| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
pKi(uM) |
- |
- |
- |
| P07862 |
BXGT006691 |
D-alanine--D-alanine ligase B |
reviewed |
- |
ddlB |
IC50 |
'=' |
163000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
35481 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
7 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
'=' |
39810 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Activity |
'=' |
83 |
% |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Activity |
'=' |
91 |
% |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Activity |
'=' |
95 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
305000 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
1400 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
IC50 |
'=' |
1400 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
17782 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
5 |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
1200 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
pKi(uM) |
'=' |
0 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
1253 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
176200 |
nM |
| P09874 |
BXGT006934 |
Poly [ADP-ribose] polymerase 1 |
reviewed |
- |
PARP1 |
IC50 |
'=' |
100000 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
38500 |
nM |
| P06760 |
BXGT006500 |
Beta-glucuronidase |
reviewed |
- |
Gusb |
IC50 |
'=' |
2800 |
nM |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
GABA ratio |
'=' |
1 |
- |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
GABA ratio |
'=' |
1 |
- |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
GABA ratio |
'=' |
1 |
- |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
GABA ratio |
'=' |
1 |
- |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
GABA ratio |
'=' |
1 |
- |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
GABA ratio |
'=' |
1 |
- |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
GABA ratio |
'=' |
1 |
- |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
GABA ratio |
'=' |
1 |
- |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
GABA ratio |
'=' |
1 |
- |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
GABA ratio |
'=' |
1 |
- |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
GABA ratio |
'=' |
1 |
- |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
GABA ratio |
'=' |
1 |
- |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
GABA ratio |
'=' |
1 |
- |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
GABA ratio |
'=' |
1 |
- |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
GABA ratio |
'=' |
1 |
- |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
GABA ratio |
'=' |
1 |
- |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Vmax |
'=' |
0 |
uM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Vmax |
'=' |
0 |
uM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
360 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
562 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
CC50 |
'=' |
63 |
ug.mL-1 |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
'=' |
12589 |
nM |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
'=' |
280000 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
25118 |
nM |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
39810 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
- |
35481 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
24336 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Thermal melting change |
'=' |
5 |
degrees C |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
47754 |
nM |
| P08659 |
BXGT006805 |
Luciferin 4-monooxygenase |
reviewed |
- |
|
Potency |
'=' |
39810 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
4900 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
28183 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
800 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
800 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
800 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
TIME |
'=' |
8 |
hr |
| P13569 |
BXGT007923 |
Cystic fibrosis transmembrane conductance regulator |
reviewed |
Ion channel |
CFTR |
EC50 |
'=' |
9000 |
nM |
| Q27686 |
BXGT013930 |
Pyruvate kinase |
reviewed |
- |
PYK |
Potency |
'=' |
12589 |
nM |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Thermal melting change |
'=' |
1 |
degrees C |
| O00506 |
BXGT003932 |
Serine/threonine-protein kinase 25 |
reviewed |
Kinase |
STK25 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
845 |
pm/min/mg |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
574 |
pm/min/mg |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Inhibition |
'=' |
65 |
% |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Activity |
'=' |
80 |
% |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Activity |
'=' |
59 |
% |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Activity |
'=' |
18 |
% |
| P41240 |
BXGT010242 |
Tyrosine-protein kinase CSK |
reviewed |
Kinase |
CSK |
Activity |
'=' |
77 |
% |
| P68871 |
BXGT011615 |
Hemoglobin subunit beta |
reviewed |
- |
HBB |
Potency |
'=' |
31622 |
nM |
| P0AES4 |
BXGT007329 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'=' |
67 |
ug.mL-1 |
| P0AES6 |
BXGT007331 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'=' |
67 |
ug.mL-1 |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
3981 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Inhibition |
- |
- |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
Inhibition |
- |
- |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Activity |
- |
- |
- |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
14125 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Activity |
- |
- |
- |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
11220 |
nM |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Activity |
'=' |
87 |
% |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Ki |
'=' |
390 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Thermal melting change |
'=' |
3 |
degrees C |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
25118 |
nM |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Inhibition |
'=' |
12 |
% |
| Q03431 |
BXGT012714 |
Parathyroid hormone/parathyroid hormone-related peptide receptor |
reviewed |
G-protein coupled receptor |
PTH1R |
Potency |
- |
50118 |
nM |
| P0C6X7 |
BXGT007440 |
Replicase polyprotein 1ab |
reviewed |
- |
rep |
IC50 |
'=' |
280800 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
33400 |
nM |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Thermal melting change |
'=' |
0 |
degrees C |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Thermal melting change |
'=' |
2 |
degrees C |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q96KB5 |
BXGT019685 |
Lymphokine-activated killer T-cell-originated protein kinase |
reviewed |
Kinase |
PBK |
Thermal melting change |
'=' |
0 |
degrees C |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
12589 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
7943 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Inhibition |
- |
- |
- |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Activity |
'=' |
21 |
% |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
28183 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
22387 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
'=' |
121600 |
nM |
| O94925 |
BXGT005342 |
Glutaminase kidney isoform, mitochondrial |
reviewed |
Enzyme |
GLS |
Potency |
- |
35481 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
31622 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
8912 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
795 |
nM |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
31622 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
39810 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
39810 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
39810 |
nM |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
35481 |
nM |
| P05979 |
BXGT006400 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
IC50 |
'>' |
100 |
ug.mL-1 |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
25 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
1 |
- |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
461 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
KSV |
'=' |
1 |
10'5/M |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Kcat |
'=' |
0 |
10'3/s |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Kcat |
'=' |
0 |
10'3/s |
| O15118 |
BXGT004127 |
NPC intracellular cholesterol transporter 1 |
reviewed |
Transporter |
NPC1 |
Potency |
'=' |
5804 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
398 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
15848 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
15848 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
19952 |
nM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
8 |
ug.mL-1 |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
12589 |
nM |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
107 |
% |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Ratio |
'=' |
0 |
- |
| Q4Q090 |
BXGT014858 |
2,3-bisphosphoglycerate-independent phosphoglycerate mutase |
unreviewed |
- |
PGAM |
Potency |
- |
19011 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Ki |
'=' |
178300 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
17400 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
IC50 |
'=' |
14000 |
nM |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
14000 |
nM |
| P04839 |
BXGT006273 |
Cytochrome b-245 heavy chain |
reviewed |
Ion channel |
CYBB |
Inhibition |
- |
- |
- |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
45700 |
nM |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
16833 |
nM |
| P90584 |
BXGT012110 |
MO15-related protein kinase Pfmrk |
unreviewed |
- |
Pfmrk |
IC50 |
'=' |
7000 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
2400 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
3162 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
8000 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
2 |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
10000 |
nM |
| P14618 |
BXGT008027 |
Pyruvate kinase PKM |
reviewed |
Kinase |
PKM |
Potency |
'=' |
3162 |
nM |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
18 |
pm/min/mg |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
28183 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
1258 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
12589 |
nM |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
50000 |
nM |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Intrinsic activity |
- |
- |
- |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Ratio |
'=' |
1 |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
'=' |
34 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
37100 |
nM |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Activity |
'=' |
102 |
% |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Activity |
'=' |
100 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Activity |
'=' |
54 |
% |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Activity |
'=' |
89 |
% |
| Q9Y4K4 |
BXGT022282 |
Mitogen-activated protein kinase kinase kinase kinase 5 |
reviewed |
Kinase |
MAP4K5 |
Activity |
'=' |
96 |
% |
| Q8IV63 |
BXGT018341 |
Inactive serine/threonine-protein kinase VRK3 |
reviewed |
Kinase |
VRK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
Inhibition |
'<' |
50 |
% |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
7943 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
8912 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
44668 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
12589 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
700 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
1995 |
nM |
| Q9H2K2 |
BXGT020454 |
Poly [ADP-ribose] polymerase tankyrase-2 |
reviewed |
- |
TNKS2 |
IC50 |
'=' |
2951 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
Ki |
'=' |
37100 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Activity |
'=' |
50 |
% |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
IC50 |
'=' |
5200 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
'=' |
5 |
uM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
19952 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
12589 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
8912 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
8912 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
12589 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
3162 |
nM |
| P00697 |
BXGT005616 |
Lysozyme C-1 |
reviewed |
- |
Lyz1 |
IC50 |
'=' |
17700 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
12589 |
nM |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
2393 |
nM |
| Q16659 |
BXGT013652 |
Mitogen-activated protein kinase 6 |
reviewed |
Kinase |
MAPK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9BVS4 |
BXGT020147 |
Serine/threonine-protein kinase RIO2 |
reviewed |
Kinase |
RIOK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
IC50 |
'=' |
130 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
EC50 |
'=' |
3000 |
nM |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
Inhibition |
- |
- |
- |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
6294 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
Potency |
- |
44668 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
7580 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
8 |
% |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'>' |
20000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
3100 |
nM |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
IC50 |
'>' |
100 |
ug.mL-1 |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
134 |
% |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
5900 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
30 |
ug.mL-1 |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
12800 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
35481 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
31622 |
nM |
| Q07869 |
BXGT012945 |
Peroxisome proliferator-activated receptor alpha |
reviewed |
Nuclear receptor |
PPARA |
FC |
'=' |
2 |
- |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
37400 |
nM |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Thermal melting change |
'=' |
3 |
degrees C |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
28900 |
nM |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Thermal melting change |
'=' |
4 |
degrees C |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
5011 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
3000 |
nM |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
4466 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
800 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
Potency |
- |
39810 |
nM |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
105 |
% |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
11220 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
6670 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
60119 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
22387 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
12589 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
1900 |
nM |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Km |
'=' |
530000 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
12995 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
63 |
nM |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
39810 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
8634 |
nM |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
IC50 |
'=' |
17800 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
'=' |
3800 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
7 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
23715 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
10000 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
10000 |
nM |
| P00760 |
BXGT005644 |
Cationic trypsin |
reviewed |
- |
|
IC50 |
'=' |
141500 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
10210 |
nM |
| P14916 |
BXGT008066 |
Urease subunit alpha |
reviewed |
- |
ureA |
IC50 |
'=' |
138000 |
nM |
| P69996 |
BXGT011656 |
Urease subunit beta |
reviewed |
- |
ureB |
IC50 |
'=' |
138000 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
'=' |
4 |
ug.mL-1 |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
33498 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
164 |
pm/min/mg |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Intrinsic activity |
- |
- |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
25118 |
nM |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Thermal melting change |
'=' |
5 |
degrees C |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
Potency |
- |
35481 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
- |
31622 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
7079 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
25118 |
nM |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
31622 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
19952 |
nM |
| P38398 |
BXGT010037 |
Breast cancer type 1 susceptibility protein |
reviewed |
Enzyme |
BRCA1 |
Potency |
- |
22387 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
Inhibition |
'=' |
72 |
% |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
60 |
% |
| P40225 |
BXGT010168 |
Thrombopoietin |
reviewed |
- |
THPO |
Potency |
'=' |
501 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
25118 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
'=' |
50118 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
39810 |
nM |
| Q13951 |
BXGT013407 |
Core-binding factor subunit beta |
reviewed |
- |
CBFB |
Potency |
- |
12589 |
nM |
| Q01196 |
BXGT012575 |
Runt-related transcription factor 1 |
reviewed |
Transcription factor |
RUNX1 |
Potency |
- |
12589 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
'=' |
12589 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
140 |
nM |
| Q6W5P4 |
BXGT016588 |
Neuropeptide S receptor |
reviewed |
- |
NPSR1 |
Potency |
'=' |
25118 |
nM |
| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
4 |
% |
| P12822 |
BXGT007850 |
Angiotensin-converting enzyme |
reviewed |
- |
ACE |
IC50 |
'=' |
280000000 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
18 |
% |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
IC50 |
'=' |
1700 |
nM |
| P22612 |
BXGT008785 |
cAMP-dependent protein kinase catalytic subunit gamma |
reviewed |
Kinase |
PRKACG |
Activity |
'=' |
87 |
% |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Activity |
'=' |
87 |
% |
| P22694 |
BXGT008797 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
Kinase |
PRKACB |
Activity |
'=' |
87 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
125 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
427 |
nM |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
570000 |
nM |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Activity |
'=' |
86 |
% |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Activity |
'=' |
57 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
3981 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
5011 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| Q9TU15 |
BXGT021625 |
Estrogen receptor beta |
reviewed |
- |
ESR2 |
Kd |
'=' |
660 |
nM |
| P49885 |
BXGT010755 |
Estrogen receptor |
reviewed |
- |
ESR1 |
Kd |
'=' |
660 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
IC50 |
'=' |
443000 |
nM |
| O95271 |
BXGT005369 |
Poly [ADP-ribose] polymerase tankyrase-1 |
reviewed |
- |
TNKS |
IC50 |
'=' |
3162 |
nM |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
10621 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
'=' |
7943 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Activity |
'=' |
82 |
% |
| P23443 |
BXGT008866 |
Ribosomal protein S6 kinase beta-1 |
reviewed |
Kinase |
RPS6KB1 |
Activity |
'=' |
65 |
% |
| P07948 |
BXGT006702 |
Tyrosine-protein kinase Lyn |
reviewed |
Kinase |
LYN |
Activity |
'=' |
88 |
% |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Intrinsic activity |
- |
- |
- |
| P51450 |
BXGT010847 |
Nuclear receptor ROR-gamma |
reviewed |
- |
Rorc |
Potency |
'=' |
14125 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
Ki |
- |
- |
- |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
3981 |
nM |
| P53323 |
BXGT010982 |
EKC/KEOPS complex subunit BUD32 |
reviewed |
- |
BUD32 |
Activity |
'=' |
103 |
% |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Activity |
'=' |
45 |
% |
| Q13627 |
BXGT013385 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
reviewed |
Kinase |
DYRK1A |
Activity |
'=' |
20 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
8912 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
1778 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ki |
'=' |
6000 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
Activity |
- |
- |
- |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Ki |
'=' |
520 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
'=' |
12589 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Ki |
'=' |
740 |
nM |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
Activity |
'=' |
98 |
% |
| O14757 |
BXGT004092 |
Serine/threonine-protein kinase Chk1 |
reviewed |
Kinase |
CHEK1 |
Activity |
'=' |
67 |
% |
| P48729 |
BXGT010655 |
Casein kinase I isoform alpha |
reviewed |
Kinase |
CSNK1A1 |
Activity |
'=' |
106 |
% |
| P49674 |
BXGT010725 |
Casein kinase I isoform epsilon |
reviewed |
- |
CSNK1E |
Activity |
'=' |
106 |
% |
| P48730 |
BXGT010656 |
Casein kinase I isoform delta |
reviewed |
Kinase |
CSNK1D |
Activity |
'=' |
106 |
% |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Activity |
'=' |
106 |
% |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Activity |
'=' |
106 |
% |
| P09769 |
BXGT006917 |
Tyrosine-protein kinase Fgr |
reviewed |
Kinase |
FGR |
Activity |
'=' |
48 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
1700 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
RBA |
'=' |
0 |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
- |
- |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
pKi(uM) |
'=' |
0 |
- |
| Q92731 |
BXGT019366 |
Estrogen receptor beta |
reviewed |
Nuclear receptor |
ESR2 |
Fold selectivity |
'=' |
10 |
- |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
32885 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
21 |
% |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
16 |
% |
| Q9ES14 |
BXGT020314 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
- |
Gabre |
Ki |
'=' |
770 |
nM |
| Q91ZM7 |
BXGT019327 |
GABA theta subunit |
unreviewed |
- |
Gabrq |
Ki |
'=' |
770 |
nM |
| P63138 |
BXGT011502 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
- |
Gabrb2 |
Ki |
'=' |
770 |
nM |
| P63079 |
BXGT011491 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
- |
Gabrb3 |
Ki |
'=' |
770 |
nM |
| P62813 |
BXGT011460 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
- |
Gabra1 |
Ki |
'=' |
770 |
nM |
| P30191 |
BXGT009410 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
- |
Gabra6 |
Ki |
'=' |
770 |
nM |
| P28473 |
BXGT009261 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
- |
Gabrg3 |
Ki |
'=' |
770 |
nM |
| P28471 |
BXGT009259 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
- |
Gabra4 |
Ki |
'=' |
770 |
nM |
| P23576 |
BXGT008885 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
- |
Gabra2 |
Ki |
'=' |
770 |
nM |
| P23574 |
BXGT008884 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
- |
Gabrg1 |
Ki |
'=' |
770 |
nM |
| P20236 |
BXGT008551 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
- |
Gabra3 |
Ki |
'=' |
770 |
nM |
| P19969 |
BXGT008536 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
- |
Gabra5 |
Ki |
'=' |
770 |
nM |
| P18508 |
BXGT008412 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
- |
Gabrg2 |
Ki |
'=' |
770 |
nM |
| P18506 |
BXGT008410 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
- |
Gabrd |
Ki |
'=' |
770 |
nM |
| P15431 |
BXGT008122 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
- |
Gabrb1 |
Ki |
'=' |
770 |
nM |
| O09028 |
BXGT004049 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
- |
Gabrp |
Ki |
'=' |
770 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3162 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
11220 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
53091 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
10590 |
nM |
| Q12791 |
BXGT013264 |
Calcium-activated potassium channel subunit alpha-1 |
reviewed |
Ion channel |
KCNMA1 |
Control |
'=' |
158 |
% |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
IC50 |
'=' |
18000 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Displacement |
'=' |
63 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Ratio IC50 |
'=' |
10 |
- |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'=' |
12 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| Q16445 |
BXGT013629 |
Gamma-aminobutyric acid receptor subunit alpha-6 |
reviewed |
Ion channel |
GABRA6 |
Ki |
'=' |
3019 |
nM |
| P31644 |
BXGT009557 |
Gamma-aminobutyric acid receptor subunit alpha-5 |
reviewed |
Ion channel |
GABRA5 |
Ki |
'=' |
3019 |
nM |
| P47869 |
BXGT010590 |
Gamma-aminobutyric acid receptor subunit alpha-2 |
reviewed |
Ion channel |
GABRA2 |
Ki |
'=' |
3019 |
nM |
| P78334 |
BXGT011834 |
Gamma-aminobutyric acid receptor subunit epsilon |
reviewed |
Ion channel |
GABRE |
Ki |
'=' |
3019 |
nM |
| P18505 |
BXGT008409 |
Gamma-aminobutyric acid receptor subunit beta-1 |
reviewed |
Ion channel |
GABRB1 |
Ki |
'=' |
3019 |
nM |
| Q8N1C3 |
BXGT018498 |
Gamma-aminobutyric acid receptor subunit gamma-1 |
reviewed |
Ion channel |
GABRG1 |
Ki |
'=' |
3019 |
nM |
| O14764 |
BXGT004094 |
Gamma-aminobutyric acid receptor subunit delta |
reviewed |
Ion channel |
GABRD |
Ki |
'=' |
3019 |
nM |
| O00591 |
BXGT003939 |
Gamma-aminobutyric acid receptor subunit pi |
reviewed |
Ion channel |
GABRP |
Ki |
'=' |
3019 |
nM |
| P34903 |
BXGT009769 |
Gamma-aminobutyric acid receptor subunit alpha-3 |
reviewed |
Ion channel |
GABRA3 |
Ki |
'=' |
3019 |
nM |
| Q9UN88 |
BXGT021783 |
Gamma-aminobutyric acid receptor subunit theta |
reviewed |
Ion channel |
GABRQ |
Ki |
'=' |
3019 |
nM |
| Q99928 |
BXGT019975 |
Gamma-aminobutyric acid receptor subunit gamma-3 |
reviewed |
Ion channel |
GABRG3 |
Ki |
'=' |
3019 |
nM |
| P48169 |
BXGT010622 |
Gamma-aminobutyric acid receptor subunit alpha-4 |
reviewed |
Ion channel |
GABRA4 |
Ki |
'=' |
3019 |
nM |
| P28472 |
BXGT009260 |
Gamma-aminobutyric acid receptor subunit beta-3 |
reviewed |
Ion channel |
GABRB3 |
Ki |
'=' |
3019 |
nM |
| P18507 |
BXGT008411 |
Gamma-aminobutyric acid receptor subunit gamma-2 |
reviewed |
Ion channel |
GABRG2 |
Ki |
'=' |
3019 |
nM |
| P47870 |
BXGT010591 |
Gamma-aminobutyric acid receptor subunit beta-2 |
reviewed |
Ion channel |
GABRB2 |
Ki |
'=' |
3019 |
nM |
| P14867 |
BXGT008061 |
Gamma-aminobutyric acid receptor subunit alpha-1 |
reviewed |
Ion channel |
GABRA1 |
Ki |
'=' |
3019 |
nM |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
Activity |
- |
- |
- |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
IC50 |
'=' |
6600 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
1258 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
39810 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
44668 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
19952 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
1000 |
nM |
| P35372 |
BXGT009823 |
Mu-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRM1 |
Ke |
'=' |
410 |
nM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
logIC50 |
'=' |
0 |
- |
| Q8IW41 |
BXGT018352 |
MAP kinase-activated protein kinase 5 |
reviewed |
Kinase |
MAPKAPK5 |
Activity |
'=' |
93 |
% |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
10000 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
900 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
13 |
% |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
15848 |
nM |
| P0A6C1 |
BXGT007045 |
Endonuclease 4 |
reviewed |
- |
nfo |
Potency |
'=' |
5623 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
8912 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
8912 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
8912 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
640 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
1550 |
nM |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
35481 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
1778 |
nM |
| P28593 |
BXGT009278 |
Trypanothione reductase |
reviewed |
- |
TPR |
Inhibition |
'=' |
13 |
% |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
8 |
- |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
31600 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
19952 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Ka |
'=' |
1 |
10'5/M |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Potency |
- |
39810 |
nM |
| O14924 |
BXGT004111 |
Regulator of G-protein signaling 12 |
reviewed |
- |
RGS12 |
Potency |
'=' |
25118 |
nM |
| P63096 |
BXGT011496 |
Guanine nucleotide-binding protein G(i) subunit alpha-1 |
reviewed |
Enzyme modulator |
GNAI1 |
Potency |
'=' |
25118 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
94 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5173 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q15078 |
BXGT013534 |
Cyclin-dependent kinase 5 activator 1 |
reviewed |
Enzyme modulator |
CDK5R1 |
IC50 |
'=' |
1600 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
IC50 |
'=' |
1600 |
nM |
| O95067 |
BXGT005347 |
G2/mitotic-specific cyclin-B2 |
reviewed |
Enzyme modulator |
CCNB2 |
IC50 |
'=' |
4000 |
nM |
| Q8WWL7 |
BXGT019000 |
G2/mitotic-specific cyclin-B3 |
reviewed |
Enzyme modulator |
CCNB3 |
IC50 |
'=' |
4000 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
4000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
4000 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
64 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
IC50 |
'=' |
653 |
nM |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
'=' |
46100 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
84 |
% |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
7079 |
nM |
| Q1CTD3 |
BXGT013756 |
D-alanine--D-alanine ligase |
reviewed |
- |
ddl |
IC50 |
'=' |
132700 |
nM |
| O95271 |
BXGT005369 |
Poly [ADP-ribose] polymerase tankyrase-1 |
reviewed |
- |
TNKS |
IC50 |
'=' |
3100 |
nM |
| Q1CTD3 |
BXGT013756 |
D-alanine--D-alanine ligase |
reviewed |
- |
ddl |
Ki |
'=' |
31000 |
nM |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Thermal melting change |
'=' |
2 |
degrees C |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Thermal melting change |
'=' |
1 |
degrees C |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Potency |
- |
18356 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
4200 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
31000 |
nM |
| P19793 |
BXGT008515 |
Retinoic acid receptor RXR-alpha |
reviewed |
Nuclear receptor |
RXRA |
Potency |
- |
15848 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Thermal melting change |
'=' |
7 |
degrees C |
| P10145 |
BXGT007542 |
Interleukin-8 |
reviewed |
Signaling |
CXCL8 |
Potency |
- |
66824 |
nM |
| Q16236 |
BXGT013624 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
Enzyme |
NFE2L2 |
Potency |
- |
33491 |
nM |
| Q99700 |
BXGT019949 |
Ataxin-2 |
reviewed |
Nucleic acid binding |
ATXN2 |
Potency |
- |
11220 |
nM |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
EC50 |
'=' |
24900 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Kq |
'=' |
1 |
10'12/M/s |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
2 |
degrees C |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
88 |
pm/min/mg |
| P35503 |
BXGT009840 |
UDP-glucuronosyltransferase 1-3 |
reviewed |
- |
UGT1A3 |
Activity |
'=' |
508 |
pm/min/mg |
| Q9FBZ2 |
BXGT020360 |
Prenyltransferase homolog |
unreviewed |
- |
SCO7190 |
Km |
'=' |
580000 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
3981 |
nM |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
31622 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
22387 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
3262 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
794 |
nM |
| Q96RI1 |
BXGT019727 |
Bile acid receptor |
reviewed |
Nuclear receptor |
NR1H4 |
Potency |
- |
50118 |
nM |
| O75874 |
BXGT005157 |
Isocitrate dehydrogenase [NADP] cytoplasmic |
reviewed |
- |
IDH1 |
Activity |
'=' |
97 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
19952 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Thermal melting change |
'=' |
-11 |
degrees C |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Thermal melting change |
'=' |
1 |
degrees C |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Thermal melting change |
'=' |
-1 |
degrees C |
| Q15208 |
BXGT013550 |
Serine/threonine-protein kinase 38 |
reviewed |
Kinase |
STK38 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q86Y07 |
BXGT017631 |
Serine/threonine-protein kinase VRK2 |
reviewed |
Kinase |
VRK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q03114 |
BXGT012692 |
Cyclin-dependent-like kinase 5 |
reviewed |
- |
Cdk5 |
EC50 |
'>' |
250000 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Kd |
'=' |
10000 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
31622 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Thermal melting change |
'=' |
0 |
degrees C |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9H2K2 |
BXGT020454 |
Poly [ADP-ribose] polymerase tankyrase-2 |
reviewed |
- |
TNKS2 |
IC50 |
'=' |
2900 |
nM |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
IC50 |
'=' |
1130 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
3548 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
6 |
- |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
'=' |
5 |
uM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
79432 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'>' |
20000 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
2058 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
23000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
10000 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
22387 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
- |
- |
- |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
25118 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Km |
'=' |
191000 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'<' |
1000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'<' |
1000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'<' |
1000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
6309 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
7 |
% |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
3200 |
nM |
| Q03181 |
BXGT012701 |
Peroxisome proliferator-activated receptor delta |
reviewed |
Nuclear receptor |
PPARD |
FC |
'=' |
3 |
- |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
10 |
% |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
Activity |
'=' |
25 |
% |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
'=' |
49900 |
nM |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Activity |
'=' |
101 |
% |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Activity |
'=' |
92 |
% |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Activity |
'=' |
92 |
% |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Activity |
'=' |
92 |
% |
| O00141 |
BXGT003882 |
Serine/threonine-protein kinase Sgk1 |
reviewed |
Kinase |
SGK1 |
Activity |
'=' |
41 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18356 |
nM |
| P35869 |
BXGT009877 |
Aryl hydrocarbon receptor |
reviewed |
Transcription factor |
AHR |
Potency |
- |
28183 |
nM |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| O95747 |
BXGT005393 |
Serine/threonine-protein kinase OSR1 |
reviewed |
Kinase |
OXSR1 |
Thermal melting change |
'=' |
2 |
degrees C |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Thermal melting change |
'=' |
5 |
degrees C |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Thermal melting change |
'=' |
2 |
degrees C |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Thermal melting change |
'=' |
4 |
degrees C |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
IC50 |
'=' |
1450 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Thermal melting change |
'=' |
2 |
degrees C |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Thermal melting change |
'=' |
0 |
degrees C |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Thermal melting change |
'=' |
1 |
degrees C |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Activity |
'=' |
10 |
% |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
'=' |
710 |
nM |
| Q15418 |
BXGT013569 |
Ribosomal protein S6 kinase alpha-1 |
reviewed |
Kinase |
RPS6KA1 |
Activity |
'=' |
86 |
% |
| O75116 |
BXGT005100 |
Rho-associated protein kinase 2 |
reviewed |
Kinase |
ROCK2 |
Activity |
'=' |
88 |
% |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Activity |
'=' |
57 |
% |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
5011 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
1 |
- |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
K |
'=' |
426 |
10'6/min |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
35481 |
nM |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
Emax |
'=' |
3 |
- |
| P41145 |
BXGT010225 |
Kappa-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRK1 |
Ke |
'=' |
410 |
nM |
| P41143 |
BXGT010223 |
Delta-type opioid receptor |
reviewed |
G-protein coupled receptor |
OPRD1 |
Ke |
'=' |
970 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Kic |
'=' |
11 |
uM |
| Q99972 |
BXGT019979 |
Myocilin |
reviewed |
Cellular structure |
MYOC |
Delta Tm |
'=' |
0 |
degrees C |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Km |
'=' |
191400 |
nM |
| P0C6X7 |
BXGT007440 |
Replicase polyprotein 1ab |
reviewed |
- |
rep |
Inhibition |
'=' |
40 |
% |
| Q99986 |
BXGT019980 |
Serine/threonine-protein kinase VRK1 |
reviewed |
Kinase |
VRK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
84 |
% |
| Q00532 |
BXGT012532 |
Cyclin-dependent kinase-like 1 |
reviewed |
Kinase |
CDKL1 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q09013 |
BXGT013023 |
Myotonin-protein kinase |
reviewed |
Kinase |
DMPK |
Thermal melting change |
'=' |
0 |
degrees C |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Thermal melting change |
'=' |
3 |
degrees C |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
'=' |
52 |
% |
| P02766 |
BXGT005953 |
Transthyretin |
reviewed |
Transporter |
TTR |
Kd |
'=' |
250 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
11900 |
nM |
| P51449 |
BXGT010846 |
Nuclear receptor ROR-gamma |
reviewed |
Nuclear receptor |
RORC |
Potency |
- |
4216 |
nM |
| P42582 |
BXGT010319 |
Homeobox protein Nkx-2.5 |
reviewed |
- |
Nkx2-5 |
IC50 |
'=' |
24000 |
nM |
| Q08369 |
BXGT012983 |
Transcription factor GATA-4 |
reviewed |
- |
Gata4 |
IC50 |
'=' |
24000 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| Q16769 |
BXGT013665 |
Glutaminyl-peptide cyclotransferase |
reviewed |
Enzyme |
QPCT |
Inhibition |
'=' |
75 |
% |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
11 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
'=' |
25 |
% |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
1500 |
nM |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
37933 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Activity |
'=' |
19 |
% |
| P13569 |
BXGT007923 |
Cystic fibrosis transmembrane conductance regulator |
reviewed |
Ion channel |
CFTR |
Ki |
'=' |
81000 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
TIME |
'=' |
3 |
hr |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Ke(app) |
'=' |
3697 |
/M/min |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
T1/2 |
'=' |
5 |
hr |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Tlag |
'=' |
81 |
min |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
3570 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Potency |
- |
3981 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
- |
- |
- |
| Q99972 |
BXGT019979 |
Myocilin |
reviewed |
Cellular structure |
MYOC |
Kd |
'=' |
41600 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
1120 |
nM |