| P81908 |
BXGT011959 |
Cholinesterase |
reviewed |
- |
BCHE |
Inhibition |
'=' |
6 |
% |
| O00141 |
BXGT003882 |
Serine/threonine-protein kinase Sgk1 |
reviewed |
Kinase |
SGK1 |
Inhibition |
'=' |
35 |
% |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Ki |
'=' |
23 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Activity |
'=' |
0 |
% |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
199 |
nM |
| P38918 |
BXGT010071 |
Aflatoxin B1 aldehyde reductase member 3 |
reviewed |
- |
Akr7a3 |
Inhibition |
'=' |
5 |
% |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
1500 |
nM |
| Q01279 |
BXGT012581 |
Epidermal growth factor receptor |
reviewed |
- |
Egfr |
Inhibition |
'=' |
25 |
% |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat |
'=' |
1 |
/s |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat/Km |
'=' |
0 |
/uM/s |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Activity |
'=' |
110 |
nM/s |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
FC |
'=' |
20 |
- |
| P18031 |
BXGT008369 |
Tyrosine-protein phosphatase non-receptor type 1 |
reviewed |
- |
PTPN1 |
IC50 |
'=' |
23300 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
IC50 |
'=' |
3200 |
nM |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
IC50 |
'=' |
21400 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
IC50 |
'=' |
25000 |
nM |
| P11021 |
BXGT007644 |
Endoplasmic reticulum chaperone BiP |
reviewed |
- |
HSPA5 |
Potency |
- |
50118 |
nM |
| P28907 |
BXGT009301 |
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 |
reviewed |
Enzyme |
CD38 |
IC50 |
'=' |
37900 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
AC50 |
'=' |
15848 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
2200 |
nM |
| P10584 |
BXGT007580 |
Malate dehydrogenase |
reviewed |
- |
mdh |
IC50 |
'=' |
6000 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Change in IC50 |
'>' |
50 |
fold |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
12589 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
Inhibition |
- |
- |
- |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
IC50 |
'=' |
2500 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
Ki |
'=' |
6990 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
446 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
- |
- |
- |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
IC50 |
'=' |
5730 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
IC50 |
'=' |
580 |
nM |
| Q99895 |
BXGT019974 |
Chymotrypsin-C |
reviewed |
- |
CTRC |
IC50 |
'=' |
100000 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
500 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
199 |
% |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Activity |
- |
- |
- |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
'=' |
1270 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
47 |
% |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
2377 |
nM |
| Q38C41 |
BXGT014361 |
Phosphotransferase |
unreviewed |
- |
Tb10.70.5800 |
IC50 |
'=' |
22378 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'>' |
50 |
% |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
94 |
% |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
Ki |
'=' |
30000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Activity |
'=' |
80 |
nM/s |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
Potency |
'=' |
15848 |
nM |
| Q96QE3 |
BXGT019718 |
ATPase family AAA domain-containing protein 5 |
reviewed |
- |
ATAD5 |
Potency |
- |
20587 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
- |
- |
- |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
11220 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
IC50 |
'=' |
5750 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
- |
- |
- |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
Activity |
- |
- |
- |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
Inhibition |
'=' |
102 |
% |
| P04745 |
BXGT006255 |
Alpha-amylase 1 |
reviewed |
- |
AMY1A |
Inhibition |
'=' |
82 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
631 |
nM |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q15208 |
BXGT013550 |
Serine/threonine-protein kinase 38 |
reviewed |
Kinase |
STK38 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q8IV63 |
BXGT018341 |
Inactive serine/threonine-protein kinase VRK3 |
reviewed |
Kinase |
VRK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| P00390 |
BXGT005526 |
Glutathione reductase, mitochondrial |
reviewed |
Enzyme |
GSR |
IC50 |
'=' |
218000 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Km |
'=' |
100400 |
nM |
| Q16512 |
BXGT013631 |
Serine/threonine-protein kinase N1 |
reviewed |
Kinase |
PKN1 |
IC50 |
'=' |
5800 |
nM |
| P08069 |
BXGT006723 |
Insulin-like growth factor 1 receptor |
reviewed |
Kinase |
IGF1R |
IC50 |
'=' |
300 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
14125 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
15848 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Activity |
- |
- |
- |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Kq |
'=' |
1 |
10'12/M/s |
| P29372 |
BXGT009336 |
DNA-3-methyladenine glycosylase |
reviewed |
Enzyme |
MPG |
Inhibition |
'=' |
44 |
% |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
35 |
% |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
Ki |
- |
- |
- |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
FC |
'=' |
4 |
- |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
26608 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
IC50 |
'=' |
1100 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
28183 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
1835 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
40 |
% |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
- |
- |
- |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'>' |
135000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
3162 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
IC50 |
- |
- |
- |
| O88397 |
BXGT005271 |
Solute carrier organic anion transporter family member 1A5 |
reviewed |
- |
Slco1a5 |
Activity |
'=' |
52 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1122 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'<' |
10 |
% |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
Ki |
'=' |
68000 |
nM |
| P04792 |
BXGT006264 |
Heat shock protein beta-1 |
reviewed |
- |
HSPB1 |
Activity |
- |
- |
- |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
- |
- |
- |
| P45452 |
BXGT010462 |
Collagenase 3 |
reviewed |
Enzyme |
MMP13 |
Inhibition |
'>' |
30 |
% |
| Q9Y2D0 |
BXGT022229 |
Carbonic anhydrase 5B, mitochondrial |
reviewed |
- |
CA5B |
Ki |
'=' |
11900 |
nM |
| P43166 |
BXGT010364 |
Carbonic anhydrase 7 |
reviewed |
- |
CA7 |
Ki |
'=' |
4840 |
nM |
| Q16790 |
BXGT013670 |
Carbonic anhydrase 9 |
reviewed |
- |
CA9 |
Ki |
'=' |
7000 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
200 |
nM |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
- |
- |
- |
| Q02769 |
BXGT012668 |
Squalene synthase |
reviewed |
- |
Fdft1 |
IC50 |
- |
- |
- |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat |
'=' |
12 |
/s |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
Activity |
- |
- |
- |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Ki |
'=' |
106700 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
10000 |
nM |
| P16116 |
BXGT008197 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
39900 |
nM |
| Q01453 |
BXGT012588 |
Peripheral myelin protein 22 |
reviewed |
Cellular structure |
PMP22 |
Potency |
'=' |
47754 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
39810 |
nM |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
'=' |
430 |
nM |
| P39900 |
BXGT010148 |
Macrophage metalloelastase |
reviewed |
Enzyme |
MMP12 |
IC50 |
'=' |
10230 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
56234 |
nM |
| P39900 |
BXGT010148 |
Macrophage metalloelastase |
reviewed |
Enzyme |
MMP12 |
Inhibition |
'>' |
30 |
% |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
7943 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
31622 |
nM |
| Q28731 |
BXGT013954 |
Thrombin |
unreviewed |
- |
thrombin |
TT |
'=' |
19 |
s |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
'=' |
1150 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
79432 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
7943 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
17782 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
1 |
- |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Activity |
'=' |
140 |
nM/s |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
77 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
'=' |
18800 |
nM |
| Q9HAW8 |
BXGT020509 |
UDP-glucuronosyltransferase 1-10 |
reviewed |
- |
UGT1A10 |
Activity |
'=' |
97 |
pm/min/mg |
| P22310 |
BXGT008754 |
UDP-glucuronosyltransferase 1-4 |
reviewed |
- |
UGT1A4 |
Activity |
'=' |
0 |
pm/min/mg |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Thermal melting change |
'=' |
9 |
degrees C |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Thermal melting change |
'=' |
3 |
degrees C |
| P10275 |
BXGT007552 |
Androgen receptor |
reviewed |
Nuclear receptor |
AR |
EC150 |
- |
- |
- |
| P21917 |
BXGT008707 |
D(4) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD4 |
Ki |
'=' |
7846 |
nM |
| P08908 |
BXGT006837 |
5-hydroxytryptamine receptor 1A |
reviewed |
G-protein coupled receptor |
HTR1A |
EC50 |
'>' |
100000 |
nM |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
35481 |
nM |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Potency |
'=' |
5623 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
10000 |
nM |
| P14061 |
BXGT007979 |
Estradiol 17-beta-dehydrogenase 1 |
reviewed |
Enzyme |
HSD17B1 |
Activity |
'=' |
65 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
15848 |
nM |
| Q8BRK8 |
BXGT017920 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
- |
Prkaa2 |
Activity |
- |
- |
- |
| P22513 |
BXGT008777 |
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal |
reviewed |
- |
|
IC50 |
'=' |
142000 |
nM |
| P28907 |
BXGT009301 |
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 |
reviewed |
Enzyme |
CD38 |
Ratio IC50 |
'=' |
9 |
- |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Thermal melting change |
'=' |
2 |
degrees C |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
IC50 |
- |
- |
- |
| P35503 |
BXGT009840 |
UDP-glucuronosyltransferase 1-3 |
reviewed |
- |
UGT1A3 |
Activity |
'=' |
550 |
pm/min/mg |
| O60656 |
BXGT004889 |
UDP-glucuronosyltransferase 1-9 |
reviewed |
- |
UGT1A9 |
Activity |
'=' |
1800 |
pm/min/mg |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
14125 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
IC50 |
'=' |
4000 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Inhibition |
'=' |
43 |
% |
| P08238 |
BXGT006753 |
Heat shock protein HSP 90-beta |
reviewed |
Chaperone |
HSP90AB1 |
Activity |
- |
- |
- |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Thermal melting change |
'=' |
1 |
degrees C |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
5 |
degrees C |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
4466 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'=' |
31 |
% |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'=' |
15000 |
nM |
| P0C6X7 |
BXGT007440 |
Replicase polyprotein 1ab |
reviewed |
- |
rep |
IC50 |
'>' |
50000 |
nM |
| O95067 |
BXGT005347 |
G2/mitotic-specific cyclin-B2 |
reviewed |
Enzyme modulator |
CCNB2 |
IC50 |
'=' |
75000 |
nM |
| Q8WWL7 |
BXGT019000 |
G2/mitotic-specific cyclin-B3 |
reviewed |
Enzyme modulator |
CCNB3 |
IC50 |
'=' |
75000 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
75000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
75000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat |
'=' |
3 |
/s |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Ki |
'=' |
1200 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
AC50 |
'=' |
316 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
300 |
nM |
| P21588 |
BXGT008668 |
5'-nucleotidase |
reviewed |
- |
Nt5e |
Ki |
'=' |
45 |
nM |
| P23443 |
BXGT008866 |
Ribosomal protein S6 kinase beta-1 |
reviewed |
Kinase |
RPS6KB1 |
Inhibition |
'=' |
25 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
891 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
7810 |
nM |
| P56560 |
BXGT011180 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
20000 |
nM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
IC50 |
'=' |
17 |
ug.mL-1 |
| P0C6E9 |
BXGT007427 |
Sialidase |
reviewed |
- |
nanH |
Activity |
- |
- |
- |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Kd |
'=' |
25 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Kb |
'=' |
39 |
10^6/M |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
ID50 |
'=' |
22 |
ug ml-1 |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
80 |
% |
| P42226 |
BXGT010288 |
Signal transducer and activator of transcription 6 |
reviewed |
Nucleic acid binding |
STAT6 |
Potency |
'=' |
2511 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
550 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
550 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
550 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Thermal melting change |
'=' |
2 |
degrees C |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Thermal melting change |
'=' |
5 |
degrees C |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Thermal melting change |
'=' |
3 |
degrees C |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Thermal melting change |
'=' |
7 |
degrees C |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Activity |
- |
- |
- |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
5930 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
8912 |
nM |
| Q01062 |
BXGT012563 |
cGMP-dependent 3',5'-cyclic phosphodiesterase |
reviewed |
- |
Pde2a |
IC50 |
'=' |
81300 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
1 |
ug.mL-1 |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Ki |
'=' |
473 |
nM |
| Q9Y6L6 |
BXGT022334 |
Solute carrier organic anion transporter family member 1B1 |
reviewed |
Transporter |
SLCO1B1 |
Inhibition |
'=' |
77 |
% |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Inhibition |
'=' |
72 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
2000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat/Km |
'=' |
0 |
/uM/s |
| P07861 |
BXGT006690 |
Neprilysin |
reviewed |
- |
Mme |
Inhibition |
'=' |
49 |
% |
| Q03114 |
BXGT012692 |
Cyclin-dependent-like kinase 5 |
reviewed |
- |
Cdk5 |
EC50 |
'=' |
63400 |
nM |
| P06278 |
BXGT006431 |
Alpha-amylase |
reviewed |
- |
amyS |
Activity |
- |
- |
- |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Thermal melting change |
'=' |
3 |
degrees C |
| O00506 |
BXGT003932 |
Serine/threonine-protein kinase 25 |
reviewed |
Kinase |
STK25 |
Thermal melting change |
'=' |
5 |
degrees C |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
14125 |
nM |
| O15648 |
BXGT004185 |
ATP-dependent 6-phosphofructokinase |
reviewed |
- |
pfk |
Potency |
- |
6745 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
'=' |
13000 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
7210 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
25118 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
25118 |
nM |
| Q01279 |
BXGT012581 |
Epidermal growth factor receptor |
reviewed |
- |
Egfr |
Inhibition |
'=' |
30 |
% |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
87600 |
nM |
| P04054 |
BXGT006136 |
Phospholipase A2 |
reviewed |
Enzyme |
PLA2G1B |
IC50 |
'=' |
2000 |
nM |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Activity |
'=' |
80 |
% |
| P0AEK4 |
BXGT007320 |
Enoyl-[acyl-carrier-protein] reductase [NADH] FabI |
reviewed |
- |
fabI |
IC50 |
'=' |
20000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
281 |
nM |
| P0C6X7 |
BXGT007440 |
Replicase polyprotein 1ab |
reviewed |
- |
rep |
IC50 |
'=' |
23800 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
2511 |
nM |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
15 |
% |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
19952 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
4 |
% |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Km |
'=' |
127000 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
IC50 |
'=' |
30000 |
nM |
| Q9D6N1 |
BXGT020260 |
Carbonic anhydrase 13 |
reviewed |
- |
Ca13 |
Ki |
'=' |
9030 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Increase in IC50 |
'>' |
50 |
- |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Decrease in IC50 |
'=' |
2 |
- |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
IC50 |
'=' |
590 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
28183 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Activity |
'=' |
100 |
nM/s |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
10000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
EC50 |
'>' |
100 |
mg kg-1 |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
3000 |
nM |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
Kd |
'=' |
7079 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
#NAME? |
'=' |
0 |
uM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
3000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
7079 |
nM |
| P35218 |
BXGT009796 |
Carbonic anhydrase 5A, mitochondrial |
reviewed |
- |
CA5A |
Ki |
'=' |
6810 |
nM |
| Q91WR5 |
BXGT019303 |
Aldo-keto reductase family 1 member C21 |
reviewed |
- |
Akr1c21 |
IC50 |
'=' |
6900 |
nM |
| Q91WR5 |
BXGT019303 |
Aldo-keto reductase family 1 member C21 |
reviewed |
- |
Akr1c21 |
Ki |
'=' |
11000 |
nM |
| Q9NWT6 |
BXGT021234 |
Hypoxia-inducible factor 1-alpha inhibitor |
reviewed |
- |
HIF1AN |
IC50 |
'=' |
10200 |
nM |
| Q63921 |
BXGT016082 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
Ptgs1 |
IC50 |
'>' |
50000 |
nM |
| P35355 |
BXGT009817 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
Ptgs2 |
IC50 |
'>' |
50000 |
nM |
| P11387 |
BXGT007696 |
DNA topoisomerase 1 |
reviewed |
Enzyme |
TOP1 |
Activity |
- |
- |
- |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Activity |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Inhibition |
'=' |
83 |
% |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
Inhibition |
'=' |
19 |
% |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Inhibition |
'=' |
19 |
% |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
Inhibition |
'=' |
19 |
% |
| O97447 |
BXGT005436 |
Putative fructose-1,6-bisphosphate aldolase |
unreviewed |
- |
ald |
Potency |
'=' |
15811 |
nM |
| P12527 |
BXGT007824 |
Arachidonate 5-lipoxygenase |
reviewed |
- |
Alox5 |
IC50 |
'=' |
400 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
IC50 |
'=' |
15400 |
nM |
| P10828 |
BXGT007624 |
Thyroid hormone receptor beta |
reviewed |
Nuclear receptor |
THRB |
Potency |
'=' |
44668 |
nM |
| Q965D7 |
BXGT019602 |
Beta-hydroxyacyl-ACP dehydratase |
unreviewed |
- |
fabZ |
IC50 |
'=' |
1500 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
2511 |
nM |
| Q99549 |
BXGT019932 |
M-phase phosphoprotein 8 |
reviewed |
Epigenetic regulator |
MPHOSPH8 |
Potency |
- |
39810 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
IC50 |
'=' |
220000 |
nM |
| P37238 |
BXGT009974 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
- |
Pparg |
Activity |
- |
- |
- |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Inhibition |
'=' |
90 |
% |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Inhibition |
'=' |
132 |
% |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Inhibition |
'=' |
138 |
% |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1000 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
IC50 |
'=' |
10500 |
nM |
| P16116 |
BXGT008197 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
2850 |
nM |
| O76074 |
BXGT005174 |
cGMP-specific 3',5'-cyclic phosphodiesterase |
reviewed |
- |
PDE5A |
Inhibition |
'=' |
23 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
Activity |
- |
- |
- |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Thermal melting change |
'=' |
3 |
degrees C |
| P15289 |
BXGT008102 |
Arylsulfatase A |
reviewed |
Enzyme |
ARSA |
Potency |
- |
33807 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
6900 |
nM |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| P19838 |
BXGT008526 |
Nuclear factor NF-kappa-B p105 subunit |
reviewed |
Transcription factor |
NFKB1 |
Inhibition |
- |
- |
- |
| Q00653 |
BXGT012541 |
Nuclear factor NF-kappa-B p100 subunit |
reviewed |
Transcription factor |
NFKB2 |
Inhibition |
- |
- |
- |
| P08482 |
BXGT006775 |
Muscarinic acetylcholine receptor M1 |
reviewed |
- |
Chrm1 |
Potency |
'=' |
3162 |
nM |
| P16116 |
BXGT008197 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
10340 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
1700 |
nM |
| P23280 |
BXGT008844 |
Carbonic anhydrase 6 |
reviewed |
- |
CA6 |
Ki |
'=' |
6170 |
nM |
| Q9ULX7 |
BXGT021769 |
Carbonic anhydrase 14 |
reviewed |
- |
CA14 |
Ki |
'=' |
5410 |
nM |
| P0DMS8 |
BXGT007506 |
Adenosine receptor A3 |
reviewed |
G-protein coupled receptor |
ADORA3 |
pKi(uM) |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
1000 |
nM |
| Q66HS9 |
BXGT016172 |
Monocarboxylate transporter 2 |
unreviewed |
- |
Slc16a7 |
IC50 |
'=' |
5000 |
nM |
| P14916 |
BXGT008066 |
Urease subunit alpha |
reviewed |
- |
ureA |
IC50 |
'=' |
11000 |
nM |
| P69996 |
BXGT011656 |
Urease subunit beta |
reviewed |
- |
ureB |
IC50 |
'=' |
11000 |
nM |
| P08482 |
BXGT006775 |
Muscarinic acetylcholine receptor M1 |
reviewed |
- |
Chrm1 |
Potency |
'=' |
19952 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
2400 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
IC50 |
'=' |
2100 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
IC50 |
'=' |
2100 |
nM |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
18492 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
17782 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Potency |
'=' |
794 |
nM |
| P11064 |
BXGT007646 |
Low molecular weight phosphotyrosine protein phosphatase |
reviewed |
- |
ACP1 |
FC |
'=' |
2 |
- |
| P35030 |
BXGT009784 |
Trypsin-3 |
reviewed |
Enzyme |
PRSS3 |
IC50 |
'=' |
15400 |
nM |
| P07478 |
BXGT006630 |
Trypsin-2 |
reviewed |
Enzyme |
PRSS2 |
IC50 |
'=' |
15400 |
nM |
| P07477 |
BXGT006629 |
Trypsin-1 |
reviewed |
Enzyme |
PRSS1 |
IC50 |
'=' |
15400 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Ka |
'=' |
2 |
10'7/M |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
17782 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Thermal melting change |
'=' |
4 |
degrees C |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
2 |
- |
| P41921 |
BXGT010274 |
Glutathione reductase |
reviewed |
- |
GLR1 |
IC50 |
'=' |
48800 |
nM |
| P28839 |
BXGT009296 |
Cytosol aminopeptidase |
reviewed |
- |
LAP3 |
IC50 |
'=' |
34300 |
nM |
| P50578 |
BXGT010811 |
Aldo-keto reductase family 1 member A1 |
reviewed |
- |
AKR1A1 |
IC50 |
'=' |
38400 |
nM |
| P15122 |
BXGT008084 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
Inhibition |
'=' |
52 |
% |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
IC50 |
'>' |
10000 |
nM |
| P30530 |
BXGT009431 |
Tyrosine-protein kinase receptor UFO |
reviewed |
Kinase |
AXL |
IC50 |
'=' |
960 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
90000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Km |
'=' |
3200 |
nM |
| P00915 |
BXGT005689 |
Carbonic anhydrase 1 |
reviewed |
- |
CA1 |
Ki |
'=' |
2680 |
nM |
| P0DP23 |
BXGT007520 |
Calmodulin-1 |
reviewed |
- |
CALM1 |
Inhibition |
- |
- |
- |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
Selectivity quotient |
'=' |
7 |
- |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
2620 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
39810 |
nM |
| Q16665 |
BXGT013653 |
Hypoxia-inducible factor 1-alpha |
reviewed |
Transcription factor |
HIF1A |
Potency |
'=' |
10000 |
nM |
| O75828 |
BXGT005154 |
Carbonyl reductase [NADPH] 3 |
reviewed |
- |
CBR3 |
Tm |
'<' |
2 |
degrees C |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
Ki |
'=' |
3800 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
2200 |
nM |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
14125 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
14125 |
nM |
| P37231 |
BXGT009972 |
Peroxisome proliferator-activated receptor gamma |
reviewed |
Nuclear receptor |
PPARG |
FC |
'=' |
1 |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
31000 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
1191 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
2320 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Thermal melting change |
'=' |
2 |
degrees C |
| P07451 |
BXGT006627 |
Carbonic anhydrase 3 |
reviewed |
- |
CA3 |
Ki |
'=' |
8100 |
nM |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
Activity |
- |
- |
- |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Potency |
'=' |
6309 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
251 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
1000 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
81 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
15300 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
Inhibition |
'=' |
18 |
% |
| Q86831 |
BXGT017584 |
Polyprotein II |
unreviewed |
- |
|
Inhibition |
'=' |
41 |
% |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
'>' |
100000 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
Inhibition |
'=' |
48 |
% |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
Activity |
- |
- |
- |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
10000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Ratio IC50 |
'=' |
8 |
- |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat |
'=' |
8 |
/s |
| Q9Y3R4 |
BXGT022265 |
Sialidase-2 |
reviewed |
Enzyme |
NEU2 |
IC50 |
'=' |
160000 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
2818 |
nM |
| P0AES4 |
BXGT007329 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'=' |
55 |
ug.mL-1 |
| P0AES6 |
BXGT007331 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'=' |
55 |
ug.mL-1 |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
CC50 |
'=' |
46 |
ug.mL-1 |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
14 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
12589 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
39810 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
125 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
29855 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
Potency |
'=' |
15848 |
nM |
| P15122 |
BXGT008084 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
Inhibition |
'=' |
9 |
% |
| P28845 |
BXGT009297 |
Corticosteroid 11-beta-dehydrogenase isozyme 1 |
reviewed |
- |
HSD11B1 |
Inhibition |
'=' |
27 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
25118 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
2700 |
nM |
| Q96GD4 |
BXGT019667 |
Aurora kinase B |
reviewed |
Kinase |
AURKB |
IC50 |
'=' |
910 |
nM |
| O60285 |
BXGT004867 |
NUAK family SNF1-like kinase 1 |
reviewed |
Kinase |
NUAK1 |
IC50 |
'=' |
5090 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
450 |
nM |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
'>' |
31622 |
nM |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
FC |
'=' |
1 |
- |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
- |
- |
- |
| P54855 |
BXGT011088 |
UDP-glucuronosyltransferase 2B15 |
reviewed |
- |
UGT2B15 |
Activity |
'=' |
5 |
pm/min/mg |
| P14916 |
BXGT008066 |
Urease subunit alpha |
reviewed |
- |
ureA |
IC50 |
'=' |
11200 |
nM |
| P69996 |
BXGT011656 |
Urease subunit beta |
reviewed |
- |
ureB |
IC50 |
'=' |
11200 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
IC50 |
'=' |
5390 |
nM |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Activity |
- |
- |
- |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
IC50 |
'=' |
500 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'=' |
280 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
8912 |
nM |
| P11168 |
BXGT007663 |
Solute carrier family 2, facilitated glucose transporter member 2 |
reviewed |
Transporter |
SLC2A2 |
IC50 |
'=' |
12000 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
22387 |
nM |
| P19224 |
BXGT008468 |
UDP-glucuronosyltransferase 1-6 |
reviewed |
- |
UGT1A6 |
Activity |
'=' |
0 |
pm/min/mg |
| P0C6E9 |
BXGT007427 |
Sialidase |
reviewed |
- |
nanH |
Inhibition |
'=' |
29 |
% |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
10060 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
IC50 |
'=' |
6 |
ug.mL-1 |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Activity |
- |
- |
- |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'>' |
20000 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
8000 |
nM |
| Q00796 |
BXGT012549 |
Sorbitol dehydrogenase |
reviewed |
Enzyme |
SORD |
IC50 |
'=' |
177000 |
nM |
| P19357 |
BXGT008475 |
Solute carrier family 2, facilitated glucose transporter member 4 |
reviewed |
- |
Slc2a4 |
Ki |
'=' |
16000 |
nM |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
pKi(uM) |
'=' |
0 |
- |
| P84022 |
BXGT012027 |
Mothers against decapentaplegic homolog 3 |
reviewed |
Transcription factor |
SMAD3 |
Potency |
- |
35481 |
nM |
| Q99714 |
BXGT019954 |
3-hydroxyacyl-CoA dehydrogenase type-2 |
reviewed |
Enzyme |
HSD17B10 |
Potency |
'=' |
158 |
nM |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
31622 |
nM |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Inhibition |
'=' |
13 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Inhibition |
'=' |
13 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
- |
- |
- |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
IC50 |
'=' |
440 |
nM |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'>' |
20000 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
7700 |
nM |
| P16152 |
BXGT008201 |
Carbonyl reductase [NADPH] 1 |
reviewed |
- |
CBR1 |
Tm |
'<' |
2 |
degrees C |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
15848 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
'=' |
4500 |
nM |
| Q00796 |
BXGT012549 |
Sorbitol dehydrogenase |
reviewed |
Enzyme |
SORD |
IC50 |
'=' |
35600 |
nM |
| P51570 |
BXGT010858 |
Galactokinase |
reviewed |
Kinase |
GALK1 |
Potency |
'=' |
42128 |
nM |
| Q6W5P4 |
BXGT016588 |
Neuropeptide S receptor |
reviewed |
- |
NPSR1 |
Potency |
'=' |
158 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
9800 |
nM |
| B2RXH2 |
BXGT002006 |
Lysine-specific demethylase 4E |
reviewed |
- |
KDM4E |
Potency |
'=' |
8912 |
nM |
| P00760 |
BXGT005644 |
Cationic trypsin |
reviewed |
- |
|
IC50 |
'=' |
7100 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
5600 |
nM |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
2800 |
nM |
| P50578 |
BXGT010811 |
Aldo-keto reductase family 1 member A1 |
reviewed |
- |
AKR1A1 |
Activity |
- |
- |
- |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Thermal melting change |
'=' |
7 |
degrees C |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Thermal melting change |
'=' |
1 |
degrees C |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Thermal melting change |
'=' |
7 |
degrees C |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Thermal melting change |
'=' |
5 |
degrees C |
| P07378 |
BXGT006616 |
Phosphoglycerate kinase, glycosomal |
reviewed |
- |
|
Potency |
- |
7568 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Ki |
'=' |
1180 |
nM |
| P21398 |
BXGT008645 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
10 |
nM |
| P07943 |
BXGT006700 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
Akr1b1 |
IC50 |
'=' |
8320 |
nM |
| P51635 |
BXGT010869 |
Aldo-keto reductase family 1 member A1 |
reviewed |
- |
Akr1a1 |
IC50 |
'=' |
2320 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
'=' |
28183 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
IC50 |
'=' |
40 |
ug.mL-1 |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
22387 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
22387 |
nM |
| Q76353 |
BXGT016849 |
Integrase |
unreviewed |
- |
|
IC50 |
- |
- |
- |
| P24385 |
BXGT008965 |
G1/S-specific cyclin-D1 |
reviewed |
Enzyme modulator |
CCND1 |
IC50 |
'=' |
61000 |
nM |
| P11802 |
BXGT007750 |
Cyclin-dependent kinase 4 |
reviewed |
Kinase |
CDK4 |
IC50 |
'=' |
61000 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
- |
- |
- |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
12 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
FC |
'=' |
170 |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
900 |
nM |
| P10481 |
BXGT007573 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
'=' |
25340 |
nM |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
3162 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
IC50 |
'>' |
100000 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Inhibition |
'=' |
68 |
% |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
25118 |
nM |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
'=' |
10000 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
49 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
10000 |
nM |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
2511 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
11 |
% |
| P08236 |
BXGT006752 |
Beta-glucuronidase |
reviewed |
- |
GUSB |
Inhibition |
- |
- |
- |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Activity |
- |
- |
- |
| Q62868 |
BXGT016047 |
Rho-associated protein kinase 2 |
reviewed |
- |
Rock2 |
Inhibition |
'=' |
55 |
% |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Inhibition |
'=' |
30 |
% |
| Q8IW41 |
BXGT018352 |
MAP kinase-activated protein kinase 5 |
reviewed |
Kinase |
MAPKAPK5 |
Inhibition |
'=' |
51 |
% |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Inhibition |
'=' |
101 |
% |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
1122 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
IC50 |
'=' |
1540 |
nM |
| P0C6E9 |
BXGT007427 |
Sialidase |
reviewed |
- |
nanH |
IC50 |
- |
- |
- |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
12589 |
nM |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
IC50 |
'=' |
2200 |
nM |
| Q9UNA4 |
BXGT021785 |
DNA polymerase iota |
reviewed |
- |
POLI |
Potency |
- |
562 |
nM |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
30 |
% |
| Q1CTD3 |
BXGT013756 |
D-alanine--D-alanine ligase |
reviewed |
- |
ddl |
Ki |
'=' |
4300 |
nM |
| Q965D6 |
BXGT019601 |
3-oxoacyl-acyl-carrier protein reductase |
unreviewed |
- |
fabG |
IC50 |
'=' |
5400 |
nM |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
13600 |
nM |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
'=' |
420760 |
nM |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
35481 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
35481 |
nM |
| P53987 |
BXGT011023 |
Monocarboxylate transporter 1 |
reviewed |
- |
Slc16a1 |
IC50 |
'=' |
14000 |
nM |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
Activity |
- |
- |
- |
| P23219 |
BXGT008837 |
Prostaglandin G/H synthase 1 |
reviewed |
Enzyme |
PTGS1 |
Inhibition |
'=' |
90 |
% |
| O62664 |
BXGT004924 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
PTGS1 |
Inhibition |
- |
- |
- |
| P07862 |
BXGT006691 |
D-alanine--D-alanine ligase B |
reviewed |
- |
ddlB |
IC50 |
'=' |
19900 |
nM |
| P38918 |
BXGT010071 |
Aflatoxin B1 aldehyde reductase member 3 |
reviewed |
- |
Akr7a3 |
Inhibition |
'=' |
5 |
% |
| P38918 |
BXGT010071 |
Aflatoxin B1 aldehyde reductase member 3 |
reviewed |
- |
Akr7a3 |
Inhibition |
'=' |
6 |
% |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Ki |
'=' |
22 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
790 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
Inhibition |
'=' |
14 |
% |
| P16116 |
BXGT008197 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
10300 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Inhibition |
'=' |
25 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
14 |
% |
| Q15078 |
BXGT013534 |
Cyclin-dependent kinase 5 activator 1 |
reviewed |
Enzyme modulator |
CDK5R1 |
IC50 |
'=' |
23000 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
IC50 |
'=' |
23000 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
Ki |
'=' |
38300 |
nM |
| P0AES4 |
BXGT007329 |
DNA gyrase subunit A |
reviewed |
- |
gyrA |
IC50 |
'=' |
47 |
ug.mL-1 |
| P0AES6 |
BXGT007331 |
DNA gyrase subunit B |
reviewed |
- |
gyrB |
IC50 |
'=' |
47 |
ug.mL-1 |
| Q13526 |
BXGT013369 |
Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 |
reviewed |
- |
PIN1 |
Potency |
- |
2685 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
39810 |
nM |
| P83916 |
BXGT012025 |
Chromobox protein homolog 1 |
reviewed |
Epigenetic regulator |
CBX1 |
Potency |
- |
44668 |
nM |
| Q9HAW9 |
BXGT020510 |
UDP-glucuronosyltransferase 1-8 |
reviewed |
- |
UGT1A8 |
Activity |
'=' |
548 |
pm/min/mg |
| Q28731 |
BXGT013954 |
Thrombin |
unreviewed |
- |
thrombin |
Activity |
'=' |
5 |
g/L |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
Potency |
'=' |
31622 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Inhibition |
'=' |
72 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
3 |
% |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
12589 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
190000 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'=' |
20000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'=' |
20000 |
nM |
| P07265 |
BXGT006583 |
Alpha-glucosidase MAL62 |
reviewed |
- |
MAL62 |
logIC50 |
'=' |
0 |
- |
| O43570 |
BXGT004601 |
Carbonic anhydrase 12 |
reviewed |
- |
CA12 |
Ki |
'=' |
9390 |
nM |
| P97697 |
BXGT012214 |
Inositol monophosphatase 1 |
reviewed |
- |
Impa1 |
Potency |
'=' |
11220 |
nM |
| P0DP23 |
BXGT007520 |
Calmodulin-1 |
reviewed |
- |
CALM1 |
Ratio IC50 |
'=' |
2 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
76 |
% |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Ki |
'=' |
660 |
nM |
| Q01066 |
BXGT012565 |
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B |
reviewed |
- |
Pde1b |
IC50 |
'=' |
275000 |
nM |
| Q9EPR9 |
BXGT020293 |
Phosphodiesterase |
unreviewed |
- |
Pde1a |
IC50 |
'=' |
275000 |
nM |
| Q63421 |
BXGT016070 |
Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C |
reviewed |
- |
Pde1c |
IC50 |
'=' |
275000 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Ki |
'=' |
27000 |
nM |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Thermal melting change |
'=' |
2 |
degrees C |
| P16098 |
BXGT008191 |
Beta-amylase |
reviewed |
- |
BMY1 |
Activity |
- |
- |
- |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
IC50 |
'=' |
43 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
12589 |
nM |
| Q1CTD3 |
BXGT013756 |
D-alanine--D-alanine ligase |
reviewed |
- |
ddl |
Kd |
'=' |
12900 |
nM |
| Q9F4F7 |
BXGT020344 |
4'-phosphopantetheinyl transferase ffp |
reviewed |
- |
ffp |
Potency |
'=' |
89125 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
IC50 |
'=' |
64000 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
1000 |
nM |
| Q16637 |
BXGT013646 |
Survival motor neuron protein |
reviewed |
Epigenetic regulator |
SMN1 |
Potency |
'=' |
35481 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
'>' |
32000 |
nM |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
CC50 |
'=' |
45 |
ug.mL-1 |
| P79208 |
BXGT011858 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
PTGS2 |
Inhibition |
- |
- |
- |
| Q00532 |
BXGT012532 |
Cyclin-dependent kinase-like 1 |
reviewed |
Kinase |
CDKL1 |
Thermal melting change |
'=' |
1 |
degrees C |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Thermal melting change |
'=' |
4 |
degrees C |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Thermal melting change |
'=' |
8 |
degrees C |
| O95747 |
BXGT005393 |
Serine/threonine-protein kinase OSR1 |
reviewed |
Kinase |
OXSR1 |
Thermal melting change |
'=' |
7 |
degrees C |
| Q9BVS4 |
BXGT020147 |
Serine/threonine-protein kinase RIO2 |
reviewed |
Kinase |
RIOK2 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Thermal melting change |
'=' |
5 |
degrees C |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Thermal melting change |
'=' |
5 |
degrees C |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Thermal melting change |
'=' |
4 |
degrees C |
| P0C6X7 |
BXGT007440 |
Replicase polyprotein 1ab |
reviewed |
- |
rep |
IC50 |
'=' |
8100 |
nM |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
Inhibition |
- |
- |
- |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
37800 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
58400 |
nM |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
39810 |
nM |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
'=' |
5011 |
nM |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
'=' |
100000 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Inhibition |
'=' |
99 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
'=' |
19952 |
nM |
| P15428 |
BXGT008121 |
15-hydroxyprostaglandin dehydrogenase [NAD(+)] |
reviewed |
- |
HPGD |
Potency |
'=' |
19952 |
nM |
| Q63921 |
BXGT016082 |
Prostaglandin G/H synthase 1 |
reviewed |
- |
Ptgs1 |
IC50 |
'=' |
50000 |
nM |
| P35355 |
BXGT009817 |
Prostaglandin G/H synthase 2 |
reviewed |
- |
Ptgs2 |
IC50 |
'=' |
50000 |
nM |
| O89049 |
BXGT005293 |
Thioredoxin reductase 1, cytoplasmic |
reviewed |
- |
Txnrd1 |
Potency |
- |
23778 |
nM |
| P14635 |
BXGT008031 |
G2/mitotic-specific cyclin-B1 |
reviewed |
Enzyme modulator |
CCNB1 |
IC50 |
'>' |
20000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
IC50 |
'>' |
20000 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
ID50 |
'=' |
0 |
mM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Activity |
- |
- |
- |
| P22748 |
BXGT008802 |
Carbonic anhydrase 4 |
reviewed |
- |
CA4 |
Ki |
'=' |
7890 |
nM |
| P00918 |
BXGT005690 |
Carbonic anhydrase 2 |
reviewed |
- |
CA2 |
Ki |
'=' |
2540 |
nM |
| Q9Y253 |
BXGT022216 |
DNA polymerase eta |
reviewed |
- |
POLH |
Potency |
- |
794 |
nM |
| P30543 |
BXGT009437 |
Adenosine receptor A2a |
reviewed |
- |
Adora2a |
pKi(uM) |
'=' |
0 |
- |
| P25099 |
BXGT009016 |
Adenosine receptor A1 |
reviewed |
- |
Adora1 |
Ki |
'=' |
2470 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
KSV |
'=' |
1 |
10'5/M |
| P03956 |
BXGT006120 |
Interstitial collagenase |
reviewed |
Enzyme |
MMP1 |
IC50 |
- |
- |
- |
| P35030 |
BXGT009784 |
Trypsin-3 |
reviewed |
Enzyme |
PRSS3 |
Ki |
'=' |
13100 |
nM |
| P07478 |
BXGT006630 |
Trypsin-2 |
reviewed |
Enzyme |
PRSS2 |
Ki |
'=' |
13100 |
nM |
| P07477 |
BXGT006629 |
Trypsin-1 |
reviewed |
Enzyme |
PRSS1 |
Ki |
'=' |
13100 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
IC50 |
'=' |
40000 |
nM |
| Q16659 |
BXGT013652 |
Mitogen-activated protein kinase 6 |
reviewed |
Kinase |
MAPK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
23600 |
nM |
| P14679 |
BXGT008039 |
Tyrosinase |
reviewed |
Enzyme |
TYR |
Inhibition |
'=' |
40 |
% |
| Q965D5 |
BXGT019600 |
Enoyl-acyl-carrier protein reductase |
unreviewed |
- |
fabI |
Ki |
'=' |
1090 |
nM |
| P00811 |
BXGT005666 |
Beta-lactamase |
reviewed |
- |
ampC |
Change in IC50 |
'=' |
2 |
fold |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
Potency |
'=' |
19952 |
nM |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
Activity |
'=' |
30 |
% |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
28 |
% |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
- |
- |
- |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Ki |
'=' |
8100 |
nM |
| B4URF0 |
BXGT002146 |
Neuraminidase |
unreviewed |
- |
NA |
IC50 |
'=' |
67500 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Activity |
'=' |
60 |
% |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
122 |
% |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
Activity |
- |
- |
- |
| P15145 |
BXGT008088 |
Aminopeptidase N |
reviewed |
- |
ANPEP |
Inhibition |
'=' |
73 |
% |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Activity |
- |
- |
- |
| P00352 |
BXGT005510 |
Retinal dehydrogenase 1 |
reviewed |
Enzyme |
ALDH1A1 |
Potency |
'=' |
12589 |
nM |
| P32871 |
BXGT009672 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
- |
PIK3CA |
Inhibition |
'=' |
18 |
% |
| O14757 |
BXGT004092 |
Serine/threonine-protein kinase Chk1 |
reviewed |
Kinase |
CHEK1 |
Inhibition |
'=' |
56 |
% |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Inhibition |
'=' |
37 |
% |
| Q9NPH5 |
BXGT021159 |
NADPH oxidase 4 |
reviewed |
Enzyme |
NOX4 |
IC50 |
'=' |
680 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
IC50 |
'=' |
10200 |
nM |
| Q66HS9 |
BXGT016172 |
Monocarboxylate transporter 2 |
unreviewed |
- |
Slc16a7 |
Activity |
'=' |
17 |
% |
| P17538 |
BXGT008314 |
Chymotrypsinogen B |
reviewed |
Enzyme |
CTRB1 |
IC50 |
'=' |
100000 |
nM |
| P03126 |
BXGT006024 |
Protein E6 |
reviewed |
- |
E6 |
IC50 |
'>' |
20000 |
nM |
| Q1CTD3 |
BXGT013756 |
D-alanine--D-alanine ligase |
reviewed |
- |
ddl |
IC50 |
'=' |
48500 |
nM |
| P16116 |
BXGT008197 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
32870 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
FC |
'=' |
1 |
- |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
- |
- |
- |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Activity |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Activity |
- |
- |
- |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Activity |
- |
- |
- |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Activity |
- |
- |
- |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
IC50 |
'=' |
4230 |
nM |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
EC50 |
'=' |
1100 |
nM |
| P22303 |
BXGT008751 |
Acetylcholinesterase |
reviewed |
Enzyme |
ACHE |
IC50 |
'=' |
353860 |
nM |
| P04062 |
BXGT006140 |
Lysosomal acid glucosylceramidase |
reviewed |
- |
GBA |
Potency |
- |
28183 |
nM |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
IC50 |
'=' |
1200 |
nM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Vmax |
'=' |
0 |
uM |
| P03468 |
BXGT006079 |
Neuraminidase |
reviewed |
- |
NA |
logIC50 |
'=' |
1 |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
10000 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
10000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Inhibition |
- |
- |
- |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Potency |
'=' |
31622 |
nM |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Thermal melting change |
'=' |
3 |
degrees C |
| P06737 |
BXGT006492 |
Glycogen phosphorylase, liver form |
reviewed |
Enzyme |
PYGL |
IC50 |
'=' |
4800 |
nM |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
FC |
'=' |
4 |
- |
| P04637 |
BXGT006243 |
Cellular tumor antigen p53 |
reviewed |
Transcription factor |
TP53 |
Potency |
'=' |
1000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
FC |
'=' |
4 |
- |
| P03372 |
BXGT006059 |
Estrogen receptor |
reviewed |
Nuclear receptor |
ESR1 |
Activity |
'=' |
70 |
% |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
AC50 |
- |
- |
- |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
78 |
pm/min/mg |
| P49798 |
BXGT010745 |
Regulator of G-protein signaling 4 |
reviewed |
Enzyme modulator |
RGS4 |
Potency |
- |
11917 |
nM |
| O42275 |
BXGT004559 |
Acetylcholinesterase |
reviewed |
- |
ache |
IC50 |
- |
- |
- |
| P39748 |
BXGT010134 |
Flap endonuclease 1 |
reviewed |
Enzyme |
FEN1 |
Potency |
- |
39810 |
nM |
| P35030 |
BXGT009784 |
Trypsin-3 |
reviewed |
Enzyme |
PRSS3 |
IC50 |
'=' |
19000 |
nM |
| P07478 |
BXGT006630 |
Trypsin-2 |
reviewed |
Enzyme |
PRSS2 |
IC50 |
'=' |
19000 |
nM |
| P07477 |
BXGT006629 |
Trypsin-1 |
reviewed |
Enzyme |
PRSS1 |
IC50 |
'=' |
19000 |
nM |
| Q28731 |
BXGT013954 |
Thrombin |
unreviewed |
- |
thrombin |
APTT |
'=' |
30 |
s |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
Activity |
'=' |
268 |
% |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
18356 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
5400 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
14581 |
nM |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
IC50 |
'=' |
7589 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
7600 |
nM |
| P27986 |
BXGT009216 |
Phosphatidylinositol 3-kinase regulatory subunit alpha |
reviewed |
Kinase |
PIK3R1 |
IC50 |
'=' |
3800 |
nM |
| Q9WKE8 |
BXGT021921 |
Reverse transcriptase |
unreviewed |
- |
reverse |
IC50 |
'<' |
200 |
ug.mL-1 |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Activity |
'=' |
570 |
pm/min/mg |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
15848 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
15848 |
nM |
| P0DP23 |
BXGT007520 |
Calmodulin-1 |
reviewed |
- |
CALM1 |
IC50 |
'=' |
12970 |
nM |
| P22309 |
BXGT008753 |
UDP-glucuronosyltransferase 1-1 |
reviewed |
- |
UGT1A1 |
Drug metabolism |
- |
- |
- |
| P16473 |
BXGT008234 |
Thyrotropin receptor |
reviewed |
G-protein coupled receptor |
TSHR |
Potency |
'=' |
39810 |
nM |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
IC50 |
'=' |
13790 |
nM |
| Q96KQ7 |
BXGT019687 |
Histone-lysine N-methyltransferase EHMT2 |
reviewed |
Epigenetic regulator |
EHMT2 |
Potency |
- |
28183 |
nM |
| P53987 |
BXGT011023 |
Monocarboxylate transporter 1 |
reviewed |
- |
Slc16a1 |
Activity |
'=' |
11 |
% |
| O94782 |
BXGT005332 |
Ubiquitin carboxyl-terminal hydrolase 1 |
reviewed |
Enzyme |
USP1 |
Potency |
- |
56234 |
nM |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
IC50 |
'=' |
240000 |
nM |
| Q2M2H8 |
BXGT026100 |
Probable maltase-glucoamylase 2 |
reviewed |
Enzyme |
MGAM2 |
IC50 |
'=' |
7800 |
nM |
| P14410 |
BXGT008009 |
Sucrase-isomaltase, intestinal |
reviewed |
Enzyme |
SI |
IC50 |
'=' |
7800 |
nM |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
IC50 |
'=' |
7800 |
nM |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
IC50 |
'=' |
7800 |
nM |
| P27169 |
BXGT009161 |
Serum paraoxonase/arylesterase 1 |
reviewed |
- |
PON1 |
Ka |
'=' |
1 |
10'5/M |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
5011 |
nM |
| P21728 |
BXGT008686 |
D(1A) dopamine receptor |
reviewed |
G-protein coupled receptor |
DRD1 |
Potency |
- |
4109 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
7940 |
nM |
| Q2M2H8 |
BXGT026100 |
Probable maltase-glucoamylase 2 |
reviewed |
Enzyme |
MGAM2 |
Inhibition |
'=' |
83 |
% |
| P14410 |
BXGT008009 |
Sucrase-isomaltase, intestinal |
reviewed |
Enzyme |
SI |
Inhibition |
'=' |
83 |
% |
| P10253 |
BXGT007550 |
Lysosomal alpha-glucosidase |
reviewed |
Enzyme |
GAA |
Inhibition |
'=' |
83 |
% |
| O43451 |
BXGT004594 |
Maltase-glucoamylase, intestinal |
reviewed |
Enzyme |
MGAM |
Inhibition |
'=' |
83 |
% |
| P08254 |
BXGT006758 |
Stromelysin-1 |
reviewed |
Enzyme |
MMP3 |
IC50 |
'=' |
5570 |
nM |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
Inhibition |
'>' |
30 |
% |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Thermal melting change |
'=' |
2 |
degrees C |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Thermal melting change |
'=' |
4 |
degrees C |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Thermal melting change |
'=' |
6 |
degrees C |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Thermal melting change |
'=' |
5 |
degrees C |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Efficacy |
'=' |
40 |
picometer |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
K |
'=' |
496 |
10'6/min |
| P35503 |
BXGT009840 |
UDP-glucuronosyltransferase 1-3 |
reviewed |
- |
UGT1A3 |
Drug metabolism |
- |
- |
- |
| P29372 |
BXGT009336 |
DNA-3-methyladenine glycosylase |
reviewed |
Enzyme |
MPG |
Inhibition |
- |
- |
- |
| P13267 |
BXGT007895 |
DNA polymerase III PolC-type |
reviewed |
- |
polC |
Potency |
- |
10621 |
nM |
| Q9NPD5 |
BXGT021151 |
Solute carrier organic anion transporter family member 1B3 |
reviewed |
Transporter |
SLCO1B3 |
Inhibition |
'=' |
21 |
% |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
15200 |
nM |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
1122 |
nM |
| P33527 |
BXGT009728 |
Multidrug resistance-associated protein 1 |
reviewed |
Transporter |
ABCC1 |
FC |
'=' |
1 |
- |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
Inhibition |
- |
- |
- |
| P51679 |
BXGT010877 |
C-C chemokine receptor type 4 |
reviewed |
G-protein coupled receptor |
CCR4 |
IC50 |
'=' |
10200 |
nM |
| P33261 |
BXGT009707 |
Cytochrome P450 2C19 |
reviewed |
- |
CYP2C19 |
AC50 |
- |
- |
- |
| Q03164 |
BXGT012700 |
Histone-lysine N-methyltransferase 2A |
reviewed |
- |
KMT2A |
Potency |
'=' |
12589 |
nM |
| O00255 |
BXGT003903 |
Menin |
reviewed |
- |
MEN1 |
Potency |
'=' |
12589 |
nM |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
IC50 |
'=' |
3000 |
nM |
| P54132 |
BXGT011032 |
Bloom syndrome protein |
reviewed |
- |
BLM |
Potency |
'=' |
35481 |
nM |
| P58335 |
BXGT011233 |
Anthrax toxin receptor 2 |
reviewed |
Receptor |
ANTXR2 |
IC50 |
'>' |
300000 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
6 |
degrees C |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5804 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
25118 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Inhibition |
'=' |
4 |
% |
| P35354 |
BXGT009816 |
Prostaglandin G/H synthase 2 |
reviewed |
Enzyme |
PTGS2 |
IC50 |
'=' |
28600 |
nM |
| O94956 |
BXGT005343 |
Solute carrier organic anion transporter family member 2B1 |
reviewed |
Transporter |
SLCO2B1 |
Activity |
- |
- |
- |
| P08183 |
BXGT006741 |
ATP-dependent translocase ABCB1 |
reviewed |
Transporter |
ABCB1 |
IC50 |
'=' |
52500 |
nM |
| P45452 |
BXGT010462 |
Collagenase 3 |
reviewed |
Enzyme |
MMP13 |
IC50 |
'=' |
8460 |
nM |
| P08254 |
BXGT006758 |
Stromelysin-1 |
reviewed |
Enzyme |
MMP3 |
Inhibition |
'>' |
30 |
% |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
Inhibition |
'>' |
30 |
% |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
Ki |
'=' |
14000 |
nM |
| P35030 |
BXGT009784 |
Trypsin-3 |
reviewed |
Enzyme |
PRSS3 |
Inhibition |
'=' |
84 |
% |
| P07478 |
BXGT006630 |
Trypsin-2 |
reviewed |
Enzyme |
PRSS2 |
Inhibition |
'=' |
84 |
% |
| P07477 |
BXGT006629 |
Trypsin-1 |
reviewed |
Enzyme |
PRSS1 |
Inhibition |
'=' |
84 |
% |
| P04150 |
BXGT006154 |
Glucocorticoid receptor |
reviewed |
Nuclear receptor |
NR3C1 |
EC150 |
- |
- |
- |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
IC50 |
'=' |
1390 |
nM |
| P80276 |
BXGT011888 |
Aldo-keto reductase family 1 member B1 |
reviewed |
- |
AKR1B1 |
IC50 |
'=' |
50100 |
nM |
| P18054 |
BXGT008370 |
Arachidonate 12-lipoxygenase, 12S-type |
reviewed |
Enzyme |
ALOX12 |
Potency |
'=' |
1000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
EC50 |
'=' |
278 |
nM |
| P53051 |
BXGT010971 |
Oligo-1,6-glucosidase IMA1 |
reviewed |
- |
IMA1 |
IC50 |
'=' |
530000 |
nM |
| P06746 |
BXGT006496 |
DNA polymerase beta |
reviewed |
Enzyme |
POLB |
Potency |
'=' |
199 |
nM |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Thermal melting change |
'=' |
8 |
degrees C |
| P46063 |
BXGT010501 |
ATP-dependent DNA helicase Q1 |
reviewed |
Enzyme |
RECQL |
Potency |
'=' |
1778 |
nM |
| P14780 |
BXGT008053 |
Matrix metalloproteinase-9 |
reviewed |
Enzyme |
MMP9 |
IC50 |
'=' |
1610 |
nM |
| P51589 |
BXGT010867 |
Cytochrome P450 2J2 |
reviewed |
- |
CYP2J2 |
Activity |
'=' |
29 |
% |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
1550 |
nM |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
6500 |
nM |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
'=' |
36 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
'=' |
75 |
% |
| P48147 |
BXGT010620 |
Prolyl endopeptidase |
reviewed |
Enzyme |
PREP |
IC50 |
'=' |
13000 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
130000 |
nM |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
71 |
% |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
43 |
% |
| Q9NR56 |
BXGT021179 |
Muscleblind-like protein 1 |
reviewed |
Nucleic acid binding |
MBNL1 |
Potency |
- |
28183 |
nM |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
Inhibition |
'=' |
95 |
% |
| P29477 |
BXGT009355 |
Nitric oxide synthase, inducible |
reviewed |
- |
Nos2 |
IC50 |
'=' |
16400 |
nM |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
IC50 |
'=' |
1200 |
nM |
| Q60795 |
BXGT016000 |
Nuclear factor erythroid 2-related factor 2 |
reviewed |
- |
Nfe2l2 |
FC |
'=' |
1 |
- |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
2200 |
nM |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
IC50 |
'=' |
12000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
19952 |
nM |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
7000 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
'=' |
2110 |
nM |
| Q99986 |
BXGT019980 |
Serine/threonine-protein kinase VRK1 |
reviewed |
Kinase |
VRK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| P05177 |
BXGT006336 |
Cytochrome P450 1A2 |
reviewed |
Enzyme |
CYP1A2 |
IC50 |
'=' |
4097 |
nM |
| P37059 |
BXGT009957 |
Estradiol 17-beta-dehydrogenase 2 |
reviewed |
Enzyme |
HSD17B2 |
Activity |
'=' |
6 |
% |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Emax |
'=' |
177 |
% |
| Q14576 |
BXGT013487 |
ELAV-like protein 3 |
reviewed |
- |
ELAVL3 |
IC50 |
'=' |
1800 |
nM |
| P12530 |
BXGT007827 |
Arachidonate 15-lipoxygenase |
reviewed |
- |
ALOX15 |
IC50 |
'=' |
37000 |
nM |
| P34913 |
BXGT009770 |
Bifunctional epoxide hydrolase 2 |
reviewed |
Enzyme |
EPHX2 |
Inhibition |
'>' |
40 |
% |
| P11511 |
BXGT007717 |
Aromatase |
reviewed |
Enzyme |
CYP19A1 |
Activity |
'=' |
96 |
% |
| Q09013 |
BXGT013023 |
Myotonin-protein kinase |
reviewed |
Kinase |
DMPK |
Thermal melting change |
'=' |
3 |
degrees C |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
4 |
degrees C |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q86Y07 |
BXGT017631 |
Serine/threonine-protein kinase VRK2 |
reviewed |
Kinase |
VRK2 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
'=' |
37 |
% |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
Ratio |
'=' |
2 |
- |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'=' |
120 |
nM |
| Q15717 |
BXGT013589 |
ELAV-like protein 1 |
reviewed |
- |
ELAVL1 |
IC50 |
'=' |
1400 |
nM |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
2850 |
nM |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Inhibition |
'=' |
103 |
% |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Inhibition |
'=' |
113 |
% |
| P15121 |
BXGT008083 |
Aldo-keto reductase family 1 member B1 |
reviewed |
Enzyme |
AKR1B1 |
IC50 |
'=' |
2900 |
nM |
| Q9UBT6 |
BXGT021664 |
DNA polymerase kappa |
reviewed |
- |
POLK |
Potency |
- |
946 |
nM |
| O96394 |
BXGT005423 |
Arginase |
unreviewed |
- |
|
IC50 |
'=' |
4000 |
nM |
| P51589 |
BXGT010867 |
Cytochrome P450 2J2 |
reviewed |
- |
CYP2J2 |
Activity |
'=' |
44 |
% |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
10820 |
nM |
| P11712 |
BXGT007738 |
Cytochrome P450 2C9 |
reviewed |
- |
CYP2C9 |
AC50 |
- |
- |
- |
| O75604 |
BXGT005139 |
Ubiquitin carboxyl-terminal hydrolase 2 |
reviewed |
Enzyme |
USP2 |
Potency |
'=' |
31622 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
IC50 |
'=' |
1500 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
40 |
% |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Inhibition |
'=' |
70 |
% |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Inhibition |
'=' |
150 |
% |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
1258 |
nM |
| Q04760 |
BXGT012782 |
Lactoylglutathione lyase |
reviewed |
- |
GLO1 |
Ki |
'=' |
6 |
nM |
| P10632 |
BXGT007592 |
Cytochrome P450 2C8 |
reviewed |
- |
CYP2C8 |
IC50 |
'=' |
3500 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
72 |
% |
| P21397 |
BXGT008644 |
Amine oxidase [flavin-containing] A |
reviewed |
- |
MAOA |
IC50 |
'=' |
2440 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Km |
'=' |
106000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Km |
'=' |
25000 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat/Km |
'=' |
1 |
/uM/s |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
Kcat/Km |
'=' |
0 |
/uM/s |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
Ki |
'=' |
280 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Thermal melting change |
'=' |
5 |
degrees C |
| P16050 |
BXGT008184 |
Arachidonate 15-lipoxygenase |
reviewed |
Enzyme |
ALOX15 |
Activity |
- |
- |
- |
| O15439 |
BXGT004169 |
Multidrug resistance-associated protein 4 |
reviewed |
Transporter |
ABCC4 |
IC50 |
'=' |
20800 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
1412 |
nM |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Thermal melting change |
'=' |
2 |
degrees C |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
IC50 |
'=' |
20000 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
Kd |
'=' |
38 |
nM |
| P00734 |
BXGT005630 |
Prothrombin |
reviewed |
Enzyme |
F2 |
RU |
'=' |
1882 |
- |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
IC50 |
'>' |
50000 |
nM |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Thermal melting change |
'=' |
2 |
degrees C |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Vmax |
'=' |
0 |
uM |
| P08170 |
BXGT006736 |
Seed linoleate 13S-lipoxygenase-1 |
reviewed |
- |
LOX1.1 |
Km |
'=' |
129200 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
8 |
degrees C |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
Inhibition |
- |
- |
- |
| Q96KB5 |
BXGT019685 |
Lymphokine-activated killer T-cell-originated protein kinase |
reviewed |
Kinase |
PBK |
Thermal melting change |
'=' |
0 |
degrees C |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'=' |
61 |
% |
| P00747 |
BXGT005639 |
Plasminogen |
reviewed |
Enzyme |
PLG |
Inhibition |
'=' |
30 |
% |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Vmax |
'=' |
194 |
% |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Thermal melting change |
'=' |
8 |
degrees C |
| P06276 |
BXGT006430 |
Cholinesterase |
reviewed |
- |
BCHE |
IC50 |
- |
- |
- |
| O42713 |
BXGT004563 |
Polyphenol oxidase 2 |
reviewed |
- |
PPO2 |
Inhibition |
'=' |
45 |
% |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
IC50 |
'=' |
133000 |
nM |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Thermal melting change |
'=' |
2 |
degrees C |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'=' |
133000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Vmax |
'=' |
177 |
% |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
32730 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Tlag |
'=' |
82 |
min |
| Q7ZJM1 |
BXGT017268 |
Integrase |
unreviewed |
- |
pol |
IC50 |
'=' |
600 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
IC50 |
'>' |
20000 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
'=' |
18 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
14900 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
Thermal melting change |
'=' |
1 |
degrees C |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Thermal melting change |
'=' |
8 |
degrees C |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Thermal melting change |
'=' |
7 |
degrees C |
| P00591 |
BXGT005592 |
Pancreatic triacylglycerol lipase |
reviewed |
- |
PNLIP |
IC50 |
'>' |
70000 |
nM |
| P27695 |
BXGT009199 |
DNA-(apurinic or apyrimidinic site) lyase |
reviewed |
- |
APEX1 |
Potency |
- |
707 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
IC50 |
'=' |
124600 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'=' |
5600 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'=' |
5600 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'=' |
5600 |
nM |
| P34913 |
BXGT009770 |
Bifunctional epoxide hydrolase 2 |
reviewed |
Enzyme |
EPHX2 |
IC50 |
'=' |
33540 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'=' |
1660 |
nM |
| P08253 |
BXGT006757 |
72 kDa type IV collagenase |
reviewed |
Enzyme |
MMP2 |
IC50 |
'=' |
6680 |
nM |
| Q9HC97 |
BXGT020527 |
G-protein coupled receptor 35 |
reviewed |
G-protein coupled receptor |
GPR35 |
EC50 |
'=' |
8020 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Activity |
- |
- |
- |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Potency |
- |
15410 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
T1/2 |
'=' |
4 |
hr |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
79 |
% |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
IC50 |
'=' |
3100 |
nM |
| P10635 |
BXGT007595 |
Cytochrome P450 2D6 |
reviewed |
- |
CYP2D6 |
IC50 |
'>' |
20000 |
nM |
| P09917 |
BXGT006941 |
Arachidonate 5-lipoxygenase |
reviewed |
Enzyme |
ALOX5 |
IC50 |
'=' |
4000 |
nM |
| Q9UM73 |
BXGT021773 |
ALK tyrosine kinase receptor |
reviewed |
Kinase |
ALK |
IC50 |
'=' |
3320 |
nM |
| P00749 |
BXGT005641 |
Urokinase-type plasminogen activator |
reviewed |
Enzyme |
PLAU |
IC50 |
'=' |
12100 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Thermal melting change |
'=' |
4 |
degrees C |
| O15438 |
BXGT004168 |
Canalicular multispecific organic anion transporter 2 |
reviewed |
Transporter |
ABCC3 |
IC50 |
'=' |
133000 |
nM |
| O60218 |
BXGT004858 |
Aldo-keto reductase family 1 member B10 |
reviewed |
Enzyme |
AKR1B10 |
Inhibition |
'=' |
23 |
% |
| P25024 |
BXGT009005 |
C-X-C chemokine receptor type 1 |
reviewed |
G-protein coupled receptor |
CXCR1 |
IC50 |
'>' |
100000 |
nM |
| P30518 |
BXGT009428 |
Vasopressin V2 receptor |
reviewed |
G-protein coupled receptor |
AVPR2 |
IC50 |
'=' |
6309 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
EC50 |
'=' |
35000 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
IC50 |
'<' |
1000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
IC50 |
'<' |
1000 |
nM |
| P67870 |
BXGT011566 |
Casein kinase II subunit beta |
reviewed |
Kinase |
CSNK2B |
IC50 |
'<' |
1000 |
nM |
| P05164 |
BXGT006333 |
Myeloperoxidase |
reviewed |
Enzyme |
MPO |
Activity |
'=' |
78 |
% |
| P80025 |
BXGT011867 |
Lactoperoxidase |
reviewed |
- |
LPO |
IC50 |
'=' |
6100 |
nM |
| P27487 |
BXGT009187 |
Dipeptidyl peptidase 4 |
reviewed |
Enzyme |
DPP4 |
IC50 |
'=' |
2920 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
TIME |
'=' |
8 |
hr |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
Ki |
'=' |
11900 |
nM |
| Q15118 |
BXGT013540 |
[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial |
reviewed |
Kinase |
PDK1 |
Inhibition |
- |
- |
- |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'=' |
9900 |
nM |
| P47989 |
BXGT010602 |
Xanthine dehydrogenase/oxidase |
reviewed |
Enzyme |
XDH |
IC50 |
'=' |
3500 |
nM |
| P08246 |
BXGT006756 |
Neutrophil elastase |
reviewed |
Enzyme |
ELANE |
IC50 |
'=' |
14300 |
nM |
| Q28731 |
BXGT013954 |
Thrombin |
unreviewed |
- |
thrombin |
PT |
'=' |
6 |
s |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
IC50 |
'=' |
8900 |
nM |
| P80457 |
BXGT011911 |
Xanthine dehydrogenase/oxidase |
reviewed |
- |
XDH |
IC50 |
'=' |
31900 |
nM |
| P27338 |
BXGT009172 |
Amine oxidase [flavin-containing] B |
reviewed |
- |
MAOB |
IC50 |
'=' |
38660 |
nM |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Inhibition |
'=' |
88 |
% |
| P05067 |
BXGT006306 |
Amyloid-beta precursor protein |
reviewed |
Enzyme modulator |
APP |
Ke(app) |
'=' |
6829 |
/M/min |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
Inhibition |
'=' |
67 |
% |
| Q16678 |
BXGT013656 |
Cytochrome P450 1B1 |
reviewed |
Enzyme |
CYP1B1 |
IC50 |
'=' |
1000 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
EC50 |
'=' |
8800 |
nM |
| Q00613 |
BXGT012540 |
Heat shock factor protein 1 |
reviewed |
Transcription factor |
HSF1 |
Activity |
'>' |
90 |
% |
| P07949 |
BXGT006703 |
Proto-oncogene tyrosine-protein kinase receptor Ret |
reviewed |
Kinase |
RET |
IC50 |
'=' |
78100 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
EC50 |
'=' |
30 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
IC50 |
'>' |
20000 |
nM |
| P04798 |
BXGT006265 |
Cytochrome P450 1A1 |
reviewed |
Enzyme |
CYP1A1 |
Inhibition |
'=' |
31 |
% |