| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
7079 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
7079 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
0 |
% |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
2000 |
nM |
| Q08493 |
BXGT012987 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4C |
reviewed |
- |
PDE4C |
Activity |
'=' |
3 |
pmol |
| Q07343 |
BXGT012926 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B |
reviewed |
- |
PDE4B |
Activity |
'=' |
3 |
pmol |
| Q08499 |
BXGT012988 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
reviewed |
- |
PDE4D |
Activity |
'=' |
3 |
pmol |
| P27815 |
BXGT009208 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A |
reviewed |
- |
PDE4A |
Activity |
'=' |
3 |
pmol |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
35481 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
1901 |
nM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
26 |
ug.mL-1 |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
12589 |
nM |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
10000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
12589 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
12589 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
316 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
1258 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7079 |
nM |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
CC50 |
'=' |
195 |
ug.mL-1 |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7943 |
nM |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
1258 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
3981 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
Inhibition |
- |
- |
- |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
1000 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'<' |
1000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'<' |
1000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'<' |
1000 |
nM |
| P08238 |
BXGT006753 |
Heat shock protein HSP 90-beta |
reviewed |
Chaperone |
HSP90AB1 |
IC50 |
'=' |
13500 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
1995 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
199 |
nM |
| Q15746 |
BXGT013591 |
Myosin light chain kinase, smooth muscle |
reviewed |
Kinase |
MYLK |
Ki |
'=' |
1700 |
nM |
| Q9HCT0 |
BXGT020538 |
Fibroblast growth factor 22 |
reviewed |
Signaling |
FGF22 |
AbsAC1 |
'=' |
4 |
uM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
7943 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
82600 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
3981 |
nM |
| O95398 |
BXGT005378 |
Rap guanine nucleotide exchange factor 3 |
reviewed |
Enzyme modulator |
RAPGEF3 |
Potency |
- |
15848 |
nM |
| Q9Y468 |
BXGT022270 |
Lethal(3)malignant brain tumor-like protein 1 |
reviewed |
Epigenetic regulator |
L3MBTL1 |
Potency |
'=' |
446 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
25118 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
25118 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
600 |
nM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
logIC50 |
'=' |
1 |
- |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
12589 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
3981 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
25118 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
- |
- |
- |
| Q27686 |
BXGT013930 |
Pyruvate kinase |
reviewed |
- |
PYK |
Potency |
'=' |
1995 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
3548 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
46200 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| Q03114 |
BXGT012692 |
Cyclin-dependent-like kinase 5 |
reviewed |
- |
Cdk5 |
EC50 |
'=' |
71100 |
nM |
| Q9UIF8 |
BXGT021718 |
Bromodomain adjacent to zinc finger domain protein 2B |
reviewed |
- |
BAZ2B |
Potency |
- |
22387 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
17782 |
nM |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
3162 |
nM |
| P06278 |
BXGT006431 |
Alpha-amylase |
reviewed |
- |
amyS |
Activity |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1995 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
354 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
19952 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
IC50 |
'=' |
14000 |
nM |
| P90584 |
BXGT012110 |
MO15-related protein kinase Pfmrk |
unreviewed |
- |
Pfmrk |
IC50 |
'=' |
157000 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
891 |
nM |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
5211 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
2238 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
1683 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
31622 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
1258 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
'=' |
37800 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
7943 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
158 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
84921 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
'=' |
10000 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
62 |
% |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
19952 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
19952 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
6309 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
3793 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
29000 |
nM |
| P27189 |
BXGT009163 |
DNA primase TraC |
reviewed |
- |
traC |
IC50 |
'=' |
700000 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
125 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
IC50 |
'=' |
3000 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
631 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Activity |
- |
- |
- |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
2511 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
10000 |
nM |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
IC50 |
'=' |
11 |
ug.mL-1 |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
0 |
- |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
7943 |
nM |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
3013 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
11 |
ug.mL-1 |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
56 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
12589 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
12589 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
23280 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
14125 |
nM |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
2000 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
4466 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
14700 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
IC50 |
'=' |
20000 |
nM |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
14125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
281 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
199 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
39810 |
nM |
| Q08493 |
BXGT012987 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4C |
reviewed |
- |
PDE4C |
Inhibition |
'=' |
50 |
% |
| Q07343 |
BXGT012926 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4B |
reviewed |
- |
PDE4B |
Inhibition |
'=' |
50 |
% |
| Q08499 |
BXGT012988 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4D |
reviewed |
- |
PDE4D |
Inhibition |
'=' |
50 |
% |
| P27815 |
BXGT009208 |
cAMP-specific 3',5'-cyclic phosphodiesterase 4A |
reviewed |
- |
PDE4A |
Inhibition |
'=' |
50 |
% |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
'=' |
31622 |
nM |
| P00760 |
BXGT005644 |
Cationic trypsin |
reviewed |
- |
|
IC50 |
'=' |
10200 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
75400 |
nM |
| P00530 |
BXGT005574 |
Tyrosine-protein kinase transforming protein Fps |
reviewed |
- |
V-FPS |
Ki |
'=' |
1800 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
158 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
946 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
2800 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
5011 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
7079 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
400 |
nM |
| Q14576 |
BXGT013487 |
ELAV-like protein 3 |
reviewed |
- |
ELAVL3 |
IC50 |
'=' |
1000 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
IC50 |
'=' |
2100 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
13371 |
nM |
| P0AES4 |
BXGT007329 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'=' |
225 |
ug.mL-1 |
| P0AES6 |
BXGT007331 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'=' |
225 |
ug.mL-1 |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
2400 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
IC50 |
'=' |
22000 |
nM |
| P16098 |
BXGT008191 |
Beta-amylase |
reviewed |
- |
BMY1 |
Activity |
- |
- |
- |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
28183 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
10000 |
nM |
| P05186 |
BXGT006338 |
Alkaline phosphatase, tissue-nonspecific isozyme |
reviewed |
Enzyme |
ALPL |
IC50 |
'=' |
33200 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
2238 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
920 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
920 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
920 |
nM |
| P55212 |
BXGT011112 |
Caspase-6 |
reviewed |
Enzyme |
CASP6 |
AC50 |
'=' |
461 |
nM |
| P10696 |
BXGT007603 |
Alkaline phosphatase, germ cell type |
reviewed |
Enzyme |
ALPG |
EC50 |
'=' |
32300 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
25118 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
2993 |
nM |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
Ki |
'=' |
33500 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
299 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P13267 |
BXGT007895 |
DNA polymerase III PolC-type |
reviewed |
- |
polC |
Potency |
- |
15003 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
3981 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
1995 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
5011 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
12589 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
2 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
1995 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
562 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
25118 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
6309 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
26679 |
nM |
| P09923 |
BXGT006942 |
Intestinal-type alkaline phosphatase |
reviewed |
Enzyme |
ALPI |
EC50 |
'>' |
100000 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
19952 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
150 |
nM |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Activity |
- |
- |
- |
| O75164 |
BXGT005104 |
Lysine-specific demethylase 4A |
reviewed |
- |
KDM4A |
Potency |
- |
3548 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
IC50 |
'=' |
560 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
2511 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
10000 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Potency |
'=' |
44668 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
354 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
1412 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Ki |
'=' |
2600 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
'=' |
30200 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
79 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1412 |
nM |
| Q14790 |
BXGT013505 |
Caspase-8 |
reviewed |
Enzyme |
CASP8 |
Inhibition |
- |
- |
- |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
1584 |
nM |
| Q91WR5 |
BXGT019303 |
Aldo-keto reductase family 1 member C21 |
reviewed |
- |
Akr1c21 |
IC50 |
'=' |
12300 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
7600 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
31622 |
nM |
| Q962Y6 |
BXGT019597 |
Thioredoxin glutathione reductase |
unreviewed |
- |
TGR |
Potency |
'=' |
3548 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
7079 |
nM |
| P31941 |
BXGT009585 |
DNA dC->dU-editing enzyme APOBEC-3A |
reviewed |
- |
APOBEC3A |
IC50 |
'=' |
17500 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
8912 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
19952 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
70794 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
707 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
952 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
1122 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
IC50 |
'=' |
1690 |
nM |
| Q86831 |
BXGT017584 |
Polyprotein II |
unreviewed |
- |
|
Inhibition |
'=' |
82 |
% |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
1500 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
7943 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
7943 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
37933 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
390 |
nM |
| Q8WZA2 |
BXGT019025 |
Rap guanine nucleotide exchange factor 4 |
reviewed |
Enzyme modulator |
RAPGEF4 |
Potency |
- |
8912 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
39810 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
398 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
2818 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
1995 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
19952 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
10000 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
22387 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
14125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18356 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
24 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
28183 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
25929 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
7062 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
15100 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
IC50 |
'=' |
1200 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
13300 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
2500 |
nM |
| O14924 |
BXGT004111 |
Regulator of G-protein signaling 12 |
reviewed |
- |
RGS12 |
Potency |
'=' |
10000 |
nM |
| P63096 |
BXGT011496 |
Guanine nucleotide-binding protein G(i) subunit alpha-1 |
reviewed |
Enzyme modulator |
GNAI1 |
Potency |
'=' |
10000 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
8912 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
2818 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Ki |
'=' |
370 |
nM |
| Q4GZG4 |
BXGT014813 |
Phosphoglycerate kinase |
unreviewed |
- |
PGKC |
Potency |
- |
650 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'=' |
12 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
199 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
12589 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
12589 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
39810 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
3162 |
nM |
| P28907 |
BXGT009301 |
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 |
reviewed |
Enzyme |
CD38 |
IC50 |
'=' |
24800 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
14125 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'<' |
3000 |
nM |
| Q14191 |
BXGT013452 |
Werner syndrome ATP-dependent helicase |
reviewed |
Enzyme |
WRN |
Potency |
- |
1122 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Potency |
'=' |
16481 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
794 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
95 |
% |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
3013 |
nM |
| P29372 |
BXGT009336 |
DNA-3-methyladenine glycosylase |
reviewed |
Enzyme |
MPG |
Inhibition |
'=' |
36 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
19952 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
17782 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
39810 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
8492 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
843 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
31622 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
237 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
3020 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
4 |
% |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
27 |
nM |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
2511 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
2818 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
10000 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
3981 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
31622 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
2511 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
23000 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
1062 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
8436 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
IC50 |
'=' |
320 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
29910 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
Inhibition |
'=' |
67 |
% |
| Q57TT1 |
BXGT015153 |
Uncharacterized protein |
unreviewed |
- |
Tb927.8.6820 |
Potency |
- |
50118 |
nM |
| P11064 |
BXGT007646 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
Inhibition |
'=' |
14 |
% |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
150000 |
nM |
| Q9Y468 |
BXGT022270 |
Lethal(3)malignant brain tumor-like protein 1 |
reviewed |
Epigenetic regulator |
L3MBTL1 |
Potency |
- |
150 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Ratio |
'=' |
9 |
- |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
281 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
93 |
% |
| P55210 |
BXGT011110 |
Caspase-7 |
reviewed |
Enzyme |
CASP7 |
AC50 |
'=' |
5400 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
1122 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
2380 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
9976 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
IC50 |
'=' |
2120 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
4466 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
71000 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
23934 |
nM |
| Q9HC16 |
BXGT020525 |
DNA dC->dU-editing enzyme APOBEC-3G |
reviewed |
Enzyme |
APOBEC3G |
IC50 |
'=' |
2390 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
1694 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
-3 |
% |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
6400 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
11220 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
2685 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
Ki |
'=' |
1200 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
33498 |
nM |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
15811 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
37150 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
281 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
14800 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Potency |
- |
9466 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
1000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
IC50 |
'<' |
3000 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
EC50 |
'=' |
54000 |
nM |
| P24822 |
BXGT008996 |
Intestinal-type alkaline phosphatase |
reviewed |
- |
Iap |
IC50 |
'=' |
12500 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
89125 |
nM |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
IC50 |
'=' |
4720 |
nM |
| P32929 |
BXGT009682 |
Cystathionine gamma-lyase |
reviewed |
Enzyme |
CTH |
Inhibition |
- |
- |
- |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
IC50 |
'=' |
850 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
30 |
% |
| P11168 |
BXGT007663 |
Solute carrier family 2, facilitated glucose transporter member 2 |
reviewed |
Transporter |
SLC2A2 |
IC50 |
'=' |
12000 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Efficacy |
'=' |
224 |
picometer |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
25118 |
nM |
| P35520 |
BXGT009842 |
Cystathionine beta-synthase |
reviewed |
- |
CBS |
Inhibition |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
210000 |
nM |
| Q02127 |
BXGT012635 |
Dihydroorotate dehydrogenase (quinone), mitochondrial |
reviewed |
Enzyme |
DHODH |
Inhibition |
'=' |
41 |
% |
| P35520 |
BXGT009842 |
Cystathionine beta-synthase |
reviewed |
- |
CBS |
IC50 |
'=' |
18800 |
nM |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
IC50 |
'=' |
1562 |
nM |
| Q4QEW7 |
BXGT014876 |
Dihydroorotate dehydrogenase (fumarate) |
unreviewed |
- |
DHODH |
IC50 |
'=' |
31622 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'>' |
50 |
% |