| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Kd |
- |
- |
- |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Kd |
- |
- |
- |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
- |
- |
- |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Kd |
- |
- |
- |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Kd |
- |
- |
- |
| P08631 |
BXGT006801 |
Tyrosine-protein kinase HCK |
reviewed |
Kinase |
HCK |
Ki |
'=' |
2511 |
nM |
| P22607 |
BXGT008784 |
Fibroblast growth factor receptor 3 |
reviewed |
Kinase |
FGFR3 |
Ki |
'>' |
1995 |
nM |
| Q7KZI7 |
BXGT016990 |
Serine/threonine-protein kinase MARK2 |
reviewed |
Kinase |
MARK2 |
Ki |
'>' |
7943 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Ki |
'=' |
1995 |
nM |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Ki |
'>' |
7943 |
nM |
| O14757 |
BXGT004092 |
Serine/threonine-protein kinase Chk1 |
reviewed |
Kinase |
CHEK1 |
Ki |
'>' |
6309 |
nM |
| Q9Y463 |
BXGT022269 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
reviewed |
Kinase |
DYRK1B |
Ki |
'>' |
2511 |
nM |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Kd |
'=' |
920 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
100 |
% |
| Q9Y4K4 |
BXGT022282 |
Mitogen-activated protein kinase kinase kinase kinase 5 |
reviewed |
Kinase |
MAP4K5 |
Ki |
'=' |
1584 |
nM |
| Q05513 |
BXGT012820 |
Protein kinase C zeta type |
reviewed |
Kinase |
PRKCZ |
Ki |
'>' |
7943 |
nM |
| P36894 |
BXGT009939 |
Bone morphogenetic protein receptor type-1A |
reviewed |
Kinase |
BMPR1A |
Kd |
'>' |
10000 |
nM |
| Q00532 |
BXGT012532 |
Cyclin-dependent kinase-like 1 |
reviewed |
Kinase |
CDKL1 |
Kd |
'>' |
10000 |
nM |
| Q9UM73 |
BXGT021773 |
ALK tyrosine kinase receptor |
reviewed |
Kinase |
ALK |
Kd |
'>' |
10000 |
nM |
| O75747 |
BXGT005149 |
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma |
reviewed |
Kinase |
PIK3C2G |
Kd |
'>' |
10000 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
Kd |
'>' |
10000 |
nM |
| P09769 |
BXGT006917 |
Tyrosine-protein kinase Fgr |
reviewed |
Kinase |
FGR |
Kd |
'=' |
2600 |
nM |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Kd |
'=' |
470 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
Kd |
'>' |
10000 |
nM |
| P24723 |
BXGT008989 |
Protein kinase C eta type |
reviewed |
Kinase |
PRKCH |
Kd |
'>' |
10000 |
nM |
| Q13237 |
BXGT013331 |
cGMP-dependent protein kinase 2 |
reviewed |
Kinase |
PRKG2 |
Kd |
'>' |
10000 |
nM |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Kd |
'>' |
10000 |
nM |
| O14578 |
BXGT004072 |
Citron Rho-interacting kinase |
reviewed |
Kinase |
CIT |
Kd |
'=' |
1300 |
nM |
| Q15208 |
BXGT013550 |
Serine/threonine-protein kinase 38 |
reviewed |
Kinase |
STK38 |
Kd |
'>' |
10000 |
nM |
| P57058 |
BXGT011209 |
Hormonally up-regulated neu tumor-associated kinase |
reviewed |
Kinase |
HUNK |
Kd |
'>' |
10000 |
nM |
| Q9BZL6 |
BXGT020199 |
Serine/threonine-protein kinase D2 |
reviewed |
Kinase |
PRKD2 |
Kd |
'>' |
10000 |
nM |
| Q9BX84 |
BXGT020161 |
Transient receptor potential cation channel subfamily M member 6 |
reviewed |
Kinase |
TRPM6 |
Kd |
'>' |
10000 |
nM |
| Q00537 |
BXGT012536 |
Cyclin-dependent kinase 17 |
reviewed |
Kinase |
CDK17 |
Kd |
'>' |
10000 |
nM |
| P31751 |
BXGT009576 |
RAC-beta serine/threonine-protein kinase |
reviewed |
Kinase |
AKT2 |
Kd |
'>' |
10000 |
nM |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Kd |
'>' |
10000 |
nM |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Kd |
'=' |
3200 |
nM |
| P45985 |
BXGT010496 |
Dual specificity mitogen-activated protein kinase kinase 4 |
reviewed |
Kinase |
MAP2K4 |
Kd |
'>' |
10000 |
nM |
| Q9NWZ3 |
BXGT021239 |
Interleukin-1 receptor-associated kinase 4 |
reviewed |
Kinase |
IRAK4 |
Ki |
'=' |
1000 |
nM |
| Q14012 |
BXGT013437 |
Calcium/calmodulin-dependent protein kinase type 1 |
reviewed |
Kinase |
CAMK1 |
Ki |
'>' |
6309 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
Ki |
'>' |
6309 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
22 |
nM |
| Q9NWZ3 |
BXGT021239 |
Interleukin-1 receptor-associated kinase 4 |
reviewed |
Kinase |
IRAK4 |
Kd apparent |
'>' |
30000 |
nM |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Ki |
'>' |
7943 |
nM |
| Q96SB4 |
BXGT019740 |
SRSF protein kinase 1 |
reviewed |
Kinase |
SRPK1 |
Ki |
'>' |
7943 |
nM |
| Q05655 |
BXGT012832 |
Protein kinase C delta type |
reviewed |
Kinase |
PRKCD |
Ki |
'>' |
7943 |
nM |
| P27448 |
BXGT009183 |
MAP/microtubule affinity-regulating kinase 3 |
reviewed |
Kinase |
MARK3 |
Ki |
'>' |
6309 |
nM |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Ki |
'>' |
3162 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
IC50 |
'=' |
133000 |
nM |
| Q13464 |
BXGT013357 |
Rho-associated protein kinase 1 |
reviewed |
Kinase |
ROCK1 |
Ki |
'>' |
6309 |
nM |
| Q16644 |
BXGT013647 |
MAP kinase-activated protein kinase 3 |
reviewed |
Kinase |
MAPKAPK3 |
Ki |
'>' |
10000 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Ki |
'>' |
1584 |
nM |
| P41240 |
BXGT010242 |
Tyrosine-protein kinase CSK |
reviewed |
Kinase |
CSK |
Kd |
- |
- |
- |
| P54764 |
BXGT011078 |
Ephrin type-A receptor 4 |
reviewed |
Kinase |
EPHA4 |
Kd |
- |
- |
- |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Ki |
'=' |
1258 |
nM |
| P48729 |
BXGT010655 |
Casein kinase I isoform alpha |
reviewed |
Kinase |
CSNK1A1 |
Ki |
'>' |
5011 |
nM |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Ki |
'>' |
3981 |
nM |
| P51451 |
BXGT010848 |
Tyrosine-protein kinase Blk |
reviewed |
Kinase |
BLK |
Ki |
'=' |
1000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Ki |
'>' |
2511 |
nM |
| P51817 |
BXGT010895 |
cAMP-dependent protein kinase catalytic subunit PRKX |
reviewed |
Kinase |
PRKX |
Ki |
'>' |
1584 |
nM |
| O75676 |
BXGT005144 |
Ribosomal protein S6 kinase alpha-4 |
reviewed |
Kinase |
RPS6KA4 |
Ki |
'>' |
1584 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
Ki |
'>' |
7943 |
nM |
| P50613 |
BXGT010815 |
Cyclin-dependent kinase 7 |
reviewed |
Kinase |
CDK7 |
Ki |
'>' |
3981 |
nM |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Ki |
'>' |
3981 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
39810 |
nM |
| Q9UHD2 |
BXGT021697 |
Serine/threonine-protein kinase TBK1 |
reviewed |
Kinase |
TBK1 |
Ki |
'>' |
3162 |
nM |
| Q02779 |
BXGT012670 |
Mitogen-activated protein kinase kinase kinase 10 |
reviewed |
Kinase |
MAP3K10 |
Ki |
'>' |
3162 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
33 |
nM |
| Q13976 |
BXGT013409 |
cGMP-dependent protein kinase 1 |
reviewed |
Kinase |
PRKG1 |
Ki |
'>' |
1995 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
639 |
nM |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| O95747 |
BXGT005393 |
Serine/threonine-protein kinase OSR1 |
reviewed |
Kinase |
OXSR1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
5 |
degrees C |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
Ki |
'>' |
7943 |
nM |
| Q13188 |
BXGT013324 |
Serine/threonine-protein kinase 3 |
reviewed |
Kinase |
STK3 |
Ki |
'>' |
7943 |
nM |
| Q07912 |
BXGT012947 |
Activated CDC42 kinase 1 |
reviewed |
Kinase |
TNK2 |
Kd |
- |
- |
- |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Kd |
- |
- |
- |
| P54756 |
BXGT011074 |
Ephrin type-A receptor 5 |
reviewed |
Kinase |
EPHA5 |
Kd |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
1 |
nM |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Kd |
- |
- |
- |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Ki |
'>' |
6309 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
2815 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
2815 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2815 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
2815 |
nM |
| Q16513 |
BXGT013632 |
Serine/threonine-protein kinase N2 |
reviewed |
Kinase |
PKN2 |
Ki |
'>' |
7943 |
nM |
| Q9H093 |
BXGT020433 |
NUAK family SNF1-like kinase 2 |
reviewed |
Kinase |
NUAK2 |
Kd |
'>' |
10000 |
nM |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
Kd |
'=' |
530 |
nM |
| Q96D53 |
BXGT019637 |
Atypical kinase COQ8B, mitochondrial |
reviewed |
Kinase |
COQ8B |
Kd |
'>' |
10000 |
nM |
| P57059 |
BXGT011210 |
Serine/threonine-protein kinase SIK1 |
reviewed |
- |
SIK1 |
Kd |
'>' |
10000 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd |
'=' |
4300 |
nM |
| Q14680 |
BXGT013499 |
Maternal embryonic leucine zipper kinase |
reviewed |
Kinase |
MELK |
Kd |
'>' |
10000 |
nM |
| O14976 |
BXGT004118 |
Cyclin-G-associated kinase |
reviewed |
Kinase |
GAK |
Kd |
'=' |
13 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd |
'>' |
10000 |
nM |
| O14965 |
BXGT004117 |
Aurora kinase A |
reviewed |
Kinase |
AURKA |
Kd |
'>' |
10000 |
nM |
| P04629 |
BXGT006239 |
High affinity nerve growth factor receptor |
reviewed |
Kinase |
NTRK1 |
Kd |
'>' |
10000 |
nM |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Kd |
'>' |
10000 |
nM |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Kd |
'>' |
10000 |
nM |
| P21127 |
BXGT008623 |
Cyclin-dependent kinase 11B |
reviewed |
Kinase |
CDK11B |
Kd |
'>' |
10000 |
nM |
| Q9BWU1 |
BXGT020156 |
Cyclin-dependent kinase 19 |
reviewed |
Kinase |
CDK19 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
0 |
nM |
| Q9Y616 |
BXGT022313 |
Interleukin-1 receptor-associated kinase 3 |
reviewed |
Kinase |
IRAK3 |
Kd |
'=' |
1500 |
nM |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
Kd |
'>' |
10000 |
nM |
| Q59H18 |
BXGT015278 |
Serine/threonine-protein kinase TNNI3K |
reviewed |
- |
TNNI3K |
Kd |
'>' |
10000 |
nM |
| P08069 |
BXGT006723 |
Insulin-like growth factor 1 receptor |
reviewed |
Kinase |
IGF1R |
Kd |
'>' |
10000 |
nM |
| Q86YV6 |
BXGT017636 |
Myosin light chain kinase family member 4 |
reviewed |
- |
MYLK4 |
Kd |
'>' |
10000 |
nM |
| Q02763 |
BXGT012667 |
Angiopoietin-1 receptor |
reviewed |
Kinase |
TEK |
Kd |
'>' |
10000 |
nM |
| Q9BYT3 |
BXGT020189 |
Serine/threonine-protein kinase 33 |
reviewed |
Kinase |
STK33 |
Kd |
'>' |
10000 |
nM |
| P16591 |
BXGT008246 |
Tyrosine-protein kinase Fer |
reviewed |
Kinase |
FER |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
35 |
nM |
| P50613 |
BXGT010815 |
Cyclin-dependent kinase 7 |
reviewed |
Kinase |
CDK7 |
Kd apparent |
'>' |
30000 |
nM |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Kd apparent |
'>' |
30000 |
nM |
| Q8TBX8 |
BXGT018791 |
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma |
reviewed |
Kinase |
PIP4K2C |
Kd apparent |
'>' |
30000 |
nM |
| P12268 |
BXGT007783 |
Inosine-5'-monophosphate dehydrogenase 2 |
reviewed |
Enzyme |
IMPDH2 |
Kd apparent |
'>' |
30000 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Kd |
'>' |
10000 |
nM |
| P29323 |
BXGT009334 |
Ephrin type-B receptor 2 |
reviewed |
Kinase |
EPHB2 |
Kd apparent |
'>' |
30000 |
nM |
| Q99640 |
BXGT019944 |
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
reviewed |
Kinase |
PKMYT1 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
0 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
1100 |
nM |
| Q15418 |
BXGT013569 |
Ribosomal protein S6 kinase alpha-1 |
reviewed |
Kinase |
RPS6KA1 |
Kd |
'>' |
10000 |
nM |
| O94806 |
BXGT005335 |
Serine/threonine-protein kinase D3 |
reviewed |
Kinase |
PRKD3 |
Kd |
'>' |
10000 |
nM |
| P54753 |
BXGT011073 |
Ephrin type-B receptor 3 |
reviewed |
Kinase |
EPHB3 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
1 |
nM |
| P22694 |
BXGT008797 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
Kinase |
PRKACB |
Kd |
'>' |
10000 |
nM |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9P2K8 |
BXGT021302 |
eIF-2-alpha kinase GCN2 |
reviewed |
- |
EIF2AK4 |
Kd |
'>' |
10000 |
nM |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Kd |
'>' |
10000 |
nM |
| P46734 |
BXGT010537 |
Dual specificity mitogen-activated protein kinase kinase 3 |
reviewed |
Kinase |
MAP2K3 |
Kd |
'>' |
10000 |
nM |
| O60674 |
BXGT004892 |
Tyrosine-protein kinase JAK2 |
reviewed |
Kinase |
JAK2 |
Kd |
'>' |
10000 |
nM |
| Q9BXA7 |
BXGT020164 |
Testis-specific serine/threonine-protein kinase 1 |
reviewed |
Kinase |
TSSK1B |
Kd |
'>' |
10000 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1 |
nM |
| Q92630 |
BXGT019360 |
Dual specificity tyrosine-phosphorylation-regulated kinase 2 |
reviewed |
Kinase |
DYRK2 |
Kd |
'>' |
10000 |
nM |
| P54764 |
BXGT011078 |
Ephrin type-A receptor 4 |
reviewed |
Kinase |
EPHA4 |
Kd |
'>' |
10000 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Kd |
'>' |
10000 |
nM |
| O75116 |
BXGT005100 |
Rho-associated protein kinase 2 |
reviewed |
Kinase |
ROCK2 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
2700 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
0 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Inhibition |
'=' |
28 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
4000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
240 |
nM |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Ki |
'=' |
630 |
nM |
| Q13153 |
BXGT013319 |
Serine/threonine-protein kinase PAK 1 |
reviewed |
Kinase |
PAK1 |
Ki |
'>' |
10000 |
nM |
| P41743 |
BXGT010270 |
Protein kinase C iota type |
reviewed |
Kinase |
PRKCI |
Ki |
'>' |
5011 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
941 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
941 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
941 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
941 |
nM |
| Q9P2R7 |
BXGT021304 |
Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial |
reviewed |
Enzyme |
SUCLA2 |
Kd apparent |
'>' |
30000 |
nM |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Kd apparent |
'>' |
30000 |
nM |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Kd apparent |
'>' |
30000 |
nM |
| P53671 |
BXGT011009 |
LIM domain kinase 2 |
reviewed |
Kinase |
LIMK2 |
Kd apparent |
'>' |
30000 |
nM |
| O00764 |
BXGT003948 |
Pyridoxal kinase |
reviewed |
Kinase |
PDXK |
Kd apparent |
'>' |
30000 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Kd |
'>' |
10000 |
nM |
| Q07912 |
BXGT012947 |
Activated CDC42 kinase 1 |
reviewed |
Kinase |
TNK2 |
Kd |
'>' |
10000 |
nM |
| Q8N4C8 |
BXGT018510 |
Misshapen-like kinase 1 |
reviewed |
Kinase |
MINK1 |
Kd |
'=' |
1800 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Kd |
'=' |
410 |
nM |
| Q9BUB5 |
BXGT020133 |
MAP kinase-interacting serine/threonine-protein kinase 1 |
reviewed |
Kinase |
MKNK1 |
Kd |
'=' |
290 |
nM |
| O00238 |
BXGT003900 |
Bone morphogenetic protein receptor type-1B |
reviewed |
Kinase |
BMPR1B |
Kd |
'>' |
10000 |
nM |
| P49336 |
BXGT010697 |
Cyclin-dependent kinase 8 |
reviewed |
Kinase |
CDK8 |
Kd |
'>' |
10000 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Kd |
'>' |
10000 |
nM |
| P07332 |
BXGT006601 |
Tyrosine-protein kinase Fes/Fps |
reviewed |
Kinase |
FES |
Kd |
'>' |
10000 |
nM |
| P51956 |
BXGT010909 |
Serine/threonine-protein kinase Nek3 |
reviewed |
Kinase |
NEK3 |
Kd |
'>' |
10000 |
nM |
| O00750 |
BXGT003943 |
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta |
reviewed |
Kinase |
PIK3C2B |
Kd |
'>' |
10000 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Kd |
'>' |
10000 |
nM |
| P41743 |
BXGT010270 |
Protein kinase C iota type |
reviewed |
Kinase |
PRKCI |
Kd |
'>' |
10000 |
nM |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Kd |
'>' |
10000 |
nM |
| P51957 |
BXGT010910 |
Serine/threonine-protein kinase Nek4 |
reviewed |
Kinase |
NEK4 |
Kd |
'>' |
10000 |
nM |
| P42680 |
BXGT010329 |
Tyrosine-protein kinase Tec |
reviewed |
Kinase |
TEC |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
98 |
% |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
IC50 |
'=' |
2000 |
nM |
| P51957 |
BXGT010910 |
Serine/threonine-protein kinase Nek4 |
reviewed |
Kinase |
NEK4 |
Ki |
'>' |
6309 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Thermal melting change |
'=' |
0 |
degrees C |
| Q8IV63 |
BXGT018341 |
Inactive serine/threonine-protein kinase VRK3 |
reviewed |
Kinase |
VRK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q8IW41 |
BXGT018352 |
MAP kinase-activated protein kinase 5 |
reviewed |
Kinase |
MAPKAPK5 |
Ki |
'>' |
1584 |
nM |
| Q9Y463 |
BXGT022269 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1B |
reviewed |
Kinase |
DYRK1B |
Kd |
'>' |
10000 |
nM |
| O75676 |
BXGT005144 |
Ribosomal protein S6 kinase alpha-4 |
reviewed |
Kinase |
RPS6KA4 |
Kd |
'>' |
10000 |
nM |
| P42685 |
BXGT010332 |
Tyrosine-protein kinase FRK |
reviewed |
Kinase |
FRK |
Kd |
'=' |
2000 |
nM |
| P53667 |
BXGT011008 |
LIM domain kinase 1 |
reviewed |
Kinase |
LIMK1 |
Kd |
'>' |
10000 |
nM |
| Q02779 |
BXGT012670 |
Mitogen-activated protein kinase kinase kinase 10 |
reviewed |
Kinase |
MAP3K10 |
Kd |
'>' |
10000 |
nM |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Kd |
'>' |
10000 |
nM |
| Q13177 |
BXGT013323 |
Serine/threonine-protein kinase PAK 2 |
reviewed |
Kinase |
PAK2 |
Kd |
'>' |
10000 |
nM |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Kd |
'>' |
10000 |
nM |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Kd |
'>' |
10000 |
nM |
| Q15835 |
BXGT013606 |
Rhodopsin kinase |
reviewed |
Kinase |
GRK1 |
Kd |
'>' |
10000 |
nM |
| Q96SB4 |
BXGT019740 |
SRSF protein kinase 1 |
reviewed |
Kinase |
SRPK1 |
Kd |
'>' |
10000 |
nM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Ki |
'>' |
3981 |
nM |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Kd |
'>' |
10000 |
nM |
| Q96PF2 |
BXGT019708 |
Testis-specific serine/threonine-protein kinase 2 |
reviewed |
Kinase |
TSSK2 |
Ki |
'>' |
1584 |
nM |
| Q9NR20 |
BXGT021176 |
Dual specificity tyrosine-phosphorylation-regulated kinase 4 |
reviewed |
Kinase |
DYRK4 |
Ki |
'>' |
7943 |
nM |
| Q04771 |
BXGT012783 |
Activin receptor type-1 |
reviewed |
Kinase |
ACVR1 |
Ki |
'>' |
3981 |
nM |
| P29597 |
BXGT009367 |
Non-receptor tyrosine-protein kinase TYK2 |
reviewed |
Kinase |
TYK2 |
Kd |
'>' |
10000 |
nM |
| Q15349 |
BXGT013558 |
Ribosomal protein S6 kinase alpha-2 |
reviewed |
Kinase |
RPS6KA2 |
Kd |
'>' |
10000 |
nM |
| Q9UF33 |
BXGT021676 |
Ephrin type-A receptor 6 |
reviewed |
Kinase |
EPHA6 |
Kd |
'=' |
590 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Ki |
'>' |
7943 |
nM |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Ki |
'=' |
2511 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
Inhibition |
- |
- |
- |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Inhibition |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Inhibition |
- |
- |
- |
| Q8IW41 |
BXGT018352 |
MAP kinase-activated protein kinase 5 |
reviewed |
Kinase |
MAPKAPK5 |
Kd |
'>' |
10000 |
nM |
| O15075 |
BXGT004124 |
Serine/threonine-protein kinase DCLK1 |
reviewed |
Kinase |
DCLK1 |
Ki |
'>' |
10000 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Ki |
'>' |
5011 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Potency |
'=' |
1122 |
nM |
| P49336 |
BXGT010697 |
Cyclin-dependent kinase 8 |
reviewed |
Kinase |
CDK8 |
Ki |
'>' |
3981 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
20 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
Activity |
- |
- |
- |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Activity |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Activity |
- |
- |
- |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Activity |
- |
- |
- |
| Q9Y6R4 |
BXGT022340 |
Mitogen-activated protein kinase kinase kinase 4 |
reviewed |
Kinase |
MAP3K4 |
Kd |
- |
- |
- |
| Q9HBH9 |
BXGT020521 |
MAP kinase-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
MKNK2 |
Kd |
'=' |
360 |
nM |
| Q9UIK4 |
BXGT021720 |
Death-associated protein kinase 2 |
reviewed |
Kinase |
DAPK2 |
Kd |
- |
- |
- |
| Q15349 |
BXGT013558 |
Ribosomal protein S6 kinase alpha-2 |
reviewed |
Kinase |
RPS6KA2 |
Kd |
- |
- |
- |
| P29317 |
BXGT009331 |
Ephrin type-A receptor 2 |
reviewed |
Kinase |
EPHA2 |
Kd |
- |
- |
- |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
- |
- |
- |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Thermal melting change |
'=' |
-1 |
degrees C |
| O14965 |
BXGT004117 |
Aurora kinase A |
reviewed |
Kinase |
AURKA |
Ki |
'>' |
3162 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
10480 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
10480 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
10480 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
10480 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
476 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Thermal melting change |
'=' |
0 |
degrees C |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Thermal melting change |
'=' |
7 |
degrees C |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
101 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
14 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
4 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
25118 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Kd |
'>' |
10000 |
nM |
| Q8N568 |
BXGT018516 |
Serine/threonine-protein kinase DCLK2 |
reviewed |
Kinase |
DCLK2 |
Kd |
'>' |
10000 |
nM |
| O75460 |
BXGT005127 |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
reviewed |
Kinase |
ERN1 |
Kd |
'>' |
10000 |
nM |
| P51813 |
BXGT010894 |
Cytoplasmic tyrosine-protein kinase BMX |
reviewed |
Kinase |
BMX |
Kd |
'>' |
10000 |
nM |
| P48729 |
BXGT010655 |
Casein kinase I isoform alpha |
reviewed |
Kinase |
CSNK1A1 |
Kd |
'>' |
10000 |
nM |
| P35916 |
BXGT009881 |
Vascular endothelial growth factor receptor 3 |
reviewed |
Kinase |
FLT4 |
Kd |
'>' |
10000 |
nM |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Kd |
'>' |
10000 |
nM |
| Q99759 |
BXGT019960 |
Mitogen-activated protein kinase kinase kinase 3 |
reviewed |
Kinase |
MAP3K3 |
Kd |
'=' |
2100 |
nM |
| Q13164 |
BXGT013322 |
Mitogen-activated protein kinase 7 |
reviewed |
Kinase |
MAPK7 |
Kd |
'>' |
10000 |
nM |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Kd |
'>' |
10000 |
nM |
| P54756 |
BXGT011074 |
Ephrin type-A receptor 5 |
reviewed |
Kinase |
EPHA5 |
Kd |
'>' |
10000 |
nM |
| Q2M2I8 |
BXGT014130 |
AP2-associated protein kinase 1 |
reviewed |
Kinase |
AAK1 |
Kd |
'>' |
10000 |
nM |
| P50613 |
BXGT010815 |
Cyclin-dependent kinase 7 |
reviewed |
Kinase |
CDK7 |
Kd |
'>' |
10000 |
nM |
| P07333 |
BXGT006602 |
Macrophage colony-stimulating factor 1 receptor |
reviewed |
Kinase |
CSF1R |
Selectivity |
'=' |
0 |
- |
| Q08881 |
BXGT013012 |
Tyrosine-protein kinase ITK/TSK |
reviewed |
Kinase |
ITK |
Kd |
'>' |
10000 |
nM |
| Q15831 |
BXGT013604 |
Serine/threonine-protein kinase STK11 |
reviewed |
Kinase |
STK11 |
Kd |
'>' |
10000 |
nM |
| P53667 |
BXGT011008 |
LIM domain kinase 1 |
reviewed |
Kinase |
LIMK1 |
Ki |
'=' |
3981 |
nM |
| Q14012 |
BXGT013437 |
Calcium/calmodulin-dependent protein kinase type 1 |
reviewed |
Kinase |
CAMK1 |
Kd |
'>' |
10000 |
nM |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Ki |
'>' |
6309 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ratio IC50 |
'=' |
12 |
- |
| Q16659 |
BXGT013652 |
Mitogen-activated protein kinase 6 |
reviewed |
Kinase |
MAPK6 |
Kd |
'=' |
1600 |
nM |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Ki |
'>' |
7943 |
nM |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
Ki |
'>' |
398 |
nM |
| Q96KB5 |
BXGT019685 |
Lymphokine-activated killer T-cell-originated protein kinase |
reviewed |
Kinase |
PBK |
Thermal melting change |
'=' |
0 |
degrees C |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
Ki |
'>' |
3162 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Inhibition |
- |
- |
- |
| Q04771 |
BXGT012783 |
Activin receptor type-1 |
reviewed |
Kinase |
ACVR1 |
Kd |
'>' |
10000 |
nM |
| O14730 |
BXGT004085 |
Serine/threonine-protein kinase RIO3 |
reviewed |
Kinase |
RIOK3 |
Kd |
'>' |
10000 |
nM |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Kd |
'>' |
10000 |
nM |
| Q96PY6 |
BXGT019712 |
Serine/threonine-protein kinase Nek1 |
reviewed |
Kinase |
NEK1 |
Kd |
'>' |
10000 |
nM |
| Q06187 |
BXGT012860 |
Tyrosine-protein kinase BTK |
reviewed |
Kinase |
BTK |
Kd |
'>' |
10000 |
nM |
| P50750 |
BXGT010818 |
Cyclin-dependent kinase 9 |
reviewed |
Kinase |
CDK9 |
Kd |
'>' |
10000 |
nM |
| P80192 |
BXGT011883 |
Mitogen-activated protein kinase kinase kinase 9 |
reviewed |
Kinase |
MAP3K9 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'>' |
10000 |
nM |
| O15146 |
BXGT004131 |
Muscle, skeletal receptor tyrosine-protein kinase |
reviewed |
Kinase |
MUSK |
Kd |
'>' |
10000 |
nM |
| Q15746 |
BXGT013591 |
Myosin light chain kinase, smooth muscle |
reviewed |
Kinase |
MYLK |
Kd |
'>' |
10000 |
nM |
| Q8N5S9 |
BXGT018520 |
Calcium/calmodulin-dependent protein kinase kinase 1 |
reviewed |
Kinase |
CAMKK1 |
Kd |
'>' |
10000 |
nM |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Kd |
'>' |
10000 |
nM |
| Q9UIK4 |
BXGT021720 |
Death-associated protein kinase 2 |
reviewed |
Kinase |
DAPK2 |
Kd |
'>' |
10000 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Inhibition |
- |
- |
- |
| P33981 |
BXGT009744 |
Dual specificity protein kinase TTK |
reviewed |
Kinase |
TTK |
Kd |
'>' |
10000 |
nM |
| Q9H1R3 |
BXGT020446 |
Myosin light chain kinase 2, skeletal/cardiac muscle |
reviewed |
Kinase |
MYLK2 |
Kd |
- |
- |
- |
| P09769 |
BXGT006917 |
Tyrosine-protein kinase Fgr |
reviewed |
Kinase |
FGR |
Kd |
- |
- |
- |
| P54762 |
BXGT011076 |
Ephrin type-B receptor 1 |
reviewed |
Kinase |
EPHB1 |
Kd |
'=' |
7300 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'<' |
1 |
nM |
| Q99755 |
BXGT019958 |
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha |
reviewed |
Kinase |
PIP5K1A |
Kd |
'>' |
10000 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Ki |
'>' |
3981 |
nM |
| Q96KB5 |
BXGT019685 |
Lymphokine-activated killer T-cell-originated protein kinase |
reviewed |
Kinase |
PBK |
Ki |
'>' |
10000 |
nM |
| P29317 |
BXGT009331 |
Ephrin type-A receptor 2 |
reviewed |
Kinase |
EPHA2 |
Ki |
'>' |
3162 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
Activity |
- |
- |
- |
| Q96L34 |
BXGT019689 |
MAP/microtubule affinity-regulating kinase 4 |
reviewed |
Kinase |
MARK4 |
Ki |
'>' |
5011 |
nM |
| P07333 |
BXGT006602 |
Macrophage colony-stimulating factor 1 receptor |
reviewed |
Kinase |
CSF1R |
Ki |
'>' |
2511 |
nM |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Kd |
- |
- |
- |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Kd |
- |
- |
- |
| O00418 |
BXGT003918 |
Eukaryotic elongation factor 2 kinase |
reviewed |
Kinase |
EEF2K |
Ki |
'>' |
3981 |
nM |
| P07948 |
BXGT006702 |
Tyrosine-protein kinase Lyn |
reviewed |
Kinase |
LYN |
Ki |
'=' |
158 |
nM |
| O15075 |
BXGT004124 |
Serine/threonine-protein kinase DCLK1 |
reviewed |
Kinase |
DCLK1 |
Kd |
'>' |
10000 |
nM |
| Q8TD19 |
BXGT018804 |
Serine/threonine-protein kinase Nek9 |
reviewed |
Kinase |
NEK9 |
Kd |
'>' |
10000 |
nM |
| Q16816 |
BXGT013673 |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
reviewed |
Kinase |
PHKG1 |
Kd |
'=' |
3700 |
nM |
| Q9NWZ3 |
BXGT021239 |
Interleukin-1 receptor-associated kinase 4 |
reviewed |
Kinase |
IRAK4 |
Kd |
'=' |
540 |
nM |
| Q9H2X6 |
BXGT020458 |
Homeodomain-interacting protein kinase 2 |
reviewed |
Kinase |
HIPK2 |
Kd |
'>' |
10000 |
nM |
| P49137 |
BXGT010680 |
MAP kinase-activated protein kinase 2 |
reviewed |
Kinase |
MAPKAPK2 |
Kd |
'>' |
10000 |
nM |
| Q9C098 |
BXGT020208 |
Serine/threonine-protein kinase DCLK3 |
reviewed |
Kinase |
DCLK3 |
Kd |
'=' |
2900 |
nM |
| P37023 |
BXGT009953 |
Serine/threonine-protein kinase receptor R3 |
reviewed |
Kinase |
ACVRL1 |
Kd |
'>' |
10000 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
IC50 |
'=' |
1100 |
nM |
| P54760 |
BXGT011075 |
Ephrin type-B receptor 4 |
reviewed |
Kinase |
EPHB4 |
IC50 |
'=' |
1000 |
nM |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'=' |
148000 |
nM |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Kd |
'=' |
2000 |
nM |
| P34947 |
BXGT009774 |
G protein-coupled receptor kinase 5 |
reviewed |
Kinase |
GRK5 |
Ki |
'>' |
3981 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Kd |
'>' |
10000 |
nM |
| Q8NFD2 |
BXGT018559 |
Ankyrin repeat and protein kinase domain-containing protein 1 |
reviewed |
Kinase |
ANKK1 |
Kd |
'>' |
10000 |
nM |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Kd |
- |
- |
- |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Kd |
- |
- |
- |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
Kd |
'>' |
10000 |
nM |
| Q14289 |
BXGT013459 |
Protein-tyrosine kinase 2-beta |
reviewed |
Kinase |
PTK2B |
Ki |
'>' |
1584 |
nM |
| O14965 |
BXGT004117 |
Aurora kinase A |
reviewed |
Kinase |
AURKA |
Kd |
- |
- |
- |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Kd |
- |
- |
- |
| Q8TD08 |
BXGT018803 |
Mitogen-activated protein kinase 15 |
reviewed |
Kinase |
MAPK15 |
Kd |
'>' |
10000 |
nM |
| Q15139 |
BXGT013546 |
Serine/threonine-protein kinase D1 |
reviewed |
Kinase |
PRKD1 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
10 |
nM |
| Q96L34 |
BXGT019689 |
MAP/microtubule affinity-regulating kinase 4 |
reviewed |
Kinase |
MARK4 |
Kd |
'>' |
10000 |
nM |
| O14976 |
BXGT004118 |
Cyclin-G-associated kinase |
reviewed |
Kinase |
GAK |
Kd |
'=' |
7 |
nM |
| Q92887 |
BXGT019389 |
Canalicular multispecific organic anion transporter 1 |
reviewed |
Transporter |
ABCC2 |
Activity |
'=' |
74 |
% |
| P25779 |
BXGT009067 |
Cruzipain |
reviewed |
- |
|
IC50 |
'=' |
88000 |
nM |
| P16591 |
BXGT008246 |
Tyrosine-protein kinase Fer |
reviewed |
Kinase |
FER |
Kd |
- |
- |
- |
| Q99640 |
BXGT019944 |
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
reviewed |
Kinase |
PKMYT1 |
Kd |
- |
- |
- |
| P42685 |
BXGT010332 |
Tyrosine-protein kinase FRK |
reviewed |
Kinase |
FRK |
Kd |
- |
- |
- |
| P22607 |
BXGT008784 |
Fibroblast growth factor receptor 3 |
reviewed |
Kinase |
FGFR3 |
Kd |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Kd |
'=' |
3500 |
nM |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Kd |
'=' |
800 |
nM |
| P07948 |
BXGT006702 |
Tyrosine-protein kinase Lyn |
reviewed |
Kinase |
LYN |
Kd |
'=' |
990 |
nM |
| P23443 |
BXGT008866 |
Ribosomal protein S6 kinase beta-1 |
reviewed |
Kinase |
RPS6KB1 |
Kd |
'>' |
10000 |
nM |
| Q8IWQ3 |
BXGT018355 |
Serine/threonine-protein kinase BRSK2 |
reviewed |
Kinase |
BRSK2 |
Kd |
'>' |
10000 |
nM |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Kd |
'>' |
10000 |
nM |
| Q9H4B4 |
BXGT020474 |
Serine/threonine-protein kinase PLK3 |
reviewed |
Kinase |
PLK3 |
Kd |
'>' |
10000 |
nM |
| O00329 |
BXGT003909 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform |
reviewed |
Kinase |
PIK3CD |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
40 |
nM |
| Q05655 |
BXGT012832 |
Protein kinase C delta type |
reviewed |
Kinase |
PRKCD |
Kd |
'>' |
10000 |
nM |
| Q6DT37 |
BXGT016259 |
Serine/threonine-protein kinase MRCK gamma |
reviewed |
Kinase |
CDC42BPG |
Kd |
'>' |
10000 |
nM |
| Q9H3Y6 |
BXGT020468 |
Tyrosine-protein kinase Srms |
reviewed |
Kinase |
SRMS |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
2 |
nM |
| O60674 |
BXGT004892 |
Tyrosine-protein kinase JAK2 |
reviewed |
Kinase |
JAK2 |
Activity |
- |
- |
- |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
1100 |
nM |
| P08631 |
BXGT006801 |
Tyrosine-protein kinase HCK |
reviewed |
Kinase |
HCK |
Kd |
'=' |
4400 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
Kd |
'>' |
10000 |
nM |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Kd |
'>' |
10000 |
nM |
| Q9H0K1 |
BXGT020438 |
Serine/threonine-protein kinase SIK2 |
reviewed |
Kinase |
SIK2 |
Kd |
'=' |
2100 |
nM |
| Q09013 |
BXGT013023 |
Myotonin-protein kinase |
reviewed |
Kinase |
DMPK |
Kd |
'=' |
6900 |
nM |
| P21709 |
BXGT008685 |
Ephrin type-A receptor 1 |
reviewed |
Kinase |
EPHA1 |
Kd |
'=' |
4000 |
nM |
| P29320 |
BXGT009332 |
Ephrin type-A receptor 3 |
reviewed |
Kinase |
EPHA3 |
Kd |
'>' |
10000 |
nM |
| Q00526 |
BXGT012531 |
Cyclin-dependent kinase 3 |
reviewed |
Kinase |
CDK3 |
Kd |
'>' |
10000 |
nM |
| Q13976 |
BXGT013409 |
cGMP-dependent protein kinase 1 |
reviewed |
Kinase |
PRKG1 |
Kd |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
280 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'=' |
1900 |
nM |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Ki |
'>' |
6309 |
nM |
| P19525 |
BXGT008492 |
Interferon-induced, double-stranded RNA-activated protein kinase |
reviewed |
Kinase |
EIF2AK2 |
Kd |
'>' |
10000 |
nM |
| Q8TDX7 |
BXGT018817 |
Serine/threonine-protein kinase Nek7 |
reviewed |
Kinase |
NEK7 |
Kd |
'>' |
10000 |
nM |
| P27037 |
BXGT009153 |
Activin receptor type-2A |
reviewed |
Kinase |
ACVR2A |
Kd |
'>' |
10000 |
nM |
| Q13705 |
BXGT013393 |
Activin receptor type-2B |
reviewed |
Kinase |
ACVR2B |
Kd |
'>' |
10000 |
nM |
| Q9UK32 |
BXGT021736 |
Ribosomal protein S6 kinase alpha-6 |
reviewed |
Kinase |
RPS6KA6 |
Kd |
'>' |
10000 |
nM |
| Q16620 |
BXGT013645 |
BDNF/NT-3 growth factors receptor |
reviewed |
Kinase |
NTRK2 |
Ki |
'>' |
3981 |
nM |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Kd |
'=' |
5700 |
nM |
| P30530 |
BXGT009431 |
Tyrosine-protein kinase receptor UFO |
reviewed |
Kinase |
AXL |
Kd |
'>' |
10000 |
nM |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
3500 |
nM |
| O95835 |
BXGT005400 |
Serine/threonine-protein kinase LATS1 |
reviewed |
Kinase |
LATS1 |
Kd |
'>' |
10000 |
nM |
| O43283 |
BXGT004583 |
Mitogen-activated protein kinase kinase kinase 13 |
reviewed |
Kinase |
MAP3K13 |
Kd |
'>' |
10000 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Kd |
'=' |
630 |
nM |
| Q16513 |
BXGT013632 |
Serine/threonine-protein kinase N2 |
reviewed |
Kinase |
PKN2 |
Kd |
'>' |
10000 |
nM |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Kd |
'>' |
10000 |
nM |
| O60331 |
BXGT004872 |
Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma |
reviewed |
Kinase |
PIP5K1C |
Kd |
'>' |
10000 |
nM |
| P15735 |
BXGT008151 |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
reviewed |
Kinase |
PHKG2 |
Ki |
'=' |
3162 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Inhibition |
- |
- |
- |
| O75914 |
BXGT005165 |
Serine/threonine-protein kinase PAK 3 |
reviewed |
Kinase |
PAK3 |
Kd |
- |
- |
- |
| P42338 |
BXGT010303 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform |
reviewed |
Kinase |
PIK3CB |
IC50 |
'>' |
50000 |
nM |
| P78527 |
BXGT011846 |
DNA-dependent protein kinase catalytic subunit |
reviewed |
Kinase |
PRKDC |
IC50 |
'>' |
50000 |
nM |
| P22455 |
BXGT008772 |
Fibroblast growth factor receptor 4 |
reviewed |
Kinase |
FGFR4 |
Kd |
'>' |
10000 |
nM |
| Q13882 |
BXGT013399 |
Protein-tyrosine kinase 6 |
reviewed |
Kinase |
PTK6 |
Kd |
'>' |
10000 |
nM |
| P04049 |
BXGT006133 |
RAF proto-oncogene serine/threonine-protein kinase |
reviewed |
Kinase |
RAF1 |
Kd |
'>' |
10000 |
nM |
| Q13470 |
BXGT013359 |
Non-receptor tyrosine-protein kinase TNK1 |
reviewed |
Kinase |
TNK1 |
Kd |
'>' |
10000 |
nM |
| P53671 |
BXGT011009 |
LIM domain kinase 2 |
reviewed |
Kinase |
LIMK2 |
Kd |
'>' |
10000 |
nM |
| Q9C098 |
BXGT020208 |
Serine/threonine-protein kinase DCLK3 |
reviewed |
Kinase |
DCLK3 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
380 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
13 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
39 |
nM |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Kd |
'>' |
10000 |
nM |
| P30291 |
BXGT009417 |
Wee1-like protein kinase |
reviewed |
Kinase |
WEE1 |
Kd |
'>' |
10000 |
nM |
| Q13188 |
BXGT013324 |
Serine/threonine-protein kinase 3 |
reviewed |
Kinase |
STK3 |
Kd |
'>' |
10000 |
nM |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Kd |
'>' |
10000 |
nM |
| Q5VT25 |
BXGT015887 |
Serine/threonine-protein kinase MRCK alpha |
reviewed |
Kinase |
CDC42BPA |
Kd |
'>' |
10000 |
nM |
| P29317 |
BXGT009331 |
Ephrin type-A receptor 2 |
reviewed |
Kinase |
EPHA2 |
Kd |
'>' |
10000 |
nM |
| Q04759 |
BXGT012781 |
Protein kinase C theta type |
reviewed |
Kinase |
PRKCQ |
Kd |
'>' |
10000 |
nM |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Kd |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
599 |
nM |
| Q9NSY1 |
BXGT021209 |
BMP-2-inducible protein kinase |
reviewed |
Kinase |
BMP2K |
Kd |
- |
- |
- |
| Q06187 |
BXGT012860 |
Tyrosine-protein kinase BTK |
reviewed |
Kinase |
BTK |
Kd |
- |
- |
- |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Kd |
'=' |
1100 |
nM |
| P21802 |
BXGT008691 |
Fibroblast growth factor receptor 2 |
reviewed |
Kinase |
FGFR2 |
Kd |
- |
- |
- |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Ratio |
'>' |
1 |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
99 |
% |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
343 |
nM |
| Q07002 |
BXGT012908 |
Cyclin-dependent kinase 18 |
reviewed |
Kinase |
CDK18 |
Kd |
'>' |
10000 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Kd |
- |
- |
- |
| P51813 |
BXGT010894 |
Cytoplasmic tyrosine-protein kinase BMX |
reviewed |
Kinase |
BMX |
Kd |
- |
- |
- |
| Q06418 |
BXGT012875 |
Tyrosine-protein kinase receptor TYRO3 |
reviewed |
Kinase |
TYRO3 |
Kd |
'>' |
10000 |
nM |
| P49674 |
BXGT010725 |
Casein kinase I isoform epsilon |
reviewed |
- |
CSNK1E |
Kd |
'=' |
430 |
nM |
| Q9UQB9 |
BXGT021810 |
Aurora kinase C |
reviewed |
Kinase |
AURKC |
Kd |
'>' |
10000 |
nM |
| P36896 |
BXGT009940 |
Activin receptor type-1B |
reviewed |
Kinase |
ACVR1B |
Kd |
'>' |
10000 |
nM |
| P07949 |
BXGT006703 |
Proto-oncogene tyrosine-protein kinase receptor Ret |
reviewed |
Kinase |
RET |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
1000 |
nM |
| P35590 |
BXGT009854 |
Tyrosine-protein kinase receptor Tie-1 |
reviewed |
Kinase |
TIE1 |
Kd |
'>' |
10000 |
nM |
| P36897 |
BXGT009941 |
TGF-beta receptor type-1 |
reviewed |
Kinase |
TGFBR1 |
Kd |
'>' |
10000 |
nM |
| Q86UX6 |
BXGT017614 |
Serine/threonine-protein kinase 32C |
reviewed |
Kinase |
STK32C |
Kd |
'>' |
10000 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
IC50 |
'>' |
50000 |
nM |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
IC50 |
'>' |
50000 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Inhibition |
'=' |
12 |
% |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'>' |
10000 |
nM |
| O15111 |
BXGT004126 |
Inhibitor of nuclear factor kappa-B kinase subunit alpha |
reviewed |
Kinase |
CHUK |
Ki |
'>' |
3981 |
nM |
| Q9H1R3 |
BXGT020446 |
Myosin light chain kinase 2, skeletal/cardiac muscle |
reviewed |
Kinase |
MYLK2 |
Kd |
'=' |
1900 |
nM |
| P78362 |
BXGT011839 |
SRSF protein kinase 2 |
reviewed |
Kinase |
SRPK2 |
Kd |
'>' |
10000 |
nM |
| Q8WXR4 |
BXGT019015 |
Myosin-IIIb |
reviewed |
Kinase |
MYO3B |
Kd |
'>' |
10000 |
nM |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Kd |
'>' |
10000 |
nM |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Kd |
'>' |
10000 |
nM |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Kd |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
2700 |
nM |
| P27448 |
BXGT009183 |
MAP/microtubule affinity-regulating kinase 3 |
reviewed |
Kinase |
MARK3 |
Kd |
'>' |
10000 |
nM |
| Q16584 |
BXGT013642 |
Mitogen-activated protein kinase kinase kinase 11 |
reviewed |
Kinase |
MAP3K11 |
Kd |
'>' |
10000 |
nM |
| Q16512 |
BXGT013631 |
Serine/threonine-protein kinase N1 |
reviewed |
Kinase |
PKN1 |
Kd |
'>' |
10000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
1730 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
1730 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1730 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
1730 |
nM |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Kd |
'=' |
1400 |
nM |
| P07948 |
BXGT006702 |
Tyrosine-protein kinase Lyn |
reviewed |
Kinase |
LYN |
Kd |
- |
- |
- |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Kd |
'=' |
870 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
Kd |
- |
- |
- |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Kd |
- |
- |
- |
| P35916 |
BXGT009881 |
Vascular endothelial growth factor receptor 3 |
reviewed |
Kinase |
FLT4 |
Kd |
- |
- |
- |
| O94768 |
BXGT005331 |
Serine/threonine-protein kinase 17B |
reviewed |
Kinase |
STK17B |
Kd |
'=' |
6500 |
nM |
| Q9HBY8 |
BXGT020524 |
Serine/threonine-protein kinase Sgk2 |
reviewed |
Kinase |
SGK2 |
Ki |
'>' |
7943 |
nM |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Ki |
'=' |
501 |
nM |
| P30530 |
BXGT009431 |
Tyrosine-protein kinase receptor UFO |
reviewed |
Kinase |
AXL |
Ki |
'=' |
1584 |
nM |
| Q86UE8 |
BXGT017612 |
Serine/threonine-protein kinase tousled-like 2 |
reviewed |
Kinase |
TLK2 |
Kd |
'>' |
10000 |
nM |
| O14757 |
BXGT004092 |
Serine/threonine-protein kinase Chk1 |
reviewed |
Kinase |
CHEK1 |
Kd |
'>' |
10000 |
nM |
| Q9BRS2 |
BXGT020119 |
Serine/threonine-protein kinase RIO1 |
reviewed |
Kinase |
RIOK1 |
Kd |
'>' |
10000 |
nM |
| Q9P0L2 |
BXGT021289 |
Serine/threonine-protein kinase MARK1 |
reviewed |
Kinase |
MARK1 |
Kd |
'>' |
10000 |
nM |
| Q13153 |
BXGT013319 |
Serine/threonine-protein kinase PAK 1 |
reviewed |
Kinase |
PAK1 |
Kd |
- |
- |
- |
| Q92772 |
BXGT019371 |
Cyclin-dependent kinase-like 2 |
reviewed |
Kinase |
CDKL2 |
Kd |
'>' |
10000 |
nM |
| P54756 |
BXGT011074 |
Ephrin type-A receptor 5 |
reviewed |
Kinase |
EPHA5 |
Kd |
'=' |
1500 |
nM |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Kd |
- |
- |
- |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Kd |
- |
- |
- |
| Q3U3Q1 |
BXGT014526 |
Serine/threonine-protein kinase ULK3 |
reviewed |
- |
Ulk3 |
Kd |
'=' |
1400 |
nM |
| Q9HAZ1 |
BXGT020511 |
Dual specificity protein kinase CLK4 |
reviewed |
- |
CLK4 |
Kd |
- |
- |
- |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Kd |
- |
- |
- |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Kd |
- |
- |
- |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Ki |
'>' |
5011 |
nM |
| P42685 |
BXGT010332 |
Tyrosine-protein kinase FRK |
reviewed |
Kinase |
FRK |
Ki |
'=' |
251 |
nM |
| Q96GD4 |
BXGT019667 |
Aurora kinase B |
reviewed |
Kinase |
AURKB |
Ki |
'>' |
6309 |
nM |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Ki |
'>' |
1995 |
nM |
| O75116 |
BXGT005100 |
Rho-associated protein kinase 2 |
reviewed |
Kinase |
ROCK2 |
Ki |
'>' |
6309 |
nM |
| O60674 |
BXGT004892 |
Tyrosine-protein kinase JAK2 |
reviewed |
Kinase |
JAK2 |
Kd |
- |
- |
- |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Kd |
- |
- |
- |
| Q8N5S9 |
BXGT018520 |
Calcium/calmodulin-dependent protein kinase kinase 1 |
reviewed |
Kinase |
CAMKK1 |
Kd |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Potency |
'=' |
3 |
nM |
| Q9UF33 |
BXGT021676 |
Ephrin type-A receptor 6 |
reviewed |
Kinase |
EPHA6 |
Kd |
'=' |
1400 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Kd |
'=' |
1100 |
nM |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Kd |
- |
- |
- |
| Q9Y2H1 |
BXGT022233 |
Serine/threonine-protein kinase 38-like |
reviewed |
Kinase |
STK38L |
Kd |
- |
- |
- |
| P22607 |
BXGT008784 |
Fibroblast growth factor receptor 3 |
reviewed |
Kinase |
FGFR3 |
Kd |
- |
- |
- |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
IC50 |
'>' |
50000 |
nM |
| Q07912 |
BXGT012947 |
Activated CDC42 kinase 1 |
reviewed |
Kinase |
TNK2 |
Ki |
'>' |
3162 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
23 |
nM |
| Q92918 |
BXGT019394 |
Mitogen-activated protein kinase kinase kinase kinase 1 |
reviewed |
Kinase |
MAP4K1 |
Kd |
'>' |
10000 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Kd |
'>' |
10000 |
nM |
| Q13546 |
BXGT013372 |
Receptor-interacting serine/threonine-protein kinase 1 |
reviewed |
Kinase |
RIPK1 |
Kd |
'>' |
10000 |
nM |
| P08922 |
BXGT006843 |
Proto-oncogene tyrosine-protein kinase ROS |
reviewed |
Kinase |
ROS1 |
Kd |
'>' |
10000 |
nM |
| P51813 |
BXGT010894 |
Cytoplasmic tyrosine-protein kinase BMX |
reviewed |
Kinase |
BMX |
Activity |
- |
- |
- |
| Q96GD4 |
BXGT019667 |
Aurora kinase B |
reviewed |
Kinase |
AURKB |
Kd |
'>' |
10000 |
nM |
| O60285 |
BXGT004867 |
NUAK family SNF1-like kinase 1 |
reviewed |
Kinase |
NUAK1 |
Kd |
'>' |
10000 |
nM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Kd |
- |
- |
- |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Kd |
'=' |
5000 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Ki |
'>' |
5011 |
nM |
| Q9Y2H1 |
BXGT022233 |
Serine/threonine-protein kinase 38-like |
reviewed |
Kinase |
STK38L |
Kd |
'>' |
10000 |
nM |
| P21802 |
BXGT008691 |
Fibroblast growth factor receptor 2 |
reviewed |
Kinase |
FGFR2 |
Kd |
'>' |
10000 |
nM |
| Q9NYL2 |
BXGT021259 |
Mitogen-activated protein kinase kinase kinase 20 |
reviewed |
Kinase |
MAP3K20 |
Kd |
'>' |
10000 |
nM |
| P54760 |
BXGT011075 |
Ephrin type-B receptor 4 |
reviewed |
Kinase |
EPHB4 |
Kd |
'>' |
10000 |
nM |
| Q9NRP7 |
BXGT021192 |
Serine/threonine-protein kinase 36 |
reviewed |
Kinase |
STK36 |
Kd |
'>' |
10000 |
nM |
| P07333 |
BXGT006602 |
Macrophage colony-stimulating factor 1 receptor |
reviewed |
Kinase |
CSF1R |
Kd |
'>' |
10000 |
nM |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Kd |
'>' |
10000 |
nM |
| Q9Y6E0 |
BXGT022327 |
Serine/threonine-protein kinase 24 |
reviewed |
Kinase |
STK24 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ratio |
'=' |
505 |
- |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Kd |
'>' |
10000 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Ki |
'=' |
2511 |
nM |
| P54762 |
BXGT011076 |
Ephrin type-B receptor 1 |
reviewed |
Kinase |
EPHB1 |
Kd |
'=' |
1300 |
nM |
| P14616 |
BXGT008026 |
Insulin receptor-related protein |
reviewed |
Kinase |
INSRR |
Kd |
'>' |
10000 |
nM |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Kd |
'=' |
1700 |
nM |
| Q13163 |
BXGT013321 |
Dual specificity mitogen-activated protein kinase kinase 5 |
reviewed |
Kinase |
MAP2K5 |
Kd |
'=' |
600 |
nM |
| P50613 |
BXGT010815 |
Cyclin-dependent kinase 7 |
reviewed |
Kinase |
CDK7 |
Kd |
'=' |
610 |
nM |
| Q13153 |
BXGT013319 |
Serine/threonine-protein kinase PAK 1 |
reviewed |
Kinase |
PAK1 |
Kd |
'>' |
10000 |
nM |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Kd |
'>' |
10000 |
nM |
| O15111 |
BXGT004126 |
Inhibitor of nuclear factor kappa-B kinase subunit alpha |
reviewed |
Kinase |
CHUK |
Kd |
'>' |
10000 |
nM |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Kd |
'>' |
10000 |
nM |
| P54762 |
BXGT011076 |
Ephrin type-B receptor 1 |
reviewed |
Kinase |
EPHB1 |
Kd |
'>' |
10000 |
nM |
| P53355 |
BXGT010985 |
Death-associated protein kinase 1 |
reviewed |
Kinase |
DAPK1 |
Kd |
'>' |
10000 |
nM |
| Q9Y5S2 |
BXGT022301 |
Serine/threonine-protein kinase MRCK beta |
reviewed |
Kinase |
CDC42BPB |
Kd |
'>' |
10000 |
nM |
| P37173 |
BXGT009970 |
TGF-beta receptor type-2 |
reviewed |
Kinase |
TGFBR2 |
Kd |
'>' |
10000 |
nM |
| P41240 |
BXGT010242 |
Tyrosine-protein kinase CSK |
reviewed |
Kinase |
CSK |
Kd |
'>' |
10000 |
nM |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
190 |
nM |
| Q00526 |
BXGT012531 |
Cyclin-dependent kinase 3 |
reviewed |
Kinase |
CDK3 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'<' |
1 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'<' |
1 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'<' |
1 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'<' |
1 |
nM |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Kd |
'=' |
2900 |
nM |
| O94806 |
BXGT005335 |
Serine/threonine-protein kinase D3 |
reviewed |
Kinase |
PRKD3 |
Kd apparent |
'>' |
30000 |
nM |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Kd apparent |
'>' |
30000 |
nM |
| O60674 |
BXGT004892 |
Tyrosine-protein kinase JAK2 |
reviewed |
Kinase |
JAK2 |
Ki |
'>' |
1584 |
nM |
| P07949 |
BXGT006703 |
Proto-oncogene tyrosine-protein kinase receptor Ret |
reviewed |
Kinase |
RET |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y2K2 |
BXGT022238 |
Serine/threonine-protein kinase SIK3 |
reviewed |
Kinase |
SIK3 |
Kd apparent |
'>' |
30000 |
nM |
| Q13882 |
BXGT013399 |
Protein-tyrosine kinase 6 |
reviewed |
Kinase |
PTK6 |
Kd apparent |
'>' |
30000 |
nM |
| Q13470 |
BXGT013359 |
Non-receptor tyrosine-protein kinase TNK1 |
reviewed |
Kinase |
TNK1 |
Kd apparent |
'>' |
30000 |
nM |
| P15735 |
BXGT008151 |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
reviewed |
Kinase |
PHKG2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UGJ0 |
BXGT021683 |
5'-AMP-activated protein kinase subunit gamma-2 |
reviewed |
Enzyme modulator |
PRKAG2 |
Kd apparent |
'>' |
30000 |
nM |
| O14976 |
BXGT004118 |
Cyclin-G-associated kinase |
reviewed |
Kinase |
GAK |
Kd apparent |
'=' |
951 |
nM |
| P27361 |
BXGT009176 |
Mitogen-activated protein kinase 3 |
reviewed |
Kinase |
MAPK3 |
Kd apparent |
'>' |
30000 |
nM |
| P05141 |
BXGT006325 |
ADP/ATP translocase 2 |
reviewed |
Transporter |
SLC25A5 |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
2 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
2 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
2 |
nM |
| O00506 |
BXGT003932 |
Serine/threonine-protein kinase 25 |
reviewed |
Kinase |
STK25 |
Kd |
'>' |
10000 |
nM |
| Q8IYT8 |
BXGT018370 |
Serine/threonine-protein kinase ULK2 |
reviewed |
Kinase |
ULK2 |
Kd |
'>' |
10000 |
nM |
| Q8NEV4 |
BXGT018558 |
Myosin-IIIa |
reviewed |
Kinase |
MYO3A |
Kd |
'>' |
10000 |
nM |
| Q8NI60 |
BXGT018572 |
Atypical kinase COQ8A, mitochondrial |
reviewed |
Kinase |
COQ8A |
Kd |
'>' |
10000 |
nM |
| Q13627 |
BXGT013385 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
reviewed |
Kinase |
DYRK1A |
Kd |
'>' |
10000 |
nM |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Kd |
'>' |
10000 |
nM |
| Q8WTQ7 |
BXGT018984 |
Rhodopsin kinase |
reviewed |
Kinase |
GRK7 |
Kd |
'>' |
10000 |
nM |
| Q32MK0 |
BXGT014323 |
Myosin light chain kinase 3 |
reviewed |
Kinase |
MYLK3 |
Kd |
'>' |
10000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
22 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
22 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
22 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
22 |
nM |
| Q12866 |
BXGT013273 |
Tyrosine-protein kinase Mer |
reviewed |
Kinase |
MERTK |
Kd |
'>' |
10000 |
nM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Kd |
'>' |
10000 |
nM |
| P23443 |
BXGT008866 |
Ribosomal protein S6 kinase beta-1 |
reviewed |
Kinase |
RPS6KB1 |
Ki |
'>' |
5011 |
nM |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Kd |
'>' |
10000 |
nM |
| P13861 |
BXGT007961 |
cAMP-dependent protein kinase type II-alpha regulatory subunit |
reviewed |
- |
PRKAR2A |
Kd apparent |
'>' |
30000 |
nM |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Kd apparent |
'>' |
30000 |
nM |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Kd apparent |
'>' |
30000 |
nM |
| Q16513 |
BXGT013632 |
Serine/threonine-protein kinase N2 |
reviewed |
Kinase |
PKN2 |
Kd apparent |
'>' |
30000 |
nM |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Kd |
- |
- |
- |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Kd |
- |
- |
- |
| P48729 |
BXGT010655 |
Casein kinase I isoform alpha |
reviewed |
Kinase |
CSNK1A1 |
IC50 |
'>' |
50000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
515 |
nM |
| P42684 |
BXGT010331 |
Tyrosine-protein kinase ABL2 |
reviewed |
Kinase |
ABL2 |
Kd |
- |
- |
- |
| Q9JI10 |
BXGT020811 |
Serine/threonine-protein kinase 3 |
reviewed |
- |
Stk3 |
Kd |
- |
- |
- |
| Q04206 |
BXGT012754 |
Transcription factor p65 |
reviewed |
Transcription factor |
RELA |
Inhibition |
- |
- |
- |
| Q14164 |
BXGT013451 |
Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
reviewed |
Kinase |
IKBKE |
Kd apparent |
'>' |
30000 |
nM |
| P23458 |
BXGT008868 |
Tyrosine-protein kinase JAK1 |
reviewed |
Kinase |
JAK1 |
Kd apparent |
'>' |
30000 |
nM |
| Q16584 |
BXGT013642 |
Mitogen-activated protein kinase kinase kinase 11 |
reviewed |
Kinase |
MAP3K11 |
Kd apparent |
'>' |
30000 |
nM |
| P08631 |
BXGT006801 |
Tyrosine-protein kinase HCK |
reviewed |
Kinase |
HCK |
IC50 |
'=' |
110 |
nM |
| P42679 |
BXGT010328 |
Megakaryocyte-associated tyrosine-protein kinase |
reviewed |
Kinase |
MATK |
Ki |
'>' |
1995 |
nM |
| P51451 |
BXGT010848 |
Tyrosine-protein kinase Blk |
reviewed |
Kinase |
BLK |
Kd |
'=' |
1200 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
13980 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
13980 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
13980 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
13980 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| Q15746 |
BXGT013591 |
Myosin light chain kinase, smooth muscle |
reviewed |
Kinase |
MYLK |
Kd apparent |
'>' |
30000 |
nM |
| O95382 |
BXGT005376 |
Mitogen-activated protein kinase kinase kinase 6 |
reviewed |
Kinase |
MAP3K6 |
Kd apparent |
'>' |
30000 |
nM |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Kd apparent |
'>' |
30000 |
nM |
| Q99640 |
BXGT019944 |
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase |
reviewed |
Kinase |
PKMYT1 |
Kd apparent |
'>' |
30000 |
nM |
| Q01538 |
BXGT012597 |
Myelin transcription factor 1 |
reviewed |
Transcription factor |
MYT1 |
Activity |
'<' |
5 |
% |
| Q9Y243 |
BXGT022214 |
RAC-gamma serine/threonine-protein kinase |
reviewed |
Kinase |
AKT3 |
Ki |
'>' |
10000 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Ki |
'>' |
1995 |
nM |
| Q12851 |
BXGT013271 |
Mitogen-activated protein kinase kinase kinase kinase 2 |
reviewed |
Kinase |
MAP4K2 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
400 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
520 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
1100 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Kd |
'>' |
10000 |
nM |
| P29320 |
BXGT009332 |
Ephrin type-A receptor 3 |
reviewed |
Kinase |
EPHA3 |
Kd |
'=' |
5500 |
nM |
| O95819 |
BXGT005398 |
Mitogen-activated protein kinase kinase kinase kinase 4 |
reviewed |
Kinase |
MAP4K4 |
Ki |
'=' |
1000 |
nM |
| Q86Y07 |
BXGT017631 |
Serine/threonine-protein kinase VRK2 |
reviewed |
Kinase |
VRK2 |
Kd |
'>' |
10000 |
nM |
| Q9NYY3 |
BXGT021264 |
Serine/threonine-protein kinase PLK2 |
reviewed |
Kinase |
PLK2 |
Kd |
'>' |
10000 |
nM |
| Q9UEW8 |
BXGT021675 |
STE20/SPS1-related proline-alanine-rich protein kinase |
reviewed |
Kinase |
STK39 |
Kd |
'>' |
10000 |
nM |
| Q9Y2H9 |
BXGT022234 |
Microtubule-associated serine/threonine-protein kinase 1 |
reviewed |
Kinase |
MAST1 |
Kd |
'>' |
10000 |
nM |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Kd |
'>' |
10000 |
nM |
| Q8TBX8 |
BXGT018791 |
Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma |
reviewed |
Kinase |
PIP4K2C |
Kd |
'=' |
7500 |
nM |
| P48730 |
BXGT010656 |
Casein kinase I isoform delta |
reviewed |
Kinase |
CSNK1D |
Kd |
'=' |
3200 |
nM |
| P35916 |
BXGT009881 |
Vascular endothelial growth factor receptor 3 |
reviewed |
Kinase |
FLT4 |
Ki |
'=' |
6309 |
nM |
| P29376 |
BXGT009339 |
Leukocyte tyrosine kinase receptor |
reviewed |
Kinase |
LTK |
Ki |
'>' |
1584 |
nM |
| Q9H4B4 |
BXGT020474 |
Serine/threonine-protein kinase PLK3 |
reviewed |
Kinase |
PLK3 |
Ki |
'>' |
7943 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Ki |
'>' |
2511 |
nM |
| Q8TDC3 |
BXGT018808 |
Serine/threonine-protein kinase BRSK1 |
reviewed |
Kinase |
BRSK1 |
Ki |
'=' |
3162 |
nM |
| Q8NE63 |
BXGT018551 |
Homeodomain-interacting protein kinase 4 |
reviewed |
Kinase |
HIPK4 |
Ki |
'=' |
1258 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Inhibition |
'=' |
81 |
% |
| O75460 |
BXGT005127 |
Serine/threonine-protein kinase/endoribonuclease IRE1 |
reviewed |
Kinase |
ERN1 |
Kd apparent |
'>' |
30000 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Kd apparent |
'=' |
4372 |
nM |
| Q96L34 |
BXGT019689 |
MAP/microtubule affinity-regulating kinase 4 |
reviewed |
Kinase |
MARK4 |
Kd apparent |
'>' |
30000 |
nM |
| Q13882 |
BXGT013399 |
Protein-tyrosine kinase 6 |
reviewed |
Kinase |
PTK6 |
Ki |
'>' |
1995 |
nM |
| P16591 |
BXGT008246 |
Tyrosine-protein kinase Fer |
reviewed |
Kinase |
FER |
Kd apparent |
'>' |
30000 |
nM |
| P51617 |
BXGT010868 |
Interleukin-1 receptor-associated kinase 1 |
reviewed |
Kinase |
IRAK1 |
Ki |
'=' |
316 |
nM |
| Q6DT37 |
BXGT016259 |
Serine/threonine-protein kinase MRCK gamma |
reviewed |
Kinase |
CDC42BPG |
Kd apparent |
'>' |
30000 |
nM |
| Q8N4C8 |
BXGT018510 |
Misshapen-like kinase 1 |
reviewed |
Kinase |
MINK1 |
Ki |
'=' |
5011 |
nM |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Ki |
'=' |
398 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Ki |
'>' |
7943 |
nM |
| P52333 |
BXGT010928 |
Tyrosine-protein kinase JAK3 |
reviewed |
Kinase |
JAK3 |
Ki |
'>' |
1584 |
nM |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
Kd apparent |
'>' |
30000 |
nM |
| P41743 |
BXGT010270 |
Protein kinase C iota type |
reviewed |
Kinase |
PRKCI |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y4K4 |
BXGT022282 |
Mitogen-activated protein kinase kinase kinase kinase 5 |
reviewed |
Kinase |
MAP4K5 |
Kd apparent |
'>' |
30000 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Ki |
'>' |
7943 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Kd apparent |
'>' |
30000 |
nM |
| P11802 |
BXGT007750 |
Cyclin-dependent kinase 4 |
reviewed |
Kinase |
CDK4 |
Kd apparent |
'>' |
30000 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
12 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Kd |
'>' |
10000 |
nM |
| Q14289 |
BXGT013459 |
Protein-tyrosine kinase 2-beta |
reviewed |
Kinase |
PTK2B |
Kd |
'>' |
10000 |
nM |
| P29376 |
BXGT009339 |
Leukocyte tyrosine kinase receptor |
reviewed |
Kinase |
LTK |
Kd |
'=' |
5500 |
nM |
| Q9UQ88 |
BXGT021808 |
Cyclin-dependent kinase 11A |
reviewed |
- |
CDK11A |
Kd |
'>' |
10000 |
nM |
| Q8TD19 |
BXGT018804 |
Serine/threonine-protein kinase Nek9 |
reviewed |
Kinase |
NEK9 |
Kd |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
21 |
nM |
| Q16620 |
BXGT013645 |
BDNF/NT-3 growth factors receptor |
reviewed |
Kinase |
NTRK2 |
Kd |
'>' |
10000 |
nM |
| P50750 |
BXGT010818 |
Cyclin-dependent kinase 9 |
reviewed |
Kinase |
CDK9 |
Ki |
'>' |
1584 |
nM |
| Q9NY57 |
BXGT021250 |
Serine/threonine-protein kinase 32B |
reviewed |
Kinase |
STK32B |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Ki |
'>' |
630 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Ki |
'>' |
1995 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
4 |
nM |
| P52333 |
BXGT010928 |
Tyrosine-protein kinase JAK3 |
reviewed |
Kinase |
JAK3 |
Kd |
'>' |
10000 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd |
'=' |
1800 |
nM |
| Q13418 |
BXGT013351 |
Integrin-linked protein kinase |
reviewed |
Kinase |
ILK |
Kd apparent |
'>' |
30000 |
nM |
| Q9UHD2 |
BXGT021697 |
Serine/threonine-protein kinase TBK1 |
reviewed |
Kinase |
TBK1 |
Kd |
'>' |
10000 |
nM |
| Q9UL54 |
BXGT021755 |
Serine/threonine-protein kinase TAO2 |
reviewed |
Kinase |
TAOK2 |
Kd |
'>' |
10000 |
nM |
| Q9UBE8 |
BXGT021652 |
Serine/threonine-protein kinase NLK |
reviewed |
Kinase |
NLK |
Kd |
'=' |
4200 |
nM |
| Q9HAZ1 |
BXGT020511 |
Dual specificity protein kinase CLK4 |
reviewed |
- |
CLK4 |
Kd |
'>' |
10000 |
nM |
| O15254 |
BXGT004143 |
Peroxisomal acyl-coenzyme A oxidase 3 |
reviewed |
Enzyme |
ACOX3 |
Kd apparent |
'>' |
30000 |
nM |
| P11274 |
BXGT007681 |
Breakpoint cluster region protein |
reviewed |
Enzyme modulator |
BCR |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
39 |
nM |
| P42685 |
BXGT010332 |
Tyrosine-protein kinase FRK |
reviewed |
Kinase |
FRK |
Kd apparent |
'>' |
30000 |
nM |
| P48730 |
BXGT010656 |
Casein kinase I isoform delta |
reviewed |
Kinase |
CSNK1D |
Ki |
'=' |
7943 |
nM |
| Q9UEE5 |
BXGT021671 |
Serine/threonine-protein kinase 17A |
reviewed |
Kinase |
STK17A |
Ki |
'>' |
3981 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'=' |
14800 |
nM |
| P33981 |
BXGT009744 |
Dual specificity protein kinase TTK |
reviewed |
Kinase |
TTK |
Kd apparent |
'>' |
30000 |
nM |
| P49761 |
BXGT010736 |
Dual specificity protein kinase CLK3 |
reviewed |
Kinase |
CLK3 |
Kd |
- |
- |
- |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Kd |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
173 |
nM |
| P27448 |
BXGT009183 |
MAP/microtubule affinity-regulating kinase 3 |
reviewed |
Kinase |
MARK3 |
Kd apparent |
'>' |
30000 |
nM |
| P30086 |
BXGT009400 |
Phosphatidylethanolamine-binding protein 1 |
reviewed |
Enzyme modulator |
PEBP1 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Thermal melting change |
'=' |
0 |
degrees C |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9Y6R4 |
BXGT022340 |
Mitogen-activated protein kinase kinase kinase 4 |
reviewed |
Kinase |
MAP3K4 |
Kd |
'>' |
10000 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Kd |
'>' |
10000 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Kd |
'>' |
10000 |
nM |
| Q9Y243 |
BXGT022214 |
RAC-gamma serine/threonine-protein kinase |
reviewed |
Kinase |
AKT3 |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
3000 |
nM |
| P0A0J7 |
BXGT006970 |
Quinolone resistance protein NorA |
reviewed |
- |
norA |
Inhibition |
'=' |
94 |
% |
| P0A0J7 |
BXGT006970 |
Quinolone resistance protein NorA |
reviewed |
- |
norA |
IC50 |
'=' |
9700 |
nM |
| O15197 |
BXGT004136 |
Ephrin type-B receptor 6 |
reviewed |
Kinase |
EPHB6 |
Kd apparent |
'>' |
30000 |
nM |
| P02545 |
BXGT005889 |
Prelamin-A/C |
reviewed |
- |
LMNA |
Potency |
'=' |
0 |
nM |
| Q52WX2 |
BXGT014988 |
Serine/threonine-protein kinase SBK1 |
reviewed |
- |
SBK1 |
Kd |
'=' |
560 |
nM |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Ki |
'>' |
3981 |
nM |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Kd |
- |
- |
- |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Kd |
- |
- |
- |
| P09619 |
BXGT006911 |
Platelet-derived growth factor receptor beta |
reviewed |
Kinase |
PDGFRB |
Kd |
- |
- |
- |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Kd |
- |
- |
- |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
Kd |
- |
- |
- |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Kd |
- |
- |
- |
| O43781 |
BXGT004625 |
Dual specificity tyrosine-phosphorylation-regulated kinase 3 |
reviewed |
Kinase |
DYRK3 |
Ki |
'>' |
5011 |
nM |
| P42681 |
BXGT010330 |
Tyrosine-protein kinase TXK |
reviewed |
Kinase |
TXK |
Kd |
'=' |
6000 |
nM |
| Q9BZL6 |
BXGT020199 |
Serine/threonine-protein kinase D2 |
reviewed |
Kinase |
PRKD2 |
Ki |
'=' |
2511 |
nM |
| P11802 |
BXGT007750 |
Cyclin-dependent kinase 4 |
reviewed |
Kinase |
CDK4 |
Kd |
'>' |
10000 |
nM |
| P16234 |
BXGT008209 |
Platelet-derived growth factor receptor alpha |
reviewed |
Kinase |
PDGFRA |
Kd |
'>' |
10000 |
nM |
| P15735 |
BXGT008151 |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
reviewed |
Kinase |
PHKG2 |
Kd |
'>' |
10000 |
nM |
| Q13873 |
BXGT013398 |
Bone morphogenetic protein receptor type-2 |
reviewed |
Kinase |
BMPR2 |
Kd |
'>' |
10000 |
nM |
| Q08345 |
BXGT012982 |
Epithelial discoidin domain-containing receptor 1 |
reviewed |
Kinase |
DDR1 |
Kd |
'>' |
10000 |
nM |
| Q9UQM7 |
BXGT021814 |
Calcium/calmodulin-dependent protein kinase type II subunit alpha |
reviewed |
Kinase |
CAMK2A |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3 |
nM |
| Q13627 |
BXGT013385 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
reviewed |
Kinase |
DYRK1A |
Ki |
'>' |
5011 |
nM |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Ki |
'>' |
7943 |
nM |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Kd |
'=' |
2300 |
nM |
| Q9NRP7 |
BXGT021192 |
Serine/threonine-protein kinase 36 |
reviewed |
Kinase |
STK36 |
Kd |
- |
- |
- |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Kd |
- |
- |
- |
| P29322 |
BXGT009333 |
Ephrin type-A receptor 8 |
reviewed |
Kinase |
EPHA8 |
Kd |
- |
- |
- |
| O14965 |
BXGT004117 |
Aurora kinase A |
reviewed |
Kinase |
AURKA |
Kd apparent |
'>' |
30000 |
nM |
| Q5S007 |
BXGT015650 |
Leucine-rich repeat serine/threonine-protein kinase 2 |
reviewed |
Kinase |
LRRK2 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
230 |
nM |
| P42684 |
BXGT010331 |
Tyrosine-protein kinase ABL2 |
reviewed |
Kinase |
ABL2 |
Kd |
'=' |
1600 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
0 |
nM |
| Q02156 |
BXGT012639 |
Protein kinase C epsilon type |
reviewed |
Kinase |
PRKCE |
Kd |
'>' |
10000 |
nM |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Kd |
'>' |
10000 |
nM |
| Q15569 |
BXGT013580 |
Dual specificity testis-specific protein kinase 1 |
reviewed |
Kinase |
TESK1 |
Kd |
'>' |
10000 |
nM |
| Q9UKI8 |
BXGT021743 |
Serine/threonine-protein kinase tousled-like 1 |
reviewed |
Kinase |
TLK1 |
Kd |
'>' |
10000 |
nM |
| Q96BR1 |
BXGT019627 |
Serine/threonine-protein kinase Sgk3 |
reviewed |
- |
SGK3 |
Kd |
'>' |
10000 |
nM |
| Q9UPE1 |
BXGT021796 |
SRSF protein kinase 3 |
reviewed |
Kinase |
SRPK3 |
Kd |
'>' |
10000 |
nM |
| Q9UPZ9 |
BXGT021804 |
Serine/threonine-protein kinase ICK |
reviewed |
Kinase |
CILK1 |
Kd |
'>' |
10000 |
nM |
| Q7KZI7 |
BXGT016990 |
Serine/threonine-protein kinase MARK2 |
reviewed |
Kinase |
MARK2 |
Kd |
'>' |
10000 |
nM |
| P17252 |
BXGT008294 |
Protein kinase C alpha type |
reviewed |
Kinase |
PRKCA |
Kd |
- |
- |
- |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Kd |
- |
- |
- |
| P33981 |
BXGT009744 |
Dual specificity protein kinase TTK |
reviewed |
Kinase |
TTK |
Kd |
- |
- |
- |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Kd |
- |
- |
- |
| P08069 |
BXGT006723 |
Insulin-like growth factor 1 receptor |
reviewed |
Kinase |
IGF1R |
Ki |
'>' |
1258 |
nM |
| Q16832 |
BXGT013678 |
Discoidin domain-containing receptor 2 |
reviewed |
Kinase |
DDR2 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
1 |
nM |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Kd |
'>' |
10000 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Kd |
'=' |
3800 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
5 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2753 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Kd |
'>' |
10000 |
nM |
| Q9HBH9 |
BXGT020521 |
MAP kinase-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
MKNK2 |
Kd |
'=' |
1200 |
nM |
| O75385 |
BXGT005121 |
Serine/threonine-protein kinase ULK1 |
reviewed |
Kinase |
ULK1 |
Kd |
'>' |
10000 |
nM |
| P78356 |
BXGT011837 |
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta |
reviewed |
Kinase |
PIP4K2B |
Kd |
'>' |
10000 |
nM |
| P31152 |
BXGT009511 |
Mitogen-activated protein kinase 4 |
reviewed |
Kinase |
MAPK4 |
Kd |
'=' |
3100 |
nM |
| O75914 |
BXGT005165 |
Serine/threonine-protein kinase PAK 3 |
reviewed |
Kinase |
PAK3 |
Kd |
'>' |
10000 |
nM |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
72 |
nM |
| Q9Y4K4 |
BXGT022282 |
Mitogen-activated protein kinase kinase kinase kinase 5 |
reviewed |
Kinase |
MAP4K5 |
Kd |
- |
- |
- |
| Q13882 |
BXGT013399 |
Protein-tyrosine kinase 6 |
reviewed |
Kinase |
PTK6 |
Kd |
- |
- |
- |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Kd |
- |
- |
- |
| P49674 |
BXGT010725 |
Casein kinase I isoform epsilon |
reviewed |
- |
CSNK1E |
Kd |
'=' |
2000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
54 |
nM |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Ki |
'>' |
6309 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Ki |
'=' |
158 |
nM |
| P04629 |
BXGT006239 |
High affinity nerve growth factor receptor |
reviewed |
Kinase |
NTRK1 |
Kd |
- |
- |
- |
| P29320 |
BXGT009332 |
Ephrin type-A receptor 3 |
reviewed |
Kinase |
EPHA3 |
Kd |
- |
- |
- |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
Kd |
'=' |
800 |
nM |
| P15735 |
BXGT008151 |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
reviewed |
Kinase |
PHKG2 |
Kd |
'=' |
6400 |
nM |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Potency |
- |
1373 |
nM |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P29376 |
BXGT009339 |
Leukocyte tyrosine kinase receptor |
reviewed |
Kinase |
LTK |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Inhibition |
- |
- |
- |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Kd |
'>' |
10000 |
nM |
| P10636 |
BXGT007596 |
Microtubule-associated protein tau |
reviewed |
- |
MAPT |
Potency |
'=' |
35481 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
IC50 |
'>' |
50000 |
nM |
| O00329 |
BXGT003909 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform |
reviewed |
Kinase |
PIK3CD |
IC50 |
'>' |
50000 |
nM |
| O14920 |
BXGT004110 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
reviewed |
Kinase |
IKBKB |
Ki |
'>' |
3162 |
nM |
| Q08881 |
BXGT013012 |
Tyrosine-protein kinase ITK/TSK |
reviewed |
Kinase |
ITK |
Ki |
'>' |
1584 |
nM |
| Q06187 |
BXGT012860 |
Tyrosine-protein kinase BTK |
reviewed |
Kinase |
BTK |
Ki |
'>' |
1258 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Kd |
'>' |
10000 |
nM |
| P43403 |
BXGT010385 |
Tyrosine-protein kinase ZAP-70 |
reviewed |
Kinase |
ZAP70 |
Kd |
'>' |
10000 |
nM |
| O95819 |
BXGT005398 |
Mitogen-activated protein kinase kinase kinase kinase 4 |
reviewed |
Kinase |
MAP4K4 |
Kd |
'>' |
10000 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Ki |
'>' |
7943 |
nM |
| Q15375 |
BXGT013562 |
Ephrin type-A receptor 7 |
reviewed |
Kinase |
EPHA7 |
Kd |
- |
- |
- |
| P08922 |
BXGT006843 |
Proto-oncogene tyrosine-protein kinase ROS |
reviewed |
Kinase |
ROS1 |
Ki |
'>' |
1995 |
nM |
| P08684 |
BXGT006812 |
Cytochrome P450 3A4 |
reviewed |
Enzyme |
CYP3A4 |
Activity |
- |
- |
- |
| Q6PHR2 |
BXGT016467 |
Serine/threonine-protein kinase ULK3 |
reviewed |
Kinase |
ULK3 |
Kd |
'>' |
10000 |
nM |
| Q13464 |
BXGT013357 |
Rho-associated protein kinase 1 |
reviewed |
Kinase |
ROCK1 |
Kd |
'>' |
10000 |
nM |
| P68400 |
BXGT011599 |
Casein kinase II subunit alpha |
reviewed |
Kinase |
CSNK2A1 |
Ki |
'>' |
6309 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd |
'=' |
5500 |
nM |
| Q8IVW4 |
BXGT018350 |
Cyclin-dependent kinase-like 3 |
reviewed |
Kinase |
CDKL3 |
Kd |
'>' |
10000 |
nM |
| P30530 |
BXGT009431 |
Tyrosine-protein kinase receptor UFO |
reviewed |
Kinase |
AXL |
Kd |
'=' |
1800 |
nM |
| P42679 |
BXGT010328 |
Megakaryocyte-associated tyrosine-protein kinase |
reviewed |
Kinase |
MATK |
Kd |
'>' |
10000 |
nM |
| Q04912 |
BXGT012790 |
Macrophage-stimulating protein receptor |
reviewed |
Kinase |
MST1R |
Kd |
'>' |
10000 |
nM |
| Q02763 |
BXGT012667 |
Angiopoietin-1 receptor |
reviewed |
Kinase |
TEK |
Kd |
- |
- |
- |
| Q9H2X6 |
BXGT020458 |
Homeodomain-interacting protein kinase 2 |
reviewed |
Kinase |
HIPK2 |
Ki |
'>' |
3162 |
nM |
| P16234 |
BXGT008209 |
Platelet-derived growth factor receptor alpha |
reviewed |
Kinase |
PDGFRA |
Ki |
'>' |
1995 |
nM |
| O94806 |
BXGT005335 |
Serine/threonine-protein kinase D3 |
reviewed |
Kinase |
PRKD3 |
Ki |
'=' |
1258 |
nM |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Ki |
'>' |
3981 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
35 |
% |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Kd |
'>' |
10000 |
nM |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Kd |
'>' |
10000 |
nM |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Kd |
'>' |
10000 |
nM |
| O94768 |
BXGT005331 |
Serine/threonine-protein kinase 17B |
reviewed |
Kinase |
STK17B |
Kd |
'=' |
3800 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
0 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
2 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
1 |
nM |
| Q8IVH8 |
BXGT018345 |
Mitogen-activated protein kinase kinase kinase kinase 3 |
reviewed |
Kinase |
MAP4K3 |
Kd |
'>' |
10000 |
nM |
| Q9Y4K4 |
BXGT022282 |
Mitogen-activated protein kinase kinase kinase kinase 5 |
reviewed |
Kinase |
MAP4K5 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Ki |
'=' |
3162 |
nM |
| Q5VT25 |
BXGT015887 |
Serine/threonine-protein kinase MRCK alpha |
reviewed |
Kinase |
CDC42BPA |
Ki |
'>' |
10000 |
nM |
| P53667 |
BXGT011008 |
LIM domain kinase 1 |
reviewed |
Kinase |
LIMK1 |
Kd |
- |
- |
- |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Kd |
- |
- |
- |
| Q2M2I8 |
BXGT014130 |
AP2-associated protein kinase 1 |
reviewed |
Kinase |
AAK1 |
Kd |
- |
- |
- |
| P08631 |
BXGT006801 |
Tyrosine-protein kinase HCK |
reviewed |
Kinase |
HCK |
Kd |
- |
- |
- |
| P54760 |
BXGT011075 |
Ephrin type-B receptor 4 |
reviewed |
Kinase |
EPHB4 |
Kd |
- |
- |
- |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Kd |
- |
- |
- |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Kd |
- |
- |
- |
| Q04759 |
BXGT012781 |
Protein kinase C theta type |
reviewed |
Kinase |
PRKCQ |
Ki |
'>' |
2511 |
nM |
| P07949 |
BXGT006703 |
Proto-oncogene tyrosine-protein kinase receptor Ret |
reviewed |
Kinase |
RET |
IC50 |
'=' |
1700 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
- |
- |
- |
| Q9H0K1 |
BXGT020438 |
Serine/threonine-protein kinase SIK2 |
reviewed |
Kinase |
SIK2 |
Ki |
'=' |
316 |
nM |
| P29597 |
BXGT009367 |
Non-receptor tyrosine-protein kinase TYK2 |
reviewed |
Kinase |
TYK2 |
Ki |
'>' |
1995 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Ki |
'>' |
6309 |
nM |
| Q9ULC5 |
BXGT021758 |
Long-chain-fatty-acid--CoA ligase 5 |
reviewed |
Enzyme |
ACSL5 |
Kd apparent |
'>' |
30000 |
nM |
| P31689 |
BXGT009569 |
DnaJ homolog subfamily A member 1 |
reviewed |
- |
DNAJA1 |
Kd apparent |
'>' |
30000 |
nM |
| O14920 |
BXGT004110 |
Inhibitor of nuclear factor kappa-B kinase subunit beta |
reviewed |
Kinase |
IKBKB |
Kd |
'>' |
10000 |
nM |
| Q9UK32 |
BXGT021736 |
Ribosomal protein S6 kinase alpha-6 |
reviewed |
Kinase |
RPS6KA6 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
93 |
% |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Kd apparent |
'>' |
30000 |
nM |
| P12931 |
BXGT007859 |
Proto-oncogene tyrosine-protein kinase Src |
reviewed |
Kinase |
SRC |
Kd apparent |
'>' |
30000 |
nM |
| P37173 |
BXGT009970 |
TGF-beta receptor type-2 |
reviewed |
Kinase |
TGFBR2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
80 |
nM |
| Q96PY6 |
BXGT019712 |
Serine/threonine-protein kinase Nek1 |
reviewed |
Kinase |
NEK1 |
Kd apparent |
'>' |
30000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
1604 |
nM |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Kd |
'=' |
1100 |
nM |
| P09769 |
BXGT006917 |
Tyrosine-protein kinase Fgr |
reviewed |
Kinase |
FGR |
Kd |
'>' |
10000 |
nM |
| P32298 |
BXGT009617 |
G protein-coupled receptor kinase 4 |
reviewed |
Kinase |
GRK4 |
Kd |
'>' |
10000 |
nM |
| Q9NSY1 |
BXGT021209 |
BMP-2-inducible protein kinase |
reviewed |
Kinase |
BMP2K |
Kd |
'>' |
10000 |
nM |
| Q56UN5 |
BXGT015107 |
Mitogen-activated protein kinase kinase kinase 19 |
reviewed |
Kinase |
MAP3K19 |
Kd |
'=' |
240 |
nM |
| Q96Q40 |
BXGT019714 |
Cyclin-dependent kinase 15 |
reviewed |
Kinase |
CDK15 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
480 |
nM |
| Q9H422 |
BXGT020469 |
Homeodomain-interacting protein kinase 3 |
reviewed |
Kinase |
HIPK3 |
Kd |
'>' |
10000 |
nM |
| P20794 |
BXGT008600 |
Serine/threonine-protein kinase MAK |
reviewed |
Kinase |
MAK |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
82 |
% |
| Q8N752 |
BXGT018526 |
Casein kinase I isoform alpha-like |
reviewed |
Kinase |
CSNK1A1L |
Kd |
'>' |
10000 |
nM |
| P48730 |
BXGT010656 |
Casein kinase I isoform delta |
reviewed |
Kinase |
CSNK1D |
Kd |
'>' |
10000 |
nM |
| O95342 |
BXGT005373 |
Bile salt export pump |
reviewed |
Transporter |
ABCB11 |
IC50 |
'=' |
10900 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
1260 |
nM |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Ki |
'>' |
2511 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
Inhibition |
'=' |
6 |
% |
| P54646 |
BXGT011062 |
5'-AMP-activated protein kinase catalytic subunit alpha-2 |
reviewed |
Kinase |
PRKAA2 |
Kd |
'>' |
10000 |
nM |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Kd |
'>' |
10000 |
nM |
| Q9H0K1 |
BXGT020438 |
Serine/threonine-protein kinase SIK2 |
reviewed |
Kinase |
SIK2 |
Inhibition |
'=' |
46 |
% |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Inhibition |
'=' |
46 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
70 |
nM |
| O15296 |
BXGT004148 |
Arachidonate 15-lipoxygenase B |
reviewed |
Enzyme |
ALOX15B |
Potency |
- |
19952 |
nM |
| P53778 |
BXGT011013 |
Mitogen-activated protein kinase 12 |
reviewed |
Kinase |
MAPK12 |
Kd |
- |
- |
- |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Kd |
- |
- |
- |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Kd |
- |
- |
- |
| Q9UQB9 |
BXGT021810 |
Aurora kinase C |
reviewed |
Kinase |
AURKC |
Kd |
- |
- |
- |
| P42684 |
BXGT010331 |
Tyrosine-protein kinase ABL2 |
reviewed |
Kinase |
ABL2 |
Kd |
'>' |
10000 |
nM |
| P07949 |
BXGT006703 |
Proto-oncogene tyrosine-protein kinase receptor Ret |
reviewed |
Kinase |
RET |
Ki |
'>' |
1258 |
nM |
| Q9NYL2 |
BXGT021259 |
Mitogen-activated protein kinase kinase kinase 20 |
reviewed |
Kinase |
MAP3K20 |
Ki |
'>' |
7943 |
nM |
| P05129 |
BXGT006322 |
Protein kinase C gamma type |
reviewed |
Kinase |
PRKCG |
Ki |
'>' |
7943 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd apparent |
'>' |
30000 |
nM |
| P09769 |
BXGT006917 |
Tyrosine-protein kinase Fgr |
reviewed |
Kinase |
FGR |
Kd apparent |
'>' |
30000 |
nM |
| Q6ZSR9 |
BXGT016637 |
Uncharacterized protein FLJ45252 |
reviewed |
- |
|
Kd apparent |
'>' |
30000 |
nM |
| P07332 |
BXGT006601 |
Tyrosine-protein kinase Fes/Fps |
reviewed |
Kinase |
FES |
Ki |
'>' |
1995 |
nM |
| P06241 |
BXGT006429 |
Tyrosine-protein kinase Fyn |
reviewed |
Kinase |
FYN |
Ki |
'>' |
794 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
4270 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
4270 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
4270 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
4270 |
nM |
| Q8TDC3 |
BXGT018808 |
Serine/threonine-protein kinase BRSK1 |
reviewed |
Kinase |
BRSK1 |
Kd |
'>' |
10000 |
nM |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Kd |
'>' |
10000 |
nM |
| Q6P3R8 |
BXGT016447 |
Serine/threonine-protein kinase Nek5 |
reviewed |
- |
NEK5 |
Kd |
'>' |
10000 |
nM |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Kd apparent |
'>' |
30000 |
nM |
| Q96GD4 |
BXGT019667 |
Aurora kinase B |
reviewed |
Kinase |
AURKB |
Kd apparent |
'>' |
30000 |
nM |
| Q9HBH9 |
BXGT020521 |
MAP kinase-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
MKNK2 |
Inhibition |
'=' |
46 |
% |
| Q02880 |
BXGT012677 |
DNA topoisomerase 2-beta |
reviewed |
- |
TOP2B |
Kd apparent |
'>' |
30000 |
nM |
| P22234 |
BXGT008745 |
Multifunctional protein ADE2 |
reviewed |
Enzyme |
PAICS |
Kd apparent |
'>' |
30000 |
nM |
| O75643 |
BXGT005142 |
U5 small nuclear ribonucleoprotein 200 kDa helicase |
reviewed |
- |
SNRNP200 |
Kd apparent |
'>' |
30000 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
29855 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
7 |
nM |
| Q9UBE8 |
BXGT021652 |
Serine/threonine-protein kinase NLK |
reviewed |
Kinase |
NLK |
Kd |
'>' |
10000 |
nM |
| Q14164 |
BXGT013451 |
Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
reviewed |
Kinase |
IKBKE |
Kd |
'>' |
10000 |
nM |
| P68370 |
BXGT011596 |
Tubulin alpha-1A chain |
reviewed |
- |
Tuba1a |
Kd |
'=' |
410 |
nM |
| Q04912 |
BXGT012790 |
Macrophage-stimulating protein receptor |
reviewed |
Kinase |
MST1R |
Ki |
'>' |
3981 |
nM |
| Q15375 |
BXGT013562 |
Ephrin type-A receptor 7 |
reviewed |
Kinase |
EPHA7 |
Kd |
'>' |
10000 |
nM |
| P29322 |
BXGT009333 |
Ephrin type-A receptor 8 |
reviewed |
Kinase |
EPHA8 |
Kd |
'=' |
1800 |
nM |
| P51817 |
BXGT010895 |
cAMP-dependent protein kinase catalytic subunit PRKX |
reviewed |
Kinase |
PRKX |
Kd |
'>' |
10000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
400 |
nM |
| P31751 |
BXGT009576 |
RAC-beta serine/threonine-protein kinase |
reviewed |
Kinase |
AKT2 |
Ki |
'>' |
7943 |
nM |
| P11799 |
BXGT007749 |
Myosin light chain kinase, smooth muscle |
reviewed |
- |
Mylk |
Kd |
'>' |
10000 |
nM |
| P29323 |
BXGT009334 |
Ephrin type-B receptor 2 |
reviewed |
Kinase |
EPHB2 |
Kd |
'>' |
10000 |
nM |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Ki |
'>' |
1000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
832 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
832 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
832 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
832 |
nM |
| P15735 |
BXGT008151 |
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform |
reviewed |
Kinase |
PHKG2 |
Kd |
'=' |
2700 |
nM |
| Q86V86 |
BXGT017617 |
Serine/threonine-protein kinase pim-3 |
reviewed |
- |
PIM3 |
Kd |
'=' |
5800 |
nM |
| Q8WU08 |
BXGT018990 |
Serine/threonine-protein kinase 32A |
reviewed |
Kinase |
STK32A |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1 |
nM |
| Q9BVS4 |
BXGT020147 |
Serine/threonine-protein kinase RIO2 |
reviewed |
Kinase |
RIOK2 |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
2900 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
4700 |
nM |
| Q12852 |
BXGT013272 |
Mitogen-activated protein kinase kinase kinase 12 |
reviewed |
Kinase |
MAP3K12 |
Kd |
'>' |
10000 |
nM |
| P0C264 |
BXGT007408 |
Uncharacterized serine/threonine-protein kinase SBK3 |
reviewed |
- |
SBK3 |
Kd |
'>' |
10000 |
nM |
| P62344 |
BXGT011426 |
Calcium-dependent protein kinase 1 |
reviewed |
- |
CPK1 |
Kd |
'>' |
10000 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
Kd apparent |
'>' |
30000 |
nM |
| O75716 |
BXGT005147 |
Serine/threonine-protein kinase 16 |
reviewed |
Kinase |
STK16 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q8TD19 |
BXGT018804 |
Serine/threonine-protein kinase Nek9 |
reviewed |
Kinase |
NEK9 |
Kd apparent |
'>' |
30000 |
nM |
| P46734 |
BXGT010537 |
Dual specificity mitogen-activated protein kinase kinase 3 |
reviewed |
Kinase |
MAP2K3 |
Kd apparent |
'>' |
30000 |
nM |
| Q01813 |
BXGT012618 |
ATP-dependent 6-phosphofructokinase, platelet type |
reviewed |
Kinase |
PFKP |
Kd apparent |
'>' |
30000 |
nM |
| Q9H0A0 |
BXGT020434 |
RNA cytidine acetyltransferase |
reviewed |
- |
NAT10 |
Kd apparent |
'>' |
30000 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Kd apparent |
'>' |
30000 |
nM |
| Q13177 |
BXGT013323 |
Serine/threonine-protein kinase PAK 2 |
reviewed |
Kinase |
PAK2 |
Kd apparent |
'>' |
30000 |
nM |
| P49589 |
BXGT010714 |
Cysteine--tRNA ligase, cytoplasmic |
reviewed |
Enzyme |
CARS1 |
Kd apparent |
'>' |
30000 |
nM |
| P16591 |
BXGT008246 |
Tyrosine-protein kinase Fer |
reviewed |
Kinase |
FER |
Ki |
'>' |
1584 |
nM |
| P53667 |
BXGT011008 |
LIM domain kinase 1 |
reviewed |
Kinase |
LIMK1 |
Kd apparent |
'>' |
30000 |
nM |
| P42336 |
BXGT010302 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform |
reviewed |
Kinase |
PIK3CA |
IC50 |
- |
- |
- |
| P11473 |
BXGT007709 |
Vitamin D3 receptor |
reviewed |
Nuclear receptor |
VDR |
Potency |
- |
89125 |
nM |
| P25098 |
BXGT009015 |
Beta-adrenergic receptor kinase 1 |
reviewed |
Kinase |
GRK2 |
Kd apparent |
'>' |
30000 |
nM |
| P49411 |
BXGT010703 |
Elongation factor Tu, mitochondrial |
reviewed |
Enzyme |
TUFM |
Kd apparent |
'>' |
30000 |
nM |
| Q9UM73 |
BXGT021773 |
ALK tyrosine kinase receptor |
reviewed |
Kinase |
ALK |
Ki |
'>' |
1258 |
nM |
| P49748 |
BXGT010733 |
Very long-chain specific acyl-CoA dehydrogenase, mitochondrial |
reviewed |
Enzyme |
ACADVL |
Kd apparent |
'>' |
30000 |
nM |
| P31751 |
BXGT009576 |
RAC-beta serine/threonine-protein kinase |
reviewed |
Kinase |
AKT2 |
Kd apparent |
'>' |
30000 |
nM |
| O14578 |
BXGT004072 |
Citron Rho-interacting kinase |
reviewed |
Kinase |
CIT |
Kd apparent |
'>' |
30000 |
nM |
| Q08345 |
BXGT012982 |
Epithelial discoidin domain-containing receptor 1 |
reviewed |
Kinase |
DDR1 |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
8 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
8 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
8 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
8 |
nM |
| Q16816 |
BXGT013673 |
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform |
reviewed |
Kinase |
PHKG1 |
Kd |
- |
- |
- |
| Q7KZI7 |
BXGT016990 |
Serine/threonine-protein kinase MARK2 |
reviewed |
Kinase |
MARK2 |
Kd |
- |
- |
- |
| P10721 |
BXGT007605 |
Mast/stem cell growth factor receptor Kit |
reviewed |
Kinase |
KIT |
Kd |
- |
- |
- |
| P25094 |
BXGT009014 |
Peripheral myelin protein 22 |
reviewed |
- |
Pmp22 |
Potency |
- |
36125 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3100 |
nM |
| Q16832 |
BXGT013678 |
Discoidin domain-containing receptor 2 |
reviewed |
Kinase |
DDR2 |
Kd apparent |
'>' |
30000 |
nM |
| Q05655 |
BXGT012832 |
Protein kinase C delta type |
reviewed |
Kinase |
PRKCD |
Kd apparent |
'>' |
30000 |
nM |
| P54756 |
BXGT011074 |
Ephrin type-A receptor 5 |
reviewed |
Kinase |
EPHA5 |
Kd apparent |
'>' |
30000 |
nM |
| Q9H2G2 |
BXGT020452 |
STE20-like serine/threonine-protein kinase |
reviewed |
Kinase |
SLK |
Kd apparent |
'>' |
30000 |
nM |
| O75385 |
BXGT005121 |
Serine/threonine-protein kinase ULK1 |
reviewed |
Kinase |
ULK1 |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
22 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
22 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
22 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
22 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'>' |
10000 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
11 |
nM |
| O75496 |
BXGT005132 |
Geminin |
reviewed |
- |
GMNN |
Potency |
- |
13335 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
15 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
11 |
nM |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Ki |
'>' |
2511 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
98 |
% |
| Q96RG2 |
BXGT019726 |
PAS domain-containing serine/threonine-protein kinase |
reviewed |
Kinase |
PASK |
Ki |
'>' |
1584 |
nM |
| Q7L7X3 |
BXGT016997 |
Serine/threonine-protein kinase TAO1 |
reviewed |
Kinase |
TAOK1 |
Ki |
'>' |
6309 |
nM |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Ki |
'>' |
1258 |
nM |
| Q13237 |
BXGT013331 |
cGMP-dependent protein kinase 2 |
reviewed |
Kinase |
PRKG2 |
Ki |
'>' |
1584 |
nM |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Ki |
'>' |
3981 |
nM |
| Q7Z406 |
BXGT017251 |
Myosin-14 |
reviewed |
- |
MYH14 |
Kd apparent |
'>' |
30000 |
nM |
| Q92499 |
BXGT019350 |
ATP-dependent RNA helicase DDX1 |
reviewed |
- |
DDX1 |
Kd apparent |
'>' |
30000 |
nM |
| P30085 |
BXGT009399 |
UMP-CMP kinase |
reviewed |
Kinase |
CMPK1 |
Kd apparent |
'>' |
30000 |
nM |
| Q6ZN16 |
BXGT016630 |
Mitogen-activated protein kinase kinase kinase 15 |
reviewed |
- |
MAP3K15 |
Kd |
'>' |
10000 |
nM |
| Q16288 |
BXGT013625 |
NT-3 growth factor receptor |
reviewed |
Kinase |
NTRK3 |
Kd |
'>' |
10000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
3700 |
nM |
| Q13233 |
BXGT013330 |
Mitogen-activated protein kinase kinase kinase 1 |
reviewed |
Kinase |
MAP3K1 |
Kd |
'>' |
10000 |
nM |
| Q9NRP7 |
BXGT021192 |
Serine/threonine-protein kinase 36 |
reviewed |
Kinase |
STK36 |
Kd |
'=' |
5700 |
nM |
| P0C1S8 |
BXGT007404 |
Wee1-like protein kinase 2 |
reviewed |
- |
WEE2 |
Kd |
'>' |
10000 |
nM |
| O14936 |
BXGT004114 |
Peripheral plasma membrane protein CASK |
reviewed |
Kinase |
CASK |
Kd |
'>' |
10000 |
nM |
| Q9Y2K2 |
BXGT022238 |
Serine/threonine-protein kinase SIK3 |
reviewed |
Kinase |
SIK3 |
Kd |
'>' |
10000 |
nM |
| P08581 |
BXGT006794 |
Hepatocyte growth factor receptor |
reviewed |
Kinase |
MET |
Kd |
'=' |
3500 |
nM |
| P19784 |
BXGT008513 |
Casein kinase II subunit alpha' |
reviewed |
Kinase |
CSNK2A2 |
Kd |
'>' |
10000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
Kd |
'=' |
790 |
nM |
| Q9UBF8 |
BXGT021653 |
Phosphatidylinositol 4-kinase beta |
reviewed |
Kinase |
PI4KB |
Kd |
'>' |
10000 |
nM |
| Q15139 |
BXGT013546 |
Serine/threonine-protein kinase D1 |
reviewed |
Kinase |
PRKD1 |
Kd |
'=' |
3500 |
nM |
| O15264 |
BXGT004144 |
Mitogen-activated protein kinase 13 |
reviewed |
Kinase |
MAPK13 |
Kd |
'>' |
10000 |
nM |
| O76039 |
BXGT005171 |
Cyclin-dependent kinase-like 5 |
reviewed |
Kinase |
CDKL5 |
Kd |
'>' |
10000 |
nM |
| O15530 |
BXGT004177 |
3-phosphoinositide-dependent protein kinase 1 |
reviewed |
Kinase |
PDPK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Thermal melting change |
'=' |
0 |
degrees C |
| P56817 |
BXGT011200 |
Beta-secretase 1 |
reviewed |
Enzyme |
BACE1 |
IC50 |
'=' |
20000 |
nM |
| Q9HAZ1 |
BXGT020511 |
Dual specificity protein kinase CLK4 |
reviewed |
- |
CLK4 |
Ki |
'>' |
6309 |
nM |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
IC50 |
- |
- |
- |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
0 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
0 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
0 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1080 |
nM |
| Q12851 |
BXGT013271 |
Mitogen-activated protein kinase kinase kinase kinase 2 |
reviewed |
Kinase |
MAP4K2 |
Ki |
'>' |
5011 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
0 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
0 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
0 |
nM |
| Q06418 |
BXGT012875 |
Tyrosine-protein kinase receptor TYRO3 |
reviewed |
Kinase |
TYRO3 |
Ki |
'>' |
1995 |
nM |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Ki |
'>' |
6309 |
nM |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
Kd |
'>' |
10000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
3100 |
nM |
| O95747 |
BXGT005393 |
Serine/threonine-protein kinase OSR1 |
reviewed |
Kinase |
OXSR1 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
780 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
460 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
360 |
nM |
| Q9Y2U5 |
BXGT022248 |
Mitogen-activated protein kinase kinase kinase 2 |
reviewed |
Kinase |
MAP3K2 |
Kd |
'=' |
3300 |
nM |
| O94921 |
BXGT005341 |
Cyclin-dependent kinase 14 |
reviewed |
Kinase |
CDK14 |
Kd |
'>' |
10000 |
nM |
| Q9NRH2 |
BXGT021188 |
SNF-related serine/threonine-protein kinase |
reviewed |
Kinase |
SNRK |
Kd |
'>' |
10000 |
nM |
| O14733 |
BXGT004087 |
Dual specificity mitogen-activated protein kinase kinase 7 |
reviewed |
Kinase |
MAP2K7 |
Kd |
'>' |
10000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
62 |
nM |
| P52333 |
BXGT010928 |
Tyrosine-protein kinase JAK3 |
reviewed |
Kinase |
JAK3 |
IC50 |
'>' |
1000 |
nM |
| P57078 |
BXGT011211 |
Receptor-interacting serine/threonine-protein kinase 4 |
reviewed |
Kinase |
RIPK4 |
Kd |
'>' |
10000 |
nM |
| Q9H093 |
BXGT020433 |
NUAK family SNF1-like kinase 2 |
reviewed |
Kinase |
NUAK2 |
Kd |
'=' |
4600 |
nM |
| P9WI81 |
BXGT012312 |
Serine/threonine-protein kinase PknB |
reviewed |
- |
pknB |
Kd |
'>' |
10000 |
nM |
| Q8NE63 |
BXGT018551 |
Homeodomain-interacting protein kinase 4 |
reviewed |
Kinase |
HIPK4 |
Kd |
'=' |
310 |
nM |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
Kd |
'>' |
10000 |
nM |
| P61075 |
BXGT011353 |
Cell division control protein 2 homolog |
reviewed |
- |
CRK2 |
Kd |
'>' |
10000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
173 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
173 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
173 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
173 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| Q7L7X3 |
BXGT016997 |
Serine/threonine-protein kinase TAO1 |
reviewed |
Kinase |
TAOK1 |
Kd apparent |
'>' |
30000 |
nM |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Ki |
'=' |
794 |
nM |
| P29597 |
BXGT009367 |
Non-receptor tyrosine-protein kinase TYK2 |
reviewed |
Kinase |
TYK2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
1013 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
1013 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1013 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
1013 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
- |
- |
- |
| Q04759 |
BXGT012781 |
Protein kinase C theta type |
reviewed |
Kinase |
PRKCQ |
Kd apparent |
'>' |
30000 |
nM |
| Q7KZI7 |
BXGT016990 |
Serine/threonine-protein kinase MARK2 |
reviewed |
Kinase |
MARK2 |
Kd apparent |
'>' |
30000 |
nM |
| Q96S44 |
BXGT019738 |
EKC/KEOPS complex subunit TP53RK |
reviewed |
Kinase |
TP53RK |
Kd apparent |
'>' |
30000 |
nM |
| Q14004 |
BXGT013435 |
Cyclin-dependent kinase 13 |
reviewed |
Kinase |
CDK13 |
Kd |
'>' |
10000 |
nM |
| P45983 |
BXGT010494 |
Mitogen-activated protein kinase 8 |
reviewed |
Kinase |
MAPK8 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
9 |
nM |
| Q9NU22 |
BXGT021214 |
Midasin |
reviewed |
- |
MDN1 |
Kd apparent |
'>' |
30000 |
nM |
| Q15831 |
BXGT013604 |
Serine/threonine-protein kinase STK11 |
reviewed |
Kinase |
STK11 |
Kd apparent |
'>' |
30000 |
nM |
| Q5S007 |
BXGT015650 |
Leucine-rich repeat serine/threonine-protein kinase 2 |
reviewed |
Kinase |
LRRK2 |
Ki |
'>' |
2511 |
nM |
| Q14164 |
BXGT013451 |
Inhibitor of nuclear factor kappa-B kinase subunit epsilon |
reviewed |
Kinase |
IKBKE |
Ki |
'>' |
3162 |
nM |
| Q9HBH9 |
BXGT020521 |
MAP kinase-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
MKNK2 |
Ki |
'=' |
398 |
nM |
| P04629 |
BXGT006239 |
High affinity nerve growth factor receptor |
reviewed |
Kinase |
NTRK1 |
Ki |
'>' |
2511 |
nM |
| P51617 |
BXGT010868 |
Interleukin-1 receptor-associated kinase 1 |
reviewed |
Kinase |
IRAK1 |
Kd |
'=' |
69 |
nM |
| Q13233 |
BXGT013330 |
Mitogen-activated protein kinase kinase kinase 1 |
reviewed |
Kinase |
MAP3K1 |
Kd apparent |
'>' |
30000 |
nM |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Inhibition |
'=' |
46 |
% |
| Q14839 |
BXGT013509 |
Chromodomain-helicase-DNA-binding protein 4 |
reviewed |
- |
CHD4 |
Kd apparent |
'>' |
30000 |
nM |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Ki |
'>' |
1995 |
nM |
| Q9H3Y6 |
BXGT020468 |
Tyrosine-protein kinase Srms |
reviewed |
Kinase |
SRMS |
Ki |
'>' |
1584 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Ki |
'=' |
25 |
nM |
| P08631 |
BXGT006801 |
Tyrosine-protein kinase HCK |
reviewed |
Kinase |
HCK |
Kd apparent |
'>' |
30000 |
nM |
| Q9UNQ0 |
BXGT021792 |
ATP-binding cassette sub-family G member 2 |
reviewed |
Transporter |
ABCG2 |
IC50 |
'=' |
3190 |
nM |
| Q9NQU5 |
BXGT021169 |
Serine/threonine-protein kinase PAK 6 |
reviewed |
- |
PAK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q00536 |
BXGT012535 |
Cyclin-dependent kinase 16 |
reviewed |
Kinase |
CDK16 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q99986 |
BXGT019980 |
Serine/threonine-protein kinase VRK1 |
reviewed |
Kinase |
VRK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Inhibition |
- |
- |
- |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
IC50 |
'=' |
1200 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
46 |
% |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Kd |
- |
- |
- |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Kd |
- |
- |
- |
| Q14012 |
BXGT013437 |
Calcium/calmodulin-dependent protein kinase type 1 |
reviewed |
Kinase |
CAMK1 |
Kd |
- |
- |
- |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
55 |
% |
| O75676 |
BXGT005144 |
Ribosomal protein S6 kinase alpha-4 |
reviewed |
Kinase |
RPS6KA4 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
14 |
nM |
| Q13976 |
BXGT013409 |
cGMP-dependent protein kinase 1 |
reviewed |
Kinase |
PRKG1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13131 |
BXGT013314 |
5'-AMP-activated protein kinase catalytic subunit alpha-1 |
reviewed |
Kinase |
PRKAA1 |
Kd |
'>' |
10000 |
nM |
| Q9UHD2 |
BXGT021697 |
Serine/threonine-protein kinase TBK1 |
reviewed |
Kinase |
TBK1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13464 |
BXGT013357 |
Rho-associated protein kinase 1 |
reviewed |
Kinase |
ROCK1 |
Kd apparent |
'>' |
30000 |
nM |
| P20340 |
BXGT008566 |
Ras-related protein Rab-6A |
reviewed |
- |
RAB6A |
Kd apparent |
'>' |
30000 |
nM |
| Q13554 |
BXGT013374 |
Calcium/calmodulin-dependent protein kinase type II subunit beta |
reviewed |
Kinase |
CAMK2B |
Thermal melting change |
'=' |
0 |
degrees C |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Kd |
- |
- |
- |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Ki |
'>' |
794 |
nM |
| Q00537 |
BXGT012536 |
Cyclin-dependent kinase 17 |
reviewed |
Kinase |
CDK17 |
Kd apparent |
'>' |
30000 |
nM |
| P0A0J7 |
BXGT006970 |
Quinolone resistance protein NorA |
reviewed |
- |
norA |
FC |
'=' |
16 |
- |
| Q9BUB5 |
BXGT020133 |
MAP kinase-interacting serine/threonine-protein kinase 1 |
reviewed |
Kinase |
MKNK1 |
Inhibition |
'=' |
46 |
% |
| Q86XP3 |
BXGT017630 |
ATP-dependent RNA helicase DDX42 |
reviewed |
- |
DDX42 |
Kd apparent |
'>' |
30000 |
nM |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1100 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
25 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
25 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
25 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
25 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Kd apparent |
'>' |
30000 |
nM |
| P26196 |
BXGT009089 |
Probable ATP-dependent RNA helicase DDX6 |
reviewed |
- |
DDX6 |
Kd apparent |
'>' |
30000 |
nM |
| Q13164 |
BXGT013322 |
Mitogen-activated protein kinase 7 |
reviewed |
Kinase |
MAPK7 |
Kd apparent |
'>' |
30000 |
nM |
| Q14683 |
BXGT013500 |
Structural maintenance of chromosomes protein 1A |
reviewed |
- |
SMC1A |
Kd apparent |
'>' |
30000 |
nM |
| Q07912 |
BXGT012947 |
Activated CDC42 kinase 1 |
reviewed |
Kinase |
TNK2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
76 |
nM |
| Q15418 |
BXGT013569 |
Ribosomal protein S6 kinase alpha-1 |
reviewed |
Kinase |
RPS6KA1 |
Kd apparent |
'>' |
30000 |
nM |
| Q6PHR2 |
BXGT016467 |
Serine/threonine-protein kinase ULK3 |
reviewed |
Kinase |
ULK3 |
Kd apparent |
'>' |
30000 |
nM |
| P42680 |
BXGT010329 |
Tyrosine-protein kinase Tec |
reviewed |
Kinase |
TEC |
Kd apparent |
'>' |
30000 |
nM |
| Q00535 |
BXGT012534 |
Cyclin-dependent-like kinase 5 |
reviewed |
Kinase |
CDK5 |
Kd apparent |
'>' |
30000 |
nM |
| Q86TW2 |
BXGT017609 |
Uncharacterized aarF domain-containing protein kinase 1 |
reviewed |
Kinase |
ADCK1 |
Kd apparent |
'>' |
30000 |
nM |
| P49841 |
BXGT010750 |
Glycogen synthase kinase-3 beta |
reviewed |
Kinase |
GSK3B |
Thermal melting change |
'=' |
0 |
degrees C |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Kd apparent |
'>' |
30000 |
nM |
| Q05513 |
BXGT012820 |
Protein kinase C zeta type |
reviewed |
Kinase |
PRKCZ |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| O60674 |
BXGT004892 |
Tyrosine-protein kinase JAK2 |
reviewed |
Kinase |
JAK2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
6 |
nM |
| P45984 |
BXGT010495 |
Mitogen-activated protein kinase 9 |
reviewed |
Kinase |
MAPK9 |
Kd apparent |
'>' |
30000 |
nM |
| P11216 |
BXGT007673 |
Glycogen phosphorylase, brain form |
reviewed |
Enzyme |
PYGB |
Kd apparent |
'>' |
30000 |
nM |
| P51956 |
BXGT010909 |
Serine/threonine-protein kinase Nek3 |
reviewed |
Kinase |
NEK3 |
Kd apparent |
'>' |
30000 |
nM |
| Q96RR4 |
BXGT019734 |
Calcium/calmodulin-dependent protein kinase kinase 2 |
reviewed |
Kinase |
CAMKK2 |
Kd apparent |
'>' |
30000 |
nM |
| P08574 |
BXGT006792 |
Cytochrome c1, heme protein, mitochondrial |
reviewed |
- |
CYC1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
26 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Ki |
'=' |
398 |
nM |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Potency |
- |
1729 |
nM |
| Q05397 |
BXGT012815 |
Focal adhesion kinase 1 |
reviewed |
Kinase |
PTK2 |
Ki |
'>' |
1584 |
nM |
| P48730 |
BXGT010656 |
Casein kinase I isoform delta |
reviewed |
Kinase |
CSNK1D |
Kd apparent |
'>' |
30000 |
nM |
| O00238 |
BXGT003900 |
Bone morphogenetic protein receptor type-1B |
reviewed |
Kinase |
BMPR1B |
Kd apparent |
'>' |
30000 |
nM |
| Q13523 |
BXGT013368 |
Serine/threonine-protein kinase PRP4 homolog |
reviewed |
Kinase |
PRPF4B |
Kd |
'>' |
10000 |
nM |
| O75676 |
BXGT005144 |
Ribosomal protein S6 kinase alpha-4 |
reviewed |
Kinase |
RPS6KA4 |
Kd |
'=' |
1200 |
nM |
| O15197 |
BXGT004136 |
Ephrin type-B receptor 6 |
reviewed |
Kinase |
EPHB6 |
Kd |
'=' |
3200 |
nM |
| O95382 |
BXGT005376 |
Mitogen-activated protein kinase kinase kinase 6 |
reviewed |
Kinase |
MAP3K6 |
Kd |
'>' |
10000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
2200 |
nM |
| P42338 |
BXGT010303 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform |
reviewed |
Kinase |
PIK3CB |
Kd |
'>' |
10000 |
nM |
| Q9H2K8 |
BXGT020455 |
Serine/threonine-protein kinase TAO3 |
reviewed |
Kinase |
TAOK3 |
Kd |
'>' |
10000 |
nM |
| Q7L7X3 |
BXGT016997 |
Serine/threonine-protein kinase TAO1 |
reviewed |
Kinase |
TAOK1 |
Kd |
'>' |
10000 |
nM |
| Q8NG66 |
BXGT018566 |
Serine/threonine-protein kinase Nek11 |
reviewed |
Kinase |
NEK11 |
Kd |
'>' |
10000 |
nM |
| Q8IY84 |
BXGT018364 |
Serine/threonine-protein kinase NIM1 |
reviewed |
Kinase |
NIM1K |
Kd |
'>' |
10000 |
nM |
| P04899 |
BXGT006281 |
Guanine nucleotide-binding protein G(i) subunit alpha-2 |
reviewed |
Enzyme modulator |
GNAI2 |
Kd apparent |
'>' |
30000 |
nM |
| P16083 |
BXGT008187 |
Ribosyldihydronicotinamide dehydrogenase [quinone] |
reviewed |
- |
NQO2 |
Kd apparent |
'>' |
30000 |
nM |
| Q16539 |
BXGT013634 |
Mitogen-activated protein kinase 14 |
reviewed |
Kinase |
MAPK14 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
140 |
nM |
| Q9BQI3 |
BXGT020113 |
Eukaryotic translation initiation factor 2-alpha kinase 1 |
reviewed |
Kinase |
EIF2AK1 |
Kd |
'>' |
10000 |
nM |
| Q9NRM7 |
BXGT021190 |
Serine/threonine-protein kinase LATS2 |
reviewed |
Kinase |
LATS2 |
Kd |
'>' |
10000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
100 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
100 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
100 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
100 |
nM |
| P17612 |
BXGT008322 |
cAMP-dependent protein kinase catalytic subunit alpha |
reviewed |
Kinase |
PRKACA |
Thermal melting change |
'=' |
1 |
degrees C |
| Q9HC98 |
BXGT020528 |
Serine/threonine-protein kinase Nek6 |
reviewed |
Kinase |
NEK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3 |
nM |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| O43293 |
BXGT004584 |
Death-associated protein kinase 3 |
reviewed |
Kinase |
DAPK3 |
Thermal melting change |
'=' |
3 |
degrees C |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9BVS4 |
BXGT020147 |
Serine/threonine-protein kinase RIO2 |
reviewed |
Kinase |
RIOK2 |
Thermal melting change |
'=' |
2 |
degrees C |
| Q15208 |
BXGT013550 |
Serine/threonine-protein kinase 38 |
reviewed |
Kinase |
STK38 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q86Y07 |
BXGT017631 |
Serine/threonine-protein kinase VRK2 |
reviewed |
Kinase |
VRK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
1000 |
nM |
| Q9NSY1 |
BXGT021209 |
BMP-2-inducible protein kinase |
reviewed |
Kinase |
BMP2K |
Kd apparent |
'>' |
30000 |
nM |
| Q13555 |
BXGT013375 |
Calcium/calmodulin-dependent protein kinase type II subunit gamma |
reviewed |
Kinase |
CAMK2G |
Thermal melting change |
'=' |
0 |
degrees C |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q00532 |
BXGT012532 |
Cyclin-dependent kinase-like 1 |
reviewed |
Kinase |
CDKL1 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
IC50 |
- |
- |
- |
| Q01538 |
BXGT012597 |
Myelin transcription factor 1 |
reviewed |
Transcription factor |
MYT1 |
IC50 |
- |
- |
- |
| O43683 |
BXGT004614 |
Mitotic checkpoint serine/threonine-protein kinase BUB1 |
reviewed |
Kinase |
BUB1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Thermal melting change |
'=' |
0 |
degrees C |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd |
'=' |
5100 |
nM |
| P54760 |
BXGT011075 |
Ephrin type-B receptor 4 |
reviewed |
Kinase |
EPHB4 |
Kd |
'=' |
2500 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd |
'=' |
680 |
nM |
| O43318 |
BXGT004586 |
Mitogen-activated protein kinase kinase kinase 7 |
reviewed |
Kinase |
MAP3K7 |
Kd |
'>' |
10000 |
nM |
| Q5VT25 |
BXGT015887 |
Serine/threonine-protein kinase MRCK alpha |
reviewed |
Kinase |
CDC42BPA |
Kd apparent |
'>' |
30000 |
nM |
| P22694 |
BXGT008797 |
cAMP-dependent protein kinase catalytic subunit beta |
reviewed |
Kinase |
PRKACB |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
845 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
845 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
845 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
845 |
nM |
| P31153 |
BXGT009512 |
S-adenosylmethionine synthase isoform type-2 |
reviewed |
Enzyme |
MAT2A |
Kd apparent |
'>' |
30000 |
nM |
| Q9BXA7 |
BXGT020164 |
Testis-specific serine/threonine-protein kinase 1 |
reviewed |
Kinase |
TSSK1B |
Ki |
'>' |
1584 |
nM |
| O00311 |
BXGT003908 |
Cell division cycle 7-related protein kinase |
reviewed |
Kinase |
CDC7 |
Ki |
'>' |
1258 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
'=' |
48 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
65 |
% |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
24 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
127 |
nM |
| O96017 |
BXGT005415 |
Serine/threonine-protein kinase Chk2 |
reviewed |
Kinase |
CHEK2 |
Thermal melting change |
'=' |
3 |
degrees C |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
127 |
nM |
| P30291 |
BXGT009417 |
Wee1-like protein kinase |
reviewed |
Kinase |
WEE1 |
Kd apparent |
'>' |
30000 |
nM |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q12851 |
BXGT013271 |
Mitogen-activated protein kinase kinase kinase kinase 2 |
reviewed |
Kinase |
MAP4K2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'>' |
5000 |
nM |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P286 |
BXGT021299 |
Serine/threonine-protein kinase PAK 5 |
reviewed |
Kinase |
PAK5 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Thermal melting change |
'=' |
0 |
degrees C |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Thermal melting change |
'=' |
0 |
degrees C |
| P38117 |
BXGT010027 |
Electron transfer flavoprotein subunit beta |
reviewed |
Enzyme |
ETFB |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
6 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
6 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
6 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
6 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
3300 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
3300 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3300 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
3300 |
nM |
| Q9NUW8 |
BXGT021219 |
Tyrosyl-DNA phosphodiesterase 1 |
reviewed |
Enzyme |
TDP1 |
Potency |
- |
5309 |
nM |
| Q96RG2 |
BXGT019726 |
PAS domain-containing serine/threonine-protein kinase |
reviewed |
Kinase |
PASK |
Kd apparent |
'>' |
30000 |
nM |
| P12236 |
BXGT007775 |
ADP/ATP translocase 3 |
reviewed |
Transporter |
SLC25A6 |
Kd apparent |
'>' |
30000 |
nM |
| Q16659 |
BXGT013652 |
Mitogen-activated protein kinase 6 |
reviewed |
Kinase |
MAPK6 |
Thermal melting change |
'=' |
0 |
degrees C |
| P54577 |
BXGT011055 |
Tyrosine--tRNA ligase, cytoplasmic |
reviewed |
Enzyme |
YARS1 |
Kd apparent |
'>' |
30000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
1830 |
nM |
| Q9NSE4 |
BXGT021207 |
Isoleucine--tRNA ligase, mitochondrial |
reviewed |
Enzyme |
IARS2 |
Kd apparent |
'>' |
30000 |
nM |
| P11309 |
BXGT007685 |
Serine/threonine-protein kinase pim-1 |
reviewed |
Kinase |
PIM1 |
Thermal melting change |
'=' |
3 |
degrees C |
| P52564 |
BXGT010932 |
Dual specificity mitogen-activated protein kinase kinase 6 |
reviewed |
Kinase |
MAP2K6 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9HCP0 |
BXGT020536 |
Casein kinase I isoform gamma-1 |
reviewed |
Kinase |
CSNK1G1 |
Thermal melting change |
'=' |
0 |
degrees C |
| P51955 |
BXGT010908 |
Serine/threonine-protein kinase Nek2 |
reviewed |
Kinase |
NEK2 |
Thermal melting change |
'=' |
1 |
degrees C |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q96NX5 |
BXGT019702 |
Calcium/calmodulin-dependent protein kinase type 1G |
reviewed |
Kinase |
CAMK1G |
Thermal melting change |
'=' |
1 |
degrees C |
| Q8IU85 |
BXGT018333 |
Calcium/calmodulin-dependent protein kinase type 1D |
reviewed |
Kinase |
CAMK1D |
Thermal melting change |
'=' |
0 |
degrees C |
| P24941 |
BXGT009002 |
Cyclin-dependent kinase 2 |
reviewed |
Kinase |
CDK2 |
Thermal melting change |
'=' |
0 |
degrees C |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Thermal melting change |
'=' |
1 |
degrees C |
| O00506 |
BXGT003932 |
Serine/threonine-protein kinase 25 |
reviewed |
Kinase |
STK25 |
Thermal melting change |
- |
- |
- |
| P42684 |
BXGT010331 |
Tyrosine-protein kinase ABL2 |
reviewed |
Kinase |
ABL2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
498 |
nM |
| P36894 |
BXGT009939 |
Bone morphogenetic protein receptor type-1A |
reviewed |
Kinase |
BMPR1A |
Kd apparent |
'>' |
30000 |
nM |
| Q13705 |
BXGT013393 |
Activin receptor type-2B |
reviewed |
Kinase |
ACVR2B |
Kd apparent |
'>' |
30000 |
nM |
| P07332 |
BXGT006601 |
Tyrosine-protein kinase Fes/Fps |
reviewed |
Kinase |
FES |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y6R4 |
BXGT022340 |
Mitogen-activated protein kinase kinase kinase 4 |
reviewed |
Kinase |
MAP3K4 |
Kd apparent |
'>' |
30000 |
nM |
| P61026 |
BXGT011351 |
Ras-related protein Rab-10 |
reviewed |
- |
RAB10 |
Kd apparent |
'>' |
30000 |
nM |
| Q15759 |
BXGT013595 |
Mitogen-activated protein kinase 11 |
reviewed |
Kinase |
MAPK11 |
Kd apparent |
'>' |
30000 |
nM |
| P08069 |
BXGT006723 |
Insulin-like growth factor 1 receptor |
reviewed |
Kinase |
IGF1R |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
188 |
nM |
| Q14289 |
BXGT013459 |
Protein-tyrosine kinase 2-beta |
reviewed |
Kinase |
PTK2B |
Kd apparent |
'>' |
30000 |
nM |
| Q09013 |
BXGT013023 |
Myotonin-protein kinase |
reviewed |
Kinase |
DMPK |
Thermal melting change |
'=' |
3 |
degrees C |
| P41240 |
BXGT010242 |
Tyrosine-protein kinase CSK |
reviewed |
Kinase |
CSK |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
90 |
% |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
12720 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
12720 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
12720 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
12720 |
nM |
| Q9NYV4 |
BXGT021262 |
Cyclin-dependent kinase 12 |
reviewed |
Kinase |
CDK12 |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y2W1 |
BXGT022249 |
Thyroid hormone receptor-associated protein 3 |
reviewed |
Transcription factor |
THRAP3 |
Kd apparent |
'>' |
30000 |
nM |
| P36888 |
BXGT009938 |
Receptor-type tyrosine-protein kinase FLT3 |
reviewed |
Kinase |
FLT3 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
66 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
28 |
% |
| Q9UF33 |
BXGT021676 |
Ephrin type-A receptor 6 |
reviewed |
Kinase |
EPHA6 |
Inhibition |
'=' |
46 |
% |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Inhibition |
'=' |
46 |
% |
| Q14680 |
BXGT013499 |
Maternal embryonic leucine zipper kinase |
reviewed |
Kinase |
MELK |
Ki |
'>' |
1584 |
nM |
| P31749 |
BXGT009574 |
RAC-alpha serine/threonine-protein kinase |
reviewed |
Kinase |
AKT1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13163 |
BXGT013321 |
Dual specificity mitogen-activated protein kinase kinase 5 |
reviewed |
Kinase |
MAP2K5 |
Kd apparent |
'>' |
30000 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
10620 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
10620 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
10620 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
10620 |
nM |
| Q15067 |
BXGT013532 |
Peroxisomal acyl-coenzyme A oxidase 1 |
reviewed |
Enzyme |
ACOX1 |
Kd apparent |
'>' |
30000 |
nM |
| Q99759 |
BXGT019960 |
Mitogen-activated protein kinase kinase kinase 3 |
reviewed |
Kinase |
MAP3K3 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| O95819 |
BXGT005398 |
Mitogen-activated protein kinase kinase kinase kinase 4 |
reviewed |
Kinase |
MAP4K4 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Ki |
'=' |
0 |
nM |
| Q9Y6E0 |
BXGT022327 |
Serine/threonine-protein kinase 24 |
reviewed |
Kinase |
STK24 |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y2U5 |
BXGT022248 |
Mitogen-activated protein kinase kinase kinase 2 |
reviewed |
Kinase |
MAP3K2 |
Kd apparent |
'>' |
30000 |
nM |
| Q04912 |
BXGT012790 |
Macrophage-stimulating protein receptor |
reviewed |
Kinase |
MST1R |
Kd apparent |
'>' |
30000 |
nM |
| P41250 |
BXGT010244 |
Glycine--tRNA ligase |
reviewed |
Enzyme |
GARS1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13627 |
BXGT013385 |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A |
reviewed |
Kinase |
DYRK1A |
Kd apparent |
'>' |
30000 |
nM |
| Q9NTK5 |
BXGT021213 |
Obg-like ATPase 1 |
reviewed |
Enzyme modulator |
OLA1 |
Kd apparent |
'>' |
30000 |
nM |
| P18074 |
BXGT008374 |
General transcription and DNA repair factor IIH helicase subunit XPD |
reviewed |
Enzyme |
ERCC2 |
Kd apparent |
'>' |
30000 |
nM |
| O15439 |
BXGT004169 |
Multidrug resistance-associated protein 4 |
reviewed |
Transporter |
ABCC4 |
IC50 |
'=' |
4600 |
nM |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Thermal melting change |
'=' |
1 |
degrees C |
| Q8N4C8 |
BXGT018510 |
Misshapen-like kinase 1 |
reviewed |
Kinase |
MINK1 |
IC50 |
'=' |
15000 |
nM |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
Inhibition |
'=' |
46 |
% |
| Q8TDX7 |
BXGT018817 |
Serine/threonine-protein kinase Nek7 |
reviewed |
Kinase |
NEK7 |
Kd apparent |
'>' |
30000 |
nM |
| Q02750 |
BXGT012662 |
Dual specificity mitogen-activated protein kinase kinase 1 |
reviewed |
Kinase |
MAP2K1 |
Kd apparent |
'>' |
30000 |
nM |
| Q14680 |
BXGT013499 |
Maternal embryonic leucine zipper kinase |
reviewed |
Kinase |
MELK |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P51159 |
BXGT010839 |
Ras-related protein Rab-27A |
reviewed |
- |
RAB27A |
Kd apparent |
'>' |
30000 |
nM |
| P43405 |
BXGT010386 |
Tyrosine-protein kinase SYK |
reviewed |
Kinase |
SYK |
Kd apparent |
'>' |
30000 |
nM |
| P36507 |
BXGT009923 |
Dual specificity mitogen-activated protein kinase kinase 2 |
reviewed |
Kinase |
MAP2K2 |
Kd apparent |
'>' |
30000 |
nM |
| P05771 |
BXGT006384 |
Protein kinase C beta type |
reviewed |
Kinase |
PRKCB |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
9 |
nM |
| Q9UHD8 |
BXGT021698 |
Septin-9 |
reviewed |
Enzyme modulator |
SEPTIN9 |
Kd apparent |
'>' |
30000 |
nM |
| P06493 |
BXGT006445 |
Cyclin-dependent kinase 1 |
reviewed |
Kinase |
CDK1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
EC50 |
'=' |
10733 |
nM |
| O14757 |
BXGT004092 |
Serine/threonine-protein kinase Chk1 |
reviewed |
Kinase |
CHEK1 |
Kd apparent |
'>' |
30000 |
nM |
| P51617 |
BXGT010868 |
Interleukin-1 receptor-associated kinase 1 |
reviewed |
Kinase |
IRAK1 |
Kd apparent |
'>' |
30000 |
nM |
| Q9H093 |
BXGT020433 |
NUAK family SNF1-like kinase 2 |
reviewed |
Kinase |
NUAK2 |
Kd apparent |
'>' |
30000 |
nM |
| Q58FF8 |
BXGT015229 |
Putative heat shock protein HSP 90-beta 2 |
reviewed |
- |
HSP90AB2P |
Kd apparent |
'>' |
30000 |
nM |
| P06239 |
BXGT006427 |
Tyrosine-protein kinase Lck |
reviewed |
Kinase |
LCK |
Kd apparent |
'>' |
30000 |
nM |
| O00571 |
BXGT003938 |
ATP-dependent RNA helicase DDX3X |
reviewed |
- |
DDX3X |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
27 |
nM |
| P11388 |
BXGT007697 |
DNA topoisomerase 2-alpha |
reviewed |
- |
TOP2A |
Kd apparent |
'>' |
30000 |
nM |
| Q8IYD1 |
BXGT018366 |
Eukaryotic peptide chain release factor GTP-binding subunit ERF3B |
reviewed |
Enzyme |
GSPT2 |
Kd apparent |
'>' |
30000 |
nM |
| Q99683 |
BXGT019947 |
Mitogen-activated protein kinase kinase kinase 5 |
reviewed |
Kinase |
MAP3K5 |
Kd apparent |
'>' |
30000 |
nM |
| P00519 |
BXGT005570 |
Tyrosine-protein kinase ABL1 |
reviewed |
Kinase |
ABL1 |
Kd apparent |
'>' |
30000 |
nM |
| Q969S8 |
BXGT019613 |
Polyamine deacetylase HDAC10 |
reviewed |
Epigenetic regulator |
HDAC10 |
IC50 |
- |
- |
- |
| Q9UKV0 |
BXGT021750 |
Histone deacetylase 9 |
reviewed |
Epigenetic regulator |
HDAC9 |
IC50 |
- |
- |
- |
| P56524 |
BXGT011176 |
Histone deacetylase 4 |
reviewed |
Epigenetic regulator |
HDAC4 |
IC50 |
- |
- |
- |
| Q96DB2 |
BXGT019639 |
Histone deacetylase 11 |
reviewed |
Epigenetic regulator |
HDAC11 |
IC50 |
- |
- |
- |
| Q9BY41 |
BXGT020180 |
Histone deacetylase 8 |
reviewed |
Epigenetic regulator |
HDAC8 |
IC50 |
- |
- |
- |
| Q8WUI4 |
BXGT018992 |
Histone deacetylase 7 |
reviewed |
Epigenetic regulator |
HDAC7 |
IC50 |
- |
- |
- |
| Q9UQL6 |
BXGT021813 |
Histone deacetylase 5 |
reviewed |
Epigenetic regulator |
HDAC5 |
IC50 |
- |
- |
- |
| Q92769 |
BXGT019370 |
Histone deacetylase 2 |
reviewed |
Epigenetic regulator |
HDAC2 |
IC50 |
- |
- |
- |
| Q9UBN7 |
BXGT021658 |
Histone deacetylase 6 |
reviewed |
Epigenetic regulator |
HDAC6 |
IC50 |
- |
- |
- |
| O15379 |
BXGT004159 |
Histone deacetylase 3 |
reviewed |
Epigenetic regulator |
HDAC3 |
IC50 |
- |
- |
- |
| Q13547 |
BXGT013373 |
Histone deacetylase 1 |
reviewed |
Epigenetic regulator |
HDAC1 |
IC50 |
- |
- |
- |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
Kd |
'=' |
10 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
Kd |
'=' |
10 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd |
'=' |
10 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
Kd |
'=' |
10 |
nM |
| P21709 |
BXGT008685 |
Ephrin type-A receptor 1 |
reviewed |
Kinase |
EPHA1 |
Kd apparent |
'>' |
30000 |
nM |
| P33991 |
BXGT009745 |
DNA replication licensing factor MCM4 |
reviewed |
Enzyme |
MCM4 |
Kd apparent |
'>' |
30000 |
nM |
| O96013 |
BXGT005414 |
Serine/threonine-protein kinase PAK 4 |
reviewed |
Kinase |
PAK4 |
Kd apparent |
'>' |
30000 |
nM |
| Q14004 |
BXGT013435 |
Cyclin-dependent kinase 13 |
reviewed |
Kinase |
CDK13 |
Kd apparent |
'>' |
30000 |
nM |
| Q16288 |
BXGT013625 |
NT-3 growth factor receptor |
reviewed |
Kinase |
NTRK3 |
Ki |
'>' |
1258 |
nM |
| Q06187 |
BXGT012860 |
Tyrosine-protein kinase BTK |
reviewed |
Kinase |
BTK |
Kd apparent |
'>' |
30000 |
nM |
| Q01538 |
BXGT012597 |
Myelin transcription factor 1 |
reviewed |
Transcription factor |
MYT1 |
Activity |
'=' |
6 |
% |
| P51812 |
BXGT010893 |
Ribosomal protein S6 kinase alpha-3 |
reviewed |
Kinase |
RPS6KA3 |
Kd apparent |
'>' |
30000 |
nM |
| O94804 |
BXGT005334 |
Serine/threonine-protein kinase 10 |
reviewed |
Kinase |
STK10 |
Kd apparent |
'=' |
5236 |
nM |
| Q15375 |
BXGT013562 |
Ephrin type-A receptor 7 |
reviewed |
Kinase |
EPHA7 |
Kd apparent |
'>' |
30000 |
nM |
| P54753 |
BXGT011073 |
Ephrin type-B receptor 3 |
reviewed |
Kinase |
EPHB3 |
Kd apparent |
'>' |
30000 |
nM |
| O60313 |
BXGT004871 |
Dynamin-like 120 kDa protein, mitochondrial |
reviewed |
Enzyme modulator |
OPA1 |
Kd apparent |
'>' |
30000 |
nM |
| P49759 |
BXGT010734 |
Dual specificity protein kinase CLK1 |
reviewed |
Kinase |
CLK1 |
Kd apparent |
'>' |
30000 |
nM |
| P49674 |
BXGT010725 |
Casein kinase I isoform epsilon |
reviewed |
- |
CSNK1E |
Kd apparent |
'>' |
30000 |
nM |
| P43250 |
BXGT010372 |
G protein-coupled receptor kinase 6 |
reviewed |
Kinase |
GRK6 |
Kd apparent |
'>' |
30000 |
nM |
| P54619 |
BXGT011060 |
5'-AMP-activated protein kinase subunit gamma-1 |
reviewed |
Kinase |
PRKAG1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
11 |
nM |
| P07948 |
BXGT006702 |
Tyrosine-protein kinase Lyn |
reviewed |
Kinase |
LYN |
Kd apparent |
'>' |
30000 |
nM |
| Q9P289 |
BXGT021300 |
Serine/threonine-protein kinase 26 |
reviewed |
Kinase |
STK26 |
Kd apparent |
'>' |
30000 |
nM |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
IC50 |
'=' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
7680 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
1 |
nM |
| Q16566 |
BXGT013639 |
Calcium/calmodulin-dependent protein kinase type IV |
reviewed |
Kinase |
CAMK4 |
Kd apparent |
'>' |
30000 |
nM |
| P43686 |
BXGT010409 |
26S proteasome regulatory subunit 6B |
reviewed |
Enzyme |
PSMC4 |
Kd apparent |
'>' |
30000 |
nM |
| P36896 |
BXGT009940 |
Activin receptor type-1B |
reviewed |
Kinase |
ACVR1B |
Kd apparent |
'>' |
30000 |
nM |
| Q15569 |
BXGT013580 |
Dual specificity testis-specific protein kinase 1 |
reviewed |
Kinase |
TESK1 |
Kd apparent |
'>' |
30000 |
nM |
| P06737 |
BXGT006492 |
Glycogen phosphorylase, liver form |
reviewed |
Enzyme |
PYGL |
Kd apparent |
'>' |
30000 |
nM |
| Q13188 |
BXGT013324 |
Serine/threonine-protein kinase 3 |
reviewed |
Kinase |
STK3 |
Kd apparent |
'>' |
30000 |
nM |
| P08240 |
BXGT006754 |
Signal recognition particle receptor subunit alpha |
reviewed |
Nucleic acid binding |
SRPRA |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y616 |
BXGT022313 |
Interleukin-1 receptor-associated kinase 3 |
reviewed |
Kinase |
IRAK3 |
Kd apparent |
'>' |
30000 |
nM |
| P28482 |
BXGT009263 |
Mitogen-activated protein kinase 1 |
reviewed |
Kinase |
MAPK1 |
Kd apparent |
'>' |
30000 |
nM |
| P49840 |
BXGT010749 |
Glycogen synthase kinase-3 alpha |
reviewed |
Kinase |
GSK3A |
Kd apparent |
'>' |
30000 |
nM |
| P53779 |
BXGT011014 |
Mitogen-activated protein kinase 10 |
reviewed |
Kinase |
MAPK10 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
29 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
25 |
nM |
| P21860 |
BXGT008698 |
Receptor tyrosine-protein kinase erbB-3 |
reviewed |
Kinase |
ERBB3 |
IC50 |
'=' |
6 |
nM |
| Q15303 |
BXGT013557 |
Receptor tyrosine-protein kinase erbB-4 |
reviewed |
Kinase |
ERBB4 |
IC50 |
'=' |
6 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
6 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
'=' |
6 |
nM |
| Q76MJ5 |
BXGT016871 |
Serine/threonine-protein kinase/endoribonuclease IRE2 |
reviewed |
Kinase |
ERN2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Kd apparent |
'=' |
413 |
nM |
| O00329 |
BXGT003909 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform |
reviewed |
Kinase |
PIK3CD |
IC50 |
- |
- |
- |
| Q9Y6M4 |
BXGT022335 |
Casein kinase I isoform gamma-3 |
reviewed |
Kinase |
CSNK1G3 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
823 |
nM |
| P11362 |
BXGT007693 |
Fibroblast growth factor receptor 1 |
reviewed |
Kinase |
FGFR1 |
Kd apparent |
'>' |
30000 |
nM |
| P10398 |
BXGT007564 |
Serine/threonine-protein kinase A-Raf |
reviewed |
Kinase |
ARAF |
Kd apparent |
'>' |
30000 |
nM |
| Q8NI60 |
BXGT018572 |
Atypical kinase COQ8A, mitochondrial |
reviewed |
Kinase |
COQ8A |
Kd apparent |
'>' |
30000 |
nM |
| Q3MIX3 |
BXGT014506 |
Uncharacterized aarF domain-containing protein kinase 5 |
reviewed |
- |
ADCK5 |
Kd apparent |
'>' |
30000 |
nM |
| P49760 |
BXGT010735 |
Dual specificity protein kinase CLK2 |
reviewed |
Kinase |
CLK2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
EC50 |
'=' |
2162 |
nM |
| Q9Y243 |
BXGT022214 |
RAC-gamma serine/threonine-protein kinase |
reviewed |
Kinase |
AKT3 |
Kd apparent |
'>' |
30000 |
nM |
| P27707 |
BXGT009201 |
Deoxycytidine kinase |
reviewed |
Kinase |
DCK |
Kd apparent |
'>' |
30000 |
nM |
| O75116 |
BXGT005100 |
Rho-associated protein kinase 2 |
reviewed |
Kinase |
ROCK2 |
Kd apparent |
'>' |
30000 |
nM |
| P48426 |
BXGT010630 |
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha |
reviewed |
Kinase |
PIP4K2A |
Kd apparent |
'>' |
30000 |
nM |
| P23443 |
BXGT008866 |
Ribosomal protein S6 kinase beta-1 |
reviewed |
Kinase |
RPS6KB1 |
Kd apparent |
'>' |
30000 |
nM |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
Kd apparent |
'=' |
903 |
nM |
| P07947 |
BXGT006701 |
Tyrosine-protein kinase Yes |
reviewed |
Kinase |
YES1 |
Kd apparent |
'>' |
30000 |
nM |
| P78368 |
BXGT011840 |
Casein kinase I isoform gamma-2 |
reviewed |
Kinase |
CSNK1G2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9P0J0 |
BXGT021287 |
NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 |
reviewed |
Enzyme |
NDUFA13 |
Kd apparent |
'>' |
30000 |
nM |
| Q13557 |
BXGT013376 |
Calcium/calmodulin-dependent protein kinase type II subunit delta |
reviewed |
Kinase |
CAMK2D |
Kd apparent |
'>' |
30000 |
nM |
| P07741 |
BXGT006666 |
Adenine phosphoribosyltransferase |
reviewed |
- |
APRT |
Kd apparent |
'>' |
30000 |
nM |
| P53350 |
BXGT010984 |
Serine/threonine-protein kinase PLK1 |
reviewed |
Kinase |
PLK1 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UPZ9 |
BXGT021804 |
Serine/threonine-protein kinase ICK |
reviewed |
Kinase |
CILK1 |
Kd apparent |
'>' |
30000 |
nM |
| O00311 |
BXGT003908 |
Cell division cycle 7-related protein kinase |
reviewed |
Kinase |
CDC7 |
Kd apparent |
'>' |
30000 |
nM |
| Q15392 |
BXGT013566 |
Delta(24)-sterol reductase |
reviewed |
Enzyme |
DHCR24 |
Kd apparent |
'>' |
30000 |
nM |
| Q07912 |
BXGT012947 |
Activated CDC42 kinase 1 |
reviewed |
Kinase |
TNK2 |
IC50 |
'=' |
2300 |
nM |
| P0A0J7 |
BXGT006970 |
Quinolone resistance protein NorA |
reviewed |
- |
norA |
FC |
'=' |
8 |
- |
| Q04771 |
BXGT012783 |
Activin receptor type-1 |
reviewed |
Kinase |
ACVR1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'>' |
1000 |
nM |
| Q9P1W9 |
BXGT021296 |
Serine/threonine-protein kinase pim-2 |
reviewed |
Kinase |
PIM2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9BZL6 |
BXGT020199 |
Serine/threonine-protein kinase D2 |
reviewed |
Kinase |
PRKD2 |
Kd apparent |
'>' |
30000 |
nM |
| Q7RTN6 |
BXGT017085 |
STE20-related kinase adapter protein alpha |
reviewed |
Kinase |
STRADA |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
0 |
% |
| O75582 |
BXGT005137 |
Ribosomal protein S6 kinase alpha-5 |
reviewed |
Kinase |
RPS6KA5 |
Kd apparent |
'>' |
30000 |
nM |
| Q9Y572 |
BXGT022289 |
Receptor-interacting serine/threonine-protein kinase 3 |
reviewed |
Kinase |
RIPK3 |
Kd apparent |
'=' |
2664 |
nM |
| O95347 |
BXGT005374 |
Structural maintenance of chromosomes protein 2 |
reviewed |
- |
SMC2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UL54 |
BXGT021755 |
Serine/threonine-protein kinase TAO2 |
reviewed |
Kinase |
TAOK2 |
Kd apparent |
'>' |
30000 |
nM |
| Q709F0 |
BXGT016660 |
Acyl-CoA dehydrogenase family member 11 |
reviewed |
Enzyme |
ACAD11 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
129 |
nM |
| P35968 |
BXGT009887 |
Vascular endothelial growth factor receptor 2 |
reviewed |
Kinase |
KDR |
IC50 |
- |
- |
- |
| P35916 |
BXGT009881 |
Vascular endothelial growth factor receptor 3 |
reviewed |
Kinase |
FLT4 |
IC50 |
- |
- |
- |
| P17948 |
BXGT008358 |
Vascular endothelial growth factor receptor 1 |
reviewed |
Kinase |
FLT1 |
IC50 |
- |
- |
- |
| Q8IVH8 |
BXGT018345 |
Mitogen-activated protein kinase kinase kinase kinase 3 |
reviewed |
Kinase |
MAP4K3 |
Kd apparent |
'>' |
30000 |
nM |
| P50750 |
BXGT010818 |
Cyclin-dependent kinase 9 |
reviewed |
Kinase |
CDK9 |
Kd apparent |
'>' |
30000 |
nM |
| Q8TD08 |
BXGT018803 |
Mitogen-activated protein kinase 15 |
reviewed |
Kinase |
MAPK15 |
Kd apparent |
'>' |
30000 |
nM |
| P54819 |
BXGT011084 |
Adenylate kinase 2, mitochondrial |
reviewed |
Kinase |
AK2 |
Kd apparent |
'>' |
30000 |
nM |
| P15056 |
BXGT008075 |
Serine/threonine-protein kinase B-raf |
reviewed |
Kinase |
BRAF |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
10 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
96 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
0 |
nM |
| P42285 |
BXGT010297 |
Exosome RNA helicase MTR4 |
reviewed |
- |
MTREX |
Kd apparent |
'>' |
30000 |
nM |
| P22830 |
BXGT008809 |
Ferrochelatase, mitochondrial |
reviewed |
Enzyme |
FECH |
Kd apparent |
'=' |
6682 |
nM |
| P54764 |
BXGT011078 |
Ephrin type-A receptor 4 |
reviewed |
Kinase |
EPHA4 |
Kd apparent |
'>' |
30000 |
nM |
| P06213 |
BXGT006425 |
Insulin receptor |
reviewed |
Kinase |
INSR |
Kd apparent |
'>' |
30000 |
nM |
| Q9H2K8 |
BXGT020455 |
Serine/threonine-protein kinase TAO3 |
reviewed |
Kinase |
TAOK3 |
Kd apparent |
'>' |
30000 |
nM |
| O00444 |
BXGT003921 |
Serine/threonine-protein kinase PLK4 |
reviewed |
Kinase |
PLK4 |
Kd apparent |
'>' |
30000 |
nM |
| Q9UBE8 |
BXGT021652 |
Serine/threonine-protein kinase NLK |
reviewed |
Kinase |
NLK |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'>' |
2000 |
nM |
| P29317 |
BXGT009331 |
Ephrin type-A receptor 2 |
reviewed |
Kinase |
EPHA2 |
Kd apparent |
'>' |
30000 |
nM |
| P36897 |
BXGT009941 |
TGF-beta receptor type-1 |
reviewed |
Kinase |
TGFBR1 |
Kd apparent |
'>' |
30000 |
nM |
| Q9NYL2 |
BXGT021259 |
Mitogen-activated protein kinase kinase kinase 20 |
reviewed |
Kinase |
MAP3K20 |
Kd apparent |
'>' |
30000 |
nM |
| P61160 |
BXGT011365 |
Actin-related protein 2 |
reviewed |
Cellular structure |
ACTR2 |
Kd apparent |
'>' |
30000 |
nM |
| Q9BQI3 |
BXGT020113 |
Eukaryotic translation initiation factor 2-alpha kinase 1 |
reviewed |
Kinase |
EIF2AK1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
280 |
nM |
| P62826 |
BXGT011463 |
GTP-binding nuclear protein Ran |
reviewed |
Enzyme modulator |
RAN |
Kd apparent |
'>' |
30000 |
nM |
| Q8IW41 |
BXGT018352 |
MAP kinase-activated protein kinase 5 |
reviewed |
Kinase |
MAPKAPK5 |
Kd apparent |
'>' |
30000 |
nM |
| O95835 |
BXGT005400 |
Serine/threonine-protein kinase LATS1 |
reviewed |
Kinase |
LATS1 |
Kd apparent |
'>' |
30000 |
nM |
| Q13043 |
BXGT013307 |
Serine/threonine-protein kinase 4 |
reviewed |
Kinase |
STK4 |
Kd apparent |
'>' |
30000 |
nM |
| P48729 |
BXGT010655 |
Casein kinase I isoform alpha |
reviewed |
Kinase |
CSNK1A1 |
Kd apparent |
'>' |
30000 |
nM |
| P04626 |
BXGT006238 |
Receptor tyrosine-protein kinase erbB-2 |
reviewed |
Kinase |
ERBB2 |
IC50 |
- |
- |
- |
| P45985 |
BXGT010496 |
Dual specificity mitogen-activated protein kinase kinase 4 |
reviewed |
Kinase |
MAP2K4 |
Kd apparent |
'>' |
30000 |
nM |
| P42345 |
BXGT010304 |
Serine/threonine-protein kinase mTOR |
reviewed |
Kinase |
MTOR |
Kd |
'>' |
10000 |
nM |
| Q8TDR2 |
BXGT018811 |
Serine/threonine-protein kinase 35 |
reviewed |
Kinase |
STK35 |
Kd |
'>' |
10000 |
nM |
| Q9UKE5 |
BXGT021741 |
TRAF2 and NCK-interacting protein kinase |
reviewed |
Kinase |
TNIK |
Kd |
'=' |
6900 |
nM |
| Q86Z02 |
BXGT017638 |
Homeodomain-interacting protein kinase 1 |
reviewed |
Kinase |
HIPK1 |
Kd |
'>' |
10000 |
nM |
| Q6XUX3 |
BXGT016612 |
Dual serine/threonine and tyrosine protein kinase |
reviewed |
Kinase |
DSTYK |
Kd |
'>' |
10000 |
nM |
| P61158 |
BXGT011364 |
Actin-related protein 3 |
reviewed |
Cellular structure |
ACTR3 |
Kd apparent |
'>' |
30000 |
nM |
| Q92918 |
BXGT019394 |
Mitogen-activated protein kinase kinase kinase kinase 1 |
reviewed |
Kinase |
MAP4K1 |
Kd apparent |
'>' |
30000 |
nM |
| P22612 |
BXGT008785 |
cAMP-dependent protein kinase catalytic subunit gamma |
reviewed |
Kinase |
PRKACG |
Kd apparent |
'>' |
30000 |
nM |
| Q13882 |
BXGT013399 |
Protein-tyrosine kinase 6 |
reviewed |
Kinase |
PTK6 |
IC50 |
'=' |
980 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
88 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
99 |
% |
| Q9NSD9 |
BXGT021206 |
Phenylalanine--tRNA ligase beta subunit |
reviewed |
Enzyme |
FARSB |
Kd apparent |
'>' |
30000 |
nM |
| P48736 |
BXGT010658 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform |
reviewed |
Kinase |
PIK3CG |
IC50 |
- |
- |
- |
| Q13873 |
BXGT013398 |
Bone morphogenetic protein receptor type-2 |
reviewed |
Kinase |
BMPR2 |
Kd apparent |
'>' |
30000 |
nM |
| Q16512 |
BXGT013631 |
Serine/threonine-protein kinase N1 |
reviewed |
Kinase |
PKN1 |
Kd apparent |
'>' |
30000 |
nM |
| O43353 |
BXGT004589 |
Receptor-interacting serine/threonine-protein kinase 2 |
reviewed |
Kinase |
RIPK2 |
IC50 |
'=' |
3 |
nM |
| Q9H0K1 |
BXGT020438 |
Serine/threonine-protein kinase SIK2 |
reviewed |
Kinase |
SIK2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
3 |
% |
| Q9H773 |
BXGT020489 |
dCTP pyrophosphatase 1 |
reviewed |
- |
DCTPP1 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
22800 |
nM |
| Q00534 |
BXGT012533 |
Cyclin-dependent kinase 6 |
reviewed |
Kinase |
CDK6 |
Kd apparent |
'>' |
30000 |
nM |
| Q2M2I8 |
BXGT014130 |
AP2-associated protein kinase 1 |
reviewed |
Kinase |
AAK1 |
Kd apparent |
'>' |
30000 |
nM |
| P30519 |
BXGT009429 |
Heme oxygenase 2 |
reviewed |
- |
HMOX2 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
3 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2 |
nM |
| O15438 |
BXGT004168 |
Canalicular multispecific organic anion transporter 2 |
reviewed |
Transporter |
ABCC3 |
IC50 |
'=' |
133000 |
nM |
| P54760 |
BXGT011075 |
Ephrin type-B receptor 4 |
reviewed |
Kinase |
EPHB4 |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
12 |
nM |
| Q9Y5S2 |
BXGT022301 |
Serine/threonine-protein kinase MRCK beta |
reviewed |
Kinase |
CDC42BPB |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
Inhibition |
'=' |
77 |
% |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
IC50 |
'=' |
2874 |
nM |
| Q6JQN1 |
BXGT016338 |
Acyl-CoA dehydrogenase family member 10 |
reviewed |
Enzyme |
ACAD10 |
Kd apparent |
'=' |
33795 |
nM |
| Q6P5Z2 |
BXGT016454 |
Serine/threonine-protein kinase N3 |
reviewed |
Kinase |
PKN3 |
Kd apparent |
'>' |
30000 |
nM |
| Q9BZE4 |
BXGT020197 |
Nucleolar GTP-binding protein 1 |
reviewed |
- |
GTPBP4 |
Kd apparent |
'>' |
30000 |
nM |
| P42338 |
BXGT010303 |
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform |
reviewed |
Kinase |
PIK3CB |
IC50 |
- |
- |
- |
| P55263 |
BXGT011115 |
Adenosine kinase |
reviewed |
Kinase |
ADK |
Kd apparent |
'>' |
30000 |
nM |
| P00533 |
BXGT005575 |
Epidermal growth factor receptor |
reviewed |
Kinase |
EGFR |
TIME |
'<' |
0 |
hr |