| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
10 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
10000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
50118 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
8800 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
- |
- |
- |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
35481 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Ki |
'=' |
123000 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
Ki |
- |
- |
- |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
Ki |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Ki |
- |
- |
- |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
Ki |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
Ki |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
Ki |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
Ki |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
Ki |
- |
- |
- |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio |
'=' |
32 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio |
'=' |
32 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
REP |
'=' |
0 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
'=' |
24 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
4660 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
%max |
'=' |
95 |
% |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
Fluorescence intensity |
'=' |
12723 |
- |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
IC50 |
'=' |
2610 |
nM |
| O60656 |
BXGT004889 |
UDP-glucuronosyltransferase 1-9 |
reviewed |
- |
UGT1A9 |
Activity |
'=' |
0 |
nmol/mg.min |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
10000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
6900 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
5000 |
nM |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
12589 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Thermal melting change |
'=' |
2 |
degrees C |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Thermal melting change |
'=' |
4 |
degrees C |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
36000 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
98 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Selectivity |
'=' |
47 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Selectivity |
'=' |
47 |
- |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Ki |
'=' |
2960 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
83300 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
20000 |
nM |
| Q09013 |
BXGT013023 |
Myotonin-protein kinase |
reviewed |
Kinase |
DMPK |
Thermal melting change |
'=' |
2 |
degrees C |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
Ki |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
Ki |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
IC50 |
'=' |
10469 |
nM |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
IC50 |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
IC50 |
- |
- |
- |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
21331 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
501 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
25118 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
56234 |
nM |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Thermal melting change |
'=' |
0 |
degrees C |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
IC50 |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
IC50 |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
Ki |
- |
- |
- |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
Ki |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
IC50 |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
Ki |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
IC50 |
- |
- |
- |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
Ki |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
IC50 |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
Ki |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
Ki |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
'=' |
39 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ki |
- |
- |
- |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
Ki |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
Ki |
- |
- |
- |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
'=' |
9033 |
nM |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
Ki |
- |
- |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
- |
- |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
11885 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
370000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
370000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
ug.mL-1 |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
20 |
ug.mL-1 |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
4 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
92 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
89125 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
0 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
14125 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
1122 |
nM |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Tm |
'<' |
2 |
degrees C |
| O75828 |
BXGT005154 |
Carbonyl reductase [NADPH] 3 |
reviewed |
- |
CBR3 |
Tm |
'<' |
2 |
degrees C |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
77100 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
134400 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
501 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
63 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
1 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
18 |
nM |
| Q99986 |
BXGT019980 |
Serine/threonine-protein kinase VRK1 |
reviewed |
Kinase |
VRK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Ka |
'=' |
0 |
10'5/M |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
28 |
nmol/min |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
2 |
- |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
IC50 |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
- |
- |
- |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Ki |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
Ki |
- |
- |
- |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
Ki |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
Ki |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
Ki |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
IC50 |
- |
- |
- |
| P15127 |
BXGT008085 |
Insulin receptor |
reviewed |
- |
Insr |
IC50 |
- |
- |
- |
| Q9JKC1 |
BXGT020830 |
Carboxylic ester hydrolase |
unreviewed |
- |
Bche |
Inhibition |
'<' |
5 |
% |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
Ki |
- |
- |
- |
| O00506 |
BXGT003932 |
Serine/threonine-protein kinase 25 |
reviewed |
Kinase |
STK25 |
Thermal melting change |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
'=' |
4 |
uM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
'=' |
4 |
uM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'=' |
16500 |
nM |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
Ki |
- |
- |
- |
| P13945 |
BXGT007972 |
Beta-3 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB3 |
Ki |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
44979 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
232500 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
Ki |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Ki |
- |
- |
- |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
26 |
nmol/min |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
IC50 |
- |
- |
- |
| P31645 |
BXGT009558 |
Sodium-dependent serotonin transporter |
reviewed |
Transporter |
SLC6A4 |
IC50 |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
IC50 |
'=' |
7720 |
nM |
| P07550 |
BXGT006636 |
Beta-2 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB2 |
IC50 |
- |
- |
- |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
Ki |
- |
- |
- |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
IC50 |
- |
- |
- |
| P51681 |
BXGT010878 |
C-C chemokine receptor type 5 |
reviewed |
G-protein coupled receptor |
CCR5 |
IC50 |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
- |
- |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
IC50 |
- |
- |
- |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
2520 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
16 |
% |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
Activity |
- |
- |
- |
| P56937 |
BXGT011205 |
3-keto-steroid reductase |
reviewed |
- |
HSD17B7 |
Inhibition |
'=' |
0 |
% |
| P08912 |
BXGT006840 |
Muscarinic acetylcholine receptor M5 |
reviewed |
G-protein coupled receptor |
CHRM5 |
IC50 |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
Ki |
- |
- |
- |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Ratio |
'=' |
1 |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ratio |
'=' |
23 |
- |
| Q27686 |
BXGT013930 |
Pyruvate kinase |
reviewed |
- |
PYK |
Potency |
'=' |
12589 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
10000 |
nM |
| P90584 |
BXGT012110 |
MO15-related protein kinase Pfmrk |
unreviewed |
- |
Pfmrk |
IC50 |
'=' |
93000 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
IC50 |
'=' |
1300000 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Thermal melting change |
'=' |
1 |
degrees C |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
39000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
2150 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
1000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Selectivity |
'=' |
41 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Selectivity |
'=' |
41 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Fold selectivity |
'=' |
41 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio EC50 |
'=' |
13 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio EC50 |
'=' |
13 |
- |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
35050 |
nM |
| P18825 |
BXGT008426 |
Alpha-2C adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2C |
IC50 |
- |
- |
- |
| P23975 |
BXGT008935 |
Sodium-dependent noradrenaline transporter |
reviewed |
Transporter |
SLC6A2 |
IC50 |
- |
- |
- |
| P32238 |
BXGT009611 |
Cholecystokinin receptor type A |
reviewed |
G-protein coupled receptor |
CCKAR |
IC50 |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
IC50 |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
135 |
nM |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
IC50 |
- |
- |
- |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
19952 |
nM |
| P34158 |
BXGT009754 |
Cystic fibrosis transmembrane conductance regulator |
reviewed |
- |
Cftr |
Kd |
'=' |
40000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
ug.mL-1 |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Kq |
'=' |
0 |
10'12/M/s |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Fluorescence intensity |
'=' |
148 |
% |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
15848 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
900 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
900 |
nM |
| P04035 |
BXGT006129 |
3-hydroxy-3-methylglutaryl-coenzyme A reductase |
reviewed |
- |
HMGCR |
IC50 |
- |
- |
- |
| Q9Y271 |
BXGT022222 |
Cysteinyl leukotriene receptor 1 |
reviewed |
G-protein coupled receptor |
CYSLTR1 |
Ki |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
IC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
IC50 |
- |
- |
- |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
IC50 |
- |
- |
- |
| P51151 |
BXGT010837 |
Ras-related protein Rab-9A |
reviewed |
- |
RAB9A |
Potency |
'=' |
12589 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
3162 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
9 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
ug.mL-1 |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Inhibition |
'=' |
0 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
25 |
nM |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
380000 |
nM |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
5804 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
12589 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
80 |
% |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
16353 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
48 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
IC50 |
'>' |
70000 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
95 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1000 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Fluorescence intensity |
'=' |
12 |
- |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Fluorescence intensity |
'=' |
0 |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Fluorescence intensity |
'=' |
95 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
395 |
nM |
| P20309 |
BXGT008562 |
Muscarinic acetylcholine receptor M3 |
reviewed |
G-protein coupled receptor |
CHRM3 |
Ki |
- |
- |
- |
| P49146 |
BXGT010681 |
Neuropeptide Y receptor type 2 |
reviewed |
G-protein coupled receptor |
NPY2R |
IC50 |
- |
- |
- |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Fluorescence intensity |
'=' |
0 |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Fluorescence intensity |
'=' |
7 |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
31 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
31 |
% |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
77 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
77 |
% |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
66 |
% |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
Ki |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
Ki |
- |
- |
- |
| Q99720 |
BXGT019955 |
Sigma non-opioid intracellular receptor 1 |
reviewed |
- |
SIGMAR1 |
IC50 |
- |
- |
- |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
16944 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
65 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
65 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
200 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
45900 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Selectivity |
'=' |
0 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Selectivity |
'=' |
0 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
6 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
7943 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'=' |
75000 |
nM |
| P11474 |
BXGT007710 |
Steroid hormone receptor ERR1 |
reviewed |
Nuclear receptor |
ESRRA |
IC50 |
'=' |
10 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
'=' |
80000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
12589 |
nM |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
1584 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
29 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio IC50 |
'=' |
22 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio IC50 |
'=' |
22 |
- |
| P14618 |
BXGT008027 |
Pyruvate kinase PKM |
reviewed |
Kinase |
PKM |
Potency |
'=' |
25118 |
nM |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
IC50 |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
IC50 |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
IC50 |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
IC50 |
- |
- |
- |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
35481 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
10 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
5011 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23109 |
nM |
| P04278 |
BXGT006182 |
Sex hormone-binding globulin |
reviewed |
- |
SHBG |
Kd |
'=' |
39810 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
3 |
- |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
31622 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
22387 |
nM |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Thermal melting change |
'=' |
0 |
degrees C |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
810 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
8912 |
nM |
| P02791 |
BXGT005965 |
Ferritin light chain |
reviewed |
- |
FTL |
Potency |
'=' |
39810 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
11220 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio IC50 |
'=' |
45 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio IC50 |
'=' |
45 |
- |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Inhibition |
- |
- |
- |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
12589 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio |
'=' |
19 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio |
'=' |
19 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Control |
'<' |
171 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Control |
'<' |
171 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Control |
'<' |
197 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Control |
'<' |
197 |
% |
| Q06278 |
BXGT012869 |
Aldehyde oxidase |
reviewed |
Enzyme |
AOX1 |
IC50 |
'=' |
340 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
580 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
11220 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
9688 |
nM |
| Q62986 |
BXGT016053 |
Estrogen receptor beta |
reviewed |
- |
Esr2 |
Agonistic activity |
'=' |
63 |
% |
| P06211 |
BXGT006424 |
Estrogen receptor |
reviewed |
- |
Esr1 |
Agonistic activity |
'=' |
63 |
% |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
23 |
% |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
IC50 |
'=' |
10400 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
- |
- |
- |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'>' |
20000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio |
'=' |
41 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio |
'=' |
41 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio |
'=' |
16 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio |
'=' |
16 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
950 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Ki |
'=' |
100000 |
nM |
| Q8IV63 |
BXGT018341 |
Inactive serine/threonine-protein kinase VRK3 |
reviewed |
Kinase |
VRK3 |
Thermal melting change |
'=' |
1 |
degrees C |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
1145 |
nM |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Kcat |
'=' |
0 |
10'3/s |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
4466 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
3 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
395 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
1995 |
nM |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
97 |
% |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Thermal melting change |
'=' |
0 |
degrees C |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
35481 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Activity |
'=' |
10 |
% |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
17 |
% |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Thermal melting change |
'=' |
0 |
degrees C |
| P11166 |
BXGT007661 |
Solute carrier family 2, facilitated glucose transporter member 1 |
reviewed |
Transporter |
SLC2A1 |
Ki |
'=' |
7000 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
1100 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Drug transport |
- |
- |
- |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
Inhibition |
'=' |
96 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
Inhibition |
'=' |
96 |
% |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
Control |
'=' |
43 |
% |
| P30411 |
BXGT009424 |
B2 bradykinin receptor |
reviewed |
G-protein coupled receptor |
BDKRB2 |
IC50 |
- |
- |
- |
| P35367 |
BXGT009821 |
Histamine H1 receptor |
reviewed |
G-protein coupled receptor |
HRH1 |
Ki |
- |
- |
- |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
- |
- |
- |
| P15823 |
BXGT008160 |
Alpha-1B adrenergic receptor |
reviewed |
- |
Adra1b |
IC50 |
- |
- |
- |
| P35462 |
BXGT009835 |
D(3) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD3 |
IC50 |
- |
- |
- |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
Ki |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ki |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
IC50 |
- |
- |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ki |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
IC50 |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
IC50 |
'=' |
14910 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
5308 |
nM |
| P14142 |
BXGT007989 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
IC50 |
'=' |
20000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2600 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
4 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ki |
'=' |
370 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Fluorescence intensity |
'=' |
67 |
% |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Fluorescence intensity |
'=' |
20 |
- |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
7000 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
7079 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
28 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Displacement |
'=' |
20 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
1 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
25118 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
% |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
4645 |
nM |
| P26358 |
BXGT009104 |
DNA (cytosine-5)-methyltransferase 1 |
reviewed |
Epigenetic regulator |
DNMT1 |
IC50 |
'=' |
30000 |
nM |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Thermal melting change |
'=' |
1 |
degrees C |
| P51813 |
BXGT010894 |
Cytoplasmic tyrosine-protein kinase BMX |
reviewed |
Kinase |
BMX |
IC50 |
'=' |
67990 |
nM |
| P41597 |
BXGT010268 |
C-C chemokine receptor type 2 |
reviewed |
- |
CCR2 |
Ki |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Ki |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
- |
- |
- |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Ki |
- |
- |
- |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
Ki |
- |
- |
- |
| P33032 |
BXGT009689 |
Melanocortin receptor 5 |
reviewed |
G-protein coupled receptor |
MC5R |
IC50 |
- |
- |
- |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
Ki |
- |
- |
- |
| P25929 |
BXGT009078 |
Neuropeptide Y receptor type 1 |
reviewed |
G-protein coupled receptor |
NPY1R |
Ki |
- |
- |
- |
| P25105 |
BXGT009021 |
Platelet-activating factor receptor |
reviewed |
G-protein coupled receptor |
PTAFR |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Ki |
- |
- |
- |
| P08575 |
BXGT006793 |
Receptor-type tyrosine-protein phosphatase C |
reviewed |
Enzyme |
PTPRC |
Ki |
- |
- |
- |
| P28223 |
BXGT009239 |
5-hydroxytryptamine receptor 2A |
reviewed |
G-protein coupled receptor |
HTR2A |
Ki |
'=' |
2991 |
nM |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
IC50 |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
IC50 |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
IC50 |
- |
- |
- |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
50118 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
12589 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
956 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
390 |
nM |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Fluorescence intensity |
'=' |
0 |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
7943 |
nM |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
Ki |
- |
- |
- |
| Q12809 |
BXGT013267 |
Potassium voltage-gated channel subfamily H member 2 |
reviewed |
Ion channel |
KCNH2 |
IC50 |
- |
- |
- |
| Q690N0 |
BXGT016199 |
Progesterone receptor |
unreviewed |
- |
PGR |
Ki |
- |
- |
- |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
- |
- |
- |
| P24557 |
BXGT008976 |
Thromboxane-A synthase |
reviewed |
- |
TBXAS1 |
Ki |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
IC50 |
'=' |
17442 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
398 |
nM |
| P21554 |
BXGT008662 |
Cannabinoid receptor 1 |
reviewed |
G-protein coupled receptor |
CNR1 |
IC50 |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
- |
- |
- |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
IC50 |
'=' |
16918 |
nM |
| Q01959 |
BXGT012624 |
Sodium-dependent dopamine transporter |
reviewed |
Transporter |
SLC6A3 |
Ki |
'=' |
13442 |
nM |
| O95718 |
BXGT005392 |
Steroid hormone receptor ERR2 |
reviewed |
Nuclear receptor |
ESRRB |
IC50 |
'=' |
395 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| O95747 |
BXGT005393 |
Serine/threonine-protein kinase OSR1 |
reviewed |
Kinase |
OXSR1 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9BVS4 |
BXGT020147 |
Serine/threonine-protein kinase RIO2 |
reviewed |
Kinase |
RIOK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
10 |
% |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
Ki |
'=' |
10400 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
22387 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
300 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
30 |
ug.mL-1 |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
101 |
% |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'>' |
1000000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
20 |
nM |
| P11229 |
BXGT007676 |
Muscarinic acetylcholine receptor M1 |
reviewed |
G-protein coupled receptor |
CHRM1 |
IC50 |
- |
- |
- |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
IC50 |
- |
- |
- |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
IC50 |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Ki |
- |
- |
- |
| Q08209 |
BXGT012968 |
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform |
reviewed |
- |
PPP3CA |
Ki |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
Ki |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
990 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
990 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
25118 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
6 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
15848 |
nM |
| P08173 |
BXGT006738 |
Muscarinic acetylcholine receptor M4 |
reviewed |
G-protein coupled receptor |
CHRM4 |
Ki |
- |
- |
- |
| P19327 |
BXGT008472 |
5-hydroxytryptamine receptor 1A |
reviewed |
- |
Htr1a |
IC50 |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
Ki |
- |
- |
- |
| P0AEK4 |
BXGT007320 |
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI |
reviewed |
- |
fabI |
Activity |
- |
- |
- |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
19952 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
9 |
nM |
| P24385 |
BXGT008965 |
G1/S-specific cyclin-D1 |
reviewed |
Enzyme modulator |
CCND1 |
IC50 |
'=' |
250000 |
nM |
| P11802 |
BXGT007750 |
Cyclin-dependent kinase 4 |
reviewed |
Kinase |
CDK4 |
IC50 |
'=' |
250000 |
nM |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
Activity |
'=' |
3 |
uA.cm'-2 |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
RBA |
'=' |
7 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
- |
2511 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio |
'=' |
3 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio |
'=' |
3 |
- |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'>' |
10000 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
61 |
nM |
| Q00532 |
BXGT012532 |
Cyclin-dependent kinase-like 1 |
reviewed |
Kinase |
CDKL1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
Ki |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
IC50 |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
Ki |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
IC50 |
- |
- |
- |
| P11509 |
BXGT007716 |
Cytochrome P450 2A6 |
reviewed |
- |
CYP2A6 |
Ki |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
- |
- |
- |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Ki |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
IC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
- |
- |
- |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
IC50 |
- |
- |
- |
| P25021 |
BXGT009004 |
Histamine H2 receptor |
reviewed |
G-protein coupled receptor |
HRH2 |
IC50 |
- |
- |
- |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
156 |
% |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
'=' |
2210 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
% |
| P47199 |
BXGT010568 |
Quinone oxidoreductase |
reviewed |
- |
Cryz |
CD |
'=' |
22 |
uM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
35481 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
- |
- |
- |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
1973 |
nM |
| P42684 |
BXGT010331 |
Tyrosine-protein kinase ABL2 |
reviewed |
Kinase |
ABL2 |
IC50 |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
IC50 |
'>' |
10000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
3920 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Ratio IC50 |
'=' |
32 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ratio IC50 |
'=' |
32 |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
'=' |
85113 |
nM |
| P08172 |
BXGT006737 |
Muscarinic acetylcholine receptor M2 |
reviewed |
G-protein coupled receptor |
CHRM2 |
IC50 |
- |
- |
- |
| P29476 |
BXGT009354 |
Nitric oxide synthase, brain |
reviewed |
- |
Nos1 |
IC50 |
- |
- |
- |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
IC50 |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
- |
- |
- |
| P50406 |
BXGT010796 |
5-hydroxytryptamine receptor 6 |
reviewed |
G-protein coupled receptor |
HTR6 |
Ki |
- |
- |
- |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
IC50 |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
Ki |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
11220 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'>' |
100000 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Efficacy |
'=' |
115 |
% |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Km |
'=' |
330000 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
%max |
'=' |
172 |
% |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
logIC50 |
'=' |
1 |
- |
| P11344 |
BXGT007687 |
Tyrosinase |
reviewed |
- |
Tyr |
IC50 |
'>' |
500000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
IC50 |
'=' |
10000 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
10000 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
9196 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
3 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
%max |
'=' |
93 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
4680 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
0 |
nmol/mg.min |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
191 |
% |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
12990 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
RBA |
'=' |
6 |
% |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
RBA |
'=' |
13 |
% |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Thermal melting change |
'=' |
1 |
degrees C |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Activity |
'=' |
105 |
% |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
IC50 |
'=' |
19904 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
73 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
1300 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
83 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
22387 |
nM |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Inhibition |
'=' |
67 |
% |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
19952 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
16360 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Ratio IC50 |
'=' |
1400 |
- |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Ratio |
'=' |
10000 |
- |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
3548 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
39810 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
IC50 |
- |
- |
- |
| P18089 |
BXGT008379 |
Alpha-2B adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2B |
Ki |
- |
- |
- |
| P08588 |
BXGT006795 |
Beta-1 adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRB1 |
Ki |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Ki |
- |
- |
- |
| P30988 |
BXGT009491 |
Calcitonin receptor |
reviewed |
G-protein coupled receptor |
CALCR |
IC50 |
- |
- |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
- |
- |
- |
| P05181 |
BXGT006337 |
Cytochrome P450 2E1 |
reviewed |
- |
CYP2E1 |
Ki |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Ki |
'=' |
0 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
6100 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
98000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
13335 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
REP |
'=' |
0 |
% |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
84 |
% |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
71 |
% |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
25118 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
39810 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
- |
3 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
11220 |
nM |
| P25100 |
BXGT009017 |
Alpha-1D adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA1D |
Ki |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
IC50 |
- |
- |
- |
| P50052 |
BXGT010768 |
Type-2 angiotensin II receptor |
reviewed |
G-protein coupled receptor |
AGTR2 |
Ki |
- |
- |
- |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
- |
- |
- |
| P14416 |
BXGT008011 |
D(2) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD2 |
Ki |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
2 |
nM |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
5102 |
nM |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
8 |
nmol/min |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
1584 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
15848 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
480 |
nM |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Fluorescence intensity |
'=' |
112 |
% |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
- |
9074 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
22387 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| A6XA80 |
BXGT001522 |
Leukotriene C4 synthase |
reviewed |
- |
LTC4S |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
19 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Efficacy |
'=' |
91 |
% |
| P30542 |
BXGT009436 |
Adenosine receptor A1 |
reviewed |
G-protein coupled receptor |
ADORA1 |
Ki |
'=' |
11611 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
25120 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Ki |
'=' |
5000 |
nM |
| P43140 |
BXGT010360 |
Alpha-1A adrenergic receptor |
reviewed |
- |
Adra1a |
IC50 |
- |
- |
- |
| P08913 |
BXGT006841 |
Alpha-2A adrenergic receptor |
reviewed |
G-protein coupled receptor |
ADRA2A |
Ki |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
Ki |
- |
- |
- |
| P29466 |
BXGT009349 |
Caspase-1 |
reviewed |
Enzyme |
CASP1 |
Ki |
- |
- |
- |
| P32241 |
BXGT009613 |
Vasoactive intestinal polypeptide receptor 1 |
reviewed |
G-protein coupled receptor |
VIPR1 |
Ki |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
Ki |
- |
- |
- |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
25099 |
nM |
| P25101 |
BXGT009018 |
Endothelin-1 receptor |
reviewed |
G-protein coupled receptor |
EDNRA |
Ki |
- |
- |
- |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
7 |
% |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
KSV |
'=' |
0 |
10'5/M |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
1 |
degrees C |
| P32245 |
BXGT009614 |
Melanocortin receptor 4 |
reviewed |
G-protein coupled receptor |
MC4R |
IC50 |
- |
- |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
EC50 |
'=' |
2 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Ki |
- |
- |
- |
| P25025 |
BXGT009006 |
C-X-C chemokine receptor type 2 |
reviewed |
G-protein coupled receptor |
CXCR2 |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
IC50 |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Ki |
- |
- |
- |
| P41968 |
BXGT010275 |
Melanocortin receptor 3 |
reviewed |
G-protein coupled receptor |
MC3R |
IC50 |
- |
- |
- |
| P29274 |
BXGT009327 |
Adenosine receptor A2a |
reviewed |
G-protein coupled receptor |
ADORA2A |
Ki |
'=' |
9792 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
14125 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
1000 |
nM |
| P22002 |
BXGT008717 |
Voltage-dependent L-type calcium channel subunit alpha-1C |
reviewed |
- |
Cacna1c |
IC50 |
'=' |
11000 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
15848 |
nM |
| P38398 |
BXGT010037 |
Breast cancer type 1 susceptibility protein |
reviewed |
Enzyme |
BRCA1 |
Potency |
- |
10000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
446 |
nM |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Thermal melting change |
'=' |
0 |
degrees C |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Thermal melting change |
'=' |
2 |
degrees C |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
10000 |
nM |
| P21452 |
BXGT008653 |
Substance-K receptor |
reviewed |
G-protein coupled receptor |
TACR2 |
Ki |
- |
- |
- |
| P15207 |
BXGT008096 |
Androgen receptor |
reviewed |
- |
Ar |
IC50 |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
- |
- |
- |
| P37288 |
BXGT009977 |
Vasopressin V1a receptor |
reviewed |
G-protein coupled receptor |
AVPR1A |
Ki |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
5011 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
-5 |
% |
| P15917 |
BXGT008169 |
Lethal factor |
reviewed |
- |
lef |
Potency |
'=' |
31622 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
8912 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Thermal melting change |
'=' |
1 |
degrees C |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q16659 |
BXGT013652 |
Mitogen-activated protein kinase 6 |
reviewed |
Kinase |
MAPK6 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q86Y07 |
BXGT017631 |
Serine/threonine-protein kinase VRK2 |
reviewed |
Kinase |
VRK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
IC50 |
'=' |
9120 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
0 |
- |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
25 |
% |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
IC50 |
- |
- |
- |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
13333 |
nM |
| P17405 |
BXGT008304 |
Sphingomyelin phosphodiesterase |
reviewed |
Enzyme |
SMPD1 |
Potency |
- |
562341 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
94 |
% |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'>' |
400000 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'=' |
82700 |
nM |
| P51151 |
BXGT010837 |
Ras-related protein Rab-9A |
reviewed |
- |
RAB9A |
Potency |
'=' |
3981 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Thermal melting change |
'=' |
1 |
degrees C |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
14125 |
nM |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Thermal melting change |
'=' |
2 |
degrees C |
| P20781 |
BXGT008598 |
Glycine receptor subunit beta |
reviewed |
- |
Glrb |
IC50 |
- |
- |
- |
| P07727 |
BXGT006662 |
Glycine receptor subunit alpha-1 |
reviewed |
- |
Glra1 |
IC50 |
- |
- |
- |
| P24524 |
BXGT008974 |
Glycine receptor subunit alpha-3 |
reviewed |
- |
Glra3 |
IC50 |
- |
- |
- |
| P22771 |
BXGT008806 |
Glycine receptor subunit alpha-2 |
reviewed |
- |
Glra2 |
IC50 |
- |
- |
- |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
65 |
% |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
28183 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Ratio |
'=' |
23 |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Ratio |
'=' |
10000 |
- |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Ratio IC50 |
'=' |
2 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
%max |
'=' |
232 |
% |
| Q13133 |
BXGT013315 |
Oxysterols receptor LXR-alpha |
reviewed |
Nuclear receptor |
NR1H3 |
IC50 |
'=' |
31000 |
nM |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
14 |
nmol/min |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Thermal melting change |
'=' |
0 |
degrees C |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Thermal melting change |
'=' |
0 |
degrees C |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Thermal melting change |
'=' |
0 |
degrees C |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
100000 |
nM |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Potency |
- |
30747 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
22387 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Kd |
'=' |
26302 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
5323 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Thermal melting change |
'=' |
0 |
degrees C |
| Q96KB5 |
BXGT019685 |
Lymphokine-activated killer T-cell-originated protein kinase |
reviewed |
Kinase |
PBK |
Thermal melting change |
'=' |
0 |
degrees C |
| P37136 |
BXGT009967 |
Acetylcholinesterase |
reviewed |
- |
Ache |
Inhibition |
'<' |
5 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
IC50 |
'=' |
3890 |
nM |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Ki |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
| Q53685 |
BXGT015002 |
Oleandomycin glycosyltransferase |
reviewed |
- |
oleD |
Activity |
'=' |
3 |
nmol/min |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'<' |
5 |
% |
| P55055 |
BXGT011101 |
Oxysterols receptor LXR-beta |
reviewed |
Nuclear receptor |
NR1H2 |
IC50 |
'=' |
22000 |
nM |
| P11926 |
BXGT007760 |
Ornithine decarboxylase |
reviewed |
Enzyme |
ODC1 |
IC50 |
'=' |
26000 |
nM |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
50118 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
5448 |
nM |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ki |
- |
- |
- |
| P08311 |
BXGT006762 |
Cathepsin G |
reviewed |
Enzyme |
CTSG |
Ki |
- |
- |
- |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Ki |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
IC50 |
- |
- |
- |
| P28564 |
BXGT009272 |
5-hydroxytryptamine receptor 1B |
reviewed |
- |
Htr1b |
IC50 |
- |
- |
- |
| P41595 |
BXGT010267 |
5-hydroxytryptamine receptor 2B |
reviewed |
G-protein coupled receptor |
HTR2B |
Ki |
- |
- |
- |
| O70528 |
BXGT005068 |
5-hydroxytryptamine receptor 4 |
reviewed |
- |
HTR4 |
IC50 |
- |
- |
- |
| P25103 |
BXGT009020 |
Substance-P receptor |
reviewed |
G-protein coupled receptor |
TACR1 |
Ki |
- |
- |
- |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
IC50 |
'>' |
100000 |
nM |
| P05091 |
BXGT006312 |
Aldehyde dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ALDH2 |
IC50 |
- |
- |
- |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
- |
- |
- |
| P28335 |
BXGT009255 |
5-hydroxytryptamine receptor 2C |
reviewed |
G-protein coupled receptor |
HTR2C |
Ki |
'=' |
7806 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18356 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
1 |
degrees C |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
0 |
degrees C |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Thermal melting change |
'=' |
1 |
degrees C |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Thermal melting change |
'=' |
3 |
degrees C |
| P22002 |
BXGT008717 |
Voltage-dependent L-type calcium channel subunit alpha-1C |
reviewed |
- |
Cacna1c |
IC50 |
'=' |
57500 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Inhibition |
'<' |
5 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
39 |
% |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q15208 |
BXGT013550 |
Serine/threonine-protein kinase 38 |
reviewed |
Kinase |
STK38 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Thermal melting change |
'=' |
1 |
degrees C |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
Activity |
'=' |
15 |
% |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
Ki |
- |
- |
- |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
12050 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
1730 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
IC50 |
'=' |
58180 |
nM |
| O35505 |
BXGT004533 |
Voltage-dependent L-type calcium channel subunit alpha-1C |
reviewed |
- |
CACNA1C |
IC50 |
'=' |
20000 |
nM |
| P43220 |
BXGT010367 |
Glucagon-like peptide 1 receptor |
reviewed |
G-protein coupled receptor |
GLP1R |
Potency |
- |
25118 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
25929 |
nM |
| Q9UJW3 |
BXGT021732 |
DNA (cytosine-5)-methyltransferase 3-like |
reviewed |
- |
DNMT3L |
IC50 |
'>' |
100000 |
nM |
| Q9Y6K1 |
BXGT022331 |
DNA (cytosine-5)-methyltransferase 3A |
reviewed |
- |
DNMT3A |
IC50 |
'>' |
100000 |
nM |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Thermal melting change |
'=' |
3 |
degrees C |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
Inhibition |
'=' |
29 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
3900 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
FC |
'=' |
1 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Emax |
'=' |
92 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
EC50 |
'=' |
240 |
nM |
| P40763 |
BXGT010202 |
Signal transducer and activator of transcription 3 |
reviewed |
Nucleic acid binding |
STAT3 |
IC50 |
'=' |
24800 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Emax |
'=' |
121 |
% |