosum Vegetables
BXGF00178 Spinach Spinacia oleracea Vegetables
BXGF00182 Cocoa bean Theobroma cacao Cocoa and cocoa products
BXGF00205 Corn Zea mays Cereals and cereal products
BXGF00225 Swiss chard Beta vulgaris ssp. cicla Vegetables
BXGF00246 Red beetroot Beta vulgaris var. rubra Vegetables
BXGF00315 Cottonseed Gossypium Herbs and Spices
BXGF00400 French plantain Musa X paradisiaca Fruits
BXGF00816 Fats and oils Fats and oils
BXGF00823 Fruits Fruits
BXGF00827 Green zucchini Cucurbita pepo var. cylindrica Gourds
BXGF00832 Red bell pepper Capsicum annuum Vegetables
BXGF00835 Green bean Phaseolus vulgaris Pulses
BXGF00837 Nanking cherry Prunus tomentosa Fruits
BXGF00862 Phebalium ozothamnoides Phebalium ozothamnoides Others
BXGF00977 Vitex megapotamica Vitex megapotamica Human Edible Plant
BXGF01266 Dysoxylum lenticellatum Dysoxylum lenticellatum Others
BXGF01284 Saururus cernuus Saururus cernuus Medicinal Plant
BXGF01343 Strychnos fendleri Strychnos fendleri Others
BXGF01466 Halimeda macroloba Halimeda macroloba Others
BXGF01510 Cabucala madagascariensis Cabucala madagascariensis Others
BXGF02723 Hesperocyparis macrocarpa Hesperocyparis macrocarpa Others
BXGF02848 Buxus sempervirens Buxus sempervirens Medicinal Plant
BXGF03158 Rheum officinale Rheum officinale Medicinal Plant
BXGF03270 Aruncus dioicus Aruncus dioicus Medicinal Plant
BXGF03442 Rhaponticum carthamoides Rhaponticum carthamoides Medicinal Plant
BXGF03580 Urtica dioica Urtica dioica Medicinal Plant
BXGF03924 Kochia trichophylla Kochia trichophylla Others
BXGF04191 Vicia villosa Vicia villosa Medicinal Plant
BXGF04830 Artemisia oranensis Artemisia oranensis Others
BXGF04909 Hippophae fructus Hippophae fructus Others
BXGF05193 Piper futokadsura Piper futokadsura Others
BXGF05692 Potentilla multifida Potentilla multifida Medicinal Plant
BXGF05859 Haplopappus venetus Haplopappus venetus Others
BXGF05925 Centaurea amara Centaurea amara Others
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease