Showing entry for Sb-202190


　 　 　 　 　 　 　 　 　 　 　 　 　 　 　
General Compound Information
BXGC IdBXGC0045254
Compound NameSb-202190
Structure
FormulaC20H14FN3O
InchiKeyQHKYPYXTTXKZST-UHFFFAOYSA-N
SMILESOc1ccc(cc1)c1nc(c([nH]1)c1ccc(cc1)F)c1ccncc1
InchiInChI=1S/C20H14FN3O/c21-16-5-1-13(2-6-16)18-19(14-9-11-22-12-10-14)24-20(23-18)15-3-7-17(25)8-4-15/h1-12,25H,(H,23,24)
IUPAC
Molecular Weight331.11
Pubchem Id5169
Chembl IdCHEMBL278041
Targets of Information Source
DrugBank n.a
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
PDB 2RE
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
O60885 BXGT004906 Bromodomain-containing protein 4 reviewed BRD4 Epigenetic regulator - 2500 - -
Binding DB 13531
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 30 - -
reviewed BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 - - 1100000 -
reviewed BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 - - 2200000 -
reviewed BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK - - 3100000 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - 210000 -
reviewed BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA - - 1700000 -
reviewed BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK - - 3200000 -
reviewed BXGT021250 Serine/threonine-protein kinase 32B reviewed Kinase STK32B - - 4900000 -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - 4800000 -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - 620000 -
reviewed BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT - - 510000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 2600000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1900000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 2000000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1400000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1100000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 2300000 -
reviewed BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 - - 6800000 -
reviewed BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 - - 1900000 -
reviewed BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D - - 59000 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 170000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 210000 -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 53000 -
reviewed BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 - - 2400000 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 42000 -
reviewed BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK - - 28000 -
reviewed BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB - - 530000 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 150000 -
reviewed BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 270000 - - -
reviewed BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 - - 790000 -
reviewed BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK - - 1600000 -
reviewed BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK - - 4500000 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - - 9800 -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - - 32000 -
reviewed BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 - - 3300000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1700000 -
reviewed BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 - - 4900000 -
reviewed BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 - - 9600000 -
reviewed BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG - - 640000 -
reviewed BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB - - 4200000 -
reviewed BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B - - 2700000 -
reviewed BXGT019637 Atypical kinase COQ8B, mitochondrial reviewed Kinase COQ8B - - 4900000 -
reviewed BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 170000 - - -
reviewed BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B - - 950000 -
reviewed BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B - - 4800000 -
reviewed BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK - - >1 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - >1 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - >1 -
reviewed BXGT019667 Aurora kinase B reviewed Kinase AURKB - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 91 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 26 -
reviewed BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 - - >1 -
reviewed BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 - - >1 -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - 62 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - >1 -
reviewed BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 19 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 14 -
reviewed BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 - - >1 -
reviewed BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 23 -
reviewed BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 - - >1 -
reviewed BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET - - >1 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - >1 -
reviewed BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 - - >1 -
reviewed BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA - - >1 -
reviewed BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 21 -
reviewed BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 - - 27 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 17 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 11 -
reviewed BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 - - >1 -
reviewed BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 - - >1 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 8.7 - -
reviewed BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D - 188 - -
reviewed BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 - >100000 - -
reviewed BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 - >100000 - -
reviewed BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 - >100000 - -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 9 - -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - - 120 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 4600 -
reviewed BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 - - 3100 -
reviewed BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK - - 6000 -
reviewed BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 - - 3800 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - - 13 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 400 -
reviewed BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 - - 3000 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - 120 -
reviewed BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 - - 9400 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 51 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 350 -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 650 -
reviewed BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK - - 10000 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 50 - -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 28 - -
reviewed BXGT015228 Bromodomain testis-specific protein reviewed Epigenetic regulator BRDT - 20000 - -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - 9.8 - -
reviewed BXGT004906 Bromodomain-containing protein 4 reviewed Epigenetic regulator BRD4 - 2500 - -
reviewed BXGT004906 Bromodomain-containing protein 4 reviewed Epigenetic regulator BRD4 - - 3400 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 80 - -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - 100 - -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 14 - -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - 300 - -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - 4800 -
reviewed BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 - - >10000 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - >10000 -
reviewed BXGT020119 Serine/threonine-protein kinase RIO1 reviewed Kinase RIOK1 - - >10000 -
reviewed BXGT021743 Serine/threonine-protein kinase tousled-like 1 reviewed Kinase TLK1 - - >10000 -
reviewed BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B - - >10000 -
reviewed BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 - - >10000 -
reviewed BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 - - >10000 -
reviewed BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 - - 6800 -
reviewed BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 - - 1900 -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 53 -
reviewed BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 - - >10000 -
reviewed BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D - - 59 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 170 -
reviewed BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK - - 1600 -
reviewed BXGT012536 Cyclin-dependent kinase 17 reviewed Kinase CDK17 - - >10000 -
reviewed BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 - - >10000 -
reviewed BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG - - 640 -
reviewed BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER - - >10000 -
reviewed BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 - - >10000 -
reviewed BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK - - >10000 -
reviewed BXGT018526 Casein kinase I isoform alpha-like reviewed Kinase CSNK1A1L - - 1900 -
reviewed BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 - - >10000 -
reviewed BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 - - 3300 -
reviewed BXGT013331 cGMP-dependent protein kinase 2 reviewed Kinase PRKG2 - - >10000 -
reviewed BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK - - >10000 -
reviewed BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 - - >10000 -
reviewed BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 - - >10000 -
reviewed BXGT005341 Cyclin-dependent kinase 14 reviewed Kinase CDK14 - - >10000 -
reviewed BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 - - >10000 -
reviewed BXGT013322 Mitogen-activated protein kinase 7 reviewed Kinase MAPK7 - - >10000 -
reviewed BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 - - >10000 -
reviewed BXGT008492 Interferon-induced, double-stranded RNA-activated protein kinase reviewed Kinase EIF2AK2 - - >10000 -
reviewed BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 - - >10000 -
reviewed BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 - - >10000 -
reviewed BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD - - >10000 -
reviewed BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 - - >10000 -
reviewed BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 - - >10000 -
reviewed BXGT018572 Atypical kinase COQ8A, mitochondrial reviewed Kinase COQ8A - - >10000 -
reviewed BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 - - >10000 -
reviewed BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE - - >10000 -
reviewed BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 - - >10000 -
reviewed BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK - - >10000 -
reviewed BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 - - >10000 -
reviewed BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R - - >10000 -
reviewed BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 - - >10000 -
reviewed BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A - - >10000 -
reviewed BXGT017617 Serine/threonine-protein kinase pim-3 reviewed PIM3 - - >10000 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 42 -
reviewed BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 - - >10000 -
reviewed BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 - - 1100 -
reviewed BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 - - 1600 -
reviewed BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 - - >10000 -
reviewed BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A - - >10000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 2000 -
reviewed BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 - - >10000 -
reviewed BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT - - 510 -
reviewed BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D - - >10000 -
reviewed BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ - - >10000 -
reviewed BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK - - >10000 -
reviewed BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN - - >10000 -
reviewed BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 - - >10000 -
reviewed BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 - - >10000 -
reviewed BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 - - >10000 -
reviewed BXGT020156 Cyclin-dependent kinase 19 reviewed Kinase CDK19 - - >10000 -
reviewed BXGT004117 Aurora kinase A reviewed Kinase AURKA - - >10000 -
reviewed BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 - - >10000 -
reviewed BXGT007749 Myosin light chain kinase, smooth muscle reviewed Mylk - - >10000 -
reviewed BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 - - >10000 -
reviewed BXGT009511 Mitogen-activated protein kinase 4 reviewed Kinase MAPK4 - - >10000 -
reviewed BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 - - >10000 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - >10000 -
reviewed BXGT004124 Serine/threonine-protein kinase DCLK1 reviewed Kinase DCLK1 - - >10000 -
reviewed BXGT019958 Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha reviewed Kinase PIP5K1A - - >10000 -
reviewed BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 - - >10000 -
reviewed BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES - - >10000 -
reviewed BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 - - >10000 -
reviewed BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 - - >10000 -
reviewed BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 - - >10000 -
reviewed BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L - - >10000 -
reviewed BXGT017636 Myosin light chain kinase family member 4 reviewed MYLK4 - - >10000 -
reviewed BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 - - >10000 -
reviewed BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 - - >10000 -
reviewed BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 - - >10000 -
reviewed BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 - - >10000 -
reviewed BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 - - >10000 -
reviewed BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET - - >10000 -
reviewed BXGT008623 Cyclin-dependent kinase 11B reviewed Kinase CDK11B - - >10000 -
reviewed BXGT020468 Tyrosine-protein kinase Srms reviewed Kinase SRMS - - >10000 -
reviewed BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 - - 790 -
reviewed BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK - - >10000 -
reviewed BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 - - >10000 -
reviewed BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 - - >10000 -
reviewed BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 - - >10000 -
reviewed BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R - - >10000 -
reviewed BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 - - >10000 -
reviewed BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 - - >10000 -
reviewed BXGT005400 Serine/threonine-protein kinase LATS1 reviewed Kinase LATS1 - - >10000 -
reviewed BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 - - 2400 -
reviewed BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 - - >10000 -
reviewed BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G - - >10000 -
reviewed BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 - - >10000 -
reviewed BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 - - >10000 -
reviewed BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA - - >10000 -
reviewed BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB - - >10000 -
reviewed BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 - - >10000 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - 210 -
reviewed BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 - - >10000 -
reviewed BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK - - >10000 -
reviewed BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 - - >10000 -
reviewed BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 - - >10000 -
reviewed BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 - - >10000 -
reviewed BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 - - >10000 -
reviewed BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK - - >10000 -
reviewed BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 - - >10000 -
reviewed BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA - - >10000 -
reviewed BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 - - >10000 -
reviewed BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 - - >10000 -
reviewed BXGT018558 Myosin-IIIa reviewed Kinase MYO3A - - >10000 -
reviewed BXGT019015 Myosin-IIIb reviewed Kinase MYO3B - - >10000 -
reviewed BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR - - >10000 -
reviewed BXGT006425 Insulin receptor reviewed Kinase INSR - - >10000 -
reviewed BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B - - 4800 -
reviewed BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA - - 1700 -
reviewed BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 - - >10000 -
reviewed BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 - - >10000 -
reviewed BXGT013642 Mitogen-activated protein kinase kinase kinase 11 reviewed Kinase MAP3K11 - - >10000 -
reviewed BXGT011009 LIM domain kinase 2 reviewed Kinase LIMK2 - - >10000 -
reviewed BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA - - >10000 -
reviewed BXGT019712 Serine/threonine-protein kinase Nek1 reviewed Kinase NEK1 - - >10000 -
reviewed BXGT017614 Serine/threonine-protein kinase 32C reviewed Kinase STK32C - - >10000 -
reviewed BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE - - >10000 -
reviewed BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 - - >10000 -
reviewed BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK - - >10000 -
reviewed BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 - - >10000 -
reviewed BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 - - >10000 -
reviewed BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 - - >10000 -
reviewed BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 - - >10000 -
reviewed BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 - - >10000 -
reviewed BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 - - >10000 -
reviewed BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL - - >10000 -
reviewed BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K - - >10000 -
reviewed BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 - - >10000 -
reviewed BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 - - >10000 -
reviewed BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B - - 950 -
reviewed BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 - - >10000 -
reviewed BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 - - >10000 -
reviewed BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK - - 4500 -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - - >10000 -
reviewed BXGT009417 Wee1-like protein kinase reviewed Kinase WEE1 - - >10000 -
reviewed BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 - - >10000 -
reviewed BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK - - >10000 -
reviewed BXGT009939 Bone morphogenetic protein receptor type-1A reviewed Kinase BMPR1A - - >10000 -
reviewed BXGT013398 Bone morphogenetic protein receptor type-2 reviewed Kinase BMPR2 - - >10000 -
reviewed BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A - - >10000 -
reviewed BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B - - 2700 -
reviewed BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 - - >10000 -
reviewed BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 - - >10000 -
reviewed BXGT013372 Receptor-interacting serine/threonine-protein kinase 1 reviewed Kinase RIPK1 - - >10000 -
reviewed BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR - - >10000 -
reviewed BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 - - 170 -
reviewed BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 - - >10000 -
reviewed BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK - - >10000 -
reviewed BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 - - >10000 -
reviewed BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 - - >10000 -
reviewed BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 - - >10000 -
reviewed BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed PAK6 - - >10000 -
reviewed BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 - - >10000 -
reviewed BXGT010496 Dual specificity mitogen-activated protein kinase kinase 4 reviewed Kinase MAP2K4 - - >10000 -
reviewed BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 - - >10000 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 150 -
reviewed BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 - - >10000 -
reviewed BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 - - >10000 -
reviewed BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB - - 4200 -
reviewed BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 - - >10000 -
reviewed BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 - - >10000 -
reviewed BXGT011210 Serine/threonine-protein kinase SIK1 reviewed SIK1 - - >10000 -
reviewed BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC - - >10000 -
reviewed BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 - - >10000 -
reviewed BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 - - >10000 -
reviewed BXGT009153 Activin receptor type-2A reviewed Kinase ACVR2A - - >10000 -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - - 32 -
reviewed BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 - - >10000 -
reviewed BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 - - >10000 -
reviewed BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B - - >10000 -
reviewed BXGT011837 Phosphatidylinositol 5-phosphate 4-kinase type-2 beta reviewed Kinase PIP4K2B - - >10000 -
reviewed BXGT019637 Atypical kinase COQ8B, mitochondrial reviewed Kinase COQ8B - - 4900 -
reviewed BXGT021810 Aurora kinase C reviewed Kinase AURKC - - >10000 -
reviewed BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC - - >10000 -
reviewed BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 - - >10000 -
reviewed BXGT004085 Serine/threonine-protein kinase RIO3 reviewed Kinase RIOK3 - - >10000 -
reviewed BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 - - >10000 -
reviewed BXGT009953 Serine/threonine-protein kinase receptor R3 reviewed Kinase ACVRL1 - - >10000 -
reviewed BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 - - >10000 -
reviewed BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX - - >10000 -
reviewed BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B - - >10000 -
reviewed BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 - - >10000 -
reviewed BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D - - >10000 -
reviewed BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G - - >10000 -
reviewed BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK - - >10000 -
reviewed BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 - - >10000 -
reviewed BXGT019394 Mitogen-activated protein kinase kinase kinase kinase 1 reviewed Kinase MAP4K1 - - >10000 -
reviewed BXGT018345 Mitogen-activated protein kinase kinase kinase kinase 3 reviewed Kinase MAP4K3 - - >10000 -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - - >10000 -
reviewed BXGT011596 Tubulin alpha-1A chain reviewed Tuba1a - - 4900 -
reviewed BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX - - >10000 -
reviewed BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 - - >10000 -
reviewed BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK - - >10000 -
reviewed BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 - - >10000 -
reviewed BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 - - >10000 -
reviewed BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B - - >10000 -
reviewed BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK - - 3200 -
reviewed BXGT016447 Serine/threonine-protein kinase Nek5 reviewed NEK5 - - >10000 -
reviewed BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 - - >10000 -
reviewed BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 - - >10000 -
reviewed BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 - - >10000 -
reviewed BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 - - >10000 -
reviewed BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 - - >10000 -
reviewed BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 - - >10000 -
reviewed BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK - - 28 -
reviewed BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 - - >10000 -
reviewed BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 - - >10000 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - - 9.8 -
reviewed BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 - - >10000 -
reviewed BXGT021302 eIF-2-alpha kinase GCN2 reviewed EIF2AK4 - - >10000 -
reviewed BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 - - >10000 -
reviewed BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 - - 9600 -
reviewed BXGT010537 Dual specificity mitogen-activated protein kinase kinase 3 reviewed Kinase MAP2K3 - - >10000 -
reviewed BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 - - >10000 -
reviewed BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 - - >10000 -
reviewed BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET - - >10000 -
reviewed BXGT021190 Serine/threonine-protein kinase LATS2 reviewed Kinase LATS2 - - 1700 -
reviewed BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - >10000 -
reviewed BXGT021808 Cyclin-dependent kinase 11A reviewed CDK11A - - >10000 -
reviewed BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 - - >10000 -
reviewed BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK - - 3100 -
reviewed BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 - - >10000 -
reviewed BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 - - >10000 -
reviewed BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B - - >10000 -
reviewed BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 - - >10000 -
reviewed BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 - - >10000 -
reviewed BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 - - 2200 -
reviewed BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - >10000 -
reviewed BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 - - >10000 -
reviewed BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 - - >10000 -
reviewed BXGT021250 Serine/threonine-protein kinase 32B reviewed Kinase STK32B - - 4900 -
reviewed BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN - - >10000 -
reviewed BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 - - >10000 -
reviewed BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 - - >10000 -
reviewed BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 - - >10000 -
reviewed BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 - - >10000 -
reviewed BXGT009854 Tyrosine-protein kinase receptor Tie-1 reviewed Kinase TIE1 - - >10000 -
reviewed BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 - - >10000 -
reviewed BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 - - >10000 -
reviewed BXGT020511 Dual specificity protein kinase CLK4 reviewed CLK4 - - >10000 -
reviewed BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 - - >10000 -
reviewed BXGT013359 Non-receptor tyrosine-protein kinase TNK1 reviewed Kinase TNK1 - - >10000 -
reviewed BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK - - >10000 -
reviewed BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB - - 530 -
reviewed BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK - - >10000 -
reviewed BXGT013580 Dual specificity testis-specific protein kinase 1 reviewed Kinase TESK1 - - >10000 -
reviewed BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 - - >10000 -
reviewed BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 - - >10000 -
reviewed BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 - - >10000 -
reviewed BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 - - >10000 -
reviewed BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 - - >10000 -
reviewed BXGT009970 TGF-beta receptor type-2 reviewed Kinase TGFBR2 - - >10000 -
reviewed BXGT013631 Serine/threonine-protein kinase N1 reviewed Kinase PKN1 - - >10000 -
reviewed BXGT018559 Ankyrin repeat and protein kinase domain-containing protein 1 reviewed Kinase ANKK1 - - >10000 -
reviewed BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 - - >10000 -
reviewed BXGT015278 Serine/threonine-protein kinase TNNI3K reviewed TNNI3K - - >10000 -
reviewed BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 - - >10000 -
reviewed BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 - - >10000 -
reviewed BXGT006941 Arachidonate 5-lipoxygenase reviewed Enzyme ALOX5 - 50 - -
reviewed BXGT010592 Glucagon receptor reviewed G-protein coupled receptor GCGR - 80 - -
CHEMBL CHEMBL278041
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Kd - - -
Q16816 BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 Kd - - -
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Kd - - -
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 8 nM
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Residual Activity '=' 55 %
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Residual Activity '=' 81 %
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Residual Activity '=' 88 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Residual Activity '=' 113 %
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Residual Activity '=' 101 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Inhibition '=' 93 %
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Inhibition '=' 93 %
P67870 BXGT011566 Casein kinase II subunit beta reviewed Kinase CSNK2B Inhibition '=' 93 %
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 Potency '=' 5011 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Ki '>' 3981 nM
Q16236 BXGT013624 Nuclear factor erythroid 2-related factor 2 reviewed Enzyme NFE2L2 Potency - 6513 nM
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Ki '>' 1995 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Kd '=' 9 nM
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Kd '>' 10000 nM
P05177 BXGT006336 Cytochrome P450 1A2 reviewed Enzyme CYP1A2 AC50 '=' 15848 nM
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Kd '=' 4200 nM
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Kd '>' 10000 nM
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Kd '>' 10000 nM
P40225 BXGT010168 Thrombopoietin reviewed - THPO Potency '=' 31622 nM
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Ki '>' 3981 nM
Q9UIF8 BXGT021718 Bromodomain adjacent to zinc finger domain protein 2B reviewed - BAZ2B Potency - 79432 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Ki '>' 3981 nM
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 105 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 105 %
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Residual Activity '=' 104 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Residual Activity '=' 103 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Residual Activity '=' 101 %
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Residual Activity '=' 103 %
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd - - -
P48729 BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 Ki '=' 1000 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Kd '=' 350 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Ki '>' 2511 nM
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Residual Activity '=' 94 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Residual Activity '=' 96 %
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Residual Activity '=' 117 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Residual Activity '=' 111 %
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Residual Activity '=' 97 %
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Residual Activity '=' 20 %
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Residual Activity '=' 10 %
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Residual Activity '=' 105 %
P47871 BXGT010592 Glucagon receptor reviewed G-protein coupled receptor GCGR Inhibition '<' 20 %
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Kd - - -
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Kd - - -
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Residual Activity '=' 87 %
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Residual Activity '=' 105 %
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Residual Activity '=' 25 %
O43318 BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 Residual Activity '=' 101 %
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Residual Activity '=' 110 %
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Residual Activity '=' 102 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 81 %
Q9UF33 BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 Kd '=' 2200 nM
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '>' 10000 nM
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Kd '>' 10000 nM
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Kd '>' 10000 nM
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Activity '=' 84 %
P78396 BXGT011842 Cyclin-A1 reviewed Enzyme modulator CCNA1 Activity '=' 82 %
P20248 BXGT008554 Cyclin-A2 reviewed Enzyme modulator CCNA2 Activity '=' 82 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Activity '=' 82 %
Q9BUB5 BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 Kd '>' 10000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd '>' 10000 nM
Q9Y6R4 BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 Kd '>' 10000 nM
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Kd '>' 10000 nM
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Kd '>' 10000 nM
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Activity '=' 85 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Activity '=' 89 %
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Kd '>' 10000 nM
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Kd '>' 10000 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd '>' 10000 nM
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Activity '=' 65 %
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Kd '>' 10000 nM
Q8WTQ7 BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 Residual Activity '=' 121 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Potency '=' 39810 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 14125 nM
Q92918 BXGT019394 Mitogen-activated protein kinase kinase kinase kinase 1 reviewed Kinase MAP4K1 Kd '>' 10000 nM
O00506 BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1700 nM
Q9H1R3 BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 Kd '>' 10000 nM
Q9BUB5 BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 Activity '=' 87 %
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Kd '>' 10000 nM
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Kd '>' 10000 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Kd '>' 10000 nM
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Residual Activity '=' 77 %
Q13153 BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 Kd '>' 10000 nM
Q96D53 BXGT019637 Atypical kinase COQ8B, mitochondrial reviewed Kinase COQ8B Kd '=' 4900 nM
Q9H093 BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 Kd '>' 10000 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Kd '>' 10000 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Potency '=' 1000 nM
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Kd '=' 170 nM
O14730 BXGT004085 Serine/threonine-protein kinase RIO3 reviewed Kinase RIOK3 Kd '>' 10000 nM
Q13705 BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B Kd '=' 4800 nM
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Kd '>' 10000 nM
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Kd '>' 10000 nM
P22694 BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB Kd '=' 530 nM
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Kd '>' 10000 nM
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Residual Activity '=' 90 %
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Residual Activity '=' 69 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 61 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1100 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Kd '>' 10000 nM
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Kd '>' 10000 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Inhibition - - -
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 Potency '=' 7943 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Residual Activity '=' 99 %
Q8NG66 BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 Residual Activity '=' 66 %
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Residual Activity '=' 135 %
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Residual Activity '=' 89 %
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Residual Activity '=' 84 %
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Residual Activity '=' 107 %
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Residual Activity '=' 51 %
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Residual Activity '=' 90 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Residual Activity '=' 1 %
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Residual Activity '=' 105 %
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Residual Activity '=' 105 %
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Residual Activity '=' 89 %
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Residual Activity '=' 99 %
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Residual Activity '=' 80 %
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Residual Activity '=' 124 %
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Thermal melting change '=' -1 degrees C
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Thermal melting change '=' -1 degrees C
P02545 BXGT005889 Prelamin-A/C reviewed - LMNA Potency '=' 1122 nM
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Residual Activity '=' 57 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Residual Activity '=' 98 %
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Residual Activity '=' 96 %
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Residual Activity '=' 111 %
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Residual Activity '=' 83 %
Q99549 BXGT019932 M-phase phosphoprotein 8 reviewed Epigenetic regulator MPHOSPH8 Potency - 31622 nM
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Residual Activity '=' 110 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 98 %
Q8IYT8 BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 Residual Activity '=' 112 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 6513 nM
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Thermal melting change '=' 0 degrees C
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Thermal melting change '=' 0 degrees C
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Inhibition '=' 8 %
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Residual Activity '=' 113 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Residual Activity '=' 67 %
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Residual Activity '=' 123 %
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Residual Activity '=' 83 %
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 19952 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Thermal melting change '=' 0 degrees C
Q9JI10 BXGT020811 Serine/threonine-protein kinase 3 reviewed - Stk3 Kd - - -
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Kd '>' 10000 nM
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Ki '>' 3162 nM
O14578 BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT Kd '=' 510 nM
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Kd '>' 10000 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Ki '=' 63 nM
Q13873 BXGT013398 Bone morphogenetic protein receptor type-2 reviewed Kinase BMPR2 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Ki '>' 2511 nM
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Residual Activity '=' 90 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 IC50 '=' 100 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Inhibition '=' 93 %
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Residual Activity '=' 110 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Residual Activity '=' 102 %
O43318 BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 Residual Activity '=' 104 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Residual Activity '=' 12 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Thermal melting change '=' 0 degrees C
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Residual Activity '=' 95 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Kd - - -
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Kd - - -
Q8TD19 BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 Kd - - -
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Kd - - -
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Kd - - -
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd - - -
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Kd - - -
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Kd '>' 10000 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Kd '>' 10000 nM
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Kd '>' 10000 nM
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Kd '>' 10000 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Ki '>' 3981 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Ki '>' 3981 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 97 %
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Residual Activity '=' 103 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency '=' 63095 nM
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Residual Activity '=' 87 %
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Thermal melting change '=' 0 degrees C
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Thermal melting change '=' 4 degrees C
P02545 BXGT005889 Prelamin-A/C reviewed - LMNA Potency '=' 5011 nM
P08659 BXGT006805 Luciferin 4-monooxygenase reviewed - Potency '=' 1258 nM
O94782 BXGT005332 Ubiquitin carboxyl-terminal hydrolase 1 reviewed Enzyme USP1 Potency - 63095 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Inhibition '=' 79 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Kd '>' 10000 nM
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Kd '>' 10000 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Kd '>' 10000 nM
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Kd '>' 10000 nM
O94768 BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B Kd '>' 10000 nM
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Kd '>' 10000 nM
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Kd '=' 3200 nM
P16050 BXGT008184 Arachidonate 15-lipoxygenase reviewed Enzyme ALOX15 Potency '=' 15848 nM
Q9UKI8 BXGT021743 Serine/threonine-protein kinase tousled-like 1 reviewed Kinase TLK1 Kd '>' 10000 nM
Q59H18 BXGT015278 Serine/threonine-protein kinase TNNI3K reviewed - TNNI3K Kd '>' 10000 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Kd '>' 10000 nM
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF IC50 - - -
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Ki '>' 3162 nM
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Ki '>' 3981 nM
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Inhibition '=' 13 %
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Inhibition '=' 39 %
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Ki '>' 3981 nM
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Residual Activity '=' 114 %
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Residual Activity '=' 90 %
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Residual Activity '=' 66 %
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Residual Activity '=' 95 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Kd '>' 10000 nM
P00523 BXGT005572 Proto-oncogene tyrosine-protein kinase Src reviewed - SRC Activity '=' 79 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Activity '=' 5 %
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Activity '=' 87 %
Q96PY6 BXGT019712 Serine/threonine-protein kinase Nek1 reviewed Kinase NEK1 Kd '>' 10000 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Kd '>' 10000 nM
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Kd '>' 10000 nM
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Kd '>' 10000 nM
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Kd '>' 10000 nM
Q9Y616 BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 Kd '>' 10000 nM
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Kd '>' 10000 nM
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd '>' 10000 nM
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Kd '>' 10000 nM
Q15569 BXGT013580 Dual specificity testis-specific protein kinase 1 reviewed Kinase TESK1 Kd '>' 10000 nM
Q99640 BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 Kd '>' 10000 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Activity '=' 85 %
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Kd '>' 10000 nM
Q8N752 BXGT018526 Casein kinase I isoform alpha-like reviewed Kinase CSNK1A1L Kd '=' 1900 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Kd - - -
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Activity '=' 109 %
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Activity '=' 98 %
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Activity '=' 92 %
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Kd '>' 10000 nM
Q99986 BXGT019980 Serine/threonine-protein kinase VRK1 reviewed Kinase VRK1 Thermal melting change '=' 0 degrees C
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Inhibition '=' 0 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Inhibition '=' 100 %
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Kd '>' 10000 nM
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Kd '>' 10000 nM
Q9Y463 BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B Kd '>' 10000 nM
P06240 BXGT006428 Proto-oncogene tyrosine-protein kinase LCK reviewed - Lck Activity '=' 44 %
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Kd '>' 10000 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Selectivity '=' 0 -
Q9Y463 BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B Ki '>' 2511 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Ki '>' 6309 nM
Q96L34 BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 Ki '>' 5011 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Kd - - -
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Kd - - -
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Residual Activity '=' 109 %
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Kd '>' 10000 nM
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Kd '>' 10000 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Thermal melting change '=' 1 degrees C
Q15118 BXGT013540 [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial reviewed Kinase PDK1 Inhibition '=' 87 %
Q8NFD2 BXGT018559 Ankyrin repeat and protein kinase domain-containing protein 1 reviewed Kinase ANKK1 Kd '>' 10000 nM
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Kd '>' 10000 nM
Q13627 BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A Ki '>' 1995 nM
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 Potency '=' 794 nM
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Kd '>' 10000 nM
Q9H1R3 BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 Kd - - -
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Ki '>' 3162 nM
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Kd '>' 10000 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd '>' 10000 nM
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF Kd '=' 620 nM
P19838 BXGT008526 Nuclear factor NF-kappa-B p105 subunit reviewed Transcription factor NFKB1 Potency '=' 11220 nM
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Ki '>' 5011 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Residual Activity '=' 7 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Kd - - -
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 Potency '=' 15848 nM
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Inhibition - - -
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Residual Activity '=' 59 %
Q9UGI9 BXGT021682 5'-AMP-activated protein kinase subunit gamma-3 reviewed Enzyme modulator PRKAG3 Residual Activity '=' 109 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 109 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 109 %
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Residual Activity '=' 109 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 109 %
O43741 BXGT004620 5'-AMP-activated protein kinase subunit beta-2 reviewed Enzyme modulator PRKAB2 Residual Activity '=' 109 %
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Residual Activity '=' 109 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 86 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 86 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 86 %
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Residual Activity '=' 120 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Residual Activity '=' 2 %
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Residual Activity '=' 101 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Kd - - -
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Kd '>' 10000 nM
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Kd '>' 10000 nM
Q9BWU1 BXGT020156 Cyclin-dependent kinase 19 reviewed Kinase CDK19 Kd '>' 10000 nM
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Kd '>' 10000 nM
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Activity '=' 95 %
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Kd '>' 10000 nM
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Residual Activity '=' 112 %
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Residual Activity '=' 103 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 110 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Residual Activity '=' 1 %
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Residual Activity '=' 64 %
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Residual Activity '=' 94 %
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Residual Activity '=' 58 %
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Kd - - -
Q13153 BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 Kd - - -
Q8N5S9 BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 Kd - - -
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Thermal melting change '=' 0 degrees C
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Thermal melting change '=' 0 degrees C
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Thermal melting change '=' 0 degrees C
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Thermal melting change '=' 0 degrees C
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Thermal melting change '=' 0 degrees C
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Thermal melting change '=' 0 degrees C
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Kd - - -
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Kd - - -
O60885 BXGT004906 Bromodomain-containing protein 4 reviewed Epigenetic regulator BRD4 IC50 '=' 2500 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Activity '=' 103 %
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Kd '>' 10000 nM
Q8TD19 BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 Kd '>' 10000 nM
P53671 BXGT011009 LIM domain kinase 2 reviewed Kinase LIMK2 Kd '>' 10000 nM
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Kd '>' 10000 nM
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Kd '>' 10000 nM
P16473 BXGT008234 Thyrotropin receptor reviewed G-protein coupled receptor TSHR Potency '=' 12589 nM
P54132 BXGT011032 Bloom syndrome protein reviewed - BLM Potency '=' 50118 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Activity '=' 86 %
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Kd '=' 28 nM
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 910 nM
Q02779 BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 Kd '>' 10000 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 50 nM
Q62868 BXGT016047 Rho-associated protein kinase 2 reviewed - Rock2 Inhibition '=' 61 %
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 22387 nM
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Kd '>' 10000 nM
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Kd '>' 10000 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Kd '>' 10000 nM
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Kd '>' 10000 nM
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Activity '=' 104 %
Q8IVH8 BXGT018345 Mitogen-activated protein kinase kinase kinase kinase 3 reviewed Kinase MAP4K3 Kd '>' 10000 nM
Q13546 BXGT013372 Receptor-interacting serine/threonine-protein kinase 1 reviewed Kinase RIPK1 Kd '>' 10000 nM
P37023 BXGT009953 Serine/threonine-protein kinase receptor R3 reviewed Kinase ACVRL1 Kd '>' 10000 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Activity '=' 49 %
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Kd '>' 10000 nM
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Activity '=' 87 %
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Ki '>' 3981 nM
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Inhibition '=' 87 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Residual Activity '=' 100 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Potency '=' 7943 nM
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Residual Activity '=' 41 %
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Residual Activity '=' 44 %
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Activity '=' 70 %
P27037 BXGT009153 Activin receptor type-2A reviewed Kinase ACVR2A Kd '>' 10000 nM
Q00537 BXGT012536 Cyclin-dependent kinase 17 reviewed Kinase CDK17 Kd '>' 10000 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Kd '>' 10000 nM
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Kd '>' 10000 nM
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Kd '>' 10000 nM
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Kd '>' 10000 nM
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 2300 nM
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 Potency '=' 12589 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 30 nM
P16473 BXGT008234 Thyrotropin receptor reviewed G-protein coupled receptor TSHR Potency '=' 7943 nM
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Kd '=' 3800 nM
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Kd '>' 10000 nM
P36894 BXGT009939 Bone morphogenetic protein receptor type-1A reviewed Kinase BMPR1A Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Ki '>' 6309 nM
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Kd '>' 10000 nM
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Kd '=' 1900 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Kd '>' 10000 nM
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Activity '=' 69 %
O94921 BXGT005341 Cyclin-dependent kinase 14 reviewed Kinase CDK14 Kd '>' 10000 nM
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Activity '=' 70 %
Q07002 BXGT012908 Cyclin-dependent kinase 18 reviewed Kinase CDK18 Kd '>' 10000 nM
Q86YV6 BXGT017636 Myosin light chain kinase family member 4 reviewed - MYLK4 Kd '>' 10000 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 12589 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Thermal melting change '=' 0 degrees C
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Kd '>' 10000 nM
P0A6C1 BXGT007045 Endonuclease 4 reviewed - nfo Potency '=' 25118 nM
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Kd '>' 10000 nM
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Residual Activity '=' 94 %
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Residual Activity '=' 112 %
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Residual Activity '=' 123 %
P78396 BXGT011842 Cyclin-A1 reviewed Enzyme modulator CCNA1 Residual Activity '=' 88 %
P20248 BXGT008554 Cyclin-A2 reviewed Enzyme modulator CCNA2 Residual Activity '=' 88 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 88 %
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Residual Activity '=' 117 %
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Residual Activity '=' 92 %
Q01453 BXGT012588 Peripheral myelin protein 22 reviewed Cellular structure PMP22 Potency '=' 26854 nM
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd '=' 1600 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Kd '>' 10000 nM
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Kd '>' 10000 nM
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Kd '>' 10000 nM
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Kd '>' 10000 nM
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Kd '>' 10000 nM
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Kd '>' 10000 nM
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Kd '>' 10000 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Inhibition '=' 80 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Ki '>' 2511 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Kd - - -
Q9UF33 BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 4600 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Kd - - -
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Kd '>' 10000 nM
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Kd '>' 10000 nM
Q8NI60 BXGT018572 Atypical kinase COQ8A, mitochondrial reviewed Kinase COQ8A Kd '>' 10000 nM
O95149 BXGT005350 Snurportin-1 reviewed - SNUPN Potency - 125892 nM
Q14974 BXGT013516 Importin subunit beta-1 reviewed Transporter KPNB1 Potency - 125892 nM
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Residual Activity '=' 89 %
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Residual Activity '=' 117 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Residual Activity '=' 19 %
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Ki '>' 6309 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 15848 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Activity '=' 89 %
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Kd '>' 10000 nM
P33981 BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK Kd '=' 4500 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Kd '>' 10000 nM
O95835 BXGT005400 Serine/threonine-protein kinase LATS1 reviewed Kinase LATS1 Kd '>' 10000 nM
Q96L34 BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 Kd '>' 10000 nM
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Activity '=' 86 %
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Activity '=' 92 %
P00352 BXGT005510 Retinal dehydrogenase 1 reviewed Enzyme ALDH1A1 Potency '=' 35481 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '>' 10000 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Kd '>' 10000 nM
Q13237 BXGT013331 cGMP-dependent protein kinase 2 reviewed Kinase PRKG2 Kd '>' 10000 nM
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Kd '>' 10000 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Kd '>' 10000 nM
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Ki '>' 1995 nM
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Kd '=' 950 nM
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Kd '>' 10000 nM
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Activity '=' 107 %
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Kd '>' 10000 nM
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Kd '>' 10000 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Activity '=' 122 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Activity '=' 83 %
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Kd '=' 270 nM
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Activity '=' 91 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Kd '=' 2400 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Kd '=' 42 nM
O15075 BXGT004124 Serine/threonine-protein kinase DCLK1 reviewed Kinase DCLK1 Kd '>' 10000 nM
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Kd '>' 10000 nM
Q14164 BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE Ki '>' 3162 nM
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Activity '=' 104 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Activity '=' 73 %
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Kd '>' 10000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Kd - - -
Q2M2I8 BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 Kd - - -
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Kd - - -
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Kd - - -
P11799 BXGT007749 Myosin light chain kinase, smooth muscle reviewed - Mylk Kd '>' 10000 nM
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Kd '>' 10000 nM
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Kd '>' 10000 nM
P45985 BXGT010496 Dual specificity mitogen-activated protein kinase kinase 4 reviewed Kinase MAP2K4 Kd '>' 10000 nM
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1900 nM
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Kd '>' 10000 nM
B2RXH2 BXGT002006 Lysine-specific demethylase 4E reviewed - KDM4E Potency '=' 14125 nM
P15917 BXGT008169 Lethal factor reviewed - lef Potency '=' 794 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Kd - - -
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Kd - - -
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Kd - - -
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Residual Activity '=' 79 %
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Residual Activity '=' 96 %
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Residual Activity '=' 94 %
O60563 BXGT004883 Cyclin-T1 reviewed Enzyme modulator CCNT1 Residual Activity '=' 94 %
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Ki '>' 2511 nM
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Residual Activity '=' 78 %
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Kd - - -
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Kd - - -
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Kd - - -
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Kd - - -
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Kd - - -
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Residual Activity '=' 92 %
O94768 BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B Kd - - -
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Kd - - -
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Ki '>' 2511 nM
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Ki '>' 3162 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Ki '>' 1995 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Kd - - -
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Kd - - -
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Kd - - -
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Kd - - -
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Kd - - -
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Kd - - -
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Kd - - -
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Residual Activity '=' 111 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 108 %
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Residual Activity '=' 103 %
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Residual Activity '=' 105 %
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Residual Activity '=' 47 %
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Kd - - -
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Residual Activity '=' 83 %
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Residual Activity '=' 81 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Residual Activity '=' 109 %
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Residual Activity '=' 91 %
Q9UNA4 BXGT021785 DNA polymerase iota reviewed - POLI Potency - 1584 nM
P04062 BXGT006140 Lysosomal acid glucosylceramidase reviewed - GBA Potency - 14125 nM
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Kd '>' 10000 nM
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Kd - - -
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd '=' 10000 nM
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Ki '=' 2511 nM
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Kd '>' 10000 nM
Q9P2K8 BXGT021302 eIF-2-alpha kinase GCN2 reviewed - EIF2AK4 Kd '>' 10000 nM
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Activity '=' 61 %
Q2M2I8 BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 Kd '>' 10000 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Kd '=' 9600 nM
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Activity '=' 84 %
Q16659 BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 Kd '>' 10000 nM
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Kd '>' 10000 nM
P19525 BXGT008492 Interferon-induced, double-stranded RNA-activated protein kinase reviewed Kinase EIF2AK2 Kd '>' 10000 nM
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Activity '=' 63 %
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Residual Activity '=' 108 %
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd - - -
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Kd '=' 9400 nM
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Kd '=' 400 nM
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Thermal melting change '=' 0 degrees C
Q16512 BXGT013631 Serine/threonine-protein kinase N1 reviewed Kinase PKN1 Kd '>' 10000 nM
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Kd '>' 10000 nM
Q9H3Y6 BXGT020468 Tyrosine-protein kinase Srms reviewed Kinase SRMS Kd '>' 10000 nM
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Kd '=' 790 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Kd '>' 10000 nM
P31152 BXGT009511 Mitogen-activated protein kinase 4 reviewed Kinase MAPK4 Kd '>' 10000 nM
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Activity '=' 102 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Kd '>' 10000 nM
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF Kd '=' 4800 nM
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Kd '>' 10000 nM
Q9UQ88 BXGT021808 Cyclin-dependent kinase 11A reviewed - CDK11A Kd '>' 10000 nM
O43781 BXGT004625 Dual specificity tyrosine-phosphorylation-regulated kinase 3 reviewed Kinase DYRK3 Activity '=' 96 %
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Kd '>' 10000 nM
Q13164 BXGT013322 Mitogen-activated protein kinase 7 reviewed Kinase MAPK7 Kd '>' 10000 nM
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Inhibition '=' 75 %
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Activity '=' 66 %
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Residual Activity '=' 121 %
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Residual Activity '=' 41 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Residual Activity '=' 107 %
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Residual Activity '=' 43 %
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Residual Activity '=' 102 %
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Residual Activity '=' 93 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 93 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 93 %
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Residual Activity '=' 90 %
P04062 BXGT006140 Lysosomal acid glucosylceramidase reviewed - GBA Potency - 39810 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Residual Activity '=' 101 %
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Residual Activity '=' 61 %
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Activity '=' 113 %
P30291 BXGT009417 Wee1-like protein kinase reviewed Kinase WEE1 Kd '>' 10000 nM
P78362 BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Residual Activity '=' 122 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Kd '>' 10000 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Activity '=' 27 %
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Kd '=' 53 nM
P11712 BXGT007738 Cytochrome P450 2C9 reviewed - CYP2C9 AC50 '=' 15848 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 300 nM
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Residual Activity '=' 83 %
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Residual Activity '=' 92 %
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Residual Activity '=' 65 %
O60563 BXGT004883 Cyclin-T1 reviewed Enzyme modulator CCNT1 Residual Activity '=' 65 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 91 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 91 %
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Kd '>' 10000 nM
Q6DT37 BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG Kd '=' 640 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 2600 nM
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Residual Activity '=' 98 %
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Residual Activity '=' 46 %
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Residual Activity '=' 47 %
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Kd '=' 150 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Kd '=' 170 nM
Q9BYP7 BXGT020188 Serine/threonine-protein kinase WNK3 reviewed Kinase WNK3 Residual Activity '=' 75 %
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Activity '=' 0 %
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Kd '>' 10000 nM
Q13627 BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A Activity '=' 99 %
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Kd '>' 10000 nM
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Kd '>' 10000 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Kd '>' 10000 nM
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Kd '>' 10000 nM
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Activity '=' 83 %
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Residual Activity '=' 102 %
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Residual Activity '=' 87 %
Q96BR1 BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed - SGK3 Residual Activity '=' 109 %
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Residual Activity '=' 117 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 123 %
Q8IYT8 BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 Residual Activity '=' 104 %
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Residual Activity '=' 92 %
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Residual Activity '=' 92 %
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Residual Activity '=' 108 %
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Residual Activity '=' 109 %
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Residual Activity '=' 92 %
Q9NSY1 BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K Kd - - -
Q9BYP7 BXGT020188 Serine/threonine-protein kinase WNK3 reviewed Kinase WNK3 Residual Activity '=' 109 %
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Residual Activity '=' 117 %
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Residual Activity '=' 69 %
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Residual Activity '=' 111 %
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Residual Activity '=' 90 %
Q96PF2 BXGT019708 Testis-specific serine/threonine-protein kinase 2 reviewed Kinase TSSK2 Residual Activity '=' 113 %
P10635 BXGT007595 Cytochrome P450 2D6 reviewed - CYP2D6 AC50 '=' 5011 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Inhibition '=' 37 %
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Inhibition '=' 53 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Inhibition '=' 88 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Residual Activity '=' 112 %
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Residual Activity '=' 91 %
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Residual Activity '=' 105 %
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Residual Activity '=' 94 %
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Residual Activity '=' 116 %
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Residual Activity '=' 88 %
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Residual Activity '=' 109 %
P30281 BXGT009416 G1/S-specific cyclin-D3 reviewed Enzyme modulator CCND3 Residual Activity '=' 109 %
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Residual Activity '=' 52 %
Q8NEV4 BXGT018558 Myosin-IIIa reviewed Kinase MYO3A Kd '>' 10000 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Ki '>' 5011 nM
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Ki '>' 3981 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Ki '>' 2511 nM
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Ki '=' 794 nM
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Ki '>' 3981 nM
P46734 BXGT010537 Dual specificity mitogen-activated protein kinase kinase 3 reviewed Kinase MAP2K3 Kd '>' 10000 nM
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Kd '>' 10000 nM
P29376 BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK Kd '>' 10000 nM
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Ki '>' 3162 nM
Q13470 BXGT013359 Non-receptor tyrosine-protein kinase TNK1 reviewed Kinase TNK1 Kd '>' 10000 nM
Q9BRS2 BXGT020119 Serine/threonine-protein kinase RIO1 reviewed Kinase RIOK1 Kd '>' 10000 nM
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Kd - - -
Q3U3Q1 BXGT014526 Serine/threonine-protein kinase ULK3 reviewed - Ulk3 Kd - - -
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Kd - - -
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Kd '=' 13 nM
P00352 BXGT005510 Retinal dehydrogenase 1 reviewed Enzyme ALDH1A1 Potency '=' 17782 nM
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 107 %
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Residual Activity '=' 107 %
P67870 BXGT011566 Casein kinase II subunit beta reviewed Kinase CSNK2B Residual Activity '=' 107 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 122 %
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Residual Activity '=' 90 %
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Residual Activity '=' 114 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 59 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Kd '=' 3000 nM
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Kd - - -
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Residual Activity '=' 102 %
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Residual Activity '=' 119 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Kd - - -
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Kd '=' 6000 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 IC50 '=' 80 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 80 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 IC50 '=' 80 nM
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 IC50 '=' 80 nM
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Kd '>' 10000 nM
P27695 BXGT009199 DNA-(apurinic or apyrimidinic site) lyase reviewed - APEX1 Potency - 44668 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Residual Activity '=' 27 %
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Ki '>' 3162 nM
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Residual Activity '=' 57 %
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Residual Activity '=' 63 %
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Residual Activity '=' 94 %
B2RXH2 BXGT002006 Lysine-specific demethylase 4E reviewed - KDM4E Potency '=' 31622 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Residual Activity '=' 49 %
P11308 BXGT007684 Transcriptional regulator ERG reviewed Transcription factor ERG Potency - 50118 nM
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Residual Activity '=' 99 %
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Residual Activity '=' 112 %
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Residual Activity '=' 112 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 99 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 99 %
O14733 BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 Residual Activity '=' 80 %
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 794 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Ki '>' 1995 nM
Q96KQ7 BXGT019687 Histone-lysine N-methyltransferase EHMT2 reviewed Epigenetic regulator EHMT2 Potency - 843 nM
Q99714 BXGT019954 3-hydroxyacyl-CoA dehydrogenase type-2 reviewed Enzyme HSD17B10 Potency '=' 31622 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Residual Activity '=' 109 %
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Ki '>' 6309 nM
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 29092 nM
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Residual Activity '=' 111 %
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Residual Activity '=' 45 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Residual Activity '=' 123 %
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Ki '>' 5011 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Inhibition '=' 20 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Ki '=' 251 nM
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Ki '=' 2511 nM
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Ki '>' 3162 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Ki '>' 6309 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 16 nM
P78356 BXGT011837 Phosphatidylinositol 5-phosphate 4-kinase type-2 beta reviewed Kinase PIP4K2B Kd '>' 10000 nM
Q99755 BXGT019958 Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha reviewed Kinase PIP5K1A Kd '>' 10000 nM
P29597 BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 Kd '>' 10000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Kd '>' 10000 nM
Q8N5S9 BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 Activity '=' 94 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Kd '>' 10000 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Residual Activity '=' 77 %
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Residual Activity '=' 88 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Residual Activity '=' 69 %
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Residual Activity '=' 110 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Residual Activity '=' 110 %
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Kd '=' 3300 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Activity '=' 78 %
Q86UX6 BXGT017614 Serine/threonine-protein kinase 32C reviewed Kinase STK32C Kd '>' 10000 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Kd '=' 32 nM
P29376 BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK Ki '>' 1584 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd '=' 210 nM
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Kd '>' 10000 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Kd '>' 10000 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Kd '=' 2700 nM
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Thermal melting change '=' 0 degrees C
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Thermal melting change '=' 4 degrees C
Q9Y3S1 BXGT022266 Serine/threonine-protein kinase WNK2 reviewed Kinase WNK2 Residual Activity '=' 84 %
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Residual Activity '=' 103 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Residual Activity '=' 93 %
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Residual Activity '=' 109 %
Q86Z02 BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 Residual Activity '=' 96 %
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Residual Activity '=' 78 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 122 %
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Residual Activity '=' 101 %
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Residual Activity '=' 72 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 124 %
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Residual Activity '=' 115 %
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Inhibition - - -
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Inhibition - - -
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Inhibition - - -
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Residual Activity '=' 49 %
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Residual Activity '=' 93 %
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Kd - - -
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Kd - - -
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Kd - - -
Q9Y253 BXGT022216 DNA polymerase eta reviewed - POLH Potency - 22387 nM
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Kd '>' 10000 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Kd '>' 10000 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Kd '>' 10000 nM
P21127 BXGT008623 Cyclin-dependent kinase 11B reviewed Kinase CDK11B Kd '>' 10000 nM
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Kd '=' 1600 nM
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Kd '>' 10000 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Ki '=' 1000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Kd - - -
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Kd - - -
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Kd - - -
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd - - -
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Kd - - -
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Kd - - -
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Kd - - -
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Inhibition '=' 63 %
Q16288 BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 Kd '>' 10000 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Kd '>' 10000 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Kd '>' 10000 nM
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 15067 nM
Q6P3R8 BXGT016447 Serine/threonine-protein kinase Nek5 reviewed - NEK5 Kd '>' 10000 nM
P42336 BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA Kd '>' 10000 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Kd '>' 10000 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Activity '=' 42 %
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Kd '>' 10000 nM
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Residual Activity '=' 85 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Residual Activity '=' 14 %
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Residual Activity '=' 94 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Kd - - -
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd - - -
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd '=' 120 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Kd - - -
P00352 BXGT005510 Retinal dehydrogenase 1 reviewed Enzyme ALDH1A1 Potency '=' 39810 nM
P00811 BXGT005666 Beta-lactamase reviewed - ampC Potency '=' 7079 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Kd - - -
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Kd - - -
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Kd - - -
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Kd - - -
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Kd - - -
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Ki '>' 5011 nM
Q08345 BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 Kd '=' 1100 nM
Q9NSY1 BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K Kd '>' 10000 nM
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Kd '>' 10000 nM
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Kd '>' 10000 nM
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Kd '>' 10000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Ki '>' 3162 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Inhibition '=' 61 %
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Kd '>' 10000 nM
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Kd '>' 10000 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Activity '=' 21 %
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Kd '>' 10000 nM
P49336 BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 Kd '>' 10000 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Inhibition '=' 11 %
Q8TD08 BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 Kd '>' 10000 nM
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Kd '>' 10000 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Activity '=' 90 %
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Activity '=' 90 %
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Activity '=' 71 %
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Residual Activity '=' 117 %
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Residual Activity '=' 88 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Residual Activity '=' 19 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 37847 nM
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Residual Activity '=' 95 %
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 44668 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Residual Activity '=' 40 %
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 20596 nM
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 123 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Residual Activity '=' 49 %
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Residual Activity '=' 83 %
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Residual Activity '=' 98 %
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd - - -
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Kd - - -
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Kd - - -
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Kd - - -
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Kd - - -
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Kd '=' 3100 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Kd - - -
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Kd - - -
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Kd '=' 120 nM
P12527 BXGT007824 Arachidonate 5-lipoxygenase reviewed - Alox5 Inhibition '=' 68 %
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Residual Activity '=' 12 %
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Residual Activity '=' 87 %
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Residual Activity '=' 36 %
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Thermal melting change '=' 0 degrees C
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Thermal melting change '=' 0 degrees C
Q8WXR4 BXGT019015 Myosin-IIIb reviewed Kinase MYO3B Kd '>' 10000 nM
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Kd '>' 10000 nM
P37173 BXGT009970 TGF-beta receptor type-2 reviewed Kinase TGFBR2 Kd '>' 10000 nM
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Kd '>' 10000 nM
Q9NRM7 BXGT021190 Serine/threonine-protein kinase LATS2 reviewed Kinase LATS2 Kd '=' 1700 nM
P84022 BXGT012027 Mothers against decapentaplegic homolog 3 reviewed Transcription factor SMAD3 Potency - 35481 nM
P15917 BXGT008169 Lethal factor reviewed - lef FC '=' 4 -
Q9C098 BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 Kd '>' 10000 nM
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Kd '>' 10000 nM
Q5SC61 BXGT015659 Mitogen-activated protein kinase unreviewed - MAPK-1 IC50 - - -
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Residual Activity '=' 101 %
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Residual Activity '=' 68 %
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Residual Activity '=' 29 %
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Residual Activity '=' 87 %
Q9NYY3 BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 Residual Activity '=' 104 %
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Residual Activity '=' 117 %
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Residual Activity '=' 54 %
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Residual Activity '=' 110 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Ki '=' 1258 nM
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Inhibition - - -
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Residual Activity '=' 97 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 80 %
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Residual Activity '=' 34 %
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Residual Activity '=' 85 %
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Residual Activity '=' 11 %
O75496 BXGT005132 Geminin reviewed - GMNN Potency '=' 22387 nM
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Residual Activity '=' 5 %
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd '>' 10000 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Ki '=' 501 nM
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 35481 nM
Q16236 BXGT013624 Nuclear factor erythroid 2-related factor 2 reviewed Enzyme NFE2L2 Potency - 7307 nM
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Kd '=' 650 nM
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Kd - - -
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Kd - - -
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 AC50 '=' 501 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Ki '>' 3162 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Activity '=' 83 %
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Kd '>' 10000 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Kd '>' 10000 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Kd '>' 10000 nM
Q9NY57 BXGT021250 Serine/threonine-protein kinase 32B reviewed Kinase STK32B Kd '=' 4900 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Kd '>' 10000 nM
Q04771 BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 Kd '>' 10000 nM
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Kd '>' 10000 nM
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Activity '=' 86 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Kd '>' 10000 nM
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Kd '>' 10000 nM
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Kd '>' 10000 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Kd '>' 10000 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Ki '=' 5 nM
P68370 BXGT011596 Tubulin alpha-1A chain reviewed - Tuba1a Kd '=' 4900 nM
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Activity '=' 89 %
Q8NG66 BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 Residual Activity '=' 85 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Inhibition '=' 97 %
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Residual Activity '=' 92 %
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Residual Activity '=' 92 %
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Residual Activity '=' 84 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Inhibition - - -
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Residual Activity '=' 70 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 24 %
P33981 BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK Kd - - -
Q9Y6R4 BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 Kd - - -
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Kd - - -
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Kd - - -
Q99640 BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 Kd - - -
P15428 BXGT008121 15-hydroxyprostaglandin dehydrogenase [NAD(+)] reviewed - HPGD Potency '=' 15848 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Residual Activity '=' 108 %
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Residual Activity '=' 104 %
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Residual Activity '=' 58 %
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Residual Activity '=' 113 %
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Residual Activity '=' 98 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Residual Activity '=' 98 %
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Residual Activity '=' 111 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 14 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Residual Activity '=' 83 %
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Residual Activity '=' 76 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition - - -
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Residual Activity '=' 92 %
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Residual Activity '=' 85 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 90 %
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Residual Activity '=' 59 %
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Residual Activity '=' 92 %
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Residual Activity '=' 68 %
Q9UPE1 BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 Residual Activity '=' 110 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Residual Activity '=' 49 %
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Ki '>' 2511 nM
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Residual Activity '=' 65 %
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Residual Activity '=' 77 %
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Residual Activity '=' 108 %
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Residual Activity '=' 80 %
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Residual Activity '=' 90 %
O94806 BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 Ki '=' 2511 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Ki '>' 2511 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Ki '>' 6309 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Residual Activity '=' 92 %
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Ki '>' 2511 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 26 %
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Residual Activity '=' 112 %
P83916 BXGT012025 Chromobox protein homolog 1 reviewed Epigenetic regulator CBX1 Potency - 56234 nM
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Residual Activity '=' 92 %
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Residual Activity '=' 125 %
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Residual Activity '=' 107 %
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Residual Activity '=' 99 %
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Residual Activity '=' -1 %
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Residual Activity '=' 92 %
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Residual Activity '=' 121 %
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Residual Activity '=' 34 %
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Residual Activity '=' 85 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 113 %
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Residual Activity '=' 103 %
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Residual Activity '=' 59 %
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Residual Activity '=' 49 %
P14635 BXGT008031 G2/mitotic-specific cyclin-B1 reviewed Enzyme modulator CCNB1 Residual Activity '=' 92 %
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Residual Activity '=' 92 %
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Residual Activity '=' 16 %
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Residual Activity '=' 87 %
O94806 BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 Kd '>' 10000 nM
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Kd '>' 10000 nM
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 AC50 '=' 10000 nM
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Activity '=' 84 %
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Kd '=' 59 nM
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Residual Activity '=' 93 %
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Residual Activity '=' 117 %
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Residual Activity '=' 41 %
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Residual Activity '=' 98 %
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Residual Activity '=' 85 %
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Residual Activity '=' 100 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Activity '=' 82 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Activity '=' 3 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Kd '=' 3100 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Inhibition - - -
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Inhibition - - -
Q8TD08 BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 Activity '=' 106 %
Q8N5S9 BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 Kd '>' 10000 nM
Q8IV63 BXGT018341 Inactive serine/threonine-protein kinase VRK3 reviewed Kinase VRK3 Thermal melting change '=' 0 degrees C
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Residual Activity '=' 96 %
Q96PF2 BXGT019708 Testis-specific serine/threonine-protein kinase 2 reviewed Kinase TSSK2 Residual Activity '=' 103 %
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Inhibition '=' 95 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Inhibition '=' 88 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Inhibition '=' 105 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Inhibition - - -
Q8TF76 BXGT018826 Serine/threonine-protein kinase haspin reviewed Kinase HASPIN Residual Activity '=' 10 %
P05129 BXGT006322 Protein kinase C gamma type reviewed Kinase PRKCG Residual Activity '=' 106 %
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Residual Activity '=' 113 %
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Residual Activity '=' 121 %
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Residual Activity '=' 107 %
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Kd - - -
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Kd - - -
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Kd - - -
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Kd - - -
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Kd '>' 10000 nM
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Kd '>' 10000 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Kd '>' 10000 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 10000 nM
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Activity '=' 93 %
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Activity '=' 103 %
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Activity '=' 103 %
P67870 BXGT011566 Casein kinase II subunit beta reviewed Kinase CSNK2B Activity '=' 103 %
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Kd '>' 10000 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Inhibition '=' 39 %
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Ki '>' 3162 nM
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Ki '>' 6309 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Ki '>' 3981 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Inhibition - - -
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Residual Activity '=' -2 %
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Residual Activity '=' 102 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 210 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1400 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Kd '>' 10000 nM
Q9Y2H1 BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L Kd '>' 10000 nM
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Activity '=' 86 %
Q86Z02 BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 Residual Activity '=' 103 %
Q16584 BXGT013642 Mitogen-activated protein kinase kinase kinase 11 reviewed Kinase MAP3K11 Kd '>' 10000 nM
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Residual Activity '=' 77 %
P78362 BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 Residual Activity '=' 118 %
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Residual Activity '=' 88 %
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Residual Activity '=' 127 %
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Residual Activity '=' 8 %
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Residual Activity '=' 95 %
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Ki '>' 3981 nM
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Residual Activity '=' 110 %
Q96QE3 BXGT019718 ATPase family AAA domain-containing protein 5 reviewed - ATAD5 Potency - 29081 nM
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Ki '>' 3162 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Residual Activity '=' 113 %
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Residual Activity '=' 115 %
Q15078 BXGT013534 Cyclin-dependent kinase 5 activator 1 reviewed Enzyme modulator CDK5R1 Residual Activity '=' 127 %
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Residual Activity '=' 127 %
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Residual Activity '=' 86 %
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Residual Activity '=' 14 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd - - -
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Residual Activity '=' 83 %
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Residual Activity '=' 99 %
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Residual Activity '=' 111 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 66 %
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Residual Activity '=' 103 %
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Residual Activity '=' 104 %
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Kd '>' 10000 nM
Q14164 BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE Kd '>' 10000 nM
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Activity '=' 107 %
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Activity '=' 92 %
Q9NYL2 BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 Kd '>' 10000 nM
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Kd '>' 10000 nM
O95819 BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 Kd '>' 10000 nM
O95819 BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 Ki '=' 1000 nM
P49336 BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 Ki '>' 3981 nM
Q16659 BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 Thermal melting change '=' 0 degrees C
P15428 BXGT008121 15-hydroxyprostaglandin dehydrogenase [NAD(+)] reviewed - HPGD Potency '=' 25118 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Residual Activity '=' 55 %
O75496 BXGT005132 Geminin reviewed - GMNN Potency - 3548 nM
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Thermal melting change '=' 0 degrees C
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Thermal melting change '=' 0 degrees C
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Thermal melting change '=' 0 degrees C
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Thermal melting change '=' 0 degrees C
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Residual Activity '=' 69 %
Q8WTQ7 BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 Residual Activity '=' 96 %
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Residual Activity '=' 84 %
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Residual Activity '=' 68 %
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Residual Activity '=' 67 %
P05129 BXGT006322 Protein kinase C gamma type reviewed Kinase PRKCG Residual Activity '=' 103 %
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Ki '>' 3981 nM
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Residual Activity '=' 58 %
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Residual Activity '=' 108 %
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Residual Activity '=' 106 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Residual Activity '=' 65 %
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Residual Activity '=' 122 %
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Residual Activity '=' 93 %
P43250 BXGT010372 G protein-coupled receptor kinase 6 reviewed Kinase GRK6 Residual Activity '=' 97 %
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Residual Activity '=' 122 %
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Residual Activity '=' 105 %
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Residual Activity '=' 13 %
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Residual Activity '=' 141 %
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Residual Activity '=' 104 %
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Residual Activity '=' 81 %
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Residual Activity '=' 100 %
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Residual Activity '=' 92 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Residual Activity '=' 99 %
Q16288 BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 Ki '=' 2511 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Residual Activity '=' 76 %
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Residual Activity '=' 105 %
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Residual Activity '=' 19 %
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Residual Activity '=' 99 %
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Thermal melting change '=' 0 degrees C
P09917 BXGT006941 Arachidonate 5-lipoxygenase reviewed Enzyme ALOX5 IC50 '=' 50 nM
O60885 BXGT004906 Bromodomain-containing protein 4 reviewed Epigenetic regulator BRD4 Kd '=' 3400 nM
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Activity '=' 97 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 2000 nM
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Kd '>' 10000 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Kd '>' 10000 nM
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Kd '>' 10000 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Kd '=' 1700 nM
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Ki '>' 10000 nM
P47871 BXGT010592 Glucagon receptor reviewed G-protein coupled receptor GCGR IC50 '=' 80 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Residual Activity '=' 83 %
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Residual Activity '=' 93 %
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Residual Activity '=' 109 %
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Residual Activity '=' 41 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Inhibition - - -
Q5S007 BXGT015650 Leucine-rich repeat serine/threonine-protein kinase 2 reviewed Kinase LRRK2 Ki '>' 2511 nM
Q9Y3S1 BXGT022266 Serine/threonine-protein kinase WNK2 reviewed Kinase WNK2 Residual Activity '=' 118 %
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Residual Activity '=' 82 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Residual Activity '=' 55 %
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Residual Activity '=' 36 %
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 126 %
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Residual Activity '=' 100 %
Q9NYY3 BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 Residual Activity '=' 105 %
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Residual Activity '=' 90 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Inhibition - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Residual Activity '=' 74 %
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Residual Activity '=' 72 %
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Residual Activity '=' 81 %
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Residual Activity '=' 93 %
P04062 BXGT006140 Lysosomal acid glucosylceramidase reviewed - GBA Potency - 19952 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 102 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 102 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 102 %
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 IC50 '>' 100000 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Ki '>' 3981 nM
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Thermal melting change '=' 0 degrees C
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Thermal melting change '=' 1 degrees C
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Thermal melting change '=' 0 degrees C
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Thermal melting change '=' 0 degrees C
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Residual Activity '=' -1 %
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Residual Activity '=' 94 %
O14733 BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 Residual Activity '=' 57 %
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Residual Activity '=' 97 %
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Residual Activity '=' 99 %
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Residual Activity '=' 113 %
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Residual Activity '=' 91 %
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Residual Activity '=' 109 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 109 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 109 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 91 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 91 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 91 %
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Residual Activity '=' 32 %
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Residual Activity '=' 98 %
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Residual Activity '=' 12 %
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Residual Activity '=' 109 %
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Residual Activity '=' 80 %
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Thermal melting change '=' 0 degrees C
P03070 BXGT006016 Large T antigen reviewed - IC50 - 4870 nM
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Residual Activity '=' 100 %
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Residual Activity '=' 12 %
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Ki '>' 1584 nM
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Ki '>' 1584 nM
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Residual Activity '=' 43 %
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Residual Activity '=' 37 %
Q96BR1 BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed - SGK3 Residual Activity '=' 73 %
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Residual Activity '=' 45 %
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Kd '=' 6800 nM
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Activity '=' 93 %
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Activity '=' 85 %
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Activity '=' 76 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd '>' 10000 nM
Q02779 BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 Ki '>' 3162 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Residual Activity '=' 136 %
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Residual Activity '=' 96 %
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Residual Activity '=' 95 %
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Residual Activity '=' 110 %
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Residual Activity '=' 76 %
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Thermal melting change '=' 1 degrees C
P33261 BXGT009707 Cytochrome P450 2C19 reviewed - CYP2C19 Potency '=' 10000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Residual Activity '=' 69 %
Q04771 BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 Ki '>' 3162 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Ki '>' 3162 nM
Q8TF76 BXGT018826 Serine/threonine-protein kinase haspin reviewed Kinase HASPIN Residual Activity '=' 55 %
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Residual Activity '=' 106 %
Q9Y2H1 BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L Kd - - -
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Kd - - -
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Residual Activity '=' 26 %
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Residual Activity '=' 115 %
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Residual Activity '=' 92 %
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Thermal melting change '=' 4 degrees C
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Residual Activity '=' 108 %
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Residual Activity '=' 108 %
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Residual Activity '=' 104 %
P51946 BXGT010907 Cyclin-H reviewed Enzyme modulator CCNH Residual Activity '=' 104 %
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Activity '=' 7 %
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Thermal melting change '=' 0 degrees C
Q15208 BXGT013550 Serine/threonine-protein kinase 38 reviewed Kinase STK38 Thermal melting change '=' 0 degrees C
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Inhibition '=' 92 %
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Inhibition '=' 97 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Inhibition '=' 3 %
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Kd '=' 51 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd - - -
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Kd - - -
O75164 BXGT005104 Lysine-specific demethylase 4A reviewed - KDM4A Potency - 50118 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Residual Activity '=' 24 %
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Residual Activity '=' 107 %
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Residual Activity '=' 100 %
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Residual Activity '=' 40 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Inhibition '=' 4 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Ki '>' 3162 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Ki '>' 3981 nM
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Residual Activity '=' 99 %
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Residual Activity '=' 79 %
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Residual Activity '=' 75 %
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Residual Activity '=' 53 %
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 98 %
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Residual Activity '=' 123 %
P30281 BXGT009416 G1/S-specific cyclin-D3 reviewed Enzyme modulator CCND3 Residual Activity '=' 123 %
O94782 BXGT005332 Ubiquitin carboxyl-terminal hydrolase 1 reviewed Enzyme USP1 Potency - 3548133 nM
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Inhibition '=' 98 %
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Residual Activity '=' 74 %
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Residual Activity '=' 88 %
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Residual Activity '=' 91 %
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Residual Activity '=' 126 %
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Residual Activity '=' 107 %
P43250 BXGT010372 G protein-coupled receptor kinase 6 reviewed Kinase GRK6 Residual Activity '=' 109 %
P14635 BXGT008031 G2/mitotic-specific cyclin-B1 reviewed Enzyme modulator CCNB1 Residual Activity '=' 101 %
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Residual Activity '=' 101 %
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Residual Activity '=' 92 %
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Residual Activity '=' 27 %
O96020 BXGT005416 G1/S-specific cyclin-E2 reviewed Enzyme modulator CCNE2 Residual Activity '=' 108 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 108 %
P24864 BXGT009000 G1/S-specific cyclin-E1 reviewed Enzyme modulator CCNE1 Residual Activity '=' 108 %
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Residual Activity '=' 95 %
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Residual Activity '=' 114 %
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Residual Activity '=' 105 %
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Residual Activity '=' 78 %
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Ki '>' 5011 nM
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Ki '>' 3981 nM
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Residual Activity '=' 43 %
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Residual Activity '=' 117 %
P78362 BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 Residual Activity '=' 76 %
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Residual Activity '=' 79 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Residual Activity '=' -1 %
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Activity '=' 99 %
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Activity '=' 91 %
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Thermal melting change '=' 0 degrees C
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Thermal melting change '=' 0 degrees C
P35590 BXGT009854 Tyrosine-protein kinase receptor Tie-1 reviewed Kinase TIE1 Kd '>' 10000 nM
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Kd '>' 10000 nM
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Kd '>' 10000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Thermal melting change '=' 0 degrees C
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Thermal melting change '=' 0 degrees C
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Residual Activity '=' 45 %
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Residual Activity '=' 56 %
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Ki '>' 2511 nM
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Residual Activity '=' 106 %
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Residual Activity '=' 76 %
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Residual Activity '=' 127 %
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Residual Activity '=' 65 %
O00141 BXGT003882 Serine/threonine-protein kinase Sgk1 reviewed Kinase SGK1 Residual Activity '=' 99 %
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Residual Activity '=' 107 %
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Residual Activity '=' 104 %
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Residual Activity '=' 28 %
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Residual Activity '=' 82 %
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Kd '>' 10000 nM
Q16816 BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 Kd '>' 10000 nM
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Residual Activity '=' 77 %
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Residual Activity '=' 102 %
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 IC50 - - -
Q92830 BXGT019379 Histone acetyltransferase KAT2A reviewed - KAT2A Potency - 631 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 9 nM
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Thermal melting change '=' 1 degrees C
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Residual Activity '=' 87 %
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Residual Activity '=' 112 %
Q9BVS4 BXGT020147 Serine/threonine-protein kinase RIO2 reviewed Kinase RIOK2 Thermal melting change '=' 0 degrees C
Q96KB5 BXGT019685 Lymphokine-activated killer T-cell-originated protein kinase reviewed Kinase PBK Thermal melting change '=' 0 degrees C
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Thermal melting change '=' 0 degrees C
O95747 BXGT005393 Serine/threonine-protein kinase OSR1 reviewed Kinase OXSR1 Thermal melting change '=' 0 degrees C
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Residual Activity '=' 95 %
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Residual Activity '=' 93 %
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Residual Activity '=' 99 %
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Residual Activity '=' 107 %
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 IC50 '=' 9 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 28 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Thermal melting change '=' 2 degrees C
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Thermal melting change '=' 0 degrees C
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Thermal melting change '=' 4 degrees C
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Thermal melting change '=' 0 degrees C
Q00532 BXGT012532 Cyclin-dependent kinase-like 1 reviewed Kinase CDKL1 Thermal melting change '=' 0 degrees C
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Thermal melting change '=' 10 degrees C
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Residual Activity '=' 112 %
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Residual Activity '=' 105 %
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Residual Activity '=' 85 %
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Residual Activity '=' 106 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Residual Activity '=' 45 %
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Residual Activity '=' 93 %
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Inhibition '=' 0 %
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Inhibition '=' 89 %
P78396 BXGT011842 Cyclin-A1 reviewed Enzyme modulator CCNA1 Residual Activity '=' 95 %
P20248 BXGT008554 Cyclin-A2 reviewed Enzyme modulator CCNA2 Residual Activity '=' 95 %
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Residual Activity '=' 95 %
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Kd '>' 10000 nM
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Kd '>' 10000 nM
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Residual Activity '=' 109 %
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Residual Activity '=' 102 %
P51946 BXGT010907 Cyclin-H reviewed Enzyme modulator CCNH Residual Activity '=' 102 %
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Residual Activity '=' 109 %
Q9UGI9 BXGT021682 5'-AMP-activated protein kinase subunit gamma-3 reviewed Enzyme modulator PRKAG3 Residual Activity '=' 86 %
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Residual Activity '=' 86 %
Q9Y478 BXGT022271 5'-AMP-activated protein kinase subunit beta-1 reviewed Kinase PRKAB1 Residual Activity '=' 86 %
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Residual Activity '=' 86 %
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Residual Activity '=' 86 %
O43741 BXGT004620 5'-AMP-activated protein kinase subunit beta-2 reviewed Enzyme modulator PRKAB2 Residual Activity '=' 86 %
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Residual Activity '=' 86 %
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D IC50 '=' 188 nM
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Thermal melting change '=' 0 degrees C
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Thermal melting change '=' 0 degrees C
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Thermal melting change '=' 0 degrees C
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Thermal melting change '=' 1 degrees C
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Thermal melting change '=' 1 degrees C
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Residual Activity '=' 100 %
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Residual Activity '=' 95 %
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Residual Activity '=' 104 %
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Residual Activity '=' 98 %
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Residual Activity '=' 105 %
Q9UPE1 BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 Residual Activity '=' 120 %
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Residual Activity '=' 76 %
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Residual Activity '=' 45 %
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 IC50 '>' 100000 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Inhibition - - -
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Inhibition - - -
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Inhibition - - -
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Thermal melting change '=' 0 degrees C
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Residual Activity '=' 95 %
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Residual Activity '=' 98 %
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Potency - 17290 nM
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Residual Activity '=' 90 %
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Residual Activity '=' 86 %
O60885 BXGT004906 Bromodomain-containing protein 4 reviewed Epigenetic regulator BRD4 IC50 '=' 3400 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Residual Activity '=' 42 %
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Residual Activity '=' 79 %
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Residual Activity '=' 117 %
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Residual Activity '=' 75 %
O00506 BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 Thermal melting change '=' 0 degrees C
Q58F21 BXGT015228 Bromodomain testis-specific protein reviewed Epigenetic regulator BRDT IC50 '=' 20000 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Residual Activity '=' 97 %
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Residual Activity '=' 99 %
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Residual Activity '=' 107 %
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Residual Activity '=' 115 %
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Residual Activity '=' 113 %
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Residual Activity '=' 99 %
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Residual Activity '=' 68 %
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 IC50 '>' 100000 nM
O15296 BXGT004148 Arachidonate 15-lipoxygenase B reviewed Enzyme ALOX15B Potency - 7943 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 IC50 '=' 300 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 IC50 '=' 300 nM
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF05043 mammea siamensis mammea siamensis Medicinal Plant
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease