Showing entry for Chelerythrine


　 　 　 　 　 　 　 　 　 　 　 　 　 　 　
General Compound Information
BXGC IdBXGC0012352
Compound NameChelerythrine
Structure
FormulaC21H18NO4
InchiKeyLLEJIEBFSOEYIV-UHFFFAOYSA-N
SMILESCOc1c(OC)ccc2c1c[n+](C)c1c2ccc2c1cc1OCOc1c2
InchiInChI=1S/C21H18NO4/c1-22-10-16-13(6-7-17(23-2)21(16)24-3)14-5-4-12-8-18-19(26-11-25-18)9-15(12)20(14)22/h4-10H,11H2,1-3H3/q+1
IUPAC1,2-dimethoxy-12-methyl-[1,3]benzodioxolo[5,6-c]phenanthridin-12-ium
Molecular Weight348.12
Pubchem Id2703
Chembl IdCHEMBL13045
Targets of Information Source
DrugBank n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
PDB CTI
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Q9AMP1 BXGT020080 Chitinase A unreviewed chiA - - - - -
P02638 BXGT005906 Protein S100-B reviewed S100B - - - - -
P37231 BXGT009972 Peroxisome proliferator-activated receptor gamma reviewed PPARG Nuclear receptor - 566 - -
Binding DB 25524
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT012941 Bcl-2-like protein 1 reviewed Signaling BCL2L1 - 100000 - -
reviewed BXGT006379 Protein kinase C alpha type reviewed Prkca 660 - - -
reviewed BXGT008594 Aromatic-L-amino-acid decarboxylase reviewed DDC - 1280000 - -
reviewed BXGT011342 Cell division control protein 42 homolog reviewed Enzyme modulator CDC42 - >100000 - -
reviewed BXGT011481 Ras-related C3 botulinum toxin substrate 1 reviewed Enzyme modulator RAC1 - >100000 - -
reviewed BXGT007567 Apoptosis regulator Bcl-2 reviewed Signaling BCL2 171000 - - -
reviewed BXGT019384 Bcl-2-like protein 2 reviewed Signaling BCL2L2 106000 - - -
reviewed BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE - 24 - -
reviewed BXGT008751 Acetylcholinesterase reviewed Enzyme ACHE 1120 - - -
reviewed BXGT008751 Acetylcholinesterase reviewed Enzyme ACHE 320 - - -
reviewed BXGT004559 Acetylcholinesterase reviewed ache 920 - - -
reviewed BXGT004559 Acetylcholinesterase reviewed ache 480 - - -
reviewed BXGT008751 Acetylcholinesterase reviewed Enzyme ACHE - 1540 - -
reviewed BXGT004559 Acetylcholinesterase reviewed ache - 3780 - -
reviewed BXGT006430 Cholinesterase reviewed BCHE - 10340 - -
reviewed BXGT011959 Cholinesterase reviewed BCHE - 6330 - -
CHEMBL CHEMBL13045
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Residual Activity '=' 101 %
P00352 BXGT005510 Retinal dehydrogenase 1 reviewed Enzyme ALDH1A1 Potency '=' 22387 nM
Q99700 BXGT019949 Ataxin-2 reviewed Nucleic acid binding ATXN2 Potency - 5623 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Potency '=' 31622 nM
P83916 BXGT012025 Chromobox protein homolog 1 reviewed Epigenetic regulator CBX1 Potency - 50118 nM
P08659 BXGT006805 Luciferin 4-monooxygenase reviewed - Potency '=' 31622 nM
O14733 BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 Residual Activity '=' 71 %
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Residual Activity '=' 94 %
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Residual Activity '=' 44 %
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Residual Activity '=' 94 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 92 %
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Residual Activity '=' 92 %
P67870 BXGT011566 Casein kinase II subunit beta reviewed Kinase CSNK2B Residual Activity '=' 92 %
P78362 BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 Residual Activity '=' 96 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Residual Activity '=' 103 %
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Residual Activity '=' 110 %
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Residual Activity '=' 90 %
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Residual Activity '=' 80 %
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Residual Activity '=' 125 %
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Residual Activity '=' 108 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 92 %
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Residual Activity '=' 130 %
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Residual Activity '=' 101 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Residual Activity '=' 117 %
O15118 BXGT004127 NPC intracellular cholesterol transporter 1 reviewed Transporter NPC1 Potency '=' 58047 nM
Q99714 BXGT019954 3-hydroxyacyl-CoA dehydrogenase type-2 reviewed Enzyme HSD17B10 Potency '=' 25118 nM
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Residual Activity '=' 60 %
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Residual Activity '=' 68 %
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Residual Activity '=' 82 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 60 %
O43318 BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 Residual Activity '=' 92 %
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Residual Activity '=' 85 %
Q96BR1 BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed - SGK3 Residual Activity '=' 102 %
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Residual Activity '=' 92 %
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Residual Activity '=' 93 %
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Residual Activity '=' 80 %
Q8WTQ7 BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 Residual Activity '=' 91 %
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Residual Activity '=' 96 %
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Residual Activity '=' 116 %
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Residual Activity '=' 97 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Residual Activity '=' 130 %
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Residual Activity '=' 94 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Residual Activity '=' 80 %
P05129 BXGT006322 Protein kinase C gamma type reviewed Kinase PRKCG Residual Activity '=' 97 %
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Residual Activity '=' 113 %
O60563 BXGT004883 Cyclin-T1 reviewed Enzyme modulator CCNT1 Residual Activity '=' 113 %
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Residual Activity '=' 105 %
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Residual Activity '=' 107 %
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Residual Activity '=' 103 %
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 AC50 '=' 10000 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Residual Activity '=' 86 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 88 %
P14635 BXGT008031 G2/mitotic-specific cyclin-B1 reviewed Enzyme modulator CCNB1 Residual Activity '=' 97 %
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Residual Activity '=' 97 %
Q8IYT8 BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 Residual Activity '=' 104 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 110 %
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Residual Activity '=' 94 %
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Residual Activity '=' 96 %
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Residual Activity '=' 81 %
P39748 BXGT010134 Flap endonuclease 1 reviewed Enzyme FEN1 Potency - 15003 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Residual Activity '=' 66 %
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Residual Activity '=' 100 %
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Residual Activity '=' 76 %
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Residual Activity '=' 99 %
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Residual Activity '=' 99 %
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Residual Activity '=' 96 %
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Residual Activity '=' 75 %
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Residual Activity '=' 108 %
Q9UPE1 BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 Residual Activity '=' 110 %
Q9NYY3 BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 Residual Activity '=' 103 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Residual Activity '=' 100 %
P19838 BXGT008526 Nuclear factor NF-kappa-B p105 subunit reviewed Transcription factor NFKB1 Potency '=' 11220 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Residual Activity '=' 99 %
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Residual Activity '=' 106 %
P16473 BXGT008234 Thyrotropin receptor reviewed G-protein coupled receptor TSHR Potency '=' 25118 nM
P97697 BXGT012214 Inositol monophosphatase 1 reviewed - Impa1 Potency '=' 5011 nM
Q16637 BXGT013646 Survival motor neuron protein reviewed Epigenetic regulator SMN1 Potency '=' 7079 nM
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Residual Activity '=' 61 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 66 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 66 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 66 %
Q9F4F7 BXGT020344 4'-phosphopantetheinyl transferase ffp reviewed - ffp Potency '=' 25118 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 17782 nM
O15296 BXGT004148 Arachidonate 15-lipoxygenase B reviewed Enzyme ALOX15B Potency - 15848 nM
P15917 BXGT008169 Lethal factor reviewed - lef Potency '=' 25118 nM
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Residual Activity '=' 102 %
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Residual Activity '=' 93 %
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Residual Activity '=' 102 %
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Residual Activity '=' 101 %
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Residual Activity '=' 86 %
P78396 BXGT011842 Cyclin-A1 reviewed Enzyme modulator CCNA1 Residual Activity '=' 103 %
P20248 BXGT008554 Cyclin-A2 reviewed Enzyme modulator CCNA2 Residual Activity '=' 103 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 103 %
O15648 BXGT004185 ATP-dependent 6-phosphofructokinase reviewed - pfk Potency - 19011 nM
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Residual Activity '=' 83 %
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Residual Activity '=' 115 %
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Residual Activity '=' 107 %
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Residual Activity '=' 99 %
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Residual Activity '=' 132 %
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Residual Activity '=' 98 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Residual Activity '=' 106 %
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Residual Activity '=' 68 %
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Residual Activity '=' 91 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Potency '=' 31622 nM
Q96QE3 BXGT019718 ATPase family AAA domain-containing protein 5 reviewed - ATAD5 Potency - 16353 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 501 nM
P13267 BXGT007895 DNA polymerase III PolC-type reviewed - polC Potency - 26679 nM
P40225 BXGT010168 Thrombopoietin reviewed - THPO Potency '=' 1995 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Residual Activity '=' 92 %
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Residual Activity '=' 107 %
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Residual Activity '=' 106 %
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Residual Activity '=' 96 %
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Residual Activity '=' 69 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Residual Activity '=' 94 %
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 Potency '=' 39810 nM
Q99714 BXGT019954 3-hydroxyacyl-CoA dehydrogenase type-2 reviewed Enzyme HSD17B10 Potency '=' 19952 nM
P39748 BXGT010134 Flap endonuclease 1 reviewed Enzyme FEN1 Potency - 29934 nM
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Residual Activity '=' 76 %
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Residual Activity '=' 93 %
O60563 BXGT004883 Cyclin-T1 reviewed Enzyme modulator CCNT1 Residual Activity '=' 93 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 114 %
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Residual Activity '=' 132 %
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Residual Activity '=' 85 %
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 Potency '=' 10000 nM
O15296 BXGT004148 Arachidonate 15-lipoxygenase B reviewed Enzyme ALOX15B Potency - 12589 nM
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Potency '=' 2930 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Residual Activity '=' 103 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 138 %
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Residual Activity '=' 103 %
P30281 BXGT009416 G1/S-specific cyclin-D3 reviewed Enzyme modulator CCND3 Residual Activity '=' 103 %
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Residual Activity '=' 80 %
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Residual Activity '=' 130 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 91 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 91 %
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Residual Activity '=' 101 %
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Residual Activity '=' 89 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Residual Activity '=' 92 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Residual Activity '=' 52 %
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Residual Activity '=' 102 %
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Residual Activity '=' 94 %
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Residual Activity '=' 87 %
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 AC50 '=' 31622 nM
O89049 BXGT005293 Thioredoxin reductase 1, cytoplasmic reviewed - Txnrd1 Potency - 39810 nM
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Residual Activity '=' 92 %
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Residual Activity '=' 95 %
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Residual Activity '=' 114 %
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Residual Activity '=' 103 %
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Residual Activity '=' 92 %
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 14125 nM
Q16236 BXGT013624 Nuclear factor erythroid 2-related factor 2 reviewed Enzyme NFE2L2 Potency - 16360 nM
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 AC50 '=' 39810 nM
P16050 BXGT008184 Arachidonate 15-lipoxygenase reviewed Enzyme ALOX15 Potency '=' 19952 nM
P04637 BXGT006243 Cellular tumor antigen p53 reviewed Transcription factor TP53 Potency '=' 12589 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Residual Activity '=' 105 %
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Residual Activity '=' 92 %
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Residual Activity '=' 100 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Residual Activity '=' 84 %
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Residual Activity '=' 78 %
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Residual Activity '=' 100 %
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Residual Activity '=' 75 %
Q8IYT8 BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 Residual Activity '=' 94 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Residual Activity '=' 91 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Residual Activity '=' 90 %
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Residual Activity '=' 86 %
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Residual Activity '=' 91 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency '=' 63095 nM
P08482 BXGT006775 Muscarinic acetylcholine receptor M1 reviewed - Chrm1 Potency '=' 35481 nM
Q9BYP7 BXGT020188 Serine/threonine-protein kinase WNK3 reviewed Kinase WNK3 Residual Activity '=' 84 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 92 %
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Residual Activity '=' 75 %
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Residual Activity '=' 101 %
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Residual Activity '=' 107 %
P43250 BXGT010372 G protein-coupled receptor kinase 6 reviewed Kinase GRK6 Residual Activity '=' 96 %
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Residual Activity '=' 126 %
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Residual Activity '=' 62 %
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Residual Activity '=' 91 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Residual Activity '=' 101 %
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Residual Activity '=' 77 %
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Residual Activity '=' 94 %
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Residual Activity '=' 89 %
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Residual Activity '=' 108 %
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Residual Activity '=' 65 %
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Residual Activity '=' 92 %
Q96PF2 BXGT019708 Testis-specific serine/threonine-protein kinase 2 reviewed Kinase TSSK2 Residual Activity '=' 102 %
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 Potency '=' 25118 nM
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Residual Activity '=' 100 %
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Residual Activity '=' 123 %
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Residual Activity '=' 86 %
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Residual Activity '=' 81 %
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Residual Activity '=' 60 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 117 %
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Residual Activity '=' 98 %
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Residual Activity '=' 97 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Residual Activity '=' 115 %
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Residual Activity '=' 130 %
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Residual Activity '=' 120 %
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Residual Activity '=' 73 %
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Residual Activity '=' 101 %
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Residual Activity '=' 79 %
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Residual Activity '=' 102 %
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Residual Activity '=' 94 %
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Residual Activity '=' 61 %
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Residual Activity '=' 103 %
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Residual Activity '=' 114 %
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 AC50 '=' 25118 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Residual Activity '=' 103 %
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Residual Activity '=' 102 %
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Residual Activity '=' 53 %
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Residual Activity '=' 65 %
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Residual Activity '=' 83 %
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Residual Activity '=' 130 %
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Residual Activity '=' 87 %
P51946 BXGT010907 Cyclin-H reviewed Enzyme modulator CCNH Residual Activity '=' 87 %
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Residual Activity '=' 96 %
P49798 BXGT010745 Regulator of G-protein signaling 4 reviewed Enzyme modulator RGS4 Potency - 6701 nM
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Residual Activity '=' 63 %
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Residual Activity '=' 87 %
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Residual Activity '=' 90 %
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Residual Activity '=' 84 %
P14635 BXGT008031 G2/mitotic-specific cyclin-B1 reviewed Enzyme modulator CCNB1 Residual Activity '=' 103 %
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Residual Activity '=' 103 %
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Residual Activity '=' 85 %
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Residual Activity '=' 90 %
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Residual Activity '=' 71 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 110 %
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Residual Activity '=' 110 %
P67870 BXGT011566 Casein kinase II subunit beta reviewed Kinase CSNK2B Residual Activity '=' 110 %
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Residual Activity '=' 84 %
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Residual Activity '=' 81 %
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 15848 nM
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Residual Activity '=' 79 %
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Residual Activity '=' 76 %
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Residual Activity '=' 106 %
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Residual Activity '=' 90 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 126 %
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Residual Activity '=' 111 %
Q86Z02 BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 Residual Activity '=' 95 %
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Residual Activity '=' 85 %
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Residual Activity '=' 82 %
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Residual Activity '=' 82 %
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Residual Activity '=' 55 %
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Residual Activity '=' 98 %
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Residual Activity '=' 90 %
Q96BR1 BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed - SGK3 Residual Activity '=' 79 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Residual Activity '=' 109 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Residual Activity '=' 115 %
O94956 BXGT005343 Solute carrier organic anion transporter family member 2B1 reviewed Transporter SLCO2B1 Inhibition '=' 13 %
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Residual Activity '=' 84 %
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Residual Activity '=' 107 %
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Residual Activity '=' 108 %
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Residual Activity '=' 88 %
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Residual Activity '=' 85 %
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Residual Activity '=' 84 %
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Residual Activity '=' 69 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Residual Activity '=' 73 %
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Residual Activity '=' 119 %
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Residual Activity '=' 110 %
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Residual Activity '=' 95 %
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Residual Activity '=' 103 %
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Residual Activity '=' 81 %
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Residual Activity '=' 79 %
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Residual Activity '=' 77 %
P00352 BXGT005510 Retinal dehydrogenase 1 reviewed Enzyme ALDH1A1 Potency '=' 15848 nM
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Residual Activity '=' 81 %
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Residual Activity '=' 92 %
P78396 BXGT011842 Cyclin-A1 reviewed Enzyme modulator CCNA1 Residual Activity '=' 137 %
P20248 BXGT008554 Cyclin-A2 reviewed Enzyme modulator CCNA2 Residual Activity '=' 137 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 137 %
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Residual Activity '=' 92 %
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Residual Activity '=' 96 %
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Residual Activity '=' 68 %
O97447 BXGT005436 Putative fructose-1,6-bisphosphate aldolase unreviewed - ald Potency '=' 17740 nM
P11473 BXGT007709 Vitamin D3 receptor reviewed Nuclear receptor VDR Potency - 28183 nM
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Residual Activity '=' 112 %
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Residual Activity '=' 66 %
Q9UGI9 BXGT021682 5'-AMP-activated protein kinase subunit gamma-3 reviewed Enzyme modulator PRKAG3 Residual Activity '=' 60 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 60 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 60 %
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Residual Activity '=' 60 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 60 %
O43741 BXGT004620 5'-AMP-activated protein kinase subunit beta-2 reviewed Enzyme modulator PRKAB2 Residual Activity '=' 60 %
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Residual Activity '=' 60 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 95 %
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Residual Activity '=' 101 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Residual Activity '=' 81 %
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Residual Activity '=' 94 %
O43318 BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 Residual Activity '=' 94 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 1263 nM
P51450 BXGT010847 Nuclear receptor ROR-gamma reviewed - Rorc Potency '=' 8912 nM
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 93 %
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Residual Activity '=' 101 %
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Residual Activity '=' 110 %
P15289 BXGT008102 Arylsulfatase A reviewed Enzyme ARSA Potency - 8492 nM
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Residual Activity '=' 98 %
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Residual Activity '=' 90 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 110 %
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Residual Activity '=' 94 %
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Residual Activity '=' 102 %
Q9F4F7 BXGT020344 4'-phosphopantetheinyl transferase ffp reviewed - ffp Potency '=' 50118 nM
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Residual Activity '=' 82 %
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Residual Activity '=' 102 %
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Residual Activity '=' 75 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 87 %
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Residual Activity '=' 95 %
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Residual Activity '=' 89 %
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Residual Activity '=' 59 %
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Residual Activity '=' 103 %
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Residual Activity '=' 86 %
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Residual Activity '=' 75 %
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Residual Activity '=' 115 %
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Residual Activity '=' 114 %
Q8TF76 BXGT018826 Serine/threonine-protein kinase haspin reviewed Kinase HASPIN Residual Activity '=' 69 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 82 %
Q16665 BXGT013653 Hypoxia-inducible factor 1-alpha reviewed Transcription factor HIF1A Potency '=' 31622 nM
P10828 BXGT007624 Thyroid hormone receptor beta reviewed Nuclear receptor THRB Potency '=' 70794 nM
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Residual Activity '=' 73 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Residual Activity '=' 112 %
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Residual Activity '=' 93 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 98 %
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Residual Activity '=' 95 %
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Residual Activity '=' 106 %
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Residual Activity '=' 140 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 84 %
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Residual Activity '=' 82 %
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Residual Activity '=' 94 %
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Residual Activity '=' 114 %
P51946 BXGT010907 Cyclin-H reviewed Enzyme modulator CCNH Residual Activity '=' 114 %
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Residual Activity '=' 93 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 101 %
Q9NYY3 BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 Residual Activity '=' 71 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 107 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Residual Activity '=' 112 %
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Residual Activity '=' 107 %
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Residual Activity '=' 102 %
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Residual Activity '=' 97 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Residual Activity '=' 100 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Residual Activity '=' 112 %
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Residual Activity '=' 94 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Residual Activity '=' 64 %
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Residual Activity '=' 48 %
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Residual Activity '=' 93 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Residual Activity '=' 121 %
Q8TF76 BXGT018826 Serine/threonine-protein kinase haspin reviewed Kinase HASPIN Residual Activity '=' 109 %
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Residual Activity '=' 83 %
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Residual Activity '=' 107 %
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Residual Activity '=' 44 %
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Residual Activity '=' 113 %
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Residual Activity '=' 108 %
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Residual Activity '=' 93 %
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Residual Activity '=' 47 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 131 %
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Residual Activity '=' 97 %
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Residual Activity '=' 102 %
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Residual Activity '=' 92 %
O97447 BXGT005436 Putative fructose-1,6-bisphosphate aldolase unreviewed - ald Potency '=' 5000 nM
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Residual Activity '=' 108 %
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Residual Activity '=' 91 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 80 %
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Residual Activity '=' 107 %
Q9NPD5 BXGT021151 Solute carrier organic anion transporter family member 1B3 reviewed Transporter SLCO1B3 Inhibition '=' 24 %
P51450 BXGT010847 Nuclear receptor ROR-gamma reviewed - Rorc Potency '=' 3981 nM
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Residual Activity '=' 85 %
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Residual Activity '=' 89 %
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Residual Activity '=' 101 %
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Residual Activity '=' 90 %
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Residual Activity '=' 95 %
Q03164 BXGT012700 Histone-lysine N-methyltransferase 2A reviewed - KMT2A Potency '=' 25118 nM
O00255 BXGT003903 Menin reviewed - MEN1 Potency '=' 25118 nM
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Residual Activity '=' 121 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 130 %
P05129 BXGT006322 Protein kinase C gamma type reviewed Kinase PRKCG Residual Activity '=' 101 %
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Residual Activity '=' 97 %
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Residual Activity '=' 94 %
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Residual Activity '=' 78 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Residual Activity '=' 110 %
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Residual Activity '=' 93 %
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Residual Activity '=' 80 %
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Residual Activity '=' 67 %
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Residual Activity '=' 105 %
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Residual Activity '=' 74 %
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Residual Activity '=' 108 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Residual Activity '=' 86 %
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Residual Activity '=' 93 %
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Residual Activity '=' 115 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 93 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 93 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 93 %
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Residual Activity '=' 121 %
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Residual Activity '=' 103 %
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Residual Activity '=' 82 %
P30281 BXGT009416 G1/S-specific cyclin-D3 reviewed Enzyme modulator CCND3 Residual Activity '=' 82 %
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Residual Activity '=' 133 %
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Residual Activity '=' 84 %
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Residual Activity '=' 110 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Residual Activity '=' 98 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Residual Activity '=' 105 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 103 %
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Residual Activity '=' 85 %
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Residual Activity '=' 88 %
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Residual Activity '=' 108 %
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Residual Activity '=' 67 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Residual Activity '=' 100 %
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Residual Activity '=' 77 %
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Residual Activity '=' 96 %
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Residual Activity '=' 86 %
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Residual Activity '=' 101 %
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Residual Activity '=' 130 %
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 16833 nM
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Residual Activity '=' 113 %
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Residual Activity '=' 87 %
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Residual Activity '=' 101 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 87 %
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Residual Activity '=' 86 %
P43250 BXGT010372 G protein-coupled receptor kinase 6 reviewed Kinase GRK6 Residual Activity '=' 93 %
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Residual Activity '=' 90 %
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Residual Activity '=' 76 %
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Residual Activity '=' 98 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 106 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 106 %
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Residual Activity '=' 83 %
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Residual Activity '=' 100 %
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Residual Activity '=' 75 %
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Residual Activity '=' 115 %
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Residual Activity '=' 97 %
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Residual Activity '=' 63 %
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Residual Activity '=' 91 %
P04637 BXGT006243 Cellular tumor antigen p53 reviewed Transcription factor TP53 Potency '=' 5011 nM
P15428 BXGT008121 15-hydroxyprostaglandin dehydrogenase [NAD(+)] reviewed - HPGD Potency '=' 19952 nM
P18054 BXGT008370 Arachidonate 12-lipoxygenase, 12S-type reviewed Enzyme ALOX12 Potency '=' 12589 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 96 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 96 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 96 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Residual Activity '=' 101 %
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Residual Activity '=' 104 %
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Residual Activity '=' 99 %
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Residual Activity '=' 110 %
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Residual Activity '=' 71 %
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Residual Activity '=' 137 %
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Residual Activity '=' 96 %
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Residual Activity '=' 126 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 89 %
Q9Y3S1 BXGT022266 Serine/threonine-protein kinase WNK2 reviewed Kinase WNK2 Residual Activity '=' 76 %
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Residual Activity '=' 90 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 101 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 101 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 101 %
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Residual Activity '=' 104 %
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Residual Activity '=' 65 %
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Residual Activity '=' 108 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Residual Activity '=' 3 %
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Residual Activity '=' 85 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 85 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 85 %
P20711 BXGT008594 Aromatic-L-amino-acid decarboxylase reviewed - DDC IC50 '=' 1280000 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Residual Activity '=' 97 %
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Residual Activity '=' 81 %
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Residual Activity '=' 96 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 107 %
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Residual Activity '=' 107 %
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Residual Activity '=' 83 %
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Residual Activity '=' 81 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Residual Activity '=' 104 %
O14733 BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 Residual Activity '=' 110 %
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Residual Activity '=' 110 %
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Residual Activity '=' 92 %
Q9UPE1 BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 Residual Activity '=' 66 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Residual Activity '=' 107 %
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Residual Activity '=' 102 %
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Residual Activity '=' 103 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 103 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 103 %
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Residual Activity '=' 104 %
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Residual Activity '=' 61 %
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Residual Activity '=' 72 %
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Residual Activity '=' 112 %
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Residual Activity '=' 120 %
Q92830 BXGT019379 Histone acetyltransferase KAT2A reviewed - KAT2A Potency - 31622 nM
Q03164 BXGT012700 Histone-lysine N-methyltransferase 2A reviewed - KMT2A Potency '=' 22387 nM
O00255 BXGT003903 Menin reviewed - MEN1 Potency '=' 22387 nM
Q9F4F7 BXGT020344 4'-phosphopantetheinyl transferase ffp reviewed - ffp Potency '=' 56234 nM
P05177 BXGT006336 Cytochrome P450 1A2 reviewed Enzyme CYP1A2 AC50 '=' 10000 nM
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Residual Activity '=' 72 %
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Residual Activity '=' 96 %
Q9Y6L6 BXGT022334 Solute carrier organic anion transporter family member 1B1 reviewed Transporter SLCO1B1 Inhibition '=' 0 %
P11021 BXGT007644 Endoplasmic reticulum chaperone BiP reviewed - HSPA5 Potency - 20749 nM
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Residual Activity '=' 126 %
P27338 BXGT009172 Amine oxidase [flavin-containing] B reviewed - MAOB IC50 '>' 20000 nM
P51450 BXGT010847 Nuclear receptor ROR-gamma reviewed - Rorc Potency '=' 7079 nM
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Residual Activity '=' 83 %
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Residual Activity '=' 31 %
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Residual Activity '=' 91 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 107 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 107 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 79 %
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA IC50 '=' 550 nM
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 89 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 89 %
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Residual Activity '=' 111 %
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Residual Activity '=' 97 %
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Residual Activity '=' 105 %
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Residual Activity '=' 119 %
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Residual Activity '=' 92 %
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Residual Activity '=' 90 %
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Residual Activity '=' 87 %
Q86Z02 BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 Residual Activity '=' 103 %
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Residual Activity '=' 115 %
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Residual Activity '=' 133 %
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Residual Activity '=' 70 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Residual Activity '=' 69 %
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Residual Activity '=' 89 %
Q63120 BXGT016061 Canalicular multispecific organic anion transporter 1 reviewed - Abcc2 Activity - - -
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Residual Activity '=' 47 %
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Residual Activity '=' 96 %
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Residual Activity '=' 94 %
Q8NG66 BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 Residual Activity '=' 113 %
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Residual Activity '=' 97 %
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Residual Activity '=' 117 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 99 %
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Residual Activity '=' 119 %
Q8WTQ7 BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 Residual Activity '=' 99 %
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Residual Activity '=' 74 %
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Residual Activity '=' 101 %
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Residual Activity '=' 110 %
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Residual Activity '=' 82 %
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Residual Activity '=' 92 %
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Residual Activity '=' 94 %
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Residual Activity '=' 98 %
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Residual Activity '=' 100 %
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Residual Activity '=' 82 %
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Residual Activity '=' 105 %
P51151 BXGT010837 Ras-related protein Rab-9A reviewed - RAB9A Potency '=' 46109 nM
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Residual Activity '=' 88 %
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Residual Activity '=' 102 %
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Residual Activity '=' 93 %
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Residual Activity '=' 113 %
P27695 BXGT009199 DNA-(apurinic or apyrimidinic site) lyase reviewed - APEX1 Potency - 10000 nM
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Residual Activity '=' 57 %
Q4Q090 BXGT014858 2,3-bisphosphoglycerate-independent phosphoglycerate mutase unreviewed - PGAM Potency - 15101 nM
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Residual Activity '=' 115 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Residual Activity '=' 107 %
Q9Y3S1 BXGT022266 Serine/threonine-protein kinase WNK2 reviewed Kinase WNK2 Residual Activity '=' 114 %
Q96PF2 BXGT019708 Testis-specific serine/threonine-protein kinase 2 reviewed Kinase TSSK2 Residual Activity '=' 108 %
Q9BYP7 BXGT020188 Serine/threonine-protein kinase WNK3 reviewed Kinase WNK3 Residual Activity '=' 117 %
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Residual Activity '=' 98 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 98 %
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Residual Activity '=' 99 %
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Residual Activity '=' 114 %
O75604 BXGT005139 Ubiquitin carboxyl-terminal hydrolase 2 reviewed Enzyme USP2 Potency '=' 25118 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Residual Activity '=' 104 %
P27695 BXGT009199 DNA-(apurinic or apyrimidinic site) lyase reviewed - APEX1 Potency - 25118 nM
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Residual Activity '=' 53 %
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Residual Activity '=' 97 %
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Residual Activity '=' 79 %
Q8NG66 BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 Residual Activity '=' 104 %
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Residual Activity '=' 74 %
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Residual Activity '=' 104 %
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Residual Activity '=' 87 %
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Residual Activity '=' 106 %
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Residual Activity '=' 95 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Residual Activity '=' 12 %
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Residual Activity '=' 81 %
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Residual Activity '=' 65 %
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA Activity '=' 75 %
Q9UGI9 BXGT021682 5'-AMP-activated protein kinase subunit gamma-3 reviewed Enzyme modulator PRKAG3 Residual Activity '=' 89 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 89 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 89 %
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Residual Activity '=' 89 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 89 %
O43741 BXGT004620 5'-AMP-activated protein kinase subunit beta-2 reviewed Enzyme modulator PRKAB2 Residual Activity '=' 89 %
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Residual Activity '=' 89 %
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Residual Activity '=' 72 %
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Residual Activity '=' 98 %
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Residual Activity '=' 63 %
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Residual Activity '=' 94 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Residual Activity '=' 99 %
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Residual Activity '=' 63 %
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Residual Activity '=' 105 %
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Residual Activity '=' 75 %
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Residual Activity '=' 83 %
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Residual Activity '=' 92 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Residual Activity '=' 104 %
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Residual Activity '=' 70 %
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Residual Activity '=' 101 %
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA Ki '=' 220 nM
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA Inhibition - - -
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA Activity '=' 28 %
P21397 BXGT008644 Amine oxidase [flavin-containing] A reviewed - MAOA Activity '=' 28 %
P27338 BXGT009172 Amine oxidase [flavin-containing] B reviewed - MAOB Activity '=' 94 %
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF01052 Artabotrys maingayi Artabotrys maingayi Medicinal Plant
BXGF01147 Chelidonium majus Chelidonium majus Medicinal Plant
BXGF01445 Acronychia laurifolia Acronychia laurifolia Medicinal Plant
BXGF01587 Talipariti tiliaceum Talipariti tiliaceum Medicinal Plant
BXGF02193 Broussonetia kazinoki Broussonetia kazinoki Medicinal Plant
BXGF02254 Thuja plicata Thuja plicata Medicinal Plant
BXGF02557 Lamprocapnos spectabilis Lamprocapnos spectabilis Others
BXGF02672 Papaver commutatum Papaver commutatum Medicinal Plant
BXGF02860 Macleaya cordata Macleaya cordata Medicinal Plant
BXGF02933 Hosta sieboldiana Hosta sieboldiana Medicinal Plant
BXGF03260 Garcinia xanthochymus Garcinia xanthochymus Medicinal Plant
BXGF03381 Hylomecon japonica Hylomecon japonica Medicinal Plant
BXGF03433 Inula salsoloides Inula salsoloides Others
BXGF03464 Senna spectabilis Senna spectabilis Medicinal Plant
BXGF03557 Eutrochium purpureum Eutrochium purpureum Medicinal Plant
BXGF03612 Symphytum officinale Symphytum officinale Medicinal Plant
BXGF03764 Psacalium peltatum Psacalium peltatum Medicinal Plant
BXGF03829 Morinda coreia Morinda coreia Medicinal Plant
BXGF03830 Diospyros ebenum Diospyros ebenum Medicinal Plant
BXGF03888 Angelica dahurica Angelica dahurica Medicinal Plant
BXGF03914 Jacobaea cannabifolia Jacobaea cannabifolia Others
BXGF03960 Conium maculatum Conium maculatum Medicinal Plant
BXGF03971 Corydalis ophiocarpa Corydalis ophiocarpa Medicinal Plant
BXGF03979 Aglaia pyramidata Aglaia pyramidata Others
BXGF03992 Schrebera swietenoides Schrebera swietenoides Human Edible Plant
BXGF04006 Corydalis ternata Corydalis ternata Others
BXGF04008 Senecio gilliesi Senecio gilliesi Others
BXGF04020 Celastrus monospermus Celastrus monospermus Others
BXGF04055 Teclea sudanica Teclea sudanica Others
BXGF04063 Mezzettia leptopoda Mezzettia leptopoda Others
BXGF04078 Solanum spirale Solanum spirale Medicinal Plant
BXGF04101 Agave deserti Agave deserti Human Edible Plant
BXGF04111 Asclepias subulata Asclepias subulata Medicinal Plant
BXGF04119 Stachys plumosa Stachys plumosa Others
BXGF04178 Piper methysticum Piper methysticum Medicinal Plant
BXGF04190 Lappula echinata Lappula echinata Medicinal Plant
BXGF04201 Zanthoxylum simulans Zanthoxylum simulans Medicinal Plant
BXGF04237 Ligularia sagitta Ligularia sagitta Medicinal Plant
BXGF04354 Sophora leachiana Sophora leachiana Medicinal Plant
BXGF04702 Vernonia lilacina Vernonia lilacina Others
BXGF04806 Ulex airensis Ulex airensis Others
BXGF04929 Passiflora morifolia Passiflora morifolia Human Edible Plant
BXGF05074 Chaetomorpha moniligera Chaetomorpha moniligera Others
BXGF05103 Argemone mexicana Argemone mexicana Medicinal Plant
BXGF05186 Hortonia floribunda Hortonia floribunda Others
BXGF05442 Zanthoxylum bungeanum Zanthoxylum bungeanum Medicinal Plant
BXGF05476 Broussonetia papyrifera Broussonetia papyrifera Medicinal Plant
BXGF05482 Cephalocroton cordofanus Cephalocroton cordofanus Human Edible Plant
BXGF05622 Corydalis incisa Corydalis incisa Medicinal Plant
BXGF05805 Toddalia asiatica Toddalia asiatica Medicinal Plant
BXGF06182 Ventilago madraspatana Ventilago madraspatana Medicinal Plant
BXGF06268 Zanthoxylum nitidum Zanthoxylum nitidum Medicinal Plant
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease