| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
1258 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
EC50 |
'=' |
30 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
8 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Intrinsic activity |
'=' |
1 |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
120 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Kd |
'=' |
9690 |
nM |
| P30939 |
BXGT009483 |
5-hydroxytryptamine receptor 1F |
reviewed |
G-protein coupled receptor |
HTR1F |
EC50 |
'=' |
7 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
EC50 |
'=' |
523 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
8 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
4 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Efficacy |
'=' |
98 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
11 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Inhibition |
- |
- |
- |
| Q9P8Q7 |
BXGT021317 |
Isocitrate lyase |
reviewed |
- |
ICL1 |
IC50 |
'=' |
301000 |
nM |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
66 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
66 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
pD2 |
'=' |
7 |
- |
| P28565 |
BXGT009273 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
Htr1d |
IC50 |
'=' |
5 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
5 |
nM |
| P30940 |
BXGT009484 |
5-hydroxytryptamine receptor 1F |
reviewed |
- |
Htr1f |
IC50 |
'=' |
5 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
'=' |
5 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Activity |
'=' |
100 |
% |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Emax |
'=' |
100 |
% |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
Activity |
'=' |
1 |
- |
| P19224 |
BXGT008468 |
UDP-glucuronosyltransferase 1-6 |
reviewed |
- |
UGT1A6 |
Activity |
- |
- |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Activity |
'=' |
99 |
% |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
2 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Emax |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
EC50 |
- |
- |
- |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
KA |
'=' |
0 |
uM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
30600 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
'=' |
100 |
nM |
| P31652 |
BXGT009565 |
Sodium-dependent serotonin transporter |
reviewed |
- |
Slc6a4 |
Activity |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
2 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
ED50 |
'=' |
1 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
1 |
nM |
| Q9Z0E8 |
BXGT022397 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Activity |
'=' |
51 |
% |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
- |
- |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
15848 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
1 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
5 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IA |
'=' |
1 |
- |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
KA |
'=' |
19 |
uM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
KA |
'=' |
50 |
uM |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Km |
'=' |
37600 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
0 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Emax |
'=' |
91 |
% |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
15811 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Emax |
'=' |
100 |
% |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
Ki |
'=' |
1049 |
nM |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
EC50 |
'=' |
12 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IC50 |
'=' |
29 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
120 |
nM |
| P28565 |
BXGT009273 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
Htr1d |
EC50 |
'=' |
5 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Emax |
'=' |
100 |
% |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
93 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
KA |
'=' |
45 |
uM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Activity |
- |
- |
- |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
23 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
'=' |
81 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
43 |
nM |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
KA |
'=' |
0 |
uM |
| Q9S446 |
BXGT021560 |
Class A sortase SrtA |
unreviewed |
- |
srtA |
IC50 |
'>' |
100 |
ug.mL-1 |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Ki |
'=' |
242000 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Max |
'=' |
100 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
1 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
6 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
1 |
nM |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
Ki |
'=' |
109 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
2 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Activity |
'=' |
15 |
% |
| P16662 |
BXGT008253 |
UDP-glucuronosyltransferase 2B7 |
reviewed |
- |
UGT2B7 |
Activity |
'=' |
0 |
pm/min/mg |
| P06133 |
BXGT006414 |
UDP-glucuronosyltransferase 2B4 |
reviewed |
- |
UGT2B4 |
Activity |
'=' |
0 |
pm/min/mg |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
13000 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Imax |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
320 |
nM |
| Q3I4V7 |
BXGT014421 |
Carbonic anhydrase |
unreviewed |
- |
CAN2 |
KA |
'=' |
46 |
uM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IC50 |
'=' |
16 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
5 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
- |
- |
- |
| Q5AJ71 |
BXGT015288 |
Carbonic anhydrase |
reviewed |
- |
NCE103 |
KA |
'=' |
28 |
uM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
- |
- |
- |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
20900 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
5100 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
1 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
1 |
nM |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
Activity |
'=' |
99 |
% |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ka |
'=' |
3 |
uM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
18 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
180 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
170000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
90000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
63000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
15000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
140000 |
nM |
| Q99N23 |
BXGT019994 |
Carbonic anhydrase 15 |
reviewed |
- |
Ca15 |
KA |
'=' |
7 |
uM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Activity |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
11 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
2350 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
7 |
nM |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
IC50 |
- |
- |
- |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
IC50 |
- |
- |
- |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
IC50 |
- |
- |
- |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
IC50 |
- |
- |
- |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
IC50 |
- |
- |
- |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
IC50 |
- |
- |
- |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
IC50 |
- |
- |
- |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
IC50 |
- |
- |
- |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
IC50 |
- |
- |
- |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
IC50 |
- |
- |
- |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
IC50 |
- |
- |
- |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
IC50 |
- |
- |
- |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
IC50 |
- |
- |
- |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
IC50 |
- |
- |
- |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
IC50 |
- |
- |
- |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
IC50 |
- |
- |
- |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
IC50 |
'=' |
550000 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
21192 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
'=' |
13 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Activity |
'=' |
100 |
% |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
1 |
nM |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Intrinsic activity |
- |
- |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Intrinsic activity |
- |
- |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Intrinsic activity |
- |
- |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Intrinsic activity |
- |
- |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Intrinsic activity |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
2 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
'=' |
5 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
3600 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
3600 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
IC50 |
'=' |
3600 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
2 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
1 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
37000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
4400 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
49000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
6200 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
1300 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
EC50 |
'=' |
4 |
nM |
| P31652 |
BXGT009565 |
Sodium-dependent serotonin transporter |
reviewed |
- |
Slc6a4 |
Ki |
'=' |
740 |
nM |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
120 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
120 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
IC50 |
'=' |
3 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
'=' |
2 |
nM |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
KA |
'=' |
0 |
uM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
EC50 |
'=' |
5 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
930 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
930 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
930 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
KA |
'=' |
33 |
uM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
78 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
pD2 |
'=' |
7 |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
8 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
'=' |
12 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Emax |
'=' |
100 |
% |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
0 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
126 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
pKD |
'=' |
5 |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
pKD |
'=' |
5 |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
pKD |
'=' |
5 |
- |
| Q7Z2W7 |
BXGT017248 |
Transient receptor potential cation channel subfamily M member 8 |
reviewed |
Ion channel |
TRPM8 |
Inhibition |
- |
- |
- |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
Ki |
'=' |
29 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
IC50 |
'=' |
147 |
nM |
| Q9P8Q7 |
BXGT021317 |
Isocitrate lyase |
reviewed |
- |
ICL1 |
IC50 |
'=' |
53 |
ug.mL-1 |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
560 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
560 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
560 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
3 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
10 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
10 |
nM |
| Q50565 |
BXGT014936 |
Carbonic anhydrase |
unreviewed |
- |
MTH_1582 |
Ka |
'=' |
62 |
uM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
0 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
0 |
nM |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
398 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
398 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
2 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
31 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
4 |
nM |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
81 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
5 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
10 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
4 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
3 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
1 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Km |
'=' |
80000 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
214 |
nM |
| P79400 |
BXGT011863 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
IC50 |
'=' |
10 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
EC50 |
'=' |
457 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
1 |
nM |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
EC50 |
'=' |
500 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
EC50 |
'=' |
10 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
pKD |
'=' |
7 |
- |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
390 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
390 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
2 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
7 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
IA |
'=' |
1 |
- |
| O15244 |
BXGT004140 |
Solute carrier family 22 member 2 |
reviewed |
Transporter |
SLC22A2 |
Activity |
- |
- |
- |
| P79400 |
BXGT011863 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
Relative maximum |
'=' |
1 |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
70 |
nM |
| P28565 |
BXGT009273 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
Htr1d |
IC50 |
'=' |
3 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
3 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
42 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
690 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
17 |
nM |
| O70212 |
BXGT005060 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
HTR3A |
Intrinsic activity |
'=' |
1 |
- |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
17200 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
15 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
0 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Emax |
'=' |
98 |
% |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Emax |
'=' |
97 |
% |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Efficacy |
'=' |
101 |
% |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
1 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Intrinsic activity |
'=' |
1 |
% |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
229 |
nM |
| P36544 |
BXGT009926 |
Neuronal acetylcholine receptor subunit alpha-7 |
reviewed |
- |
CHRNA7 |
EC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
14 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
'=' |
1 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Emax |
'=' |
100 |
% |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
4256 |
nM |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
EC50 |
'=' |
178 |
nM |
| Q9R0W2 |
BXGT021408 |
Solute carrier family 22 member 2 |
reviewed |
- |
Slc22a2 |
Km |
'=' |
3600000 |
nM |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
EC50 |
'=' |
141 |
nM |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Agonist activity |
'=' |
0 |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Agonist activity |
'=' |
0 |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Agonist activity |
'=' |
0 |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Agonist activity |
'=' |
0 |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Agonist activity |
'=' |
0 |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
3 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
31622 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
130 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
19952 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
6 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
160 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
2 |
nM |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
EC50 |
'=' |
100 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
180 |
nM |
| O70212 |
BXGT005060 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
HTR3A |
pD2 |
'=' |
6 |
- |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
361 |
nM |
| Q9JHJ5 |
BXGT020810 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
361 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
3 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
'=' |
13 |
nM |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Activity |
'>' |
10000 |
% |
| P32305 |
BXGT009621 |
5-hydroxytryptamine receptor 7 |
reviewed |
- |
Htr7 |
Ki |
'=' |
10 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
65 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
125 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
25 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
50 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Emax |
'=' |
94 |
% |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
250 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
42000 |
nM |
| O70212 |
BXGT005060 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
HTR3A |
pD2 |
'=' |
5 |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
pKD |
'=' |
8 |
- |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
KA |
'=' |
0 |
uM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
20 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
7100 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
7943 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
51000 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
130 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
10000 |
nM |
| O70212 |
BXGT005060 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
HTR3A |
pD2 |
'=' |
4 |
- |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
24000 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
2900 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Inhibition |
'=' |
71 |
% |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
100 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
EC50 |
'=' |
55 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
Ki |
'=' |
187 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
5 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
EC50 |
'=' |
4 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Activity |
'=' |
100 |
% |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
Activity |
'=' |
22 |
% |
| P49286 |
BXGT010691 |
Melatonin receptor type 1B |
reviewed |
G-protein coupled receptor |
MTNR1B |
Ki |
'>' |
100000 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
600 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
2 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Relative efficacy |
'=' |
99 |
% |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
0 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
EC50 |
'=' |
351 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
2950 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
2950 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
2950 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
977 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
977 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
977 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
600 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
600 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
IC50 |
'=' |
3 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
'=' |
230 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
4 |
nM |
| O70212 |
BXGT005060 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
HTR3A |
pD2 |
'=' |
5 |
- |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
4 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
6 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
6 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
EC50 |
'=' |
2 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
39810 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
100 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
0 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
4600 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
4600 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
IC50 |
'=' |
4600 |
nM |
| P18090 |
BXGT008380 |
Beta-1 adrenergic receptor |
reviewed |
- |
Adrb1 |
Ki |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
2 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
4 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
ED50 |
'=' |
16 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Intrinsic activity |
'=' |
1 |
- |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
14 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
70 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Inhibition |
'=' |
28 |
% |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
4739 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
25118 |
nM |
| P28565 |
BXGT009273 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
Htr1d |
Ki |
'=' |
2 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
2 |
nM |
| P30940 |
BXGT009484 |
5-hydroxytryptamine receptor 1F |
reviewed |
- |
Htr1f |
Ki |
'=' |
2 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
2 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
IC50 |
'>' |
300000 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
nH |
'=' |
0 |
- |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
nH |
'=' |
0 |
- |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
pIC50 |
- |
- |
- |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
3 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
'=' |
5 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
3 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Emax |
'=' |
224 |
- |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Agonist activity |
'=' |
76 |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Agonist activity |
'=' |
76 |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Agonist activity |
'=' |
76 |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Agonist activity |
'=' |
76 |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Agonist activity |
'=' |
76 |
- |
| P23415 |
BXGT008864 |
Glycine receptor subunit alpha-1 |
reviewed |
Ion channel |
GLRA1 |
EC50 |
- |
- |
- |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
3 |
nM |
| P32305 |
BXGT009621 |
5-hydroxytryptamine receptor 7 |
reviewed |
- |
Htr7 |
Ki |
'=' |
7 |
nM |
| P61169 |
BXGT011367 |
D(2) dopamine receptor |
reviewed |
- |
Drd2 |
KL |
'=' |
183000 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
0 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
pEC50 |
- |
- |
- |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
EC50 |
'=' |
3 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
150 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
log(ratio) |
'=' |
7 |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
pD2 |
'=' |
7 |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
5 |
nM |
| P28566 |
BXGT009274 |
5-hydroxytryptamine receptor 1E |
reviewed |
G-protein coupled receptor |
HTR1E |
Ki |
'=' |
11 |
nM |
| P21398 |
BXGT008645 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Activity |
- |
- |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Stimulation |
'=' |
126 |
% |
| Q64264 |
BXGT016110 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
262 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
EC50 |
'=' |
17 |
nM |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
KA |
'=' |
6 |
uM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
1 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Simulation |
'=' |
219 |
% |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
210000 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
Ki |
'=' |
5 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
7 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
7 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
7 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IA |
'=' |
1 |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
10 |
nM |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
EC50 |
'=' |
6 |
nM |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
320 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
320 |
nM |
| Q9P8Q7 |
BXGT021317 |
Isocitrate lyase |
reviewed |
- |
ICL1 |
IC50 |
'=' |
301300 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
2 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
9600 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Relative efficacy |
'=' |
101 |
% |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
200 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
27000 |
nM |
| Q6FTL6 |
BXGT016286 |
Carbonic anhydrase |
unreviewed |
- |
NCE103 |
Ka |
'=' |
16 |
uM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'<' |
50 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
8 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
25 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IC50 |
'=' |
5 |
nM |
| Q60484 |
BXGT015984 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
EC50 |
'=' |
5 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
pD2 |
'=' |
8 |
- |
| Q64264 |
BXGT016110 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
5 |
nM |
| P35363 |
BXGT009818 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
500 |
nM |
| P34968 |
BXGT009776 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
500 |
nM |
| Q02152 |
BXGT012637 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
500 |
nM |
| P35363 |
BXGT009818 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
680 |
nM |
| P34968 |
BXGT009776 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
680 |
nM |
| Q02152 |
BXGT012637 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
IC50 |
'=' |
680 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
170 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
0 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
5 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
50 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
3 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
950 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
950 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
950 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Inhibition |
'<' |
50 |
% |
| P23944 |
BXGT008930 |
Alpha-1D adrenergic receptor |
reviewed |
- |
Adra1d |
Inhibition |
'<' |
50 |
% |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Inhibition |
'<' |
50 |
% |
| Q62758 |
BXGT016041 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
Htr4 |
Ki |
'=' |
37 |
nM |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
IC50 |
'=' |
727 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
IC50 |
'=' |
727 |
nM |
| P53615 |
BXGT011003 |
Carbonic anhydrase |
reviewed |
- |
NCE103 |
Ka |
'=' |
15 |
uM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
3 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
0 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
IC50 |
'=' |
97000 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Imax |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
25 |
nM |
| P19020 |
BXGT008448 |
D(3) dopamine receptor |
reviewed |
- |
Drd3 |
Ki |
'=' |
2338 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
'=' |
6 |
nM |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Activity |
'=' |
100 |
% |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Agonist activity |
'=' |
41 |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Agonist activity |
'=' |
41 |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Agonist activity |
'=' |
41 |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Agonist activity |
'=' |
41 |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Agonist activity |
'=' |
41 |
- |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Agonist activity |
'=' |
90 |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Agonist activity |
'=' |
90 |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Agonist activity |
'=' |
90 |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Agonist activity |
'=' |
90 |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Agonist activity |
'=' |
90 |
- |
| P48039 |
BXGT010607 |
Melatonin receptor type 1A |
reviewed |
G-protein coupled receptor |
MTNR1A |
Ki |
'>' |
100000 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
160 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
9 |
nM |
| Q60484 |
BXGT015984 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
EC50 |
'=' |
16 |
nM |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
0 |
pm/min/mg |
| O75795 |
BXGT005152 |
UDP-glucuronosyltransferase 2B17 |
reviewed |
- |
UGT2B17 |
Activity |
'=' |
0 |
pm/min/mg |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
12000 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
39810 |
nM |
| P08482 |
BXGT006775 |
Muscarinic acetylcholine receptor M1 |
reviewed |
- |
Chrm1 |
Potency |
'=' |
22387 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
147 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
5 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
33 |
nM |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
KA |
'=' |
6 |
uM |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Ki |
'=' |
120 |
nM |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Ki |
'=' |
120 |
nM |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Ki |
'=' |
120 |
nM |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Ki |
'=' |
120 |
nM |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Ki |
'=' |
120 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
1258 |
nM |
| P30966 |
BXGT009486 |
5-hydroxytryptamine receptor 5A |
reviewed |
- |
Htr5a |
Ki |
'=' |
150 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'>' |
400000 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
'=' |
4 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
75 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
84 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
10000 |
nM |
| P28566 |
BXGT009274 |
5-hydroxytryptamine receptor 1E |
reviewed |
G-protein coupled receptor |
HTR1E |
Ki |
'=' |
4 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Selectivity |
'=' |
0 |
- |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
0 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
Inhibition |
'=' |
25 |
% |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
445 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
510 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
35 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
6 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Ki |
'=' |
6 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Ki |
'=' |
6 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
EC50 |
'=' |
57 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Efficacy |
'=' |
99 |
% |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
'=' |
25 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
IC50 |
'=' |
5 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
1 |
nM |
| P18901 |
BXGT008440 |
D(1A) dopamine receptor |
reviewed |
- |
Drd1 |
KL |
'=' |
6543 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| Q92830 |
BXGT019379 |
Histone acetyltransferase KAT2A |
reviewed |
- |
KAT2A |
Potency |
- |
11220 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Emax |
'=' |
99 |
% |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Ki |
'=' |
87 |
nM |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Ki |
'=' |
87 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
11000 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
Ki |
'=' |
2 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'>' |
350000 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
184 |
nM |
| P30939 |
BXGT009483 |
5-hydroxytryptamine receptor 1F |
reviewed |
G-protein coupled receptor |
HTR1F |
Emax |
'=' |
100 |
% |
| Q13639 |
BXGT013389 |
5-hydroxytryptamine receptor 4 |
reviewed |
G-protein coupled receptor |
HTR4 |
Ki |
'=' |
500 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Imax |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
1 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
1 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
51 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
EC50 |
'=' |
4 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
10000 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
IC50 |
'=' |
20 |
nM |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
IC50 |
'=' |
20 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
IC50 |
'=' |
20 |
nM |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Activity |
'=' |
30 |
uM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
2 |
nM |
| Q60484 |
BXGT015984 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
EC50 |
'=' |
8 |
nM |
| P32305 |
BXGT009621 |
5-hydroxytryptamine receptor 7 |
reviewed |
- |
Htr7 |
Ki |
'=' |
0 |
nM |
| P32305 |
BXGT009621 |
5-hydroxytryptamine receptor 7 |
reviewed |
- |
Htr7 |
Increase |
- |
- |
- |
| P18417 |
BXGT008401 |
Strictosidine synthase |
reviewed |
- |
STR1 |
Km |
'=' |
1200000 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
EC50 |
'=' |
26 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
15848 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Emax |
'=' |
100 |
% |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Activity |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
1995 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Log 1/Kd |
'=' |
-3 |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
1 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Kd |
'=' |
3 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Inhibition |
'=' |
97 |
% |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
0 |
nM |
| P31652 |
BXGT009565 |
Sodium-dependent serotonin transporter |
reviewed |
- |
Slc6a4 |
Ki |
- |
- |
- |
| O75751 |
BXGT005150 |
Solute carrier family 22 member 3 |
reviewed |
Transporter |
SLC22A3 |
Activity |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
24 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
15 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
44 |
nM |
| Q60484 |
BXGT015984 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
HTR1D |
IC50 |
'=' |
3 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
'=' |
0 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
9 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
'=' |
4 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
2 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Activity |
'=' |
100 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
16 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
0 |
pm/min/mg |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
43 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Inhibition |
- |
- |
- |
| Q9JJ16 |
BXGT020824 |
5-hydroxytryptamine receptor 3B |
reviewed |
- |
Htr3b |
Intrinsic efficacy |
- |
- |
- |
| P35563 |
BXGT009849 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
Intrinsic efficacy |
- |
- |
- |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Ki |
'=' |
390000 |
nM |
| O88446 |
BXGT005272 |
Solute carrier family 22 member 3 |
reviewed |
- |
Slc22a3 |
Activity |
'=' |
30 |
% |
| Q05940 |
BXGT012846 |
Synaptic vesicular amine transporter |
reviewed |
Transporter |
SLC18A2 |
Ki |
'=' |
640000 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Inhibition |
'=' |
100 |
% |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
EC50 |
'=' |
10 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
15848 |
nM |
| P08482 |
BXGT006775 |
Muscarinic acetylcholine receptor M1 |
reviewed |
- |
Chrm1 |
Potency |
'=' |
100 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
3400 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
3300 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
980 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Emax |
'=' |
0 |
% |
| Q63089 |
BXGT016060 |
Solute carrier family 22 member 1 |
reviewed |
- |
Slc22a1 |
Activity |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Relative efficacy |
'=' |
98 |
% |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
0 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
150 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
- |
- |
- |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
0 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
0 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
323 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
147 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
79 |
nM |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
KA |
'=' |
0 |
uM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
0 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
1 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
1 |
nM |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
#NAME? |
'=' |
7 |
- |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
#NAME? |
'=' |
7 |
- |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
#NAME? |
'=' |
7 |
- |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
#NAME? |
'=' |
7 |
- |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
#NAME? |
'=' |
7 |
- |
| Q8WXA8 |
BXGT019008 |
5-hydroxytryptamine receptor 3C |
reviewed |
Ion channel |
HTR3C |
Ki |
'=' |
144 |
nM |
| Q70Z44 |
BXGT016686 |
5-hydroxytryptamine receptor 3D |
reviewed |
Ion channel |
HTR3D |
Ki |
'=' |
144 |
nM |
| O95264 |
BXGT005367 |
5-hydroxytryptamine receptor 3B |
reviewed |
Ion channel |
HTR3B |
Ki |
'=' |
144 |
nM |
| A5X5Y0 |
BXGT001376 |
5-hydroxytryptamine receptor 3E |
reviewed |
Ion channel |
HTR3E |
Ki |
'=' |
144 |
nM |
| P46098 |
BXGT010507 |
5-hydroxytryptamine receptor 3A |
reviewed |
Ion channel |
HTR3A |
Ki |
'=' |
144 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
150 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IC50 |
'=' |
6 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
EC50 |
'=' |
323 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
79 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
61 |
nM |
| P30994 |
BXGT009493 |
5-hydroxytryptamine receptor 2B |
reviewed |
- |
Htr2b |
Emax |
'=' |
74 |
% |
| Q05940 |
BXGT012846 |
Synaptic vesicular amine transporter |
reviewed |
Transporter |
SLC18A2 |
IC50 |
'=' |
1430 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
1 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
27 |
nM |
| P28221 |
BXGT009237 |
5-hydroxytryptamine receptor 1D |
reviewed |
G-protein coupled receptor |
HTR1D |
pKD |
'=' |
7 |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Activity |
'=' |
99 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
1 |
nM |
| Q8BRU6 |
BXGT026111 |
Synaptic vesicular amine transporter |
reviewed |
- |
Slc18a2 |
IC50 |
'=' |
98 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
15 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Activity |
'=' |
102 |
% |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
79 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
39 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Inhibition |
- |
- |
- |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
110 |
nM |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Activity |
'>' |
75 |
% |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
0 |
nM |
| Q4CVY4 |
BXGT026093 |
Carbonic anhydrase-like protein, putative |
unreviewed |
- |
Tc00.1047053509597.20 |
KA |
'=' |
1 |
uM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Imax |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
1 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Activity |
'>' |
75 |
% |
| P40881 |
BXGT010205 |
Carbonic anhydrase |
reviewed |
- |
|
KA |
'=' |
38 |
uM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
280 |
nM |
| P28222 |
BXGT009238 |
5-hydroxytryptamine receptor 1B |
reviewed |
G-protein coupled receptor |
HTR1B |
IC50 |
'=' |
12 |
nM |
| O70594 |
BXGT005072 |
Solute carrier family 22 member 5 |
reviewed |
- |
Slc22a5 |
Activity |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
0 |
nM |
| P23979 |
BXGT008938 |
5-hydroxytryptamine receptor 3A |
reviewed |
- |
Htr3a |
EC50 |
'=' |
1320 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
'=' |
2 |
nM |
| P12392 |
BXGT007812 |
Neuronal acetylcholine receptor subunit beta-4 |
reviewed |
- |
Chrnb4 |
EC50 |
- |
- |
- |
| P04757 |
BXGT006258 |
Neuronal acetylcholine receptor subunit alpha-3 |
reviewed |
- |
Chrna3 |
EC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
7 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
398 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
'=' |
125 |
nM |
| P28565 |
BXGT009273 |
5-hydroxytryptamine receptor 1D |
reviewed |
- |
Htr1d |
IC50 |
'=' |
20 |
nM |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
'=' |
20 |
nM |
| P30940 |
BXGT009484 |
5-hydroxytryptamine receptor 1F |
reviewed |
- |
Htr1f |
IC50 |
'=' |
20 |
nM |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
'=' |
20 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
62 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
18 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
169 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
FC |
'=' |
6 |
- |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Activity |
'=' |
52 |
% |
| P28566 |
BXGT009274 |
5-hydroxytryptamine receptor 1E |
reviewed |
G-protein coupled receptor |
HTR1E |
Ki |
'=' |
10 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
1 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
IC50 |
'=' |
0 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
190 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
IC50 |
'=' |
260 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
15 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
10 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ki |
'=' |
600 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
2 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
25118 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
EC50 |
'=' |
0 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Activity |
'>' |
75 |
% |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
5 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
0 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
302 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
47 |
nM |
| Q05940 |
BXGT012846 |
Synaptic vesicular amine transporter |
reviewed |
Transporter |
SLC18A2 |
Ki |
'=' |
2290 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
7 |
nM |
| P14842 |
BXGT008059 |
5-hydroxytryptamine receptor 2A |
reviewed |
- |
Htr2a |
Ratio Ki |
'=' |
50 |
- |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
5 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
6 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Activity |
- |
- |
- |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
82 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
1 |
nM |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
log(ratio) |
'=' |
9 |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'>' |
400000 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
'=' |
130 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
1 |
nM |
| P47898 |
BXGT010594 |
5-hydroxytryptamine receptor 5A |
reviewed |
G-protein coupled receptor |
HTR5A |
Ki |
'=' |
130 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
Ki |
'=' |
0 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
69 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Activity |
'=' |
94 |
% |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
EC50 |
'=' |
43 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
47 |
nM |
| Q05940 |
BXGT012846 |
Synaptic vesicular amine transporter |
reviewed |
Transporter |
SLC18A2 |
Ki |
'=' |
7690 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
5 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
97 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
EC50 |
'=' |
4 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
27 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Ki |
'=' |
1 |
nM |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
11 |
nM |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Activity |
'=' |
98 |
% |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
EC50 |
'=' |
1 |
nM |
| P34969 |
BXGT009777 |
5-hydroxytryptamine receptor 7 |
reviewed |
G-protein coupled receptor |
HTR7 |
EC50 |
'=' |
48 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Emax |
'=' |
2 |
% |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'=' |
19 |
nM |