| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
Ki |
'=' |
489 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Ratio |
'=' |
1 |
- |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
pKm |
'=' |
5 |
- |
| Q13002 |
BXGT013303 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
Ion channel |
GRIK2 |
Ki |
'=' |
1106 |
nM |
| Q16478 |
BXGT013630 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
Ion channel |
GRIK5 |
Ki |
'=' |
750 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
IC50 |
'=' |
1300 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
IC50 |
'=' |
1300 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
IC50 |
'=' |
1300 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
IC50 |
'=' |
1300 |
nM |
| P31422 |
BXGT009540 |
Metabotropic glutamate receptor 3 |
reviewed |
- |
Grm3 |
EC50 |
'=' |
57 |
nM |
| P31596 |
BXGT009553 |
Excitatory amino acid transporter 2 |
reviewed |
- |
Slc1a2 |
Control |
'=' |
40 |
% |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
EC50 |
'=' |
20000 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
8000 |
nM |
| P39086 |
BXGT010093 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
Ion channel |
GRIK1 |
Ki |
'=' |
701 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
EC50 |
'=' |
15000 |
nM |
| O15303 |
BXGT004150 |
Metabotropic glutamate receptor 6 |
reviewed |
G-protein coupled receptor |
GRM6 |
EC50 |
'=' |
20000 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
Ki |
'=' |
1360 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Emax |
'=' |
91 |
% |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Emax |
'=' |
94 |
% |
| P32738 |
BXGT009662 |
Choline O-acetyltransferase |
reviewed |
- |
Chat |
Control |
'=' |
78 |
% |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
Relative Potency Ratio |
'=' |
1 |
- |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
Relative Potency Ratio |
'=' |
1 |
- |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
Relative Potency Ratio |
'=' |
1 |
- |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
Relative Potency Ratio |
'=' |
1 |
- |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Relative Potency Ratio |
'=' |
1 |
- |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Relative Potency Ratio |
'=' |
1 |
- |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Relative Potency Ratio |
'=' |
1 |
- |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Relative Potency Ratio |
'=' |
1 |
- |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Relative Potency Ratio |
'=' |
1 |
- |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Relative Potency Ratio |
'=' |
1 |
- |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Relative Potency Ratio |
'=' |
1 |
- |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
Ki |
'=' |
1174897 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
3235 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
Ki |
'=' |
500 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
Ki |
'=' |
494 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
13870 |
nM |
| P70579 |
BXGT011675 |
Metabotropic glutamate receptor 8 |
reviewed |
- |
Grm8 |
EC50 |
'=' |
14010 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
Ki |
'=' |
1160 |
nM |
| Q13002 |
BXGT013303 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
Ion channel |
GRIK2 |
Activity |
- |
- |
- |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
Ki |
'=' |
140 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
EC50 |
'=' |
3660 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
331 |
nM |
| P19145 |
BXGT008463 |
General amino-acid permease GAP1 |
reviewed |
- |
GAP1 |
Activity |
- |
- |
- |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
2351 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
13650 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
Ki |
'=' |
1362 |
nM |
| P48058 |
BXGT010614 |
Glutamate receptor 4 |
reviewed |
Ion channel |
GRIA4 |
Ki |
'=' |
868 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
1800 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Ki |
'=' |
200 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Ki |
'=' |
200 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Ki |
'=' |
200 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Ki |
'=' |
200 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Ki |
'=' |
200 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Ki |
'=' |
200 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Ki |
'=' |
200 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
Ki |
'=' |
940 |
nM |
| P39086 |
BXGT010093 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
Ion channel |
GRIK1 |
EC50 |
'=' |
75000 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
EC50 |
'=' |
35200 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
2500 |
nM |
| P35349 |
BXGT009815 |
Metabotropic glutamate receptor 6 |
reviewed |
- |
Grm6 |
EC50 |
'=' |
7600 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ki |
'=' |
1400 |
nM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
Ki |
'=' |
63095 |
nM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
Ki |
'=' |
50118 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ki |
'=' |
6400 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
2880 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
EC50 |
'=' |
52000 |
nM |
| Q05BR4 |
BXGT012851 |
SLC16A10 protein |
unreviewed |
- |
SLC16A10 |
Activity |
- |
- |
- |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
16000 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
4000 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
12000 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
EC50 |
'=' |
9800 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
12589 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
EC50 |
'>' |
1000000 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
Ki |
'=' |
340 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ratio |
'=' |
5 |
- |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
EC50 |
'=' |
631000 |
nM |
| O15303 |
BXGT004150 |
Metabotropic glutamate receptor 6 |
reviewed |
G-protein coupled receptor |
GRM6 |
EC50 |
'=' |
270000 |
nM |
| P47743 |
BXGT010580 |
Metabotropic glutamate receptor 8 |
reviewed |
- |
Grm8 |
EC50 |
'=' |
22 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
3280 |
nM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
pKm |
'=' |
4 |
- |
| Q13002 |
BXGT013303 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
Ion channel |
GRIK2 |
EC50 |
'=' |
25000 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
EC50 |
'=' |
66000 |
nM |
| P31422 |
BXGT009540 |
Metabotropic glutamate receptor 3 |
reviewed |
- |
Grm3 |
EC50 |
'=' |
3000 |
nM |
| Q03469 |
BXGT012717 |
Glutamate racemase |
reviewed |
- |
murI |
Ki |
'=' |
28000 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
GSTCP activity |
- |
- |
- |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
GSTCP activity |
- |
- |
- |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
GSTCP activity |
- |
- |
- |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
GSTCP activity |
- |
- |
- |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
GSTCP activity |
- |
- |
- |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
GSTCP activity |
- |
- |
- |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
GSTCP activity |
- |
- |
- |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
Km |
'=' |
9900 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
11800 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Ki |
'=' |
870 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Ki |
'=' |
870 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Ki |
'=' |
870 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Ki |
'=' |
870 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Ki |
'=' |
870 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Ki |
'=' |
870 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Ki |
'=' |
870 |
nM |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
IC50 |
'=' |
700 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
IC50 |
'=' |
700 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
IC50 |
'=' |
700 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
IC50 |
'=' |
700 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
IC50 |
'=' |
700 |
nM |
| O15303 |
BXGT004150 |
Metabotropic glutamate receptor 6 |
reviewed |
G-protein coupled receptor |
GRM6 |
Ki |
'=' |
38000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
26000 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
Activity |
'=' |
5400000 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
EC50 |
'=' |
73000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Activity |
'=' |
4000 |
nM |
| Q836J0 |
BXGT017467 |
Glutamate racemase |
reviewed |
- |
murI |
Km |
'=' |
1200000 |
nM |
| Q836J0 |
BXGT017467 |
Glutamate racemase |
reviewed |
- |
murI |
Kcat |
'=' |
1500 |
/min |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
pKm |
'=' |
4 |
- |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
Ki |
'=' |
280 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
Ki |
'=' |
138 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
14000 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
EC50 |
'=' |
35000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
8500 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ki |
'=' |
17000 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Activity |
'=' |
1000 |
nM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
Km |
'=' |
21000 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
EC50 |
'=' |
156000 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
39810 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
2260 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
13000 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
5000 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
7300 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
Ki |
'=' |
3400 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ki |
'=' |
1200 |
nM |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
IC50 |
'=' |
270 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
IC50 |
'=' |
270 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
IC50 |
'=' |
270 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
IC50 |
'=' |
270 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
IC50 |
'=' |
270 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
EC50 |
'=' |
450 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
450 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
IC50 |
'=' |
150 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
IC50 |
'=' |
150 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
IC50 |
'=' |
150 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
IC50 |
'=' |
150 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
80 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
80 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
80 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
80 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
80 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
80 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
80 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
51000 |
nM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
pKm |
'=' |
5 |
- |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
IC50 |
'=' |
120 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
IC50 |
'=' |
120 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
IC50 |
'=' |
120 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
IC50 |
'=' |
120 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
IC50 |
'=' |
120 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Ki |
'=' |
9000 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Ki |
'=' |
570 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Ki |
'=' |
290 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Ki |
'=' |
290 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Ki |
'=' |
290 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Ki |
'=' |
290 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Ki |
'=' |
290 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Ki |
'=' |
290 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Ki |
'=' |
290 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
EC50 |
'=' |
3100 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
EC50 |
'=' |
117489 |
nM |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
Ki |
'=' |
42700 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
1 |
nM |
| P48058 |
BXGT010614 |
Glutamate receptor 4 |
reviewed |
Ion channel |
GRIA4 |
EC50 |
'=' |
3 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
140000 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
Ki |
'=' |
169 |
nM |
| Q04609 |
BXGT012768 |
Glutamate carboxypeptidase 2 |
reviewed |
Enzyme |
FOLH1 |
IC50 |
'=' |
428000 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
1200 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
EC50 |
'=' |
67000 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
18250 |
nM |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Kcat |
'=' |
107 |
/min |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
EC50 |
'=' |
2900 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
2900 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
332 |
nM |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Kcat |
'=' |
136 |
/min |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
EC50 |
'=' |
140000 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
50118 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
7400 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
172 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
172 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
172 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
172 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
172 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
172 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
172 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
EC50 |
'=' |
1 |
nM |
| P70579 |
BXGT011675 |
Metabotropic glutamate receptor 8 |
reviewed |
- |
Grm8 |
EC50 |
'=' |
8000 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Activity |
'=' |
12000 |
nM |
| P39086 |
BXGT010093 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
Ion channel |
GRIK1 |
Rmax |
'=' |
79 |
% |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
12000 |
nM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
Km |
'=' |
25000 |
nM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
pKm |
'=' |
4 |
- |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
1000 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
1000 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
1000 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
1000 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
1000 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
1000 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
1000 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
IC50 |
'=' |
214 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
IC50 |
'=' |
214 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
IC50 |
'=' |
214 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
IC50 |
'=' |
214 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
EC50 |
'=' |
19000 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
10000 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
56000 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
Km |
'=' |
9200 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
13803 |
nM |
| O15303 |
BXGT004150 |
Metabotropic glutamate receptor 6 |
reviewed |
G-protein coupled receptor |
GRM6 |
EC50 |
'=' |
4900 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
Ki |
'=' |
390 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
331 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ki |
'=' |
2400 |
nM |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Km |
'=' |
7430000 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
EC50 |
'=' |
1800 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
1800 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
1800 |
nM |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Km |
'=' |
740000 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
35000 |
nM |
| P04958 |
BXGT006288 |
Tetanus toxin |
reviewed |
- |
tetX |
Inhibition |
'=' |
0 |
% |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
IC50 |
'=' |
350 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
IC50 |
'=' |
350 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
IC50 |
'=' |
350 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
IC50 |
'=' |
350 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
IC50 |
'=' |
350 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
IC50 |
'=' |
500 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
IC50 |
'=' |
500 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
IC50 |
'=' |
500 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
IC50 |
'=' |
500 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
6200 |
nM |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
Ki |
'=' |
63 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
Ki |
'=' |
63 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
63 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
Ki |
'=' |
63 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
Ki |
'=' |
63 |
nM |
| P51907 |
BXGT010905 |
Excitatory amino acid transporter 3 |
reviewed |
- |
Slc1a1 |
Ks |
'=' |
5 |
uM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
6 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
1600 |
nM |
| P39086 |
BXGT010093 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
Ion channel |
GRIK1 |
EC50 |
'=' |
22000 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
9000 |
nM |
| Q13003 |
BXGT013304 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
Ion channel |
GRIK3 |
Ki |
'=' |
789 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
EC50 |
'=' |
140000 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
EC50 |
'=' |
190000 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
EC50 |
'=' |
130000 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
EC50 |
'=' |
16595 |
nM |
| P70579 |
BXGT011675 |
Metabotropic glutamate receptor 8 |
reviewed |
- |
Grm8 |
Ki |
'=' |
3400 |
nM |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
IC50 |
'=' |
53700 |
nM |
| Q9C0B1 |
BXGT020209 |
Alpha-ketoglutarate-dependent dioxygenase FTO |
reviewed |
- |
FTO |
IC50 |
'>' |
1000000 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
EC50 |
'=' |
21200 |
nM |
| P31422 |
BXGT009540 |
Metabotropic glutamate receptor 3 |
reviewed |
- |
Grm3 |
EC50 |
'=' |
60 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
IC50 |
'=' |
1200 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
IC50 |
'=' |
1200 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
IC50 |
'=' |
1200 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
IC50 |
'=' |
1200 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
EC50 |
'=' |
1050 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
6100 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
Ki |
'=' |
5400000 |
nM |
| O00222 |
BXGT003899 |
Metabotropic glutamate receptor 8 |
reviewed |
G-protein coupled receptor |
GRM8 |
Ki |
'=' |
9500 |
nM |
| Q13002 |
BXGT013303 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
Ion channel |
GRIK2 |
Rmax |
- |
- |
- |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
Rmax |
'=' |
51 |
% |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
Ki |
'=' |
249 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
Ki |
'=' |
4677 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
610 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
Ki |
'=' |
1100 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
Ki |
'=' |
1100 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
Ki |
'=' |
1100 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
Ki |
'=' |
1100 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Ki |
'=' |
57 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
EC50 |
'=' |
1180000 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
EC50 |
'=' |
3200 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Potency |
- |
20596 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 ratio |
'=' |
1 |
- |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
10000 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
Ki |
'=' |
490 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
EC50 |
'=' |
1778 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
1778 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
EC50 |
'=' |
1800 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
Activity |
- |
- |
- |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
IC50 |
'=' |
613 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
IC50 |
'=' |
613 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
IC50 |
'=' |
613 |
nM |
| P48058 |
BXGT010614 |
Glutamate receptor 4 |
reviewed |
Ion channel |
GRIA4 |
IC50 |
'=' |
613 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
3000 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
10621 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ki |
'=' |
11000 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
EC50 |
'=' |
120 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
EC50 |
'=' |
120 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
EC50 |
'=' |
120 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
EC50 |
'=' |
120 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
EC50 |
'=' |
120 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
EC50 |
'=' |
120 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
120 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Ki |
'=' |
250 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
EC50 |
'=' |
102329 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
69 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
69 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
69 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
69 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
69 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
69 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
69 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
171 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
171 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
171 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
171 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
171 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
171 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
171 |
nM |
| P31596 |
BXGT009553 |
Excitatory amino acid transporter 2 |
reviewed |
- |
Slc1a2 |
Control |
- |
- |
- |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
8492 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
6160 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
6160 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
EC50 |
'=' |
4900 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
3200 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
EC50 |
'=' |
4100 |
nM |
| P35349 |
BXGT009815 |
Metabotropic glutamate receptor 6 |
reviewed |
- |
Grm6 |
EC50 |
'=' |
16000 |
nM |
| P35400 |
BXGT009826 |
Metabotropic glutamate receptor 7 |
reviewed |
- |
Grm7 |
EC50 |
'=' |
1300000 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
70 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
70 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
70 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
70 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
70 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
70 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
70 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
pKm |
'=' |
5 |
- |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
12570 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ratio |
'=' |
20 |
- |
| O15303 |
BXGT004150 |
Metabotropic glutamate receptor 6 |
reviewed |
G-protein coupled receptor |
GRM6 |
Activity |
'=' |
20000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ki |
'=' |
12000 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
71000 |
nM |
| P48058 |
BXGT010614 |
Glutamate receptor 4 |
reviewed |
Ion channel |
GRIA4 |
EC50 |
'=' |
28000 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
Ki |
'=' |
281 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
4400 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
4700 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
Km |
'=' |
7900 |
nM |
| P35400 |
BXGT009826 |
Metabotropic glutamate receptor 7 |
reviewed |
- |
Grm7 |
EC50 |
'=' |
1000000 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
EC50 |
'>' |
500000 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
6400 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
IC50 |
'=' |
410 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
IC50 |
'=' |
410 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
IC50 |
'=' |
410 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
IC50 |
'=' |
410 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
IC50 |
'=' |
410 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
IC50 |
'=' |
410 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
IC50 |
'=' |
410 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
EC50 |
'=' |
17000 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
Ki |
'=' |
31622 |
nM |
| Q8TCU5 |
BXGT018802 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
Ion channel |
GRIN3A |
IC50 |
'=' |
70 |
nM |
| Q14957 |
BXGT013514 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
Ion channel |
GRIN2C |
IC50 |
'=' |
70 |
nM |
| O60391 |
BXGT004874 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
Ion channel |
GRIN3B |
IC50 |
'=' |
70 |
nM |
| O15399 |
BXGT004164 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
Ion channel |
GRIN2D |
IC50 |
'=' |
70 |
nM |
| Q13224 |
BXGT013328 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
Ion channel |
GRIN2B |
IC50 |
'=' |
70 |
nM |
| Q12879 |
BXGT013275 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
Ion channel |
GRIN2A |
IC50 |
'=' |
70 |
nM |
| Q05586 |
BXGT012826 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
Ion channel |
GRIN1 |
IC50 |
'=' |
70 |
nM |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
Relative potency |
'=' |
1 |
- |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
Relative potency |
'=' |
1 |
- |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Relative potency |
'=' |
1 |
- |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
Relative potency |
'=' |
1 |
- |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
Relative potency |
'=' |
1 |
- |
| Q63273 |
BXGT016064 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
- |
Grik5 |
IC50 |
'=' |
400 |
nM |
| P42264 |
BXGT010296 |
Glutamate receptor ionotropic, kainate 3 |
reviewed |
- |
Grik3 |
IC50 |
'=' |
400 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
IC50 |
'=' |
400 |
nM |
| Q01812 |
BXGT012617 |
Glutamate receptor ionotropic, kainate 4 |
reviewed |
- |
Grik4 |
IC50 |
'=' |
400 |
nM |
| P22756 |
BXGT008804 |
Glutamate receptor ionotropic, kainate 1 |
reviewed |
- |
Grik1 |
IC50 |
'=' |
400 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Emax |
'=' |
105 |
% |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
18000 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
18000 |
nM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
IC50 |
'=' |
52000 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
4182 |
nM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
Ki |
'=' |
51 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
33 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
Ki |
'=' |
330 |
nM |
| Q62795 |
BXGT016045 |
Sodium-dependent phosphate transport protein 1 |
reviewed |
- |
Slc17a1 |
Activity |
'=' |
29 |
% |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
Activity |
'=' |
4000 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Activity |
'=' |
9000 |
nM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
Ki |
'=' |
62000 |
nM |
| Q16478 |
BXGT013630 |
Glutamate receptor ionotropic, kainate 5 |
reviewed |
Ion channel |
GRIK5 |
Ki |
'=' |
701 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
7 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
290 |
nM |
| P42261 |
BXGT010293 |
Glutamate receptor 1 |
reviewed |
Ion channel |
GRIA1 |
EC50 |
'=' |
22000 |
nM |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
2190 |
nM |
| O00222 |
BXGT003899 |
Metabotropic glutamate receptor 8 |
reviewed |
G-protein coupled receptor |
GRM8 |
IC50 |
'=' |
5 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Ki |
'=' |
10000 |
nM |
| P42260 |
BXGT010292 |
Glutamate receptor ionotropic, kainate 2 |
reviewed |
- |
Grik2 |
EC50 |
'=' |
58884 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Emax |
'=' |
88 |
% |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
EC50 |
'=' |
19600 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
1002 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 ratio |
'=' |
1 |
- |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
IC50 |
'=' |
32000 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
Ki |
'=' |
7400 |
nM |
| P53987 |
BXGT011023 |
Monocarboxylate transporter 1 |
reviewed |
- |
Slc16a1 |
Activity |
- |
- |
- |
| Q91Y77 |
BXGT019323 |
Monocarboxylate transporter 10 |
reviewed |
- |
Slc16a10 |
Activity |
- |
- |
- |
| P42262 |
BXGT010294 |
Glutamate receptor 2 |
reviewed |
Ion channel |
GRIA2 |
EC50 |
'=' |
11000 |
nM |
| P42263 |
BXGT010295 |
Glutamate receptor 3 |
reviewed |
Ion channel |
GRIA3 |
EC50 |
'=' |
11000 |
nM |
| P35349 |
BXGT009815 |
Metabotropic glutamate receptor 6 |
reviewed |
- |
Grm6 |
EC50 |
'=' |
65090 |
nM |
| P31422 |
BXGT009540 |
Metabotropic glutamate receptor 3 |
reviewed |
- |
Grm3 |
EC50 |
'=' |
3400 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
12500 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
EC50 |
'=' |
14700 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
EC50 |
'=' |
1600 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
32359 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Emax |
'=' |
104 |
% |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
1827 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Activity |
- |
- |
- |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
60 |
nM |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Kcat |
'=' |
63 |
/min |
| P56068 |
BXGT011141 |
Glutamate racemase |
reviewed |
- |
murI |
Km |
'=' |
7360000 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
Ki |
'=' |
282 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
Ki |
'=' |
354 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
- |
- |
- |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
7079 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
EC50 |
'=' |
4700 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
14581 |
nM |
| P35400 |
BXGT009826 |
Metabotropic glutamate receptor 7 |
reviewed |
- |
Grm7 |
EC50 |
- |
- |
- |
| P08909 |
BXGT006838 |
5-hydroxytryptamine receptor 2C |
reviewed |
- |
Htr2c |
Activity |
- |
- |
- |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
EC50 |
'=' |
100000 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
Ki |
'=' |
35000 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
EC50 |
'=' |
1000 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
EC50 |
'=' |
1000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
12589 |
nM |
| P41594 |
BXGT010266 |
Metabotropic glutamate receptor 5 |
reviewed |
G-protein coupled receptor |
GRM5 |
Ki |
'=' |
11400 |
nM |
| P19492 |
BXGT008490 |
Glutamate receptor 3 |
reviewed |
- |
Gria3 |
EC50 |
'=' |
1300 |
nM |
| P19493 |
BXGT008491 |
Glutamate receptor 4 |
reviewed |
- |
Gria4 |
EC50 |
'=' |
20000 |
nM |
| Q13255 |
BXGT013332 |
Metabotropic glutamate receptor 1 |
reviewed |
G-protein coupled receptor |
GRM1 |
Ki |
'=' |
1584 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Emax |
'=' |
93 |
% |
| Q01650 |
BXGT012603 |
Large neutral amino acids transporter small subunit 1 |
reviewed |
Transporter |
SLC7A5 |
Inhibition |
'=' |
-2 |
% |
| O35921 |
BXGT026125 |
Excitatory amino acid transporter 4 |
reviewed |
- |
Slc1a6 |
IC50 |
'=' |
13000 |
nM |
| P19491 |
BXGT008489 |
Glutamate receptor 2 |
reviewed |
- |
Gria2 |
EC50 |
'=' |
7 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Inhibition |
'=' |
10 |
% |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Inhibition |
'=' |
10 |
% |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Inhibition |
'=' |
10 |
% |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Inhibition |
'=' |
10 |
% |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Inhibition |
'=' |
10 |
% |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Inhibition |
'=' |
10 |
% |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Inhibition |
'=' |
10 |
% |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
Emax |
'=' |
111 |
% |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
1767 |
nM |
| Q9R1M7 |
BXGT021417 |
Glutamate receptor ionotropic, NMDA 3A |
reviewed |
- |
Grin3a |
Ki |
'=' |
370 |
nM |
| Q8VHN2 |
BXGT018931 |
Glutamate receptor ionotropic, NMDA 3B |
reviewed |
- |
Grin3b |
Ki |
'=' |
370 |
nM |
| Q62645 |
BXGT016035 |
Glutamate receptor ionotropic, NMDA 2D |
reviewed |
- |
Grin2d |
Ki |
'=' |
370 |
nM |
| Q00961 |
BXGT012556 |
Glutamate receptor ionotropic, NMDA 2C |
reviewed |
- |
Grin2c |
Ki |
'=' |
370 |
nM |
| Q00960 |
BXGT012555 |
Glutamate receptor ionotropic, NMDA 2B |
reviewed |
- |
Grin2b |
Ki |
'=' |
370 |
nM |
| Q00959 |
BXGT012554 |
Glutamate receptor ionotropic, NMDA 2A |
reviewed |
- |
Grin2a |
Ki |
'=' |
370 |
nM |
| P35439 |
BXGT009831 |
Glutamate receptor ionotropic, NMDA 1 |
reviewed |
- |
Grin1 |
Ki |
'=' |
370 |
nM |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
IC50 |
'=' |
11000 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Ki |
'=' |
1819 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ki |
'=' |
1600 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
EC50 |
'=' |
2575 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
23160 |
nM |
| P35400 |
BXGT009826 |
Metabotropic glutamate receptor 7 |
reviewed |
- |
Grm7 |
EC50 |
'>' |
100000 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
1484 |
nM |
| P70579 |
BXGT011675 |
Metabotropic glutamate receptor 8 |
reviewed |
- |
Grm8 |
EC50 |
'=' |
21470 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
'=' |
5118 |
nM |
| Q14833 |
BXGT013508 |
Metabotropic glutamate receptor 4 |
reviewed |
G-protein coupled receptor |
GRM4 |
Ki |
'=' |
3235 |
nM |
| Q14831 |
BXGT013506 |
Metabotropic glutamate receptor 7 |
reviewed |
G-protein coupled receptor |
GRM7 |
EC50 |
'=' |
1180 |
nM |
| P23385 |
BXGT008861 |
Metabotropic glutamate receptor 1 |
reviewed |
- |
Grm1 |
EC50 |
'=' |
1584 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
4677 |
nM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
8990 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
13080 |
nM |
| Q14832 |
BXGT013507 |
Metabotropic glutamate receptor 3 |
reviewed |
G-protein coupled receptor |
GRM3 |
EC50 |
- |
- |
- |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
16090 |
nM |
| P31421 |
BXGT009539 |
Metabotropic glutamate receptor 2 |
reviewed |
- |
Grm2 |
EC50 |
'=' |
1819 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
KA |
'=' |
6 |
uM |
| P43004 |
BXGT010348 |
Excitatory amino acid transporter 2 |
reviewed |
Transporter |
SLC1A2 |
IC50 |
'=' |
52480 |
nM |
| Q01650 |
BXGT012603 |
Large neutral amino acids transporter small subunit 1 |
reviewed |
Transporter |
SLC7A5 |
Activity |
'=' |
27 |
% |
| P43003 |
BXGT010347 |
Excitatory amino acid transporter 1 |
reviewed |
Transporter |
SLC1A3 |
IC50 |
'=' |
11481 |
nM |
| P16638 |
BXGT008250 |
ATP-citrate synthase |
reviewed |
- |
Acly |
Ki |
'=' |
300000 |
nM |
| P19490 |
BXGT008488 |
Glutamate receptor 1 |
reviewed |
- |
Gria1 |
EC50 |
'=' |
3400 |
nM |
| Q4CVY4 |
BXGT026093 |
Carbonic anhydrase-like protein, putative |
unreviewed |
- |
Tc00.1047053509597.20 |
KA |
'>' |
100 |
uM |
| P31424 |
BXGT009542 |
Metabotropic glutamate receptor 5 |
reviewed |
- |
Grm5 |
EC50 |
'=' |
4700 |
nM |
| Q14416 |
BXGT013468 |
Metabotropic glutamate receptor 2 |
reviewed |
G-protein coupled receptor |
GRM2 |
Activity |
- |
- |
- |
| P35349 |
BXGT009815 |
Metabotropic glutamate receptor 6 |
reviewed |
- |
Grm6 |
EC50 |
'=' |
82210 |
nM |
| O35921 |
BXGT026125 |
Excitatory amino acid transporter 4 |
reviewed |
- |
Slc1a6 |
IC50 |
'=' |
13182 |
nM |
| P31423 |
BXGT009541 |
Metabotropic glutamate receptor 4 |
reviewed |
- |
Grm4 |
EC50 |
'=' |
9490 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
KA |
'>' |
100 |
uM |
| P43005 |
BXGT010349 |
Excitatory amino acid transporter 3 |
reviewed |
Transporter |
SLC1A1 |
IC50 |
'=' |
32359 |
nM |