Showing entry for Gefitinib



                             
General Compound Information
BXGC IdBXGC0047692
Compound NameGefitinib
Structure
FormulaC22H24ClFN4O3
InchiKeyXGALLCVXEZPNRQ-UHFFFAOYSA-N
SMILESCOc1cc2ncnc(c2cc1OCCCN1CCOCC1)Nc1ccc(c(c1)Cl)F
InchiInChI=1S/C22H24ClFN4O3/c1-29-20-13-19-16(12-21(20)31-8-2-5-28-6-9-30-10-7-28)22(26-14-25-19)27-15-3-4-18(24)17(23)11-15/h3-4,11-14H,2,5-10H2,1H3,(H,25,26,27)
IUPACN-(3-chloro-4-fluorophenyl)-7-methoxy-6-(3-morpholin-4-ylpropoxy)quinazolin-4-amine
Molecular Weight446.15
Pubchem Id123631
Chembl IdCHEMBL939
Targets of Information Source
DrugBank DB00317
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
Uniport Id BXGT Id Protein Name Status Protein Class Gene Groups Target Type
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR approved; investigational antagonist
PDB IRE
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM Ka M-1
P00533 BXGT005575 Epidermal growth factor receptor reviewed EGFR Kinase - - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed EGFR Kinase - - 5.6 -
O14976 BXGT004118 Cyclin-G-associated kinase reviewed GAK Kinase - - - -
O14976 BXGT004118 Cyclin-G-associated kinase reviewed GAK Kinase - - 1.62 -
Binding DB 5447
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
Uniport Id BXGT Id Protein Name Status Protein Class Gene Ki nM ic50 nM Kd nM EC50 nM
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 1 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 240 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 53.5 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 35.3 -
reviewed BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 - - 590000 -
reviewed BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK - - 2000000 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT 4300000 - - -
reviewed BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 - - 290000 -
reviewed BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 - - 1200000 -
reviewed BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK - - 920000 -
reviewed BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK - - 1200000 -
reviewed BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT - - 1300000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1100 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 570 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 520 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1400 -
reviewed BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK - - 630000 -
reviewed BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN - - 990000 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 430000 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - 5700000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 540 -
reviewed BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 - - 1800000 -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 13000 -
reviewed BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK - - 4400000 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 3200000 -
reviewed BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 - - 1900000 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 530000 -
reviewed BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC - - 3800000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 980 -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - - 3500000 -
reviewed BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 - - 410000 -
reviewed BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 - - 4000000 -
reviewed BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A - - 2000000 -
reviewed BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 - - 1600000 -
reviewed BXGT009511 Mitogen-activated protein kinase 4 reviewed Kinase MAPK4 - - 3100000 -
reviewed BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 - - 3700000 -
reviewed BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B - - 3800000 -
reviewed BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 - - 2100000 -
reviewed BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK - - 6000000 -
reviewed BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK - - 6900000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 92300 - -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - 10800 - -
reviewed BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 - 2300 - -
reviewed BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 - 980 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 1.4 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 3 - -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - 3.8 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 6.3 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 0.1 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 20 - -
reviewed BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 - - 1400 -
reviewed BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A - - 2900 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 33 - -
reviewed BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 - 1100 - -
reviewed BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 1100 -
reviewed BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET - - >10000 -
reviewed BXGT006425 Insulin receptor reviewed Kinase INSR - - >10000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 140 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1 -
reviewed BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A - - 2000 -
reviewed BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 - - 1800 -
reviewed BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 - - >10000 -
reviewed BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 - - 590 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 0.94 -
reviewed BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - >10000 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - >10000 -
reviewed BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK - - 6900 -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 460 -
reviewed BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 - - >10000 -
reviewed BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET - - >10000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 0.52 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - 1800 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 2 -
reviewed BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 - - >10000 -
reviewed BXGT019667 Aurora kinase B reviewed Kinase AURKB - - >10000 -
reviewed BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 - - >10000 -
reviewed BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 - - >10000 -
reviewed BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 - - 1200 -
reviewed BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R - - >10000 -
reviewed BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 3000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 0.98 -
reviewed BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 680 -
reviewed BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A - - >10000 -
reviewed BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 - - >10000 -
reviewed BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 - - >10000 -
reviewed BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 230 -
reviewed BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 1100 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 2700 -
reviewed BXGT019015 Myosin-IIIb reviewed Kinase MYO3B - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 360 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - 4300 -
reviewed BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 2200 -
reviewed BXGT015278 Serine/threonine-protein kinase TNNI3K reviewed TNNI3K - - >10000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 0.57 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 3100 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1.1 -
reviewed BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 1000 -
reviewed BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 - - >10000 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - 5500 -
reviewed BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 - - >10000 -
reviewed BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 - - >10000 -
reviewed BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 780 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 4700 -
reviewed BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 - - >10000 -
reviewed BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 - - 1500 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 40 -
reviewed BXGT015650 Leucine-rich repeat serine/threonine-protein kinase 2 reviewed Kinase LRRK2 - - >10000 -
reviewed BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 - - >10000 -
reviewed BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 - - >10000 -
reviewed BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 480 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 0.54 -
reviewed BXGT007750 Cyclin-dependent kinase 4 reviewed Kinase CDK4 - - >10000 -
reviewed BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 2900 -
reviewed BXGT021302 eIF-2-alpha kinase GCN2 reviewed EIF2AK4 - - >10000 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 400 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - 520 -
reviewed BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 - - 4000 -
reviewed BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 3500 -
reviewed BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET - - 3500 -
reviewed BXGT021808 Cyclin-dependent kinase 11A reviewed CDK11A - - >10000 -
reviewed BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 - - >1 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1.4 -
reviewed BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 - - >1 -
reviewed BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT - - >1 -
reviewed BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH - - >1 -
reviewed BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 - - >1 -
reviewed BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 - - >1 -
reviewed BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 - - >1 -
reviewed BXGT019667 Aurora kinase B reviewed Kinase AURKB - - >1 -
reviewed BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 - - >1 -
reviewed BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 - - >1 -
reviewed BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 - - >1 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 1 -
reviewed BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF - - >1 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - 57 -
reviewed BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 - - >1 -
reviewed BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK - - 69 -
reviewed BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET - - >1 -
reviewed BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA - - >1 -
reviewed BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 - - 15 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 11 -
reviewed BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 - - >1 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 76 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 1000 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 1730 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 0.45 - -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 7 -
reviewed BXGT014526 Serine/threonine-protein kinase ULK3 reviewed Ulk3 - - 1400 -
reviewed BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B - - 6500 -
reviewed BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK - - 1100 -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - - 1100 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - 1400 -
reviewed BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 - - 870 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 2300 -
reviewed BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK - - 1100 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - - 1.8 -
reviewed BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 - - 360 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 800 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 2000 -
reviewed BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 - - 6400 -
reviewed BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 - - 7300 -
reviewed BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC - - 5000 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 380 - -
reviewed BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK - - 13 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 54 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 23 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - <1.000000 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 39 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 26 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 22 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 832 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 16 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 12 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 25 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 2.6 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 23 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 127 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 22 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - >10000 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 0.509 - -
reviewed BXGT011200 Beta-secretase 1 reviewed Enzyme BACE1 - 20000 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 173 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 0.585 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 0.637 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 1013 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 1830 - -
reviewed BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 - 476 - -
reviewed BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 - >1000 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 343 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 14 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 3700 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 9.6 - -
reviewed BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 - 1260 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 21 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 70 - -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - 14800 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 4.2 - -
reviewed BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 - - >10000 -
reviewed BXGT008600 Serine/threonine-protein kinase MAK reviewed Kinase MAK - - >10000 -
reviewed BXGT013330 Mitogen-activated protein kinase kinase kinase 1 reviewed Kinase MAP3K1 - - >10000 -
reviewed BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 - - >10000 -
reviewed BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 - - >10000 -
reviewed BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 - - 470 -
reviewed BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB - - >10000 -
reviewed BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 - - >10000 -
reviewed BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 - - >10000 -
reviewed BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA - - >10000 -
reviewed BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 - - 3700 -
reviewed BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 - - >10000 -
reviewed BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 - - >10000 -
reviewed BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 - - >10000 -
reviewed BXGT017636 Myosin light chain kinase family member 4 reviewed MYLK4 - - >10000 -
reviewed BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 - - >10000 -
reviewed BXGT014988 Serine/threonine-protein kinase SBK1 reviewed SBK1 - - 560 -
reviewed BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 - - >10000 -
reviewed BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 - - 410 -
reviewed BXGT019394 Mitogen-activated protein kinase kinase kinase kinase 1 reviewed Kinase MAP4K1 - - >10000 -
reviewed BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 - - >10000 -
reviewed BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 - - >10000 -
reviewed BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B - - >10000 -
reviewed BXGT018990 Serine/threonine-protein kinase 32A reviewed Kinase STK32A - - >10000 -
reviewed BXGT018350 Cyclin-dependent kinase-like 3 reviewed Kinase CDKL3 - - >10000 -
reviewed BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 - - 290 -
reviewed BXGT019958 Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha reviewed Kinase PIP5K1A - - >10000 -
reviewed BXGT003900 Bone morphogenetic protein receptor type-1B reviewed Kinase BMPR1B - - >10000 -
reviewed BXGT013398 Bone morphogenetic protein receptor type-2 reviewed Kinase BMPR2 - - >10000 -
reviewed BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 - - >10000 -
reviewed BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 - - >10000 -
reviewed BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 - - >10000 -
reviewed BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 - - >10000 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - 5700 -
reviewed BXGT005127 Serine/threonine-protein kinase/endoribonuclease IRE1 reviewed Kinase ERN1 - - >10000 -
reviewed BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB - - >10000 -
reviewed BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 - - 69 -
reviewed BXGT009153 Activin receptor type-2A reviewed Kinase ACVR2A - - >10000 -
reviewed BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 - - >10000 -
reviewed BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL - - 1800 -
reviewed BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK - - 1200 -
reviewed BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX - - >10000 -
reviewed BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 - - >10000 -
reviewed BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 - - >10000 -
reviewed BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 - - 610 -
reviewed BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 - - >10000 -
reviewed BXGT010725 Casein kinase I isoform epsilon reviewed CSNK1E - - 430 -
reviewed BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 - - >10000 -
reviewed BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 - - >10000 -
reviewed BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 - - >10000 -
reviewed BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 - - 790 -
reviewed BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES - - >10000 -
reviewed BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 - - >10000 -
reviewed BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK - - 2000 -
reviewed BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B - - >10000 -
reviewed BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK - - 4400 -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - - >10000 -
reviewed BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 - - >10000 -
reviewed BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN - - 990 -
reviewed BXGT010328 Megakaryocyte-associated tyrosine-protein kinase reviewed Kinase MATK - - >10000 -
reviewed BXGT019960 Mitogen-activated protein kinase kinase kinase 3 reviewed Kinase MAP3K3 - - 2100 -
reviewed BXGT013642 Mitogen-activated protein kinase kinase kinase 11 reviewed Kinase MAP3K11 - - >10000 -
reviewed BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 - - >10000 -
reviewed BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 - - >10000 -
reviewed BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 - - >10000 -
reviewed BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 - - >10000 -
reviewed BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 - - >10000 -
reviewed BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 - - >10000 -
reviewed BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB - - >10000 -
reviewed BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 - - >10000 -
reviewed BXGT003943 Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta reviewed Kinase PIK3C2B - - >10000 -
reviewed BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 - - >10000 -
reviewed BXGT010658 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform reviewed Kinase PIK3CG - - >10000 -
reviewed BXGT021653 Phosphatidylinositol 4-kinase beta reviewed Kinase PI4KB - - >10000 -
reviewed BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA - - >10000 -
reviewed BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB - - >10000 -
reviewed BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI - - >10000 -
reviewed BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 - - 3500 -
reviewed BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 - - >10000 -
reviewed BXGT009511 Mitogen-activated protein kinase 4 reviewed Kinase MAPK4 - - 3100 -
reviewed BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 - - 1600 -
reviewed BXGT013322 Mitogen-activated protein kinase 7 reviewed Kinase MAPK7 - - >10000 -
reviewed BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 - - >10000 -
reviewed BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 - - >10000 -
reviewed BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 - - 3200 -
reviewed BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 - - >10000 -
reviewed BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 - - >10000 -
reviewed BXGT010537 Dual specificity mitogen-activated protein kinase kinase 3 reviewed Kinase MAP2K3 - - >10000 -
reviewed BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 - - >10000 -
reviewed BXGT008492 Interferon-induced, double-stranded RNA-activated protein kinase reviewed Kinase EIF2AK2 - - >10000 -
reviewed BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 - - >10000 -
reviewed BXGT013606 Rhodopsin kinase reviewed Kinase GRK1 - - >10000 -
reviewed BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 - - >10000 -
reviewed BXGT010496 Dual specificity mitogen-activated protein kinase kinase 4 reviewed Kinase MAP2K4 - - >10000 -
reviewed BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 - - >10000 -
reviewed BXGT010910 Serine/threonine-protein kinase Nek4 reviewed Kinase NEK4 - - >10000 -
reviewed BXGT005171 Cyclin-dependent kinase-like 5 reviewed Kinase CDKL5 - - >10000 -
reviewed BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 - - >10000 -
reviewed BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK - - >10000 -
reviewed BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC - - >10000 -
reviewed BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 - - 5500 -
reviewed BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER - - >10000 -
reviewed BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR - - 2600 -
reviewed BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK - - 630 -
reviewed BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE - - >10000 -
reviewed BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 - - >10000 -
reviewed BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC - - 3800 -
reviewed BXGT009854 Tyrosine-protein kinase receptor Tie-1 reviewed Kinase TIE1 - - >10000 -
reviewed BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 - - >10000 -
reviewed BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 - - >10000 -
reviewed BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK - - >10000 -
reviewed BXGT011009 LIM domain kinase 2 reviewed Kinase LIMK2 - - >10000 -
reviewed BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK - - >10000 -
reviewed BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 - - >10000 -
reviewed BXGT010303 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform reviewed Kinase PIK3CB - - >10000 -
reviewed BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 - - >10000 -
reviewed BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD - - >10000 -
reviewed BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 - - >10000 -
reviewed BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ - - >10000 -
reviewed BXGT013331 cGMP-dependent protein kinase 2 reviewed Kinase PRKG2 - - >10000 -
reviewed BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 - - >10000 -
reviewed BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 - - >10000 -
reviewed BXGT013580 Dual specificity testis-specific protein kinase 1 reviewed Kinase TESK1 - - >10000 -
reviewed BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 - - >10000 -
reviewed BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 - - >10000 -
reviewed BXGT013272 Mitogen-activated protein kinase kinase kinase 12 reviewed Kinase MAP3K12 - - >10000 -
reviewed BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 - - >10000 -
reviewed BXGT022248 Mitogen-activated protein kinase kinase kinase 2 reviewed Kinase MAP3K2 - - 3300 -
reviewed BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 - - >10000 -
reviewed BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 - - >10000 -
reviewed BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT - - 1300 -
reviewed BXGT013550 Serine/threonine-protein kinase 38 reviewed Kinase STK38 - - >10000 -
reviewed BXGT019712 Serine/threonine-protein kinase Nek1 reviewed Kinase NEK1 - - >10000 -
reviewed BXGT021743 Serine/threonine-protein kinase tousled-like 1 reviewed Kinase TLK1 - - >10000 -
reviewed BXGT005341 Cyclin-dependent kinase 14 reviewed Kinase CDK14 - - >10000 -
reviewed BXGT004872 Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma reviewed Kinase PIP5K1C - - >10000 -
reviewed BXGT021675 STE20/SPS1-related proline-alanine-rich protein kinase reviewed Kinase STK39 - - >10000 -
reviewed BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 - - >10000 -
reviewed BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed SGK3 - - >10000 -
reviewed BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE - - >10000 -
reviewed BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR - - >10000 -
reviewed BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 - - >10000 -
reviewed BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 - - >10000 -
reviewed BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 - - >10000 -
reviewed BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 - - >10000 -
reviewed BXGT020113 Eukaryotic translation initiation factor 2-alpha kinase 1 reviewed Kinase EIF2AK1 - - >10000 -
reviewed BXGT021190 Serine/threonine-protein kinase LATS2 reviewed Kinase LATS2 - - >10000 -
reviewed BXGT011209 Hormonally up-regulated neu tumor-associated kinase reviewed Kinase HUNK - - >10000 -
reviewed BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 - - >10000 -
reviewed BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK - - 920 -
reviewed BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK - - >10000 -
reviewed BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 - - >10000 -
reviewed BXGT021804 Serine/threonine-protein kinase ICK reviewed Kinase ICK - - >10000 -
reviewed BXGT022234 Microtubule-associated serine/threonine-protein kinase 1 reviewed Kinase MAST1 - - >10000 -
reviewed BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L - - >10000 -
reviewed BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK - - 6900 -
reviewed BXGT020156 Cyclin-dependent kinase 19 reviewed Kinase CDK19 - - >10000 -
reviewed BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 - - 2100 -
reviewed BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 - - 5700 -
reviewed BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 - - 540 -
reviewed BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 - - >10000 -
reviewed BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK - - 4200 -
reviewed BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 - - >10000 -
reviewed BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 - - >10000 -
reviewed BXGT018558 Myosin-IIIa reviewed Kinase MYO3A - - >10000 -
reviewed BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 - - >10000 -
reviewed BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 - - >10000 -
reviewed BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 - - 1200 -
reviewed BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K - - >10000 -
reviewed BXGT020161 Transient receptor potential cation channel subfamily M member 6 reviewed Kinase TRPM6 - - >10000 -
reviewed BXGT021188 SNF-related serine/threonine-protein kinase reviewed Kinase SNRK - - >10000 -
reviewed BXGT020147 Serine/threonine-protein kinase RIO2 reviewed Kinase RIOK2 - - >10000 -
reviewed BXGT021250 Serine/threonine-protein kinase 32B reviewed Kinase STK32B - - >10000 -
reviewed BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 - - >10000 -
reviewed BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A - - >10000 -
reviewed BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed PAK6 - - >10000 -
reviewed BXGT018572 Atypical kinase COQ8A, mitochondrial reviewed Kinase COQ8A - - >10000 -
reviewed BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 - - >10000 -
reviewed BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D - - >10000 -
reviewed BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G - - >10000 -
reviewed BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 - - 1800 -
reviewed BXGT011211 Receptor-interacting serine/threonine-protein kinase 4 reviewed Kinase RIPK4 - - >10000 -
reviewed BXGT020511 Dual specificity protein kinase CLK4 reviewed CLK4 - - >10000 -
reviewed BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 - - >10000 -
reviewed BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 - - >10000 -
reviewed BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 - - >10000 -
reviewed BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 - - >10000 -
reviewed BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 - - >10000 -
reviewed BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 - - >10000 -
reviewed BXGT018791 Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma reviewed Kinase PIP4K2C - - 7500 -
reviewed BXGT019637 Atypical kinase COQ8B, mitochondrial reviewed Kinase COQ8B - - >10000 -
reviewed BXGT015107 Mitogen-activated protein kinase kinase kinase 19 reviewed Kinase MAP3K19 - - 240 -
reviewed BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 - - >10000 -
reviewed BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 - - >10000 -
reviewed BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 - - 4600 -
reviewed BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 - - >10000 -
reviewed BXGT020119 Serine/threonine-protein kinase RIO1 reviewed Kinase RIOK1 - - >10000 -
reviewed BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B - - >10000 -
reviewed BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 - - >10000 -
reviewed BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 - - >10000 -
reviewed BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 - - >10000 -
reviewed BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 - - 1900 -
reviewed BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 - - >10000 -
reviewed BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 - - 2900 -
reviewed BXGT012312 Serine/threonine-protein kinase PknB reviewed pknB - - >10000 -
reviewed BXGT008623 Cyclin-dependent kinase 11B reviewed Kinase CDK11B - - >10000 -
reviewed BXGT020468 Tyrosine-protein kinase Srms reviewed Kinase SRMS - - >10000 -
reviewed BXGT018811 Serine/threonine-protein kinase 35 reviewed Kinase STK35 - - >10000 -
reviewed BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A - - >10000 -
reviewed BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 - - >10000 -
reviewed BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 - - >10000 -
reviewed BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 - - >10000 -
reviewed BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 - - >10000 -
reviewed BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 - - >10000 -
reviewed BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D - - 3200 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - 1700 -
reviewed BXGT019714 Cyclin-dependent kinase 15 reviewed Kinase CDK15 - - >10000 -
reviewed BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 - - >10000 -
reviewed BXGT018551 Homeodomain-interacting protein kinase 4 reviewed Kinase HIPK4 - - 310 -
reviewed BXGT013321 Dual specificity mitogen-activated protein kinase kinase 5 reviewed Kinase MAP2K5 - - 600 -
reviewed BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 - - >10000 -
reviewed BXGT018526 Casein kinase I isoform alpha-like reviewed Kinase CSNK1A1L - - >10000 -
reviewed BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 - - >10000 -
reviewed BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 - - >10000 -
reviewed BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 - - >10000 -
reviewed BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 - - >10000 -
reviewed BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN - - >10000 -
reviewed BXGT018364 Serine/threonine-protein kinase NIM1 reviewed Kinase NIM1K - - >10000 -
reviewed BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 - - >10000 -
reviewed BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G - - >10000 -
reviewed BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B - - >10000 -
reviewed BXGT011210 Serine/threonine-protein kinase SIK1 reviewed SIK1 - - >10000 -
reviewed BXGT017614 Serine/threonine-protein kinase 32C reviewed Kinase STK32C - - >10000 -
reviewed BXGT018559 Ankyrin repeat and protein kinase domain-containing protein 1 reviewed Kinase ANKK1 - - >10000 -
reviewed BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 - - 1500 -
reviewed BXGT014323 Myosin light chain kinase 3 reviewed Kinase MYLK3 - - >10000 -
reviewed BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 - - >10000 -
reviewed BXGT009617 G protein-coupled receptor kinase 4 reviewed Kinase GRK4 - - >10000 -
reviewed BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 - - 1600 -
reviewed BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 - - >10000 -
reviewed BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R - - >10000 -
reviewed BXGT016447 Serine/threonine-protein kinase Nek5 reviewed NEK5 - - >10000 -
reviewed BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK - - 5500 -
reviewed BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 - - >10000 -
reviewed BXGT013631 Serine/threonine-protein kinase N1 reviewed Kinase PKN1 - - >10000 -
reviewed BXGT007404 Wee1-like protein kinase 2 reviewed WEE2 - - >10000 -
reviewed BXGT007408 Uncharacterized serine/threonine-protein kinase SBK3 reviewed SBK3 - - >10000 -
reviewed BXGT016612 Dual serine/threonine and tyrosine protein kinase reviewed Kinase DSTYK - - >10000 -
reviewed BXGT011425 Calcium-dependent protein kinase 1 reviewed CPK1 - - >10000 -
reviewed BXGT011353 Cell division control protein 2 homolog reviewed CRK2 - - >10000 -
reviewed BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 - - >10000 -
reviewed BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 - - >10000 -
reviewed BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 - - >10000 -
reviewed BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK - - >10000 -
reviewed BXGT021810 Aurora kinase C reviewed Kinase AURKC - - >10000 -
reviewed BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D - - >10000 -
reviewed BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 - - >10000 -
reviewed BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 - - >10000 -
reviewed BXGT009970 TGF-beta receptor type-2 reviewed Kinase TGFBR2 - - >10000 -
reviewed BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK - - >10000 -
reviewed BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK - - 6000 -
reviewed BXGT009417 Wee1-like protein kinase reviewed Kinase WEE1 - - >10000 -
reviewed BXGT011837 Phosphatidylinositol 5-phosphate 4-kinase type-2 beta reviewed Kinase PIP4K2B - - >10000 -
reviewed BXGT005121 Serine/threonine-protein kinase ULK1 reviewed Kinase ULK1 - - >10000 -
reviewed BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 - - >10000 -
reviewed BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 - - >10000 -
reviewed BXGT004117 Aurora kinase A reviewed Kinase AURKA - - >10000 -
reviewed BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA - - >10000 -
reviewed BXGT018345 Mitogen-activated protein kinase kinase kinase kinase 3 reviewed Kinase MAP4K3 - - >10000 -
reviewed BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 - - >10000 -
reviewed BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 - - >10000 -
reviewed BXGT004114 Peripheral plasma membrane protein CASK reviewed Kinase CASK - - >10000 -
reviewed BXGT013435 Cyclin-dependent kinase 13 reviewed Kinase CDK13 - - >10000 -
reviewed BXGT013372 Receptor-interacting serine/threonine-protein kinase 1 reviewed Kinase RIPK1 - - >10000 -
reviewed BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 - - 530 -
reviewed BXGT004085 Serine/threonine-protein kinase RIO3 reviewed Kinase RIOK3 - - >10000 -
reviewed BXGT013368 Serine/threonine-protein kinase PRP4 homolog reviewed Kinase PRPF4B - - >10000 -
reviewed BXGT019371 Cyclin-dependent kinase-like 2 reviewed Kinase CDKL2 - - >10000 -
reviewed BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 - - >10000 -
reviewed BXGT013359 Non-receptor tyrosine-protein kinase TNK1 reviewed Kinase TNK1 - - >10000 -
reviewed BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 - - >10000 -
reviewed BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 - - >10000 -
reviewed BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 - - >10000 -
reviewed BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 - - 5100 -
reviewed BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B - - 3800 -
reviewed BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B - - >10000 -
reviewed BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK - - >10000 -
reviewed BXGT009939 Bone morphogenetic protein receptor type-1A reviewed Kinase BMPR1A - - >10000 -
reviewed BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK - - >10000 -
reviewed BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 - - >10000 -
reviewed BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 - - >10000 -
reviewed BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 - - >10000 -
reviewed BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 - - >10000 -
reviewed BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 - - 1300 -
reviewed BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 - - >10000 -
reviewed BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 - - 2500 -
reviewed BXGT004136 Ephrin type-B receptor 6 reviewed Kinase EPHB6 - - 3200 -
reviewed BXGT005149 Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma reviewed Kinase PIK3C2G - - >10000 -
reviewed BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 - - >10000 -
reviewed BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 - - >10000 -
reviewed BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 - - >10000 -
reviewed BXGT005376 Mitogen-activated protein kinase kinase kinase 6 reviewed Kinase MAP3K6 - - >10000 -
reviewed BXGT005400 Serine/threonine-protein kinase LATS1 reviewed Kinase LATS1 - - >10000 -
reviewed BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B - - >10000 -
reviewed BXGT004583 Mitogen-activated protein kinase kinase kinase 13 reviewed Kinase MAP3K13 - - >10000 -
reviewed BXGT004124 Serine/threonine-protein kinase DCLK1 reviewed Kinase DCLK1 - - >10000 -
reviewed BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 - - >10000 -
reviewed BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR - - >10000 -
reviewed BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 - - >10000 -
reviewed BXGT003909 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform reviewed Kinase PIK3CD - - >10000 -
reviewed BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 - - >10000 -
reviewed BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX - - >10000 -
reviewed BXGT005393 Serine/threonine-protein kinase OSR1 reviewed Kinase OXSR1 - - >10000 -
reviewed BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 - - >10000 -
reviewed BXGT012536 Cyclin-dependent kinase 17 reviewed Kinase CDK17 - - >10000 -
reviewed BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 - - >10000 -
reviewed BXGT009953 Serine/threonine-protein kinase receptor R3 reviewed Kinase ACVRL1 - - >10000 -
reviewed BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK - - >10000 -
reviewed BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 - - >10000 -
reviewed BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 - - 2700 -
reviewed BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 - - >10000 -
reviewed BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK - - >10000 -
reviewed BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R - - >10000 -
reviewed BXGT016630 Mitogen-activated protein kinase kinase kinase 15 reviewed MAP3K15 - - >10000 -
reviewed BXGT017617 Serine/threonine-protein kinase pim-3 reviewed PIM3 - - 5800 -
reviewed BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 - - 800 -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - - 3500 -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 7.3 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 1604 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 515 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 14.4 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 3.1 - -
reviewed BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 - 599 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 5.4 - -
reviewed BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR - >10000 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 2753 - -
reviewed BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK - - >10000 -
reviewed BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 - - >10000 -
reviewed BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 - - >10000 -
reviewed BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK - - >10000 -
reviewed BXGT007749 Myosin light chain kinase, smooth muscle reviewed Mylk - - >10000 -
reviewed BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D - - >10000 -
reviewed BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 - - >10000 -
reviewed BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 - - >10000 -
reviewed BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL - - >10000 -
reviewed BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 - - >10000 -
reviewed BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR - - >10000 -
reviewed BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 - - >10000 -
reviewed BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 - - >10000 -
reviewed BXGT011596 Tubulin alpha-1A chain reviewed Tuba1a - - 410 -
reviewed BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 - - >10000 -
reviewed BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK - - >10000 -
reviewed BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 - - >10000 -
reviewed BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 - - >10000 -
reviewed BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 - - >10000 -
reviewed BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 - - >10000 -
reviewed BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 - - >10000 -
reviewed BXGT009067 Cruzipain reviewed - - 148000 - -
reviewed BXGT009067 Cruzipain reviewed - - 88000 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR 0.4 - - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 1080 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 72 - -
reviewed BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 - 400 - -
reviewed BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 - 3190 - -
reviewed BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR - 25 - -
CHEMBL CHEMBL939
Uniport Id BXGT Id Protein Name Status Protein Class Gene width="10%">Type Relation value Units
Uniport Id BXGT Id Protein Name Status Protein Class Gene Type Relation value Units
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Kd - - -
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Kd - - -
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd - - -
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Kd - - -
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Kd - - -
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Ki '=' 2511 nM
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Ki '>' 1995 nM
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Ki '>' 7943 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Ki '=' 1995 nM
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Ki '>' 7943 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Ki '>' 6309 nM
Q9Y463 BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B Ki '>' 2511 nM
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Kd '=' 920 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 100 %
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Ki '=' 1584 nM
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Ki '>' 7943 nM
P36894 BXGT009939 Bone morphogenetic protein receptor type-1A reviewed Kinase BMPR1A Kd '>' 10000 nM
Q00532 BXGT012532 Cyclin-dependent kinase-like 1 reviewed Kinase CDKL1 Kd '>' 10000 nM
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Kd '>' 10000 nM
O75747 BXGT005149 Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit gamma reviewed Kinase PIK3C2G Kd '>' 10000 nM
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Kd '>' 10000 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd '=' 2600 nM
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Kd '=' 470 nM
P42336 BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA Kd '>' 10000 nM
P24723 BXGT008989 Protein kinase C eta type reviewed Kinase PRKCH Kd '>' 10000 nM
Q13237 BXGT013331 cGMP-dependent protein kinase 2 reviewed Kinase PRKG2 Kd '>' 10000 nM
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Kd '>' 10000 nM
O14578 BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT Kd '=' 1300 nM
Q15208 BXGT013550 Serine/threonine-protein kinase 38 reviewed Kinase STK38 Kd '>' 10000 nM
P57058 BXGT011209 Hormonally up-regulated neu tumor-associated kinase reviewed Kinase HUNK Kd '>' 10000 nM
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Kd '>' 10000 nM
Q9BX84 BXGT020161 Transient receptor potential cation channel subfamily M member 6 reviewed Kinase TRPM6 Kd '>' 10000 nM
Q00537 BXGT012536 Cyclin-dependent kinase 17 reviewed Kinase CDK17 Kd '>' 10000 nM
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Kd '>' 10000 nM
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Kd '>' 10000 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Kd '=' 3200 nM
P45985 BXGT010496 Dual specificity mitogen-activated protein kinase kinase 4 reviewed Kinase MAP2K4 Kd '>' 10000 nM
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Ki '=' 1000 nM
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Ki '>' 6309 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Ki '>' 6309 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 22 nM
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Kd apparent '>' 30000 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Ki '>' 7943 nM
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Ki '>' 7943 nM
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Ki '>' 7943 nM
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Ki '>' 6309 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Ki '>' 3162 nM
Q92887 BXGT019389 Canalicular multispecific organic anion transporter 1 reviewed Transporter ABCC2 IC50 '=' 133000 nM
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Ki '>' 6309 nM
Q16644 BXGT013647 MAP kinase-activated protein kinase 3 reviewed Kinase MAPKAPK3 Ki '>' 10000 nM
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Ki '>' 1584 nM
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Kd - - -
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Kd - - -
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Ki '=' 1258 nM
P48729 BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 Ki '>' 5011 nM
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Ki '>' 3981 nM
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Ki '=' 1000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Ki '>' 2511 nM
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Ki '>' 1584 nM
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Ki '>' 1584 nM
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Ki '>' 7943 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Ki '>' 3981 nM
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Ki '>' 3981 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 39810 nM
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Ki '>' 3162 nM
Q02779 BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 Ki '>' 3162 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 33 nM
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Ki '>' 1995 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 639 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Thermal melting change '=' 0 degrees C
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Thermal melting change '=' 0 degrees C
O95747 BXGT005393 Serine/threonine-protein kinase OSR1 reviewed Kinase OXSR1 Thermal melting change '=' 0 degrees C
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Thermal melting change '=' 5 degrees C
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Ki '>' 7943 nM
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Ki '>' 7943 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Kd - - -
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Kd - - -
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Kd - - -
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Ki '>' 6309 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 2815 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 2815 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2815 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 2815 nM
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Ki '>' 7943 nM
Q9H093 BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 Kd '>' 10000 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Kd '=' 530 nM
Q96D53 BXGT019637 Atypical kinase COQ8B, mitochondrial reviewed Kinase COQ8B Kd '>' 10000 nM
P57059 BXGT011210 Serine/threonine-protein kinase SIK1 reviewed - SIK1 Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd '=' 4300 nM
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Kd '>' 10000 nM
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Kd '=' 13 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd '>' 10000 nM
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Kd '>' 10000 nM
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Kd '>' 10000 nM
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Kd '>' 10000 nM
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Kd '>' 10000 nM
P21127 BXGT008623 Cyclin-dependent kinase 11B reviewed Kinase CDK11B Kd '>' 10000 nM
Q9BWU1 BXGT020156 Cyclin-dependent kinase 19 reviewed Kinase CDK19 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 0 nM
Q9Y616 BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 Kd '=' 1500 nM
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Kd '>' 10000 nM
Q59H18 BXGT015278 Serine/threonine-protein kinase TNNI3K reviewed - TNNI3K Kd '>' 10000 nM
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Kd '>' 10000 nM
Q86YV6 BXGT017636 Myosin light chain kinase family member 4 reviewed - MYLK4 Kd '>' 10000 nM
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Kd '>' 10000 nM
Q9BYT3 BXGT020189 Serine/threonine-protein kinase 33 reviewed Kinase STK33 Kd '>' 10000 nM
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 35 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Kd apparent '>' 30000 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Kd apparent '>' 30000 nM
Q8TBX8 BXGT018791 Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma reviewed Kinase PIP4K2C Kd apparent '>' 30000 nM
P12268 BXGT007783 Inosine-5'-monophosphate dehydrogenase 2 reviewed Enzyme IMPDH2 Kd apparent '>' 30000 nM
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Kd '>' 10000 nM
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Kd apparent '>' 30000 nM
Q99640 BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 0 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 1100 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Kd '>' 10000 nM
O94806 BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 Kd '>' 10000 nM
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1 nM
P22694 BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB Kd '>' 10000 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Thermal melting change '=' 1 degrees C
Q9P2K8 BXGT021302 eIF-2-alpha kinase GCN2 reviewed - EIF2AK4 Kd '>' 10000 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Kd '>' 10000 nM
P46734 BXGT010537 Dual specificity mitogen-activated protein kinase kinase 3 reviewed Kinase MAP2K3 Kd '>' 10000 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Kd '>' 10000 nM
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Kd '>' 10000 nM
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1 nM
Q92630 BXGT019360 Dual specificity tyrosine-phosphorylation-regulated kinase 2 reviewed Kinase DYRK2 Kd '>' 10000 nM
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Kd '>' 10000 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Kd '>' 10000 nM
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 2700 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 0 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Inhibition '=' 28 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 4000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 240 nM
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Ki '=' 630 nM
Q13153 BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 Ki '>' 10000 nM
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Ki '>' 5011 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 941 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 941 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 941 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 941 nM
Q9P2R7 BXGT021304 Succinate--CoA ligase [ADP-forming] subunit beta, mitochondrial reviewed Enzyme SUCLA2 Kd apparent '>' 30000 nM
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Kd apparent '>' 30000 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Kd apparent '>' 30000 nM
P53671 BXGT011009 LIM domain kinase 2 reviewed Kinase LIMK2 Kd apparent '>' 30000 nM
O00764 BXGT003948 Pyridoxal kinase reviewed Kinase PDXK Kd apparent '>' 30000 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Kd '>' 10000 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Kd '>' 10000 nM
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Kd '=' 1800 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Kd '=' 410 nM
Q9BUB5 BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 Kd '=' 290 nM
O00238 BXGT003900 Bone morphogenetic protein receptor type-1B reviewed Kinase BMPR1B Kd '>' 10000 nM
P49336 BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 Kd '>' 10000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Kd '>' 10000 nM
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Kd '>' 10000 nM
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Kd '>' 10000 nM
O00750 BXGT003943 Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta reviewed Kinase PIK3C2B Kd '>' 10000 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Kd '>' 10000 nM
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Kd '>' 10000 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Kd '>' 10000 nM
P51957 BXGT010910 Serine/threonine-protein kinase Nek4 reviewed Kinase NEK4 Kd '>' 10000 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 98 %
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF IC50 '=' 2000 nM
P51957 BXGT010910 Serine/threonine-protein kinase Nek4 reviewed Kinase NEK4 Ki '>' 6309 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Thermal melting change '=' 0 degrees C
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Thermal melting change '=' 0 degrees C
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Thermal melting change '=' 0 degrees C
Q8IV63 BXGT018341 Inactive serine/threonine-protein kinase VRK3 reviewed Kinase VRK3 Thermal melting change '=' 0 degrees C
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Ki '>' 1584 nM
Q9Y463 BXGT022269 Dual specificity tyrosine-phosphorylation-regulated kinase 1B reviewed Kinase DYRK1B Kd '>' 10000 nM
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Kd '>' 10000 nM
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Kd '=' 2000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Kd '>' 10000 nM
Q02779 BXGT012670 Mitogen-activated protein kinase kinase kinase 10 reviewed Kinase MAP3K10 Kd '>' 10000 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Kd '>' 10000 nM
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Kd '>' 10000 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Kd '>' 10000 nM
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Kd '>' 10000 nM
Q15835 BXGT013606 Rhodopsin kinase reviewed Kinase GRK1 Kd '>' 10000 nM
Q96SB4 BXGT019740 SRSF protein kinase 1 reviewed Kinase SRPK1 Kd '>' 10000 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Ki '>' 3981 nM
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Kd '>' 10000 nM
Q96PF2 BXGT019708 Testis-specific serine/threonine-protein kinase 2 reviewed Kinase TSSK2 Ki '>' 1584 nM
Q9NR20 BXGT021176 Dual specificity tyrosine-phosphorylation-regulated kinase 4 reviewed Kinase DYRK4 Ki '>' 7943 nM
Q04771 BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 Ki '>' 3981 nM
P29597 BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 Kd '>' 10000 nM
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Kd '>' 10000 nM
Q9UF33 BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 Kd '=' 590 nM
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Ki '>' 7943 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Ki '=' 2511 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 Inhibition - - -
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Inhibition - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition - - -
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Inhibition - - -
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Kd '>' 10000 nM
O15075 BXGT004124 Serine/threonine-protein kinase DCLK1 reviewed Kinase DCLK1 Ki '>' 10000 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Ki '>' 5011 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Potency '=' 1122 nM
P49336 BXGT010697 Cyclin-dependent kinase 8 reviewed Kinase CDK8 Ki '>' 3981 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 20 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 Activity - - -
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Activity - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Activity - - -
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Activity - - -
Q9Y6R4 BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 Kd - - -
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Kd '=' 360 nM
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Kd - - -
Q15349 BXGT013558 Ribosomal protein S6 kinase alpha-2 reviewed Kinase RPS6KA2 Kd - - -
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Kd - - -
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd - - -
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Thermal melting change '=' 0 degrees C
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Thermal melting change '=' -1 degrees C
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Ki '>' 3162 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 10480 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 10480 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 10480 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 10480 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 476 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Thermal melting change '=' 0 degrees C
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Thermal melting change '=' 1 degrees C
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Thermal melting change '=' 1 degrees C
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Thermal melting change '=' 7 degrees C
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 101 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 14 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 4 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 25118 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Kd '>' 10000 nM
Q8N568 BXGT018516 Serine/threonine-protein kinase DCLK2 reviewed Kinase DCLK2 Kd '>' 10000 nM
O75460 BXGT005127 Serine/threonine-protein kinase/endoribonuclease IRE1 reviewed Kinase ERN1 Kd '>' 10000 nM
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Kd '>' 10000 nM
P48729 BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 Kd '>' 10000 nM
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Kd '>' 10000 nM
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Kd '>' 10000 nM
Q99759 BXGT019960 Mitogen-activated protein kinase kinase kinase 3 reviewed Kinase MAP3K3 Kd '=' 2100 nM
Q13164 BXGT013322 Mitogen-activated protein kinase 7 reviewed Kinase MAPK7 Kd '>' 10000 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Kd '>' 10000 nM
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd '>' 10000 nM
Q2M2I8 BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 Kd '>' 10000 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Kd '>' 10000 nM
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Selectivity '=' 0 -
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Kd '>' 10000 nM
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Kd '>' 10000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Ki '=' 3981 nM
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Kd '>' 10000 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Ki '>' 6309 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Ratio IC50 '=' 12 -
Q16659 BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 Kd '=' 1600 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Ki '>' 7943 nM
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 Ki '>' 398 nM
Q96KB5 BXGT019685 Lymphokine-activated killer T-cell-originated protein kinase reviewed Kinase PBK Thermal melting change '=' 0 degrees C
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Ki '>' 3162 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Inhibition - - -
Q04771 BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 Kd '>' 10000 nM
O14730 BXGT004085 Serine/threonine-protein kinase RIO3 reviewed Kinase RIOK3 Kd '>' 10000 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Kd '>' 10000 nM
Q96PY6 BXGT019712 Serine/threonine-protein kinase Nek1 reviewed Kinase NEK1 Kd '>' 10000 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Kd '>' 10000 nM
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Kd '>' 10000 nM
P80192 BXGT011883 Mitogen-activated protein kinase kinase kinase 9 reviewed Kinase MAP3K9 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '>' 10000 nM
O15146 BXGT004131 Muscle, skeletal receptor tyrosine-protein kinase reviewed Kinase MUSK Kd '>' 10000 nM
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Kd '>' 10000 nM
Q8N5S9 BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 Kd '>' 10000 nM
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Kd '>' 10000 nM
Q9UIK4 BXGT021720 Death-associated protein kinase 2 reviewed Kinase DAPK2 Kd '>' 10000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Inhibition - - -
P33981 BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK Kd '>' 10000 nM
Q9H1R3 BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 Kd - - -
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd - - -
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Kd '=' 7300 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '<' 1 nM
Q99755 BXGT019958 Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha reviewed Kinase PIP5K1A Kd '>' 10000 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Ki '>' 3981 nM
Q96KB5 BXGT019685 Lymphokine-activated killer T-cell-originated protein kinase reviewed Kinase PBK Ki '>' 10000 nM
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Ki '>' 3162 nM
Q9UNQ0 BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 Activity - - -
Q96L34 BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 Ki '>' 5011 nM
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Ki '>' 2511 nM
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Kd - - -
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Kd - - -
O00418 BXGT003918 Eukaryotic elongation factor 2 kinase reviewed Kinase EEF2K Ki '>' 3981 nM
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Ki '=' 158 nM
O15075 BXGT004124 Serine/threonine-protein kinase DCLK1 reviewed Kinase DCLK1 Kd '>' 10000 nM
Q8TD19 BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 Kd '>' 10000 nM
Q16816 BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 Kd '=' 3700 nM
Q9NWZ3 BXGT021239 Interleukin-1 receptor-associated kinase 4 reviewed Kinase IRAK4 Kd '=' 540 nM
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Kd '>' 10000 nM
P49137 BXGT010680 MAP kinase-activated protein kinase 2 reviewed Kinase MAPKAPK2 Kd '>' 10000 nM
Q9C098 BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 Kd '=' 2900 nM
P37023 BXGT009953 Serine/threonine-protein kinase receptor R3 reviewed Kinase ACVRL1 Kd '>' 10000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC IC50 '=' 1100 nM
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 IC50 '=' 1000 nM
P25779 BXGT009067 Cruzipain reviewed - IC50 '=' 148000 nM
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Kd '=' 2000 nM
P34947 BXGT009774 G protein-coupled receptor kinase 5 reviewed Kinase GRK5 Ki '>' 3981 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Kd '>' 10000 nM
Q8NFD2 BXGT018559 Ankyrin repeat and protein kinase domain-containing protein 1 reviewed Kinase ANKK1 Kd '>' 10000 nM
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Kd - - -
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Kd - - -
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF Kd '>' 10000 nM
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Ki '>' 1584 nM
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Kd - - -
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Kd - - -
Q8TD08 BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 Kd '>' 10000 nM
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 10 nM
Q96L34 BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 Kd '>' 10000 nM
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Kd '=' 7 nM
Q92887 BXGT019389 Canalicular multispecific organic anion transporter 1 reviewed Transporter ABCC2 Activity '=' 74 %
P25779 BXGT009067 Cruzipain reviewed - IC50 '=' 88000 nM
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Kd - - -
Q99640 BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 Kd - - -
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Kd - - -
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Kd '=' 3500 nM
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Kd '=' 800 nM
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Kd '=' 990 nM
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Kd '>' 10000 nM
Q8IWQ3 BXGT018355 Serine/threonine-protein kinase BRSK2 reviewed Kinase BRSK2 Kd '>' 10000 nM
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Kd '>' 10000 nM
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Kd '>' 10000 nM
O00329 BXGT003909 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform reviewed Kinase PIK3CD Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 40 nM
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Kd '>' 10000 nM
Q6DT37 BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG Kd '>' 10000 nM
Q9H3Y6 BXGT020468 Tyrosine-protein kinase Srms reviewed Kinase SRMS Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 2 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Activity - - -
Q9UNQ0 BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 IC50 '=' 1100 nM
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Kd '=' 4400 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Kd '>' 10000 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Kd '>' 10000 nM
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Kd '=' 2100 nM
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Kd '=' 6900 nM
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Kd '=' 4000 nM
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Kd '>' 10000 nM
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Kd '>' 10000 nM
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 280 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 '=' 1900 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Ki '>' 6309 nM
P19525 BXGT008492 Interferon-induced, double-stranded RNA-activated protein kinase reviewed Kinase EIF2AK2 Kd '>' 10000 nM
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Kd '>' 10000 nM
P27037 BXGT009153 Activin receptor type-2A reviewed Kinase ACVR2A Kd '>' 10000 nM
Q13705 BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B Kd '>' 10000 nM
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Kd '>' 10000 nM
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Ki '>' 3981 nM
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Kd '=' 5700 nM
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Kd '>' 10000 nM
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 3500 nM
O95835 BXGT005400 Serine/threonine-protein kinase LATS1 reviewed Kinase LATS1 Kd '>' 10000 nM
O43283 BXGT004583 Mitogen-activated protein kinase kinase kinase 13 reviewed Kinase MAP3K13 Kd '>' 10000 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Kd '=' 630 nM
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Kd '>' 10000 nM
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Kd '>' 10000 nM
O60331 BXGT004872 Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma reviewed Kinase PIP5K1C Kd '>' 10000 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Ki '=' 3162 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Inhibition - - -
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Kd - - -
P42338 BXGT010303 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform reviewed Kinase PIK3CB IC50 '>' 50000 nM
P78527 BXGT011846 DNA-dependent protein kinase catalytic subunit reviewed Kinase PRKDC IC50 '>' 50000 nM
P22455 BXGT008772 Fibroblast growth factor receptor 4 reviewed Kinase FGFR4 Kd '>' 10000 nM
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Kd '>' 10000 nM
P04049 BXGT006133 RAF proto-oncogene serine/threonine-protein kinase reviewed Kinase RAF1 Kd '>' 10000 nM
Q13470 BXGT013359 Non-receptor tyrosine-protein kinase TNK1 reviewed Kinase TNK1 Kd '>' 10000 nM
P53671 BXGT011009 LIM domain kinase 2 reviewed Kinase LIMK2 Kd '>' 10000 nM
Q9C098 BXGT020208 Serine/threonine-protein kinase DCLK3 reviewed Kinase DCLK3 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 380 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 13 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 39 nM
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Kd '>' 10000 nM
P30291 BXGT009417 Wee1-like protein kinase reviewed Kinase WEE1 Kd '>' 10000 nM
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Kd '>' 10000 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Kd '>' 10000 nM
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Kd '>' 10000 nM
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Kd '>' 10000 nM
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Kd '>' 10000 nM
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 599 nM
Q9NSY1 BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K Kd - - -
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Kd - - -
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Kd '=' 1100 nM
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Kd - - -
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Ratio '>' 1 -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 99 %
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 343 nM
Q07002 BXGT012908 Cyclin-dependent kinase 18 reviewed Kinase CDK18 Kd '>' 10000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Kd - - -
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Kd - - -
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Kd '>' 10000 nM
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Kd '=' 430 nM
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Kd '>' 10000 nM
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Kd '>' 10000 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 1000 nM
P35590 BXGT009854 Tyrosine-protein kinase receptor Tie-1 reviewed Kinase TIE1 Kd '>' 10000 nM
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Kd '>' 10000 nM
Q86UX6 BXGT017614 Serine/threonine-protein kinase 32C reviewed Kinase STK32C Kd '>' 10000 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR IC50 '>' 50000 nM
P48736 BXGT010658 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform reviewed Kinase PIK3CG IC50 '>' 50000 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Inhibition '=' 12 %
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 '>' 10000 nM
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Ki '>' 3981 nM
Q9H1R3 BXGT020446 Myosin light chain kinase 2, skeletal/cardiac muscle reviewed Kinase MYLK2 Kd '=' 1900 nM
P78362 BXGT011839 SRSF protein kinase 2 reviewed Kinase SRPK2 Kd '>' 10000 nM
Q8WXR4 BXGT019015 Myosin-IIIb reviewed Kinase MYO3B Kd '>' 10000 nM
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Kd '>' 10000 nM
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Kd '>' 10000 nM
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 2700 nM
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Kd '>' 10000 nM
Q16584 BXGT013642 Mitogen-activated protein kinase kinase kinase 11 reviewed Kinase MAP3K11 Kd '>' 10000 nM
Q16512 BXGT013631 Serine/threonine-protein kinase N1 reviewed Kinase PKN1 Kd '>' 10000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 1730 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 1730 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1730 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 1730 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd '=' 1400 nM
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Kd - - -
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Kd '=' 870 nM
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Kd - - -
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Kd - - -
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Kd - - -
O94768 BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B Kd '=' 6500 nM
Q9HBY8 BXGT020524 Serine/threonine-protein kinase Sgk2 reviewed Kinase SGK2 Ki '>' 7943 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Ki '=' 501 nM
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Ki '=' 1584 nM
Q86UE8 BXGT017612 Serine/threonine-protein kinase tousled-like 2 reviewed Kinase TLK2 Kd '>' 10000 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Kd '>' 10000 nM
Q9BRS2 BXGT020119 Serine/threonine-protein kinase RIO1 reviewed Kinase RIOK1 Kd '>' 10000 nM
Q9P0L2 BXGT021289 Serine/threonine-protein kinase MARK1 reviewed Kinase MARK1 Kd '>' 10000 nM
Q13153 BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 Kd - - -
Q92772 BXGT019371 Cyclin-dependent kinase-like 2 reviewed Kinase CDKL2 Kd '>' 10000 nM
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd '=' 1500 nM
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Kd - - -
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Kd - - -
Q3U3Q1 BXGT014526 Serine/threonine-protein kinase ULK3 reviewed - Ulk3 Kd '=' 1400 nM
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Kd - - -
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Kd - - -
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Kd - - -
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Ki '>' 5011 nM
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Ki '=' 251 nM
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Ki '>' 6309 nM
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Ki '>' 1995 nM
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Ki '>' 6309 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Kd - - -
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Kd - - -
Q8N5S9 BXGT018520 Calcium/calmodulin-dependent protein kinase kinase 1 reviewed Kinase CAMKK1 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Potency '=' 3 nM
Q9UF33 BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 Kd '=' 1400 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Kd '=' 1100 nM
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd - - -
Q9Y2H1 BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L Kd - - -
P22607 BXGT008784 Fibroblast growth factor receptor 3 reviewed Kinase FGFR3 Kd - - -
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR IC50 '>' 50000 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Ki '>' 3162 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 23 nM
Q92918 BXGT019394 Mitogen-activated protein kinase kinase kinase kinase 1 reviewed Kinase MAP4K1 Kd '>' 10000 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Kd '>' 10000 nM
Q13546 BXGT013372 Receptor-interacting serine/threonine-protein kinase 1 reviewed Kinase RIPK1 Kd '>' 10000 nM
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Kd '>' 10000 nM
P51813 BXGT010894 Cytoplasmic tyrosine-protein kinase BMX reviewed Kinase BMX Activity - - -
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Kd '>' 10000 nM
O60285 BXGT004867 NUAK family SNF1-like kinase 1 reviewed Kinase NUAK1 Kd '>' 10000 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Kd - - -
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Kd '=' 5000 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Ki '>' 5011 nM
Q9Y2H1 BXGT022233 Serine/threonine-protein kinase 38-like reviewed Kinase STK38L Kd '>' 10000 nM
P21802 BXGT008691 Fibroblast growth factor receptor 2 reviewed Kinase FGFR2 Kd '>' 10000 nM
Q9NYL2 BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 Kd '>' 10000 nM
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd '>' 10000 nM
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Kd '>' 10000 nM
P07333 BXGT006602 Macrophage colony-stimulating factor 1 receptor reviewed Kinase CSF1R Kd '>' 10000 nM
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Kd '>' 10000 nM
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Ratio '=' 505 -
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Kd '>' 10000 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Ki '=' 2511 nM
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Kd '=' 1300 nM
P14616 BXGT008026 Insulin receptor-related protein reviewed Kinase INSRR Kd '>' 10000 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd '=' 1700 nM
Q13163 BXGT013321 Dual specificity mitogen-activated protein kinase kinase 5 reviewed Kinase MAP2K5 Kd '=' 600 nM
P50613 BXGT010815 Cyclin-dependent kinase 7 reviewed Kinase CDK7 Kd '=' 610 nM
Q13153 BXGT013319 Serine/threonine-protein kinase PAK 1 reviewed Kinase PAK1 Kd '>' 10000 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Kd '>' 10000 nM
O15111 BXGT004126 Inhibitor of nuclear factor kappa-B kinase subunit alpha reviewed Kinase CHUK Kd '>' 10000 nM
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Kd '>' 10000 nM
P54762 BXGT011076 Ephrin type-B receptor 1 reviewed Kinase EPHB1 Kd '>' 10000 nM
P53355 BXGT010985 Death-associated protein kinase 1 reviewed Kinase DAPK1 Kd '>' 10000 nM
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Kd '>' 10000 nM
P37173 BXGT009970 TGF-beta receptor type-2 reviewed Kinase TGFBR2 Kd '>' 10000 nM
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Kd '>' 10000 nM
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 190 nM
Q00526 BXGT012531 Cyclin-dependent kinase 3 reviewed Kinase CDK3 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '<' 1 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '<' 1 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '<' 1 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '<' 1 nM
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Kd '=' 2900 nM
O94806 BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 Kd apparent '>' 30000 nM
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Kd apparent '>' 30000 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Ki '>' 1584 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Kd apparent '>' 30000 nM
Q9Y2K2 BXGT022238 Serine/threonine-protein kinase SIK3 reviewed Kinase SIK3 Kd apparent '>' 30000 nM
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Kd apparent '>' 30000 nM
Q13470 BXGT013359 Non-receptor tyrosine-protein kinase TNK1 reviewed Kinase TNK1 Kd apparent '>' 30000 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd apparent '>' 30000 nM
Q9UGJ0 BXGT021683 5'-AMP-activated protein kinase subunit gamma-2 reviewed Enzyme modulator PRKAG2 Kd apparent '>' 30000 nM
O14976 BXGT004118 Cyclin-G-associated kinase reviewed Kinase GAK Kd apparent '=' 951 nM
P27361 BXGT009176 Mitogen-activated protein kinase 3 reviewed Kinase MAPK3 Kd apparent '>' 30000 nM
P05141 BXGT006325 ADP/ATP translocase 2 reviewed Transporter SLC25A5 Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 2 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 2 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 2 nM
O00506 BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 Kd '>' 10000 nM
Q8IYT8 BXGT018370 Serine/threonine-protein kinase ULK2 reviewed Kinase ULK2 Kd '>' 10000 nM
Q8NEV4 BXGT018558 Myosin-IIIa reviewed Kinase MYO3A Kd '>' 10000 nM
Q8NI60 BXGT018572 Atypical kinase COQ8A, mitochondrial reviewed Kinase COQ8A Kd '>' 10000 nM
Q13627 BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A Kd '>' 10000 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Kd '>' 10000 nM
Q8WTQ7 BXGT018984 Rhodopsin kinase reviewed Kinase GRK7 Kd '>' 10000 nM
Q32MK0 BXGT014323 Myosin light chain kinase 3 reviewed Kinase MYLK3 Kd '>' 10000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 22 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 22 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 22 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 22 nM
Q12866 BXGT013273 Tyrosine-protein kinase Mer reviewed Kinase MERTK Kd '>' 10000 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Kd '>' 10000 nM
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Ki '>' 5011 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd '>' 10000 nM
P13861 BXGT007961 cAMP-dependent protein kinase type II-alpha regulatory subunit reviewed - PRKAR2A Kd apparent '>' 30000 nM
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Kd apparent '>' 30000 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Kd apparent '>' 30000 nM
Q16513 BXGT013632 Serine/threonine-protein kinase N2 reviewed Kinase PKN2 Kd apparent '>' 30000 nM
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Kd - - -
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Kd - - -
P48729 BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 IC50 '>' 50000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 515 nM
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd - - -
Q9JI10 BXGT020811 Serine/threonine-protein kinase 3 reviewed - Stk3 Kd - - -
Q04206 BXGT012754 Transcription factor p65 reviewed Transcription factor RELA Inhibition - - -
Q14164 BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE Kd apparent '>' 30000 nM
P23458 BXGT008868 Tyrosine-protein kinase JAK1 reviewed Kinase JAK1 Kd apparent '>' 30000 nM
Q16584 BXGT013642 Mitogen-activated protein kinase kinase kinase 11 reviewed Kinase MAP3K11 Kd apparent '>' 30000 nM
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK IC50 '=' 110 nM
P42679 BXGT010328 Megakaryocyte-associated tyrosine-protein kinase reviewed Kinase MATK Ki '>' 1995 nM
P51451 BXGT010848 Tyrosine-protein kinase Blk reviewed Kinase BLK Kd '=' 1200 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 13980 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 13980 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 13980 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 13980 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
Q15746 BXGT013591 Myosin light chain kinase, smooth muscle reviewed Kinase MYLK Kd apparent '>' 30000 nM
O95382 BXGT005376 Mitogen-activated protein kinase kinase kinase 6 reviewed Kinase MAP3K6 Kd apparent '>' 30000 nM
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Kd apparent '>' 30000 nM
Q99640 BXGT019944 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase reviewed Kinase PKMYT1 Kd apparent '>' 30000 nM
Q01538 BXGT012597 Myelin transcription factor 1 reviewed Transcription factor MYT1 Activity '<' 5 %
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Ki '>' 10000 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Ki '>' 1995 nM
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 400 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 520 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 1100 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Kd '>' 10000 nM
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Kd '=' 5500 nM
O95819 BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 Ki '=' 1000 nM
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Kd '>' 10000 nM
Q9NYY3 BXGT021264 Serine/threonine-protein kinase PLK2 reviewed Kinase PLK2 Kd '>' 10000 nM
Q9UEW8 BXGT021675 STE20/SPS1-related proline-alanine-rich protein kinase reviewed Kinase STK39 Kd '>' 10000 nM
Q9Y2H9 BXGT022234 Microtubule-associated serine/threonine-protein kinase 1 reviewed Kinase MAST1 Kd '>' 10000 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Kd '>' 10000 nM
Q8TBX8 BXGT018791 Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma reviewed Kinase PIP4K2C Kd '=' 7500 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Kd '=' 3200 nM
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 Ki '=' 6309 nM
P29376 BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK Ki '>' 1584 nM
Q9H4B4 BXGT020474 Serine/threonine-protein kinase PLK3 reviewed Kinase PLK3 Ki '>' 7943 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Ki '>' 2511 nM
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Ki '=' 3162 nM
Q8NE63 BXGT018551 Homeodomain-interacting protein kinase 4 reviewed Kinase HIPK4 Ki '=' 1258 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Inhibition '=' 81 %
O75460 BXGT005127 Serine/threonine-protein kinase/endoribonuclease IRE1 reviewed Kinase ERN1 Kd apparent '>' 30000 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Kd apparent '=' 4372 nM
Q96L34 BXGT019689 MAP/microtubule affinity-regulating kinase 4 reviewed Kinase MARK4 Kd apparent '>' 30000 nM
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Ki '>' 1995 nM
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Kd apparent '>' 30000 nM
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Ki '=' 316 nM
Q6DT37 BXGT016259 Serine/threonine-protein kinase MRCK gamma reviewed Kinase CDC42BPG Kd apparent '>' 30000 nM
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 Ki '=' 5011 nM
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Ki '=' 398 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Ki '>' 7943 nM
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Ki '>' 1584 nM
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Kd apparent '>' 30000 nM
P41743 BXGT010270 Protein kinase C iota type reviewed Kinase PRKCI Kd apparent '>' 30000 nM
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Kd apparent '>' 30000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Ki '>' 7943 nM
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Kd apparent '>' 30000 nM
P11802 BXGT007750 Cyclin-dependent kinase 4 reviewed Kinase CDK4 Kd apparent '>' 30000 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 12 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Kd '>' 10000 nM
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Kd '>' 10000 nM
P29376 BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK Kd '=' 5500 nM
Q9UQ88 BXGT021808 Cyclin-dependent kinase 11A reviewed - CDK11A Kd '>' 10000 nM
Q8TD19 BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 21 nM
Q16620 BXGT013645 BDNF/NT-3 growth factors receptor reviewed Kinase NTRK2 Kd '>' 10000 nM
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Ki '>' 1584 nM
Q9NY57 BXGT021250 Serine/threonine-protein kinase 32B reviewed Kinase STK32B Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Ki '>' 630 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Ki '>' 1995 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 4 nM
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd '=' 1800 nM
Q13418 BXGT013351 Integrin-linked protein kinase reviewed Kinase ILK Kd apparent '>' 30000 nM
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Kd '>' 10000 nM
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Kd '>' 10000 nM
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Kd '=' 4200 nM
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Kd '>' 10000 nM
O15254 BXGT004143 Peroxisomal acyl-coenzyme A oxidase 3 reviewed Enzyme ACOX3 Kd apparent '>' 30000 nM
P11274 BXGT007681 Breakpoint cluster region protein reviewed Enzyme modulator BCR Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 39 nM
P42685 BXGT010332 Tyrosine-protein kinase FRK reviewed Kinase FRK Kd apparent '>' 30000 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Ki '=' 7943 nM
Q9UEE5 BXGT021671 Serine/threonine-protein kinase 17A reviewed Kinase STK17A Ki '>' 3981 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 '=' 14800 nM
P33981 BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK Kd apparent '>' 30000 nM
P49761 BXGT010736 Dual specificity protein kinase CLK3 reviewed Kinase CLK3 Kd - - -
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 173 nM
P27448 BXGT009183 MAP/microtubule affinity-regulating kinase 3 reviewed Kinase MARK3 Kd apparent '>' 30000 nM
P30086 BXGT009400 Phosphatidylethanolamine-binding protein 1 reviewed Enzyme modulator PEBP1 Kd apparent '>' 30000 nM
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Thermal melting change '=' 0 degrees C
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Thermal melting change '=' 0 degrees C
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Thermal melting change '=' 0 degrees C
Q9Y6R4 BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 Kd '>' 10000 nM
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Kd '>' 10000 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Kd '>' 10000 nM
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 3000 nM
P0A0J7 BXGT006970 Quinolone resistance protein NorA reviewed - norA Inhibition '=' 94 %
P0A0J7 BXGT006970 Quinolone resistance protein NorA reviewed - norA IC50 '=' 9700 nM
O15197 BXGT004136 Ephrin type-B receptor 6 reviewed Kinase EPHB6 Kd apparent '>' 30000 nM
P02545 BXGT005889 Prelamin-A/C reviewed - LMNA Potency '=' 0 nM
Q52WX2 BXGT014988 Serine/threonine-protein kinase SBK1 reviewed - SBK1 Kd '=' 560 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Ki '>' 3981 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Kd - - -
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Kd - - -
P09619 BXGT006911 Platelet-derived growth factor receptor beta reviewed Kinase PDGFRB Kd - - -
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Kd - - -
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Kd - - -
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Kd - - -
O43781 BXGT004625 Dual specificity tyrosine-phosphorylation-regulated kinase 3 reviewed Kinase DYRK3 Ki '>' 5011 nM
P42681 BXGT010330 Tyrosine-protein kinase TXK reviewed Kinase TXK Kd '=' 6000 nM
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Ki '=' 2511 nM
P11802 BXGT007750 Cyclin-dependent kinase 4 reviewed Kinase CDK4 Kd '>' 10000 nM
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Kd '>' 10000 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd '>' 10000 nM
Q13873 BXGT013398 Bone morphogenetic protein receptor type-2 reviewed Kinase BMPR2 Kd '>' 10000 nM
Q08345 BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 Kd '>' 10000 nM
Q9UQM7 BXGT021814 Calcium/calmodulin-dependent protein kinase type II subunit alpha reviewed Kinase CAMK2A Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3 nM
Q13627 BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A Ki '>' 5011 nM
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Ki '>' 7943 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Kd '=' 2300 nM
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Kd - - -
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Kd - - -
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Kd - - -
O14965 BXGT004117 Aurora kinase A reviewed Kinase AURKA Kd apparent '>' 30000 nM
Q5S007 BXGT015650 Leucine-rich repeat serine/threonine-protein kinase 2 reviewed Kinase LRRK2 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 230 nM
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd '=' 1600 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 0 nM
Q02156 BXGT012639 Protein kinase C epsilon type reviewed Kinase PRKCE Kd '>' 10000 nM
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Kd '>' 10000 nM
Q15569 BXGT013580 Dual specificity testis-specific protein kinase 1 reviewed Kinase TESK1 Kd '>' 10000 nM
Q9UKI8 BXGT021743 Serine/threonine-protein kinase tousled-like 1 reviewed Kinase TLK1 Kd '>' 10000 nM
Q96BR1 BXGT019627 Serine/threonine-protein kinase Sgk3 reviewed - SGK3 Kd '>' 10000 nM
Q9UPE1 BXGT021796 SRSF protein kinase 3 reviewed Kinase SRPK3 Kd '>' 10000 nM
Q9UPZ9 BXGT021804 Serine/threonine-protein kinase ICK reviewed Kinase CILK1 Kd '>' 10000 nM
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Kd '>' 10000 nM
P17252 BXGT008294 Protein kinase C alpha type reviewed Kinase PRKCA Kd - - -
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Kd - - -
P33981 BXGT009744 Dual specificity protein kinase TTK reviewed Kinase TTK Kd - - -
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Kd - - -
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Ki '>' 1258 nM
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Kd '>' 10000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Kd '=' 3800 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 5 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2753 nM
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Kd '>' 10000 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Kd '=' 1200 nM
O75385 BXGT005121 Serine/threonine-protein kinase ULK1 reviewed Kinase ULK1 Kd '>' 10000 nM
P78356 BXGT011837 Phosphatidylinositol 5-phosphate 4-kinase type-2 beta reviewed Kinase PIP4K2B Kd '>' 10000 nM
P31152 BXGT009511 Mitogen-activated protein kinase 4 reviewed Kinase MAPK4 Kd '=' 3100 nM
O75914 BXGT005165 Serine/threonine-protein kinase PAK 3 reviewed Kinase PAK3 Kd '>' 10000 nM
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 72 nM
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Kd - - -
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 Kd - - -
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Kd - - -
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Kd '=' 2000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 54 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Ki '>' 6309 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Ki '=' 158 nM
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Kd - - -
P29320 BXGT009332 Ephrin type-A receptor 3 reviewed Kinase EPHA3 Kd - - -
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Kd '=' 800 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd '=' 6400 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Potency - 1373 nM
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Thermal melting change '=' 0 degrees C
P29376 BXGT009339 Leukocyte tyrosine kinase receptor reviewed Kinase LTK Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Inhibition - - -
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Kd '>' 10000 nM
P10636 BXGT007596 Microtubule-associated protein tau reviewed - MAPT Potency '=' 35481 nM
P42336 BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA IC50 '>' 50000 nM
O00329 BXGT003909 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform reviewed Kinase PIK3CD IC50 '>' 50000 nM
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Ki '>' 3162 nM
Q08881 BXGT013012 Tyrosine-protein kinase ITK/TSK reviewed Kinase ITK Ki '>' 1584 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Ki '>' 1258 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Kd '>' 10000 nM
P43403 BXGT010385 Tyrosine-protein kinase ZAP-70 reviewed Kinase ZAP70 Kd '>' 10000 nM
O95819 BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 Kd '>' 10000 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Ki '>' 7943 nM
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Kd - - -
P08922 BXGT006843 Proto-oncogene tyrosine-protein kinase ROS reviewed Kinase ROS1 Ki '>' 1995 nM
P08684 BXGT006812 Cytochrome P450 3A4 reviewed Enzyme CYP3A4 Activity - - -
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Kd '>' 10000 nM
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Kd '>' 10000 nM
P68400 BXGT011599 Casein kinase II subunit alpha reviewed Kinase CSNK2A1 Ki '>' 6309 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd '=' 5500 nM
Q8IVW4 BXGT018350 Cyclin-dependent kinase-like 3 reviewed Kinase CDKL3 Kd '>' 10000 nM
P30530 BXGT009431 Tyrosine-protein kinase receptor UFO reviewed Kinase AXL Kd '=' 1800 nM
P42679 BXGT010328 Megakaryocyte-associated tyrosine-protein kinase reviewed Kinase MATK Kd '>' 10000 nM
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Kd '>' 10000 nM
Q02763 BXGT012667 Angiopoietin-1 receptor reviewed Kinase TEK Kd - - -
Q9H2X6 BXGT020458 Homeodomain-interacting protein kinase 2 reviewed Kinase HIPK2 Ki '>' 3162 nM
P16234 BXGT008209 Platelet-derived growth factor receptor alpha reviewed Kinase PDGFRA Ki '>' 1995 nM
O94806 BXGT005335 Serine/threonine-protein kinase D3 reviewed Kinase PRKD3 Ki '=' 1258 nM
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Ki '>' 3981 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 35 %
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Kd '>' 10000 nM
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Kd '>' 10000 nM
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd '>' 10000 nM
O94768 BXGT005331 Serine/threonine-protein kinase 17B reviewed Kinase STK17B Kd '=' 3800 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 0 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 2 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 1 nM
Q8IVH8 BXGT018345 Mitogen-activated protein kinase kinase kinase kinase 3 reviewed Kinase MAP4K3 Kd '>' 10000 nM
Q9Y4K4 BXGT022282 Mitogen-activated protein kinase kinase kinase kinase 5 reviewed Kinase MAP4K5 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Ki '=' 3162 nM
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Ki '>' 10000 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Kd - - -
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Kd - - -
Q2M2I8 BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 Kd - - -
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Kd - - -
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd - - -
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Kd - - -
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Kd - - -
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Ki '>' 2511 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET IC50 '=' 1700 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 - - -
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Ki '=' 316 nM
P29597 BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 Ki '>' 1995 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Ki '>' 6309 nM
Q9ULC5 BXGT021758 Long-chain-fatty-acid--CoA ligase 5 reviewed Enzyme ACSL5 Kd apparent '>' 30000 nM
P31689 BXGT009569 DnaJ homolog subfamily A member 1 reviewed - DNAJA1 Kd apparent '>' 30000 nM
O14920 BXGT004110 Inhibitor of nuclear factor kappa-B kinase subunit beta reviewed Kinase IKBKB Kd '>' 10000 nM
Q9UK32 BXGT021736 Ribosomal protein S6 kinase alpha-6 reviewed Kinase RPS6KA6 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 93 %
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Kd apparent '>' 30000 nM
P12931 BXGT007859 Proto-oncogene tyrosine-protein kinase Src reviewed Kinase SRC Kd apparent '>' 30000 nM
P37173 BXGT009970 TGF-beta receptor type-2 reviewed Kinase TGFBR2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 80 nM
Q96PY6 BXGT019712 Serine/threonine-protein kinase Nek1 reviewed Kinase NEK1 Kd apparent '>' 30000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 1604 nM
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Kd '=' 1100 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd '>' 10000 nM
P32298 BXGT009617 G protein-coupled receptor kinase 4 reviewed Kinase GRK4 Kd '>' 10000 nM
Q9NSY1 BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K Kd '>' 10000 nM
Q56UN5 BXGT015107 Mitogen-activated protein kinase kinase kinase 19 reviewed Kinase MAP3K19 Kd '=' 240 nM
Q96Q40 BXGT019714 Cyclin-dependent kinase 15 reviewed Kinase CDK15 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 480 nM
Q9H422 BXGT020469 Homeodomain-interacting protein kinase 3 reviewed Kinase HIPK3 Kd '>' 10000 nM
P20794 BXGT008600 Serine/threonine-protein kinase MAK reviewed Kinase MAK Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 82 %
Q8N752 BXGT018526 Casein kinase I isoform alpha-like reviewed Kinase CSNK1A1L Kd '>' 10000 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Kd '>' 10000 nM
O95342 BXGT005373 Bile salt export pump reviewed Transporter ABCB11 IC50 '=' 10900 nM
Q9UNQ0 BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 IC50 '=' 1260 nM
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Ki '>' 2511 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR Inhibition '=' 6 %
P54646 BXGT011062 5'-AMP-activated protein kinase catalytic subunit alpha-2 reviewed Kinase PRKAA2 Kd '>' 10000 nM
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Kd '>' 10000 nM
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Inhibition '=' 46 %
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Inhibition '=' 46 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 70 nM
O15296 BXGT004148 Arachidonate 15-lipoxygenase B reviewed Enzyme ALOX15B Potency - 19952 nM
P53778 BXGT011013 Mitogen-activated protein kinase 12 reviewed Kinase MAPK12 Kd - - -
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Kd - - -
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Kd - - -
Q9UQB9 BXGT021810 Aurora kinase C reviewed Kinase AURKC Kd - - -
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd '>' 10000 nM
P07949 BXGT006703 Proto-oncogene tyrosine-protein kinase receptor Ret reviewed Kinase RET Ki '>' 1258 nM
Q9NYL2 BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 Ki '>' 7943 nM
P05129 BXGT006322 Protein kinase C gamma type reviewed Kinase PRKCG Ki '>' 7943 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd apparent '>' 30000 nM
P09769 BXGT006917 Tyrosine-protein kinase Fgr reviewed Kinase FGR Kd apparent '>' 30000 nM
Q6ZSR9 BXGT016637 Uncharacterized protein FLJ45252 reviewed - Kd apparent '>' 30000 nM
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Ki '>' 1995 nM
P06241 BXGT006429 Tyrosine-protein kinase Fyn reviewed Kinase FYN Ki '>' 794 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 4270 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 4270 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 4270 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 4270 nM
Q8TDC3 BXGT018808 Serine/threonine-protein kinase BRSK1 reviewed Kinase BRSK1 Kd '>' 10000 nM
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Kd '>' 10000 nM
Q6P3R8 BXGT016447 Serine/threonine-protein kinase Nek5 reviewed - NEK5 Kd '>' 10000 nM
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Kd apparent '>' 30000 nM
Q96GD4 BXGT019667 Aurora kinase B reviewed Kinase AURKB Kd apparent '>' 30000 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Inhibition '=' 46 %
Q02880 BXGT012677 DNA topoisomerase 2-beta reviewed - TOP2B Kd apparent '>' 30000 nM
P22234 BXGT008745 Multifunctional protein ADE2 reviewed Enzyme PAICS Kd apparent '>' 30000 nM
O75643 BXGT005142 U5 small nuclear ribonucleoprotein 200 kDa helicase reviewed - SNRNP200 Kd apparent '>' 30000 nM
O75496 BXGT005132 Geminin reviewed - GMNN Potency - 29855 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 7 nM
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Kd '>' 10000 nM
Q14164 BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE Kd '>' 10000 nM
P68370 BXGT011596 Tubulin alpha-1A chain reviewed - Tuba1a Kd '=' 410 nM
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Ki '>' 3981 nM
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Kd '>' 10000 nM
P29322 BXGT009333 Ephrin type-A receptor 8 reviewed Kinase EPHA8 Kd '=' 1800 nM
P51817 BXGT010895 cAMP-dependent protein kinase catalytic subunit PRKX reviewed Kinase PRKX Kd '>' 10000 nM
Q9UNQ0 BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 IC50 '=' 400 nM
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Ki '>' 7943 nM
P11799 BXGT007749 Myosin light chain kinase, smooth muscle reviewed - Mylk Kd '>' 10000 nM
P29323 BXGT009334 Ephrin type-B receptor 2 reviewed Kinase EPHB2 Kd '>' 10000 nM
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Ki '>' 1000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 832 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 832 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 832 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 832 nM
P15735 BXGT008151 Phosphorylase b kinase gamma catalytic chain, liver/testis isoform reviewed Kinase PHKG2 Kd '=' 2700 nM
Q86V86 BXGT017617 Serine/threonine-protein kinase pim-3 reviewed - PIM3 Kd '=' 5800 nM
Q8WU08 BXGT018990 Serine/threonine-protein kinase 32A reviewed Kinase STK32A Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1 nM
Q9BVS4 BXGT020147 Serine/threonine-protein kinase RIO2 reviewed Kinase RIOK2 Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 2900 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 4700 nM
Q12852 BXGT013272 Mitogen-activated protein kinase kinase kinase 12 reviewed Kinase MAP3K12 Kd '>' 10000 nM
P0C264 BXGT007408 Uncharacterized serine/threonine-protein kinase SBK3 reviewed - SBK3 Kd '>' 10000 nM
P62344 BXGT011426 Calcium-dependent protein kinase 1 reviewed - CPK1 Kd '>' 10000 nM
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Kd apparent '>' 30000 nM
O75716 BXGT005147 Serine/threonine-protein kinase 16 reviewed Kinase STK16 Thermal melting change '=' 3 degrees C
Q8TD19 BXGT018804 Serine/threonine-protein kinase Nek9 reviewed Kinase NEK9 Kd apparent '>' 30000 nM
P46734 BXGT010537 Dual specificity mitogen-activated protein kinase kinase 3 reviewed Kinase MAP2K3 Kd apparent '>' 30000 nM
Q01813 BXGT012618 ATP-dependent 6-phosphofructokinase, platelet type reviewed Kinase PFKP Kd apparent '>' 30000 nM
Q9H0A0 BXGT020434 RNA cytidine acetyltransferase reviewed - NAT10 Kd apparent '>' 30000 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Kd apparent '>' 30000 nM
Q13177 BXGT013323 Serine/threonine-protein kinase PAK 2 reviewed Kinase PAK2 Kd apparent '>' 30000 nM
P49589 BXGT010714 Cysteine--tRNA ligase, cytoplasmic reviewed Enzyme CARS1 Kd apparent '>' 30000 nM
P16591 BXGT008246 Tyrosine-protein kinase Fer reviewed Kinase FER Ki '>' 1584 nM
P53667 BXGT011008 LIM domain kinase 1 reviewed Kinase LIMK1 Kd apparent '>' 30000 nM
P42336 BXGT010302 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform reviewed Kinase PIK3CA IC50 - - -
P11473 BXGT007709 Vitamin D3 receptor reviewed Nuclear receptor VDR Potency - 89125 nM
P25098 BXGT009015 Beta-adrenergic receptor kinase 1 reviewed Kinase GRK2 Kd apparent '>' 30000 nM
P49411 BXGT010703 Elongation factor Tu, mitochondrial reviewed Enzyme TUFM Kd apparent '>' 30000 nM
Q9UM73 BXGT021773 ALK tyrosine kinase receptor reviewed Kinase ALK Ki '>' 1258 nM
P49748 BXGT010733 Very long-chain specific acyl-CoA dehydrogenase, mitochondrial reviewed Enzyme ACADVL Kd apparent '>' 30000 nM
P31751 BXGT009576 RAC-beta serine/threonine-protein kinase reviewed Kinase AKT2 Kd apparent '>' 30000 nM
O14578 BXGT004072 Citron Rho-interacting kinase reviewed Kinase CIT Kd apparent '>' 30000 nM
Q08345 BXGT012982 Epithelial discoidin domain-containing receptor 1 reviewed Kinase DDR1 Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 8 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 8 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 8 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 8 nM
Q16816 BXGT013673 Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform reviewed Kinase PHKG1 Kd - - -
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Kd - - -
P10721 BXGT007605 Mast/stem cell growth factor receptor Kit reviewed Kinase KIT Kd - - -
P25094 BXGT009014 Peripheral myelin protein 22 reviewed - Pmp22 Potency - 36125 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3100 nM
Q16832 BXGT013678 Discoidin domain-containing receptor 2 reviewed Kinase DDR2 Kd apparent '>' 30000 nM
Q05655 BXGT012832 Protein kinase C delta type reviewed Kinase PRKCD Kd apparent '>' 30000 nM
P54756 BXGT011074 Ephrin type-A receptor 5 reviewed Kinase EPHA5 Kd apparent '>' 30000 nM
Q9H2G2 BXGT020452 STE20-like serine/threonine-protein kinase reviewed Kinase SLK Kd apparent '>' 30000 nM
O75385 BXGT005121 Serine/threonine-protein kinase ULK1 reviewed Kinase ULK1 Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 22 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 22 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 22 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 22 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '>' 10000 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 11 nM
O75496 BXGT005132 Geminin reviewed - GMNN Potency - 13335 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 15 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 11 nM
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Ki '>' 2511 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 98 %
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Ki '>' 1584 nM
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Ki '>' 6309 nM
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Ki '>' 1258 nM
Q13237 BXGT013331 cGMP-dependent protein kinase 2 reviewed Kinase PRKG2 Ki '>' 1584 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Ki '>' 3981 nM
Q7Z406 BXGT017251 Myosin-14 reviewed - MYH14 Kd apparent '>' 30000 nM
Q92499 BXGT019350 ATP-dependent RNA helicase DDX1 reviewed - DDX1 Kd apparent '>' 30000 nM
P30085 BXGT009399 UMP-CMP kinase reviewed Kinase CMPK1 Kd apparent '>' 30000 nM
Q6ZN16 BXGT016630 Mitogen-activated protein kinase kinase kinase 15 reviewed - MAP3K15 Kd '>' 10000 nM
Q16288 BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 Kd '>' 10000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 3700 nM
Q13233 BXGT013330 Mitogen-activated protein kinase kinase kinase 1 reviewed Kinase MAP3K1 Kd '>' 10000 nM
Q9NRP7 BXGT021192 Serine/threonine-protein kinase 36 reviewed Kinase STK36 Kd '=' 5700 nM
P0C1S8 BXGT007404 Wee1-like protein kinase 2 reviewed - WEE2 Kd '>' 10000 nM
O14936 BXGT004114 Peripheral plasma membrane protein CASK reviewed Kinase CASK Kd '>' 10000 nM
Q9Y2K2 BXGT022238 Serine/threonine-protein kinase SIK3 reviewed Kinase SIK3 Kd '>' 10000 nM
P08581 BXGT006794 Hepatocyte growth factor receptor reviewed Kinase MET Kd '=' 3500 nM
P19784 BXGT008513 Casein kinase II subunit alpha' reviewed Kinase CSNK2A2 Kd '>' 10000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 Kd '=' 790 nM
Q9UBF8 BXGT021653 Phosphatidylinositol 4-kinase beta reviewed Kinase PI4KB Kd '>' 10000 nM
Q15139 BXGT013546 Serine/threonine-protein kinase D1 reviewed Kinase PRKD1 Kd '=' 3500 nM
O15264 BXGT004144 Mitogen-activated protein kinase 13 reviewed Kinase MAPK13 Kd '>' 10000 nM
O76039 BXGT005171 Cyclin-dependent kinase-like 5 reviewed Kinase CDKL5 Kd '>' 10000 nM
O15530 BXGT004177 3-phosphoinositide-dependent protein kinase 1 reviewed Kinase PDPK1 Thermal melting change '=' 0 degrees C
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Thermal melting change '=' 0 degrees C
P56817 BXGT011200 Beta-secretase 1 reviewed Enzyme BACE1 IC50 '=' 20000 nM
Q9HAZ1 BXGT020511 Dual specificity protein kinase CLK4 reviewed - CLK4 Ki '>' 6309 nM
Q9UBN7 BXGT021658 Histone deacetylase 6 reviewed Epigenetic regulator HDAC6 IC50 - - -
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 0 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 0 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 0 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1080 nM
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Ki '>' 5011 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 0 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 0 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 0 nM
Q06418 BXGT012875 Tyrosine-protein kinase receptor TYRO3 reviewed Kinase TYRO3 Ki '>' 1995 nM
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Ki '>' 6309 nM
P48736 BXGT010658 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform reviewed Kinase PIK3CG Kd '>' 10000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 3100 nM
O95747 BXGT005393 Serine/threonine-protein kinase OSR1 reviewed Kinase OXSR1 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 780 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 460 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 360 nM
Q9Y2U5 BXGT022248 Mitogen-activated protein kinase kinase kinase 2 reviewed Kinase MAP3K2 Kd '=' 3300 nM
O94921 BXGT005341 Cyclin-dependent kinase 14 reviewed Kinase CDK14 Kd '>' 10000 nM
Q9NRH2 BXGT021188 SNF-related serine/threonine-protein kinase reviewed Kinase SNRK Kd '>' 10000 nM
O14733 BXGT004087 Dual specificity mitogen-activated protein kinase kinase 7 reviewed Kinase MAP2K7 Kd '>' 10000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 62 nM
P52333 BXGT010928 Tyrosine-protein kinase JAK3 reviewed Kinase JAK3 IC50 '>' 1000 nM
P57078 BXGT011211 Receptor-interacting serine/threonine-protein kinase 4 reviewed Kinase RIPK4 Kd '>' 10000 nM
Q9H093 BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 Kd '=' 4600 nM
P9WI81 BXGT012312 Serine/threonine-protein kinase PknB reviewed - pknB Kd '>' 10000 nM
Q8NE63 BXGT018551 Homeodomain-interacting protein kinase 4 reviewed Kinase HIPK4 Kd '=' 310 nM
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Kd '>' 10000 nM
P61075 BXGT011353 Cell division control protein 2 homolog reviewed - CRK2 Kd '>' 10000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 173 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 173 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 173 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 173 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Kd apparent '>' 30000 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Ki '=' 794 nM
P29597 BXGT009367 Non-receptor tyrosine-protein kinase TYK2 reviewed Kinase TYK2 Kd apparent '>' 30000 nM
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 1013 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 1013 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1013 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 1013 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 - - -
Q04759 BXGT012781 Protein kinase C theta type reviewed Kinase PRKCQ Kd apparent '>' 30000 nM
Q7KZI7 BXGT016990 Serine/threonine-protein kinase MARK2 reviewed Kinase MARK2 Kd apparent '>' 30000 nM
Q96S44 BXGT019738 EKC/KEOPS complex subunit TP53RK reviewed Kinase TP53RK Kd apparent '>' 30000 nM
Q14004 BXGT013435 Cyclin-dependent kinase 13 reviewed Kinase CDK13 Kd '>' 10000 nM
P45983 BXGT010494 Mitogen-activated protein kinase 8 reviewed Kinase MAPK8 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 9 nM
Q9NU22 BXGT021214 Midasin reviewed - MDN1 Kd apparent '>' 30000 nM
Q15831 BXGT013604 Serine/threonine-protein kinase STK11 reviewed Kinase STK11 Kd apparent '>' 30000 nM
Q5S007 BXGT015650 Leucine-rich repeat serine/threonine-protein kinase 2 reviewed Kinase LRRK2 Ki '>' 2511 nM
Q14164 BXGT013451 Inhibitor of nuclear factor kappa-B kinase subunit epsilon reviewed Kinase IKBKE Ki '>' 3162 nM
Q9HBH9 BXGT020521 MAP kinase-interacting serine/threonine-protein kinase 2 reviewed Kinase MKNK2 Ki '=' 398 nM
P04629 BXGT006239 High affinity nerve growth factor receptor reviewed Kinase NTRK1 Ki '>' 2511 nM
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Kd '=' 69 nM
Q13233 BXGT013330 Mitogen-activated protein kinase kinase kinase 1 reviewed Kinase MAP3K1 Kd apparent '>' 30000 nM
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Inhibition '=' 46 %
Q14839 BXGT013509 Chromodomain-helicase-DNA-binding protein 4 reviewed - CHD4 Kd apparent '>' 30000 nM
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Ki '>' 1995 nM
Q9H3Y6 BXGT020468 Tyrosine-protein kinase Srms reviewed Kinase SRMS Ki '>' 1584 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Ki '=' 25 nM
P08631 BXGT006801 Tyrosine-protein kinase HCK reviewed Kinase HCK Kd apparent '>' 30000 nM
Q9UNQ0 BXGT021792 ATP-binding cassette sub-family G member 2 reviewed Transporter ABCG2 IC50 '=' 3190 nM
Q9NQU5 BXGT021169 Serine/threonine-protein kinase PAK 6 reviewed - PAK6 Thermal melting change '=' 0 degrees C
Q00536 BXGT012535 Cyclin-dependent kinase 16 reviewed Kinase CDK16 Thermal melting change '=' 0 degrees C
Q99986 BXGT019980 Serine/threonine-protein kinase VRK1 reviewed Kinase VRK1 Thermal melting change '=' 0 degrees C
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Inhibition - - -
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 IC50 '=' 1200 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 46 %
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Kd - - -
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Kd - - -
Q14012 BXGT013437 Calcium/calmodulin-dependent protein kinase type 1 reviewed Kinase CAMK1 Kd - - -
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 55 %
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 14 nM
Q13976 BXGT013409 cGMP-dependent protein kinase 1 reviewed Kinase PRKG1 Kd apparent '>' 30000 nM
Q13131 BXGT013314 5'-AMP-activated protein kinase catalytic subunit alpha-1 reviewed Kinase PRKAA1 Kd '>' 10000 nM
Q9UHD2 BXGT021697 Serine/threonine-protein kinase TBK1 reviewed Kinase TBK1 Kd apparent '>' 30000 nM
Q13464 BXGT013357 Rho-associated protein kinase 1 reviewed Kinase ROCK1 Kd apparent '>' 30000 nM
P20340 BXGT008566 Ras-related protein Rab-6A reviewed - RAB6A Kd apparent '>' 30000 nM
Q13554 BXGT013374 Calcium/calmodulin-dependent protein kinase type II subunit beta reviewed Kinase CAMK2B Thermal melting change '=' 0 degrees C
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Kd - - -
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Ki '>' 794 nM
Q00537 BXGT012536 Cyclin-dependent kinase 17 reviewed Kinase CDK17 Kd apparent '>' 30000 nM
P0A0J7 BXGT006970 Quinolone resistance protein NorA reviewed - norA FC '=' 16 -
Q9BUB5 BXGT020133 MAP kinase-interacting serine/threonine-protein kinase 1 reviewed Kinase MKNK1 Inhibition '=' 46 %
Q86XP3 BXGT017630 ATP-dependent RNA helicase DDX42 reviewed - DDX42 Kd apparent '>' 30000 nM
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1100 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 25 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 25 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 25 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 25 nM
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Kd apparent '>' 30000 nM
P26196 BXGT009089 Probable ATP-dependent RNA helicase DDX6 reviewed - DDX6 Kd apparent '>' 30000 nM
Q13164 BXGT013322 Mitogen-activated protein kinase 7 reviewed Kinase MAPK7 Kd apparent '>' 30000 nM
Q14683 BXGT013500 Structural maintenance of chromosomes protein 1A reviewed - SMC1A Kd apparent '>' 30000 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 76 nM
Q15418 BXGT013569 Ribosomal protein S6 kinase alpha-1 reviewed Kinase RPS6KA1 Kd apparent '>' 30000 nM
Q6PHR2 BXGT016467 Serine/threonine-protein kinase ULK3 reviewed Kinase ULK3 Kd apparent '>' 30000 nM
P42680 BXGT010329 Tyrosine-protein kinase Tec reviewed Kinase TEC Kd apparent '>' 30000 nM
Q00535 BXGT012534 Cyclin-dependent-like kinase 5 reviewed Kinase CDK5 Kd apparent '>' 30000 nM
Q86TW2 BXGT017609 Uncharacterized aarF domain-containing protein kinase 1 reviewed Kinase ADCK1 Kd apparent '>' 30000 nM
P49841 BXGT010750 Glycogen synthase kinase-3 beta reviewed Kinase GSK3B Thermal melting change '=' 0 degrees C
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Kd apparent '>' 30000 nM
Q05513 BXGT012820 Protein kinase C zeta type reviewed Kinase PRKCZ Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
O60674 BXGT004892 Tyrosine-protein kinase JAK2 reviewed Kinase JAK2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 6 nM
P45984 BXGT010495 Mitogen-activated protein kinase 9 reviewed Kinase MAPK9 Kd apparent '>' 30000 nM
P11216 BXGT007673 Glycogen phosphorylase, brain form reviewed Enzyme PYGB Kd apparent '>' 30000 nM
P51956 BXGT010909 Serine/threonine-protein kinase Nek3 reviewed Kinase NEK3 Kd apparent '>' 30000 nM
Q96RR4 BXGT019734 Calcium/calmodulin-dependent protein kinase kinase 2 reviewed Kinase CAMKK2 Kd apparent '>' 30000 nM
P08574 BXGT006792 Cytochrome c1, heme protein, mitochondrial reviewed - CYC1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 26 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Ki '=' 398 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Potency - 1729 nM
Q05397 BXGT012815 Focal adhesion kinase 1 reviewed Kinase PTK2 Ki '>' 1584 nM
P48730 BXGT010656 Casein kinase I isoform delta reviewed Kinase CSNK1D Kd apparent '>' 30000 nM
O00238 BXGT003900 Bone morphogenetic protein receptor type-1B reviewed Kinase BMPR1B Kd apparent '>' 30000 nM
Q13523 BXGT013368 Serine/threonine-protein kinase PRP4 homolog reviewed Kinase PRPF4B Kd '>' 10000 nM
O75676 BXGT005144 Ribosomal protein S6 kinase alpha-4 reviewed Kinase RPS6KA4 Kd '=' 1200 nM
O15197 BXGT004136 Ephrin type-B receptor 6 reviewed Kinase EPHB6 Kd '=' 3200 nM
O95382 BXGT005376 Mitogen-activated protein kinase kinase kinase 6 reviewed Kinase MAP3K6 Kd '>' 10000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 2200 nM
P42338 BXGT010303 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform reviewed Kinase PIK3CB Kd '>' 10000 nM
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Kd '>' 10000 nM
Q7L7X3 BXGT016997 Serine/threonine-protein kinase TAO1 reviewed Kinase TAOK1 Kd '>' 10000 nM
Q8NG66 BXGT018566 Serine/threonine-protein kinase Nek11 reviewed Kinase NEK11 Kd '>' 10000 nM
Q8IY84 BXGT018364 Serine/threonine-protein kinase NIM1 reviewed Kinase NIM1K Kd '>' 10000 nM
P04899 BXGT006281 Guanine nucleotide-binding protein G(i) subunit alpha-2 reviewed Enzyme modulator GNAI2 Kd apparent '>' 30000 nM
P16083 BXGT008187 Ribosyldihydronicotinamide dehydrogenase [quinone] reviewed - NQO2 Kd apparent '>' 30000 nM
Q16539 BXGT013634 Mitogen-activated protein kinase 14 reviewed Kinase MAPK14 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 140 nM
Q9BQI3 BXGT020113 Eukaryotic translation initiation factor 2-alpha kinase 1 reviewed Kinase EIF2AK1 Kd '>' 10000 nM
Q9NRM7 BXGT021190 Serine/threonine-protein kinase LATS2 reviewed Kinase LATS2 Kd '>' 10000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 100 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 100 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 100 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 100 nM
P17612 BXGT008322 cAMP-dependent protein kinase catalytic subunit alpha reviewed Kinase PRKACA Thermal melting change '=' 1 degrees C
Q9HC98 BXGT020528 Serine/threonine-protein kinase Nek6 reviewed Kinase NEK6 Thermal melting change '=' 0 degrees C
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Thermal melting change '=' 0 degrees C
O43293 BXGT004584 Death-associated protein kinase 3 reviewed Kinase DAPK3 Thermal melting change '=' 3 degrees C
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Thermal melting change '=' 0 degrees C
Q9BVS4 BXGT020147 Serine/threonine-protein kinase RIO2 reviewed Kinase RIOK2 Thermal melting change '=' 2 degrees C
Q15208 BXGT013550 Serine/threonine-protein kinase 38 reviewed Kinase STK38 Thermal melting change '=' 0 degrees C
Q86Y07 BXGT017631 Serine/threonine-protein kinase VRK2 reviewed Kinase VRK2 Thermal melting change '=' 0 degrees C
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 1000 nM
Q9NSY1 BXGT021209 BMP-2-inducible protein kinase reviewed Kinase BMP2K Kd apparent '>' 30000 nM
Q13555 BXGT013375 Calcium/calmodulin-dependent protein kinase type II subunit gamma reviewed Kinase CAMK2G Thermal melting change '=' 0 degrees C
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Thermal melting change '=' 0 degrees C
Q00532 BXGT012532 Cyclin-dependent kinase-like 1 reviewed Kinase CDKL1 Thermal melting change '=' 0 degrees C
Q13547 BXGT013373 Histone deacetylase 1 reviewed Epigenetic regulator HDAC1 IC50 - - -
Q01538 BXGT012597 Myelin transcription factor 1 reviewed Transcription factor MYT1 IC50 - - -
O43683 BXGT004614 Mitotic checkpoint serine/threonine-protein kinase BUB1 reviewed Kinase BUB1 Kd apparent '>' 30000 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Thermal melting change '=' 0 degrees C
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd '=' 5100 nM
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd '=' 2500 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd '=' 680 nM
O43318 BXGT004586 Mitogen-activated protein kinase kinase kinase 7 reviewed Kinase MAP3K7 Kd '>' 10000 nM
Q5VT25 BXGT015887 Serine/threonine-protein kinase MRCK alpha reviewed Kinase CDC42BPA Kd apparent '>' 30000 nM
P22694 BXGT008797 cAMP-dependent protein kinase catalytic subunit beta reviewed Kinase PRKACB Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 845 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 845 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 845 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 845 nM
P31153 BXGT009512 S-adenosylmethionine synthase isoform type-2 reviewed Enzyme MAT2A Kd apparent '>' 30000 nM
Q9BXA7 BXGT020164 Testis-specific serine/threonine-protein kinase 1 reviewed Kinase TSSK1B Ki '>' 1584 nM
O00311 BXGT003908 Cell division cycle 7-related protein kinase reviewed Kinase CDC7 Ki '>' 1258 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 '=' 48 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 65 %
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 24 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 127 nM
O96017 BXGT005415 Serine/threonine-protein kinase Chk2 reviewed Kinase CHEK2 Thermal melting change '=' 3 degrees C
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 127 nM
P30291 BXGT009417 Wee1-like protein kinase reviewed Kinase WEE1 Kd apparent '>' 30000 nM
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Thermal melting change '=' 0 degrees C
Q12851 BXGT013271 Mitogen-activated protein kinase kinase kinase kinase 2 reviewed Kinase MAP4K2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '>' 5000 nM
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Thermal melting change '=' 0 degrees C
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Thermal melting change '=' 0 degrees C
Q9P286 BXGT021299 Serine/threonine-protein kinase PAK 5 reviewed Kinase PAK5 Thermal melting change '=' 0 degrees C
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Thermal melting change '=' 0 degrees C
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Thermal melting change '=' 0 degrees C
P38117 BXGT010027 Electron transfer flavoprotein subunit beta reviewed Enzyme ETFB Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 6 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 6 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 6 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 6 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 3300 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 3300 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3300 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 3300 nM
Q9NUW8 BXGT021219 Tyrosyl-DNA phosphodiesterase 1 reviewed Enzyme TDP1 Potency - 5309 nM
Q96RG2 BXGT019726 PAS domain-containing serine/threonine-protein kinase reviewed Kinase PASK Kd apparent '>' 30000 nM
P12236 BXGT007775 ADP/ATP translocase 3 reviewed Transporter SLC25A6 Kd apparent '>' 30000 nM
Q16659 BXGT013652 Mitogen-activated protein kinase 6 reviewed Kinase MAPK6 Thermal melting change '=' 0 degrees C
P54577 BXGT011055 Tyrosine--tRNA ligase, cytoplasmic reviewed Enzyme YARS1 Kd apparent '>' 30000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 1830 nM
Q9NSE4 BXGT021207 Isoleucine--tRNA ligase, mitochondrial reviewed Enzyme IARS2 Kd apparent '>' 30000 nM
P11309 BXGT007685 Serine/threonine-protein kinase pim-1 reviewed Kinase PIM1 Thermal melting change '=' 3 degrees C
P52564 BXGT010932 Dual specificity mitogen-activated protein kinase kinase 6 reviewed Kinase MAP2K6 Thermal melting change '=' 0 degrees C
Q9HCP0 BXGT020536 Casein kinase I isoform gamma-1 reviewed Kinase CSNK1G1 Thermal melting change '=' 0 degrees C
P51955 BXGT010908 Serine/threonine-protein kinase Nek2 reviewed Kinase NEK2 Thermal melting change '=' 1 degrees C
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Thermal melting change '=' 1 degrees C
Q96NX5 BXGT019702 Calcium/calmodulin-dependent protein kinase type 1G reviewed Kinase CAMK1G Thermal melting change '=' 1 degrees C
Q8IU85 BXGT018333 Calcium/calmodulin-dependent protein kinase type 1D reviewed Kinase CAMK1D Thermal melting change '=' 0 degrees C
P24941 BXGT009002 Cyclin-dependent kinase 2 reviewed Kinase CDK2 Thermal melting change '=' 0 degrees C
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Thermal melting change '=' 1 degrees C
O00506 BXGT003932 Serine/threonine-protein kinase 25 reviewed Kinase STK25 Thermal melting change - - -
P42684 BXGT010331 Tyrosine-protein kinase ABL2 reviewed Kinase ABL2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 498 nM
P36894 BXGT009939 Bone morphogenetic protein receptor type-1A reviewed Kinase BMPR1A Kd apparent '>' 30000 nM
Q13705 BXGT013393 Activin receptor type-2B reviewed Kinase ACVR2B Kd apparent '>' 30000 nM
P07332 BXGT006601 Tyrosine-protein kinase Fes/Fps reviewed Kinase FES Kd apparent '>' 30000 nM
Q9Y6R4 BXGT022340 Mitogen-activated protein kinase kinase kinase 4 reviewed Kinase MAP3K4 Kd apparent '>' 30000 nM
P61026 BXGT011351 Ras-related protein Rab-10 reviewed - RAB10 Kd apparent '>' 30000 nM
Q15759 BXGT013595 Mitogen-activated protein kinase 11 reviewed Kinase MAPK11 Kd apparent '>' 30000 nM
P08069 BXGT006723 Insulin-like growth factor 1 receptor reviewed Kinase IGF1R Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 188 nM
Q14289 BXGT013459 Protein-tyrosine kinase 2-beta reviewed Kinase PTK2B Kd apparent '>' 30000 nM
Q09013 BXGT013023 Myotonin-protein kinase reviewed Kinase DMPK Thermal melting change '=' 3 degrees C
P41240 BXGT010242 Tyrosine-protein kinase CSK reviewed Kinase CSK Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 90 %
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 12720 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 12720 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 12720 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 12720 nM
Q9NYV4 BXGT021262 Cyclin-dependent kinase 12 reviewed Kinase CDK12 Kd apparent '>' 30000 nM
Q9Y2W1 BXGT022249 Thyroid hormone receptor-associated protein 3 reviewed Transcription factor THRAP3 Kd apparent '>' 30000 nM
P36888 BXGT009938 Receptor-type tyrosine-protein kinase FLT3 reviewed Kinase FLT3 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 66 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 28 %
Q9UF33 BXGT021676 Ephrin type-A receptor 6 reviewed Kinase EPHA6 Inhibition '=' 46 %
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Inhibition '=' 46 %
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Ki '>' 1584 nM
P31749 BXGT009574 RAC-alpha serine/threonine-protein kinase reviewed Kinase AKT1 Kd apparent '>' 30000 nM
Q13163 BXGT013321 Dual specificity mitogen-activated protein kinase kinase 5 reviewed Kinase MAP2K5 Kd apparent '>' 30000 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 10620 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 10620 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 10620 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 10620 nM
Q15067 BXGT013532 Peroxisomal acyl-coenzyme A oxidase 1 reviewed Enzyme ACOX1 Kd apparent '>' 30000 nM
Q99759 BXGT019960 Mitogen-activated protein kinase kinase kinase 3 reviewed Kinase MAP3K3 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
O95819 BXGT005398 Mitogen-activated protein kinase kinase kinase kinase 4 reviewed Kinase MAP4K4 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Ki '=' 0 nM
Q9Y6E0 BXGT022327 Serine/threonine-protein kinase 24 reviewed Kinase STK24 Kd apparent '>' 30000 nM
Q9Y2U5 BXGT022248 Mitogen-activated protein kinase kinase kinase 2 reviewed Kinase MAP3K2 Kd apparent '>' 30000 nM
Q04912 BXGT012790 Macrophage-stimulating protein receptor reviewed Kinase MST1R Kd apparent '>' 30000 nM
P41250 BXGT010244 Glycine--tRNA ligase reviewed Enzyme GARS1 Kd apparent '>' 30000 nM
Q13627 BXGT013385 Dual specificity tyrosine-phosphorylation-regulated kinase 1A reviewed Kinase DYRK1A Kd apparent '>' 30000 nM
Q9NTK5 BXGT021213 Obg-like ATPase 1 reviewed Enzyme modulator OLA1 Kd apparent '>' 30000 nM
P18074 BXGT008374 General transcription and DNA repair factor IIH helicase subunit XPD reviewed Enzyme ERCC2 Kd apparent '>' 30000 nM
O15439 BXGT004169 Multidrug resistance-associated protein 4 reviewed Transporter ABCC4 IC50 '=' 4600 nM
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Thermal melting change '=' 1 degrees C
Q8N4C8 BXGT018510 Misshapen-like kinase 1 reviewed Kinase MINK1 IC50 '=' 15000 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Inhibition '=' 46 %
Q8TDX7 BXGT018817 Serine/threonine-protein kinase Nek7 reviewed Kinase NEK7 Kd apparent '>' 30000 nM
Q02750 BXGT012662 Dual specificity mitogen-activated protein kinase kinase 1 reviewed Kinase MAP2K1 Kd apparent '>' 30000 nM
Q14680 BXGT013499 Maternal embryonic leucine zipper kinase reviewed Kinase MELK Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P51159 BXGT010839 Ras-related protein Rab-27A reviewed - RAB27A Kd apparent '>' 30000 nM
P43405 BXGT010386 Tyrosine-protein kinase SYK reviewed Kinase SYK Kd apparent '>' 30000 nM
P36507 BXGT009923 Dual specificity mitogen-activated protein kinase kinase 2 reviewed Kinase MAP2K2 Kd apparent '>' 30000 nM
P05771 BXGT006384 Protein kinase C beta type reviewed Kinase PRKCB Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 9 nM
Q9UHD8 BXGT021698 Septin-9 reviewed Enzyme modulator SEPTIN9 Kd apparent '>' 30000 nM
P06493 BXGT006445 Cyclin-dependent kinase 1 reviewed Kinase CDK1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR EC50 '=' 10733 nM
O14757 BXGT004092 Serine/threonine-protein kinase Chk1 reviewed Kinase CHEK1 Kd apparent '>' 30000 nM
P51617 BXGT010868 Interleukin-1 receptor-associated kinase 1 reviewed Kinase IRAK1 Kd apparent '>' 30000 nM
Q9H093 BXGT020433 NUAK family SNF1-like kinase 2 reviewed Kinase NUAK2 Kd apparent '>' 30000 nM
Q58FF8 BXGT015229 Putative heat shock protein HSP 90-beta 2 reviewed - HSP90AB2P Kd apparent '>' 30000 nM
P06239 BXGT006427 Tyrosine-protein kinase Lck reviewed Kinase LCK Kd apparent '>' 30000 nM
O00571 BXGT003938 ATP-dependent RNA helicase DDX3X reviewed - DDX3X Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 27 nM
P11388 BXGT007697 DNA topoisomerase 2-alpha reviewed - TOP2A Kd apparent '>' 30000 nM
Q8IYD1 BXGT018366 Eukaryotic peptide chain release factor GTP-binding subunit ERF3B reviewed Enzyme GSPT2 Kd apparent '>' 30000 nM
Q99683 BXGT019947 Mitogen-activated protein kinase kinase kinase 5 reviewed Kinase MAP3K5 Kd apparent '>' 30000 nM
P00519 BXGT005570 Tyrosine-protein kinase ABL1 reviewed Kinase ABL1 Kd apparent '>' 30000 nM
Q969S8 BXGT019613 Polyamine deacetylase HDAC10 reviewed Epigenetic regulator HDAC10 IC50 - - -
Q9UKV0 BXGT021750 Histone deacetylase 9 reviewed Epigenetic regulator HDAC9 IC50 - - -
P56524 BXGT011176 Histone deacetylase 4 reviewed Epigenetic regulator HDAC4 IC50 - - -
Q96DB2 BXGT019639 Histone deacetylase 11 reviewed Epigenetic regulator HDAC11 IC50 - - -
Q9BY41 BXGT020180 Histone deacetylase 8 reviewed Epigenetic regulator HDAC8 IC50 - - -
Q8WUI4 BXGT018992 Histone deacetylase 7 reviewed Epigenetic regulator HDAC7 IC50 - - -
Q9UQL6 BXGT021813 Histone deacetylase 5 reviewed Epigenetic regulator HDAC5 IC50 - - -
Q92769 BXGT019370 Histone deacetylase 2 reviewed Epigenetic regulator HDAC2 IC50 - - -
Q9UBN7 BXGT021658 Histone deacetylase 6 reviewed Epigenetic regulator HDAC6 IC50 - - -
O15379 BXGT004159 Histone deacetylase 3 reviewed Epigenetic regulator HDAC3 IC50 - - -
Q13547 BXGT013373 Histone deacetylase 1 reviewed Epigenetic regulator HDAC1 IC50 - - -
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 Kd '=' 10 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 Kd '=' 10 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd '=' 10 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 Kd '=' 10 nM
P21709 BXGT008685 Ephrin type-A receptor 1 reviewed Kinase EPHA1 Kd apparent '>' 30000 nM
P33991 BXGT009745 DNA replication licensing factor MCM4 reviewed Enzyme MCM4 Kd apparent '>' 30000 nM
O96013 BXGT005414 Serine/threonine-protein kinase PAK 4 reviewed Kinase PAK4 Kd apparent '>' 30000 nM
Q14004 BXGT013435 Cyclin-dependent kinase 13 reviewed Kinase CDK13 Kd apparent '>' 30000 nM
Q16288 BXGT013625 NT-3 growth factor receptor reviewed Kinase NTRK3 Ki '>' 1258 nM
Q06187 BXGT012860 Tyrosine-protein kinase BTK reviewed Kinase BTK Kd apparent '>' 30000 nM
Q01538 BXGT012597 Myelin transcription factor 1 reviewed Transcription factor MYT1 Activity '=' 6 %
P51812 BXGT010893 Ribosomal protein S6 kinase alpha-3 reviewed Kinase RPS6KA3 Kd apparent '>' 30000 nM
O94804 BXGT005334 Serine/threonine-protein kinase 10 reviewed Kinase STK10 Kd apparent '=' 5236 nM
Q15375 BXGT013562 Ephrin type-A receptor 7 reviewed Kinase EPHA7 Kd apparent '>' 30000 nM
P54753 BXGT011073 Ephrin type-B receptor 3 reviewed Kinase EPHB3 Kd apparent '>' 30000 nM
O60313 BXGT004871 Dynamin-like 120 kDa protein, mitochondrial reviewed Enzyme modulator OPA1 Kd apparent '>' 30000 nM
P49759 BXGT010734 Dual specificity protein kinase CLK1 reviewed Kinase CLK1 Kd apparent '>' 30000 nM
P49674 BXGT010725 Casein kinase I isoform epsilon reviewed - CSNK1E Kd apparent '>' 30000 nM
P43250 BXGT010372 G protein-coupled receptor kinase 6 reviewed Kinase GRK6 Kd apparent '>' 30000 nM
P54619 BXGT011060 5'-AMP-activated protein kinase subunit gamma-1 reviewed Kinase PRKAG1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 11 nM
P07948 BXGT006702 Tyrosine-protein kinase Lyn reviewed Kinase LYN Kd apparent '>' 30000 nM
Q9P289 BXGT021300 Serine/threonine-protein kinase 26 reviewed Kinase STK26 Kd apparent '>' 30000 nM
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF IC50 '=' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 7680 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 1 nM
Q16566 BXGT013639 Calcium/calmodulin-dependent protein kinase type IV reviewed Kinase CAMK4 Kd apparent '>' 30000 nM
P43686 BXGT010409 26S proteasome regulatory subunit 6B reviewed Enzyme PSMC4 Kd apparent '>' 30000 nM
P36896 BXGT009940 Activin receptor type-1B reviewed Kinase ACVR1B Kd apparent '>' 30000 nM
Q15569 BXGT013580 Dual specificity testis-specific protein kinase 1 reviewed Kinase TESK1 Kd apparent '>' 30000 nM
P06737 BXGT006492 Glycogen phosphorylase, liver form reviewed Enzyme PYGL Kd apparent '>' 30000 nM
Q13188 BXGT013324 Serine/threonine-protein kinase 3 reviewed Kinase STK3 Kd apparent '>' 30000 nM
P08240 BXGT006754 Signal recognition particle receptor subunit alpha reviewed Nucleic acid binding SRPRA Kd apparent '>' 30000 nM
Q9Y616 BXGT022313 Interleukin-1 receptor-associated kinase 3 reviewed Kinase IRAK3 Kd apparent '>' 30000 nM
P28482 BXGT009263 Mitogen-activated protein kinase 1 reviewed Kinase MAPK1 Kd apparent '>' 30000 nM
P49840 BXGT010749 Glycogen synthase kinase-3 alpha reviewed Kinase GSK3A Kd apparent '>' 30000 nM
P53779 BXGT011014 Mitogen-activated protein kinase 10 reviewed Kinase MAPK10 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 29 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 25 nM
P21860 BXGT008698 Receptor tyrosine-protein kinase erbB-3 reviewed Kinase ERBB3 IC50 '=' 6 nM
Q15303 BXGT013557 Receptor tyrosine-protein kinase erbB-4 reviewed Kinase ERBB4 IC50 '=' 6 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 6 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 '=' 6 nM
Q76MJ5 BXGT016871 Serine/threonine-protein kinase/endoribonuclease IRE2 reviewed Kinase ERN2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Kd apparent '=' 413 nM
O00329 BXGT003909 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform reviewed Kinase PIK3CD IC50 - - -
Q9Y6M4 BXGT022335 Casein kinase I isoform gamma-3 reviewed Kinase CSNK1G3 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 823 nM
P11362 BXGT007693 Fibroblast growth factor receptor 1 reviewed Kinase FGFR1 Kd apparent '>' 30000 nM
P10398 BXGT007564 Serine/threonine-protein kinase A-Raf reviewed Kinase ARAF Kd apparent '>' 30000 nM
Q8NI60 BXGT018572 Atypical kinase COQ8A, mitochondrial reviewed Kinase COQ8A Kd apparent '>' 30000 nM
Q3MIX3 BXGT014506 Uncharacterized aarF domain-containing protein kinase 5 reviewed - ADCK5 Kd apparent '>' 30000 nM
P49760 BXGT010735 Dual specificity protein kinase CLK2 reviewed Kinase CLK2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR EC50 '=' 2162 nM
Q9Y243 BXGT022214 RAC-gamma serine/threonine-protein kinase reviewed Kinase AKT3 Kd apparent '>' 30000 nM
P27707 BXGT009201 Deoxycytidine kinase reviewed Kinase DCK Kd apparent '>' 30000 nM
O75116 BXGT005100 Rho-associated protein kinase 2 reviewed Kinase ROCK2 Kd apparent '>' 30000 nM
P48426 BXGT010630 Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha reviewed Kinase PIP4K2A Kd apparent '>' 30000 nM
P23443 BXGT008866 Ribosomal protein S6 kinase beta-1 reviewed Kinase RPS6KB1 Kd apparent '>' 30000 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 Kd apparent '=' 903 nM
P07947 BXGT006701 Tyrosine-protein kinase Yes reviewed Kinase YES1 Kd apparent '>' 30000 nM
P78368 BXGT011840 Casein kinase I isoform gamma-2 reviewed Kinase CSNK1G2 Kd apparent '>' 30000 nM
Q9P0J0 BXGT021287 NADH dehydrogenase [ubiquinone] 1 alpha subcomplex subunit 13 reviewed Enzyme NDUFA13 Kd apparent '>' 30000 nM
Q13557 BXGT013376 Calcium/calmodulin-dependent protein kinase type II subunit delta reviewed Kinase CAMK2D Kd apparent '>' 30000 nM
P07741 BXGT006666 Adenine phosphoribosyltransferase reviewed - APRT Kd apparent '>' 30000 nM
P53350 BXGT010984 Serine/threonine-protein kinase PLK1 reviewed Kinase PLK1 Kd apparent '>' 30000 nM
Q9UPZ9 BXGT021804 Serine/threonine-protein kinase ICK reviewed Kinase CILK1 Kd apparent '>' 30000 nM
O00311 BXGT003908 Cell division cycle 7-related protein kinase reviewed Kinase CDC7 Kd apparent '>' 30000 nM
Q15392 BXGT013566 Delta(24)-sterol reductase reviewed Enzyme DHCR24 Kd apparent '>' 30000 nM
Q07912 BXGT012947 Activated CDC42 kinase 1 reviewed Kinase TNK2 IC50 '=' 2300 nM
P0A0J7 BXGT006970 Quinolone resistance protein NorA reviewed - norA FC '=' 8 -
Q04771 BXGT012783 Activin receptor type-1 reviewed Kinase ACVR1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '>' 1000 nM
Q9P1W9 BXGT021296 Serine/threonine-protein kinase pim-2 reviewed Kinase PIM2 Kd apparent '>' 30000 nM
Q9BZL6 BXGT020199 Serine/threonine-protein kinase D2 reviewed Kinase PRKD2 Kd apparent '>' 30000 nM
Q7RTN6 BXGT017085 STE20-related kinase adapter protein alpha reviewed Kinase STRADA Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 0 %
O75582 BXGT005137 Ribosomal protein S6 kinase alpha-5 reviewed Kinase RPS6KA5 Kd apparent '>' 30000 nM
Q9Y572 BXGT022289 Receptor-interacting serine/threonine-protein kinase 3 reviewed Kinase RIPK3 Kd apparent '=' 2664 nM
O95347 BXGT005374 Structural maintenance of chromosomes protein 2 reviewed - SMC2 Kd apparent '>' 30000 nM
Q9UL54 BXGT021755 Serine/threonine-protein kinase TAO2 reviewed Kinase TAOK2 Kd apparent '>' 30000 nM
Q709F0 BXGT016660 Acyl-CoA dehydrogenase family member 11 reviewed Enzyme ACAD11 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 129 nM
P35968 BXGT009887 Vascular endothelial growth factor receptor 2 reviewed Kinase KDR IC50 - - -
P35916 BXGT009881 Vascular endothelial growth factor receptor 3 reviewed Kinase FLT4 IC50 - - -
P17948 BXGT008358 Vascular endothelial growth factor receptor 1 reviewed Kinase FLT1 IC50 - - -
Q8IVH8 BXGT018345 Mitogen-activated protein kinase kinase kinase kinase 3 reviewed Kinase MAP4K3 Kd apparent '>' 30000 nM
P50750 BXGT010818 Cyclin-dependent kinase 9 reviewed Kinase CDK9 Kd apparent '>' 30000 nM
Q8TD08 BXGT018803 Mitogen-activated protein kinase 15 reviewed Kinase MAPK15 Kd apparent '>' 30000 nM
P54819 BXGT011084 Adenylate kinase 2, mitochondrial reviewed Kinase AK2 Kd apparent '>' 30000 nM
P15056 BXGT008075 Serine/threonine-protein kinase B-raf reviewed Kinase BRAF Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 10 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 96 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 0 nM
P42285 BXGT010297 Exosome RNA helicase MTR4 reviewed - MTREX Kd apparent '>' 30000 nM
P22830 BXGT008809 Ferrochelatase, mitochondrial reviewed Enzyme FECH Kd apparent '=' 6682 nM
P54764 BXGT011078 Ephrin type-A receptor 4 reviewed Kinase EPHA4 Kd apparent '>' 30000 nM
P06213 BXGT006425 Insulin receptor reviewed Kinase INSR Kd apparent '>' 30000 nM
Q9H2K8 BXGT020455 Serine/threonine-protein kinase TAO3 reviewed Kinase TAOK3 Kd apparent '>' 30000 nM
O00444 BXGT003921 Serine/threonine-protein kinase PLK4 reviewed Kinase PLK4 Kd apparent '>' 30000 nM
Q9UBE8 BXGT021652 Serine/threonine-protein kinase NLK reviewed Kinase NLK Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '>' 2000 nM
P29317 BXGT009331 Ephrin type-A receptor 2 reviewed Kinase EPHA2 Kd apparent '>' 30000 nM
P36897 BXGT009941 TGF-beta receptor type-1 reviewed Kinase TGFBR1 Kd apparent '>' 30000 nM
Q9NYL2 BXGT021259 Mitogen-activated protein kinase kinase kinase 20 reviewed Kinase MAP3K20 Kd apparent '>' 30000 nM
P61160 BXGT011365 Actin-related protein 2 reviewed Cellular structure ACTR2 Kd apparent '>' 30000 nM
Q9BQI3 BXGT020113 Eukaryotic translation initiation factor 2-alpha kinase 1 reviewed Kinase EIF2AK1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 280 nM
P62826 BXGT011463 GTP-binding nuclear protein Ran reviewed Enzyme modulator RAN Kd apparent '>' 30000 nM
Q8IW41 BXGT018352 MAP kinase-activated protein kinase 5 reviewed Kinase MAPKAPK5 Kd apparent '>' 30000 nM
O95835 BXGT005400 Serine/threonine-protein kinase LATS1 reviewed Kinase LATS1 Kd apparent '>' 30000 nM
Q13043 BXGT013307 Serine/threonine-protein kinase 4 reviewed Kinase STK4 Kd apparent '>' 30000 nM
P48729 BXGT010655 Casein kinase I isoform alpha reviewed Kinase CSNK1A1 Kd apparent '>' 30000 nM
P04626 BXGT006238 Receptor tyrosine-protein kinase erbB-2 reviewed Kinase ERBB2 IC50 - - -
P45985 BXGT010496 Dual specificity mitogen-activated protein kinase kinase 4 reviewed Kinase MAP2K4 Kd apparent '>' 30000 nM
P42345 BXGT010304 Serine/threonine-protein kinase mTOR reviewed Kinase MTOR Kd '>' 10000 nM
Q8TDR2 BXGT018811 Serine/threonine-protein kinase 35 reviewed Kinase STK35 Kd '>' 10000 nM
Q9UKE5 BXGT021741 TRAF2 and NCK-interacting protein kinase reviewed Kinase TNIK Kd '=' 6900 nM
Q86Z02 BXGT017638 Homeodomain-interacting protein kinase 1 reviewed Kinase HIPK1 Kd '>' 10000 nM
Q6XUX3 BXGT016612 Dual serine/threonine and tyrosine protein kinase reviewed Kinase DSTYK Kd '>' 10000 nM
P61158 BXGT011364 Actin-related protein 3 reviewed Cellular structure ACTR3 Kd apparent '>' 30000 nM
Q92918 BXGT019394 Mitogen-activated protein kinase kinase kinase kinase 1 reviewed Kinase MAP4K1 Kd apparent '>' 30000 nM
P22612 BXGT008785 cAMP-dependent protein kinase catalytic subunit gamma reviewed Kinase PRKACG Kd apparent '>' 30000 nM
Q13882 BXGT013399 Protein-tyrosine kinase 6 reviewed Kinase PTK6 IC50 '=' 980 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 88 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 99 %
Q9NSD9 BXGT021206 Phenylalanine--tRNA ligase beta subunit reviewed Enzyme FARSB Kd apparent '>' 30000 nM
P48736 BXGT010658 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform reviewed Kinase PIK3CG IC50 - - -
Q13873 BXGT013398 Bone morphogenetic protein receptor type-2 reviewed Kinase BMPR2 Kd apparent '>' 30000 nM
Q16512 BXGT013631 Serine/threonine-protein kinase N1 reviewed Kinase PKN1 Kd apparent '>' 30000 nM
O43353 BXGT004589 Receptor-interacting serine/threonine-protein kinase 2 reviewed Kinase RIPK2 IC50 '=' 3 nM
Q9H0K1 BXGT020438 Serine/threonine-protein kinase SIK2 reviewed Kinase SIK2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 3 %
Q9H773 BXGT020489 dCTP pyrophosphatase 1 reviewed - DCTPP1 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 22800 nM
Q00534 BXGT012533 Cyclin-dependent kinase 6 reviewed Kinase CDK6 Kd apparent '>' 30000 nM
Q2M2I8 BXGT014130 AP2-associated protein kinase 1 reviewed Kinase AAK1 Kd apparent '>' 30000 nM
P30519 BXGT009429 Heme oxygenase 2 reviewed - HMOX2 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 3 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2 nM
O15438 BXGT004168 Canalicular multispecific organic anion transporter 2 reviewed Transporter ABCC3 IC50 '=' 133000 nM
P54760 BXGT011075 Ephrin type-B receptor 4 reviewed Kinase EPHB4 Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 12 nM
Q9Y5S2 BXGT022301 Serine/threonine-protein kinase MRCK beta reviewed Kinase CDC42BPB Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR Inhibition '=' 77 %
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR IC50 '=' 2874 nM
Q6JQN1 BXGT016338 Acyl-CoA dehydrogenase family member 10 reviewed Enzyme ACAD10 Kd apparent '=' 33795 nM
Q6P5Z2 BXGT016454 Serine/threonine-protein kinase N3 reviewed Kinase PKN3 Kd apparent '>' 30000 nM
Q9BZE4 BXGT020197 Nucleolar GTP-binding protein 1 reviewed - GTPBP4 Kd apparent '>' 30000 nM
P42338 BXGT010303 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform reviewed Kinase PIK3CB IC50 - - -
P55263 BXGT011115 Adenosine kinase reviewed Kinase ADK Kd apparent '>' 30000 nM
P00533 BXGT005575 Epidermal growth factor receptor reviewed Kinase EGFR TIME '<' 0 hr
Foods  containing  the  compound
Foods
BXGF Id Food Name Scientific Name Food Group
BXGF Id Food Name Scientific Name Food Group
BXGF01386 Asarum heterotropoides Asarum heterotropoides Others
BXGF05627 Asarum sieboldii Asarum sieboldii Medicinal Plant
The  compound-realted  diseases
Diseases
BXGD Id Disease Name CUI Disease Id Disease Class Name Number of targets?Number of targets related to compound connecting disease, higher numbers indicate the compound is more associated with the disease